| 0.438438 |
4.572504e-47 |
975 |
Cobalt (Ii) Chloride |
LSM-5958 |
HIF1A |
10uM |
6h |
LINCSCP_17021 |
LINCSCP_17021 |
HA1E |
| 0.429537 |
4.787897e-45 |
975 |
VE-821 |
LSM-36358 |
|
1.11uM |
24h |
LINCSCP_83660 |
LINCSCP_83660 |
ASC.C |
| 0.415123 |
6.694157e-42 |
975 |
AC1Q5RFA |
LSM-43063 |
|
0.37uM |
24h |
LINCSCP_74821 |
LINCSCP_74821 |
A375 |
| 0.410455 |
6.488781e-41 |
975 |
BRD-K49553303-001-01-8 |
LSM-40022 |
|
10uM |
6h |
LINCSCP_16844 |
LINCSCP_16844 |
HA1E |
| 0.407862 |
2.255472e-40 |
975 |
CBKINASE1_008949 |
LSM-4513 |
|
10uM |
6h |
LINCSCP_22297 |
LINCSCP_22297 |
HEPG2 |
| 0.406952 |
3.484623e-40 |
975 |
BRD-K22013971 |
LSM-9761 |
|
5uM |
24h |
LINCSCP_62262 |
LINCSCP_62262 |
VCAP |
| 0.399104 |
1.400155e-38 |
975 |
BRD-K45758869-001-01-3 |
LSM-39802 |
|
10uM |
6h |
LINCSCP_212182 |
LINCSCP_212182 |
HA1E |
| 0.397207 |
3.369225e-38 |
975 |
BRD-K19593010 |
LSM-38322 |
|
10uM |
6h |
LINCSCP_16793 |
LINCSCP_16793 |
HA1E |
| 0.392695 |
2.659003e-37 |
975 |
Cytarabine |
LSM-5470 |
POLA1|POLB|POLD1|POLE |
1.11uM |
24h |
LINCSCP_74126 |
LINCSCP_74126 |
A375 |
| -0.391768 |
4.048103e-37 |
975 |
BRD-A80960055-001-01-7 |
LSM-5162 |
|
10uM |
6h |
LINCSCP_32631 |
LINCSCP_32631 |
MCF7 |
| 0.388916 |
1.463677e-36 |
975 |
FPA1_000240 |
LSM-36679 |
|
10uM |
6h |
LINCSCP_22353 |
LINCSCP_22353 |
HEPG2 |
| 0.386073 |
5.204788e-36 |
975 |
AG-205/40776311 |
LSM-4736 |
|
10uM |
6h |
LINCSCP_22426 |
LINCSCP_22426 |
HEPG2 |
| 0.382394 |
2.637945e-35 |
975 |
SCHEMBL15556278 |
LSM-1002 |
DDR1 |
10uM |
6h |
LINCSCP_22404 |
LINCSCP_22404 |
HEPG2 |
| -0.376382 |
3.580890e-34 |
975 |
MLS000564806 |
LSM-4368 |
|
10uM |
6h |
LINCSCP_218435 |
LINCSCP_218435 |
HCT116 |
| 0.375563 |
5.086809e-34 |
975 |
BRD-K99115033 |
LSM-14515 |
|
5uM |
24h |
LINCSCP_61856 |
LINCSCP_61856 |
VCAP |
| 0.374289 |
8.763524e-34 |
975 |
STK568087 |
LSM-4669 |
|
10uM |
6h |
LINCSCP_22381 |
LINCSCP_22381 |
HEPG2 |
| 0.370829 |
3.794925e-33 |
975 |
MEGXP0_001030 |
LSM-4462 |
|
10uM |
6h |
LINCSCP_22289 |
LINCSCP_22289 |
HEPG2 |
| 0.370474 |
4.406480e-33 |
975 |
Atomoxetine |
LSM-2452 |
SLC6A2|SLC6A3|SLC6A4 |
10uM |
24h |
LINCSCP_242049 |
LINCSCP_242049 |
MCF7 |
| -0.37043 |
4.488950e-33 |
975 |
BRD-K72490684 |
LSM-41201 |
|
5uM |
6h |
LINCSCP_4113 |
LINCSCP_4113 |
A375 |
| 0.370396 |
4.553074e-33 |
975 |
Alaproclate |
LSM-1333 |
SLC6A4 |
0.12uM |
24h |
LINCSCP_74486 |
LINCSCP_74486 |
A375 |
| 0.369623 |
6.299551e-33 |
975 |
CID 75060947 |
LSM-36700 |
|
10uM |
6h |
LINCSCP_16329 |
LINCSCP_16329 |
HA1E |
| 0.369451 |
6.768602e-33 |
975 |
ZINC00399124 |
LSM-5611 |
|
10uM |
6h |
LINCSCP_16972 |
LINCSCP_16972 |
HA1E |
| 0.366678 |
2.150571e-32 |
975 |
Suprofen |
LSM-4406 |
PTGS1|PTGS2 |
3.33uM |
24h |
LINCSCP_135405 |
LINCSCP_135405 |
MCF7 |
| 0.365601 |
3.360240e-32 |
975 |
BRD-K00695053 |
LSM-8478 |
|
5uM |
24h |
LINCSCP_61931 |
LINCSCP_61931 |
VCAP |
| 0.365495 |
3.510298e-32 |
975 |
Erlotinib |
LSM-1097 |
EGFR |
0.12uM |
3h |
LINCSCP_163413 |
LINCSCP_163413 |
SKBR3 |
| 0.365177 |
4.003396e-32 |
975 |
SCHEMBL13991002 |
LSM-6278 |
|
40uM |
6h |
LINCSCP_10438 |
LINCSCP_10438 |
A673 |
| 0.363928 |
6.693471e-32 |
975 |
Cyclacillin |
LSM-3987 |
|
10uM |
24h |
LINCSCP_52668 |
LINCSCP_52668 |
SKB |
| 0.363466 |
8.094380e-32 |
975 |
CHEMBL2135537 |
LSM-6149 |
|
10uM |
6h |
LINCSCP_16879 |
LINCSCP_16879 |
HA1E |
| 0.36194 |
1.510703e-31 |
975 |
Lapatinib |
LSM-1051 |
EGFR|ERBB2 |
10uM |
3h |
LINCSCP_145915 |
LINCSCP_145915 |
MDAMB231 |
| 0.360551 |
2.658580e-31 |
975 |
Crizotinib |
LSM-1027 |
ALK|MET |
0.37uM |
24h |
LINCSCP_99369 |
LINCSCP_99369 |
HCC515 |
| 0.359119 |
4.748487e-31 |
975 |
Idelalisib |
LSM-1205 |
PIK3CD|PIK3CG |
10uM |
24h |
LINCSCP_129697 |
LINCSCP_129697 |
JURKAT |
| -0.358867 |
5.256921e-31 |
975 |
nifedipine |
LSM-4176 |
CACNA1C|CACNA1D|CACNA1F|CACNA1S|CACNA2D1 |
10uM |
24h |
LINCSCP_46055 |
LINCSCP_46055 |
PC3 |
| 0.358064 |
7.264932e-31 |
975 |
Imatinib |
LSM-1023 |
ABL1|BCR|CSF1R|KIT|PDGFRA|PDGFRB |
0.12uM |
3h |
LINCSCP_130378 |
LINCSCP_130378 |
LNCAP |
| -0.356499 |
1.361166e-30 |
975 |
BRD-K99171789 |
LSM-8095 |
|
5uM |
24h |
LINCSCP_60103 |
LINCSCP_60103 |
VCAP |
| 0.355367 |
2.139856e-30 |
975 |
Tripelennamine |
LSM-3271 |
HRH1 |
10uM |
6h |
LINCSCP_225748 |
LINCSCP_225748 |
HT29 |
| 0.355291 |
2.205395e-30 |
975 |
Methyl 1-hydroxy-7-(hydroxymethyl)-1,4a,5,7a-tetrahydrocyclopenta[c]pyran-4-carboxylate |
LSM-4955 |
|
10uM |
6h |
LINCSCP_16919 |
LINCSCP_16919 |
HA1E |
| -0.354711 |
2.777345e-30 |
975 |
Temoporfin |
LSM-45995 |
|
10uM |
24h |
LINCSCP_155235 |
LINCSCP_155235 |
PC3 |
| 0.351712 |
9.093346e-30 |
975 |
HG6-64-1 |
LSM-43248 |
|
0.1uM |
24h |
LINCSCP_11850 |
LINCSCP_11850 |
BT20 |
| -0.351318 |
1.061639e-29 |
975 |
SCHEMBL2231351 |
LSM-36442 |
|
0.001uM |
24h |
LINCSCP_41941 |
LINCSCP_41941 |
NOMO1 |
| 0.350769 |
1.317077e-29 |
975 |
BRD-K30794866 |
LSM-10284 |
|
5uM |
24h |
LINCSCP_63361 |
LINCSCP_63361 |
VCAP |
| 0.350349 |
1.552523e-29 |
975 |
XAV 939 |
LSM-5303 |
TNKS|TNKS2 |
10uM |
6h |
LINCSCP_55453 |
LINCSCP_55453 |
U937 |
| 0.349448 |
2.207482e-29 |
975 |
YL-53 |
LSM-44644 |
|
10uM |
6h |
LINCSCP_16970 |
LINCSCP_16970 |
HA1E |
| 0.34901 |
2.618336e-29 |
975 |
BRD-K45735142 |
LSM-6782 |
|
10uM |
6h |
LINCSCP_16832 |
LINCSCP_16832 |
HA1E |
| 0.348814 |
2.825875e-29 |
975 |
BRD-K35868313 |
LSM-10582 |
|
5uM |
24h |
LINCSCP_62278 |
LINCSCP_62278 |
VCAP |
| 0.348741 |
2.907972e-29 |
975 |
BRD-K48598367 |
LSM-11388 |
|
5uM |
24h |
LINCSCP_63091 |
LINCSCP_63091 |
VCAP |
| 0.348421 |
3.293307e-29 |
975 |
SUGA1_008424 |
LSM-36671 |
|
10uM |
6h |
LINCSCP_22349 |
LINCSCP_22349 |
HEPG2 |
| 0.348204 |
3.582879e-29 |
975 |
BRD-K39504007 |
LSM-10828 |
|
5uM |
24h |
LINCSCP_62282 |
LINCSCP_62282 |
VCAP |
| 0.348104 |
3.724515e-29 |
975 |
SMR000178575 |
LSM-2708 |
|
10uM |
6h |
LINCSCP_16634 |
LINCSCP_16634 |
HA1E |
| 0.348055 |
3.796347e-29 |
975 |
BRD-K17686770 |
LSM-9493 |
|
5uM |
6h |
LINCSCP_62512 |
LINCSCP_62512 |
VCAP |
| 0.347319 |
5.048544e-29 |
975 |
Ticrynafen |
LSM-5478 |
CYP2C9|SLC12A1 |
10uM |
6h |
LINCSCP_16957 |
LINCSCP_16957 |
HA1E |
| 0.346314 |
7.444423e-29 |
975 |
MLS002699918 |
LSM-2263 |
|
10uM |
6h |
LINCSCP_32029 |
LINCSCP_32029 |
MCF7 |
| 0.345993 |
8.428084e-29 |
975 |
Raltitrexed |
LSM-5952 |
TYMS |
10uM |
6h |
LINCSCP_22438 |
LINCSCP_22438 |
HEPG2 |
| 0.34565 |
9.617749e-29 |
975 |
SCHEMBL6468298 |
LSM-6130 |
|
10uM |
6h |
LINCSCP_16321 |
LINCSCP_16321 |
HA1E |
| 0.345213 |
1.137685e-28 |
975 |
BRD-K41431262 |
LSM-39564 |
|
10uM |
6h |
LINCSCP_27315 |
LINCSCP_27315 |
HT29 |
| 0.344822 |
1.321833e-28 |
975 |
Pirenzepine |
LSM-4001 |
CHRM1 |
10uM |
24h |
LINCSCP_32937 |
LINCSCP_32937 |
MCF7 |
| -0.34481 |
1.327850e-28 |
975 |
Auranofin |
LSM-43136 |
|
10uM |
6h |
LINCSCP_4679 |
LINCSCP_4679 |
A549 |
| 0.343183 |
2.474629e-28 |
975 |
BIM0133 |
LSM-5621 |
|
10uM |
6h |
LINCSCP_16975 |
LINCSCP_16975 |
HA1E |
| -0.34311 |
2.544253e-28 |
975 |
GLPG0634 |
LSM-45924 |
JAK1 |
0.12uM |
24h |
LINCSCP_153233 |
LINCSCP_153233 |
PC3 |
| 0.341296 |
5.068742e-28 |
975 |
Triacsin C |
LSM-43284 |
ACSL1 |
10uM |
6h |
LINCSCP_55538 |
LINCSCP_55538 |
U937 |
| 0.340422 |
7.052695e-28 |
975 |
Alpelisib |
LSM-4256 |
PIK3CA |
0.37uM |
3h |
LINCSCP_145218 |
LINCSCP_145218 |
MDAMB231 |
| 0.340409 |
7.088225e-28 |
975 |
BRD-K33994902 |
LSM-10485 |
|
5uM |
24h |
LINCSCP_63364 |
LINCSCP_63364 |
VCAP |
| 0.340404 |
7.101246e-28 |
975 |
Imatinib |
LSM-1023 |
ABL1|BCR|CSF1R|KIT|PDGFRA|PDGFRB |
10uM |
3h |
LINCSCP_145933 |
LINCSCP_145933 |
MDAMB231 |
| -0.339978 |
8.340106e-28 |
975 |
STK249718 |
LSM-6671 |
|
3uM |
6h |
LINCSCP_23731 |
LINCSCP_23731 |
HEPG2 |
| -0.339955 |
8.413416e-28 |
975 |
Mebendazole |
LSM-3749 |
|
40uM |
24h |
LINCSCP_67596 |
LINCSCP_67596 |
MCF7 |
| -0.339738 |
9.128669e-28 |
975 |
SCHEMBL2231351 |
LSM-36442 |
|
0.001uM |
24h |
LINCSCP_55074 |
LINCSCP_55074 |
THP1 |
| 0.339484 |
1.004416e-27 |
975 |
MEGXP0_001444 |
LSM-4390 |
|
10uM |
6h |
LINCSCP_22280 |
LINCSCP_22280 |
HEPG2 |
| 0.33939 |
1.040587e-27 |
975 |
BRD-K31427141 |
LSM-10333 |
|
5uM |
24h |
LINCSCP_305786 |
LINCSCP_305786 |
VCAP |
| 0.339005 |
1.202506e-27 |
975 |
BRD-K99395085 |
LSM-42650 |
|
5uM |
24h |
LINCSCP_64344 |
LINCSCP_64344 |
VCAP |
| 0.338328 |
1.550602e-27 |
975 |
BRD-K73400194 |
LSM-12924 |
|
5uM |
24h |
LINCSCP_62031 |
LINCSCP_62031 |
VCAP |
| -0.338251 |
1.595940e-27 |
975 |
Wortmannin |
LSM-3947 |
PIK3CA|PIK3CG|PLK1 |
1uM |
24h |
LINCSCP_24123 |
LINCSCP_24123 |
HL60 |
| 0.338063 |
1.712426e-27 |
975 |
PH-797804 |
LSM-36373 |
MAPK14 |
0.04uM |
24h |
LINCSCP_162211 |
LINCSCP_162211 |
PC3 |
| 0.337086 |
2.466648e-27 |
975 |
BRD-K30802967 |
LSM-6102 |
|
10uM |
6h |
LINCSCP_16808 |
LINCSCP_16808 |
HA1E |
| 0.337074 |
2.477195e-27 |
975 |
BRD-K99756483 |
LSM-42675 |
|
10uM |
6h |
LINCSCP_16917 |
LINCSCP_16917 |
HA1E |
| -0.33673 |
2.816842e-27 |
975 |
BRD-A24396574-001-01-5 |
LSM-5006 |
|
10uM |
3h |
LINCSCP_113445 |
LINCSCP_113445 |
HME1 |
| 0.33598 |
3.722433e-27 |
975 |
SPOX1_001033 |
LSM-4552 |
|
10uM |
6h |
LINCSCP_22324 |
LINCSCP_22324 |
HEPG2 |
| 0.335214 |
4.945233e-27 |
975 |
BRD-K84120458 |
LSM-13571 |
|
5uM |
6h |
LINCSCP_62587 |
LINCSCP_62587 |
VCAP |
| 0.335057 |
5.240879e-27 |
975 |
GW7647 |
LSM-4172 |
PPARA |
10uM |
24h |
LINCSCP_240734 |
LINCSCP_240734 |
MCF7 |
| 0.334655 |
6.082334e-27 |
975 |
BRD-K21994180 |
LSM-38461 |
|
30uM |
6h |
LINCSCP_310118 |
LINCSCP_310118 |
VCAP |
| 0.334307 |
6.917234e-27 |
975 |
BRD-K78496556 |
LSM-41553 |
|
10uM |
6h |
LINCSCP_48892 |
LINCSCP_48892 |
PC3 |
| -0.333809 |
8.310766e-27 |
975 |
Tacedinaline |
LSM-19036 |
HDAC1|HDAC10|HDAC11|HDAC2|HDAC3|HDAC4|HDAC5|HDAC6|HDAC7|HDAC8|HDAC9 |
0.1uM |
24h |
LINCSCP_49312 |
LINCSCP_49312 |
PC3 |
| 0.333549 |
9.145011e-27 |
975 |
BRD-K34412705 |
LSM-39151 |
|
10uM |
6h |
LINCSCP_34010 |
LINCSCP_34010 |
MCF7 |
| 0.333323 |
9.937777e-27 |
975 |
Iloperidone |
LSM-5598 |
DRD2|HTR1A|HTR2A|HTR6|HTR7 |
10uM |
6h |
LINCSCP_20457 |
LINCSCP_20457 |
HCC515 |
| -0.3333 |
1.002195e-26 |
975 |
MLS-0315868.0001 |
LSM-4861 |
|
10uM |
6h |
LINCSCP_20353 |
LINCSCP_20353 |
HCC515 |
| 0.332501 |
1.344380e-26 |
975 |
MK-5172 |
LSM-45592 |
|
0.12uM |
24h |
LINCSCP_72379 |
LINCSCP_72379 |
A375 |
| -0.330596 |
2.695934e-26 |
975 |
SA-1939938 |
LSM-37441 |
|
1uM |
24h |
LINCSCP_41626 |
LINCSCP_41626 |
NKDBA |
| 0.329958 |
3.400120e-26 |
975 |
Emtricitabine |
LSM-45730 |
|
0.37uM |
24h |
LINCSCP_123286 |
LINCSCP_123286 |
HT29 |
| -0.32984 |
3.549181e-26 |
975 |
Metoprolol |
LSM-1259 |
ADRB1|ADRB2 |
10uM |
24h |
LINCSCP_52792 |
LINCSCP_52792 |
SKB |
| 0.329577 |
3.905384e-26 |
975 |
Cholic acid |
LSM-5541 |
CES1|FECH|PLA2G1B |
10uM |
24h |
LINCSCP_75554 |
LINCSCP_75554 |
A375 |
| 0.329435 |
4.111139e-26 |
975 |
noscapine |
|
|
10uM |
3h |
LINCSCP_133163 |
LINCSCP_133163 |
MCF7 |
| 0.328386 |
6.009967e-26 |
975 |
Genistein |
LSM-5549 |
CFTR|ESR2 |
10uM |
6h |
LINCSCP_211781 |
LINCSCP_211781 |
HA1E |
| 0.328319 |
6.155469e-26 |
975 |
CHEMBL2355186 |
LSM-8441 |
|
5uM |
24h |
LINCSCP_62427 |
LINCSCP_62427 |
VCAP |
| 0.327502 |
8.264670e-26 |
975 |
AC1O9B20 |
LSM-4696 |
|
10uM |
6h |
LINCSCP_20134 |
LINCSCP_20134 |
HCC515 |
| -0.326894 |
1.028359e-25 |
975 |
STK249718 |
LSM-6671 |
|
10uM |
6h |
LINCSCP_23730 |
LINCSCP_23730 |
HEPG2 |
| 0.326697 |
1.103613e-25 |
975 |
Verapamil |
LSM-1298 |
CACNA1C|CACNA1D|CACNA1F|CACNA1G|CACNA1S |
10uM |
6h |
LINCSCP_227330 |
LINCSCP_227330 |
HT29 |
| 0.326626 |
1.132263e-25 |
975 |
BRD-K37852224 |
LSM-6792 |
|
10uM |
6h |
LINCSCP_20106 |
LINCSCP_20106 |
HCC515 |
| 0.32631 |
1.268252e-25 |
975 |
Ilomastat |
LSM-3143 |
|
10uM |
24h |
LINCSCP_33643 |
LINCSCP_33643 |
MCF7 |
| 0.326249 |
1.296281e-25 |
975 |
BRD-K02117849 |
LSM-8563 |
|
5uM |
24h |
LINCSCP_61730 |
LINCSCP_61730 |
VCAP |
| 0.326234 |
1.302817e-25 |
975 |
Erismodegib |
LSM-4938 |
SMO |
10uM |
6h |
LINCSCP_12806 |
LINCSCP_12806 |
DV90 |
| 0.326076 |
1.379050e-25 |
975 |
BRD-K00347265 |
LSM-8447 |
|
5uM |
24h |
LINCSCP_62245 |
LINCSCP_62245 |
VCAP |
| -0.326033 |
1.400179e-25 |
975 |
Bupropion |
LSM-1267 |
SLC6A2|SLC6A3 |
10uM |
24h |
LINCSCP_269571 |
LINCSCP_269571 |
PC3 |
| 0.326017 |
1.408129e-25 |
975 |
HMS3264J07 |
LSM-1485 |
|
10uM |
24h |
LINCSCP_32826 |
LINCSCP_32826 |
MCF7 |
| -0.325849 |
1.495599e-25 |
975 |
Propylpyrazoletriol |
LSM-1978 |
ESR1 |
10uM |
24h |
LINCSCP_44352 |
LINCSCP_44352 |
PC3 |
| 0.325756 |
1.546437e-25 |
975 |
CHEMBL2141330 |
LSM-39999 |
|
0.1uM |
24h |
LINCSCP_55100 |
LINCSCP_55100 |
THP1 |
| 0.325722 |
1.565152e-25 |
975 |
Betrixaban |
LSM-45445 |
F10 |
0.04uM |
24h |
LINCSCP_161221 |
LINCSCP_161221 |
PC3 |
| 0.325222 |
1.871292e-25 |
975 |
BRD-K99803997 |
LSM-42677 |
|
5uM |
24h |
LINCSCP_63048 |
LINCSCP_63048 |
VCAP |
| -0.324817 |
2.162141e-25 |
975 |
Mebendazole |
LSM-3749 |
|
20uM |
24h |
LINCSCP_67632 |
LINCSCP_67632 |
MCF7 |
| 0.324794 |
2.179868e-25 |
975 |
BRD-M87776818 |
LSM-45074 |
|
5uM |
24h |
LINCSCP_64052 |
LINCSCP_64052 |
VCAP |
| -0.32444 |
2.472783e-25 |
975 |
PD-0325901 |
LSM-1101 |
MAP2K1|MAP2K2 |
10uM |
24h |
LINCSCP_165556 |
LINCSCP_165556 |
SKL |
| 0.324304 |
2.595077e-25 |
975 |
TG100-115 |
LSM-5731 |
PIK3CD|PIK3CG |
10uM |
6h |
LINCSCP_22397 |
LINCSCP_22397 |
HEPG2 |
| 0.323992 |
2.899161e-25 |
975 |
MLS002554298 |
LSM-3179 |
|
10uM |
24h |
LINCSCP_238371 |
LINCSCP_238371 |
MCF7 |
| -0.323349 |
3.642915e-25 |
975 |
CHEMBL1270219 |
LSM-2948 |
|
10uM |
6h |
LINCSCP_5518 |
LINCSCP_5518 |
A549 |
| -0.323321 |
3.679115e-25 |
975 |
BRD-K54285697 |
LSM-40244 |
|
10uM |
24h |
LINCSCP_33879 |
LINCSCP_33879 |
MCF7 |
| 0.323047 |
4.053358e-25 |
975 |
4-Iodo-6-phenylpyrimidine |
LSM-6233 |
MIF |
40uM |
6h |
LINCSCP_51124 |
LINCSCP_51124 |
RMUGS |
| -0.323005 |
4.114808e-25 |
975 |
Talniflumate |
LSM-1960 |
CLCA1 |
10uM |
24h |
LINCSCP_262556 |
LINCSCP_262556 |
NPC |
| 0.322133 |
5.599936e-25 |
975 |
F0605-0375 |
LSM-4554 |
|
10uM |
6h |
LINCSCP_16268 |
LINCSCP_16268 |
HA1E |
| 0.322102 |
5.661486e-25 |
975 |
BRD-K65836281 |
LSM-12443 |
|
5uM |
24h |
LINCSCP_64016 |
LINCSCP_64016 |
VCAP |
| -0.322086 |
5.692736e-25 |
975 |
Adoprazine |
LSM-45419 |
|
0.37uM |
24h |
LINCSCP_153687 |
LINCSCP_153687 |
PC3 |
| -0.321589 |
6.782641e-25 |
975 |
BRD-A24396574-001-01-5 |
LSM-5006 |
|
10uM |
3h |
LINCSCP_130206 |
LINCSCP_130206 |
LNCAP |
| 0.321545 |
6.888481e-25 |
975 |
CHEMBL2333339 |
LSM-4809 |
|
10uM |
6h |
LINCSCP_20465 |
LINCSCP_20465 |
HCC515 |
| -0.32148 |
7.047847e-25 |
975 |
Batimastat |
LSM-6276 |
|
1.11uM |
24h |
LINCSCP_101144 |
LINCSCP_101144 |
HELA |
| -0.32145 |
7.122904e-25 |
975 |
FR-180204 |
LSM-42790 |
MAPK1|MAPK3 |
0.04uM |
24h |
LINCSCP_128245 |
LINCSCP_128245 |
HUES3 |
| 0.32114 |
7.942030e-25 |
975 |
AC1MG7IW |
LSM-4330 |
|
10uM |
24h |
LINCSCP_46184 |
LINCSCP_46184 |
PC3 |
| 0.320835 |
8.842070e-25 |
975 |
BRD-K24017250 |
LSM-9878 |
|
5uM |
24h |
LINCSCP_62135 |
LINCSCP_62135 |
VCAP |
| 0.320654 |
9.420870e-25 |
975 |
BRD-K67519589 |
LSM-40951 |
|
10uM |
6h |
LINCSCP_16874 |
LINCSCP_16874 |
HA1E |
| 0.320412 |
1.025588e-24 |
975 |
BRD-K40956802-001-01-8 |
LSM-6806 |
|
10uM |
6h |
LINCSCP_16827 |
LINCSCP_16827 |
HA1E |
| 0.319849 |
1.248739e-24 |
975 |
PLX-4720 |
LSM-1049 |
BRAF |
3.33uM |
24h |
LINCSCP_130644 |
LINCSCP_130644 |
MCF10A |
| 0.319583 |
1.370620e-24 |
975 |
Imatinib |
LSM-1023 |
ABL1|BCR|CSF1R|KIT|PDGFRA|PDGFRB |
0.04uM |
3h |
LINCSCP_145938 |
LINCSCP_145938 |
MDAMB231 |
| -0.319374 |
1.474473e-24 |
975 |
Wortmannin |
LSM-3947 |
PIK3CA|PIK3CG|PLK1 |
10uM |
24h |
LINCSCP_67607 |
LINCSCP_67607 |
MCF7 |
| 0.319102 |
1.621034e-24 |
975 |
Endecaphyllin X |
LSM-3220 |
|
10uM |
6h |
LINCSCP_227235 |
LINCSCP_227235 |
HT29 |
| 0.318755 |
1.829562e-24 |
975 |
SR 33805 oxalate |
LSM-45933 |
|
0.37uM |
24h |
LINCSCP_75551 |
LINCSCP_75551 |
A375 |
| 0.318743 |
1.837309e-24 |
975 |
BRD-K51181663 |
LSM-11558 |
|
5uM |
24h |
LINCSCP_63386 |
LINCSCP_63386 |
VCAP |
| 0.31871 |
1.858833e-24 |
975 |
GSK-461364 |
LSM-1013 |
PLK1 |
10uM |
6h |
LINCSCP_22440 |
LINCSCP_22440 |
HEPG2 |
| 0.318679 |
1.878647e-24 |
975 |
BRD-K83816656 |
LSM-41851 |
|
10uM |
6h |
LINCSCP_16892 |
LINCSCP_16892 |
HA1E |
| 0.318668 |
1.885863e-24 |
975 |
HY-11007 |
LSM-1022 |
ABL1|BCR |
0.12uM |
24h |
LINCSCP_165999 |
LINCSCP_165999 |
SKL |
| 0.318654 |
1.895138e-24 |
975 |
Mitoxantrone |
LSM-2481 |
TOP2A |
0.37uM |
3h |
LINCSCP_113370 |
LINCSCP_113370 |
HME1 |
| 0.318601 |
1.930633e-24 |
975 |
BRD-K97277752 |
LSM-14407 |
|
5uM |
24h |
LINCSCP_61516 |
LINCSCP_61516 |
VCAP |
| -0.318526 |
1.981801e-24 |
975 |
Rebastinib |
LSM-6708 |
ABL1 |
0.12uM |
24h |
LINCSCP_129570 |
LINCSCP_129570 |
JURKAT |
| 0.318484 |
2.011005e-24 |
975 |
BRD-K73876582 |
LSM-12955 |
|
5uM |
24h |
LINCSCP_61818 |
LINCSCP_61818 |
VCAP |
| -0.318424 |
2.053046e-24 |
975 |
SMR000798335 |
LSM-3364 |
|
10uM |
24h |
LINCSCP_267680 |
LINCSCP_267680 |
PC3 |
| -0.318403 |
2.068257e-24 |
975 |
NSC 663284 |
LSM-2042 |
CDC25A|CDC25B |
10uM |
6h |
LINCSCP_32990 |
LINCSCP_32990 |
MCF7 |
| -0.31791 |
2.454422e-24 |
975 |
Trichostatin A, Streptomyces Sp. |
LSM-42814 |
HDAC1|HDAC10|HDAC3|HDAC4|HDAC6|HDAC7|HDAC8 |
10uM |
6h |
LINCSCP_66958 |
LINCSCP_66958 |
HCT116 |
| 0.317669 |
2.668732e-24 |
975 |
Thiothixene |
LSM-43048 |
HTR2A |
1.11uM |
24h |
LINCSCP_144091 |
LINCSCP_144091 |
MCF7 |
| -0.317393 |
2.936579e-24 |
975 |
MLS000534605 |
LSM-4827 |
|
10uM |
6h |
LINCSCP_32066 |
LINCSCP_32066 |
MCF7 |
| 0.317299 |
3.034353e-24 |
975 |
BRD-K47024121 |
LSM-11297 |
|
5uM |
24h |
LINCSCP_63382 |
LINCSCP_63382 |
VCAP |
| 0.316796 |
3.611253e-24 |
975 |
TH02453-036-P1 |
LSM-6273 |
|
10uM |
24h |
LINCSCP_236581 |
LINCSCP_236581 |
MCF7 |
| -0.316682 |
3.755440e-24 |
975 |
Pazufloxacin |
LSM-5745 |
|
10uM |
24h |
LINCSCP_46108 |
LINCSCP_46108 |
PC3 |
| -0.316483 |
4.023678e-24 |
975 |
Dichloroacetic acid |
LSM-5314 |
|
10uM |
6h |
LINCSCP_46148 |
LINCSCP_46148 |
PC3 |
| -0.316402 |
4.136939e-24 |
975 |
SPECTRUM_001418 |
LSM-1664 |
ADRB2 |
10uM |
24h |
LINCSCP_203877 |
LINCSCP_203877 |
ASC |
| 0.31624 |
4.375028e-24 |
975 |
BRD-K99785919 |
LSM-14559 |
|
5uM |
24h |
LINCSCP_62338 |
LINCSCP_62338 |
VCAP |
| 0.315999 |
4.755022e-24 |
975 |
BRD-K20332840 |
LSM-9670 |
|
5uM |
24h |
LINCSCP_62632 |
LINCSCP_62632 |
VCAP |
| 0.315952 |
4.832389e-24 |
975 |
BRD-K83509924 |
LSM-41833 |
|
10uM |
6h |
LINCSCP_16891 |
LINCSCP_16891 |
HA1E |
| 0.315892 |
4.932095e-24 |
975 |
SUGA2_000113 |
LSM-36634 |
|
10uM |
6h |
LINCSCP_22293 |
LINCSCP_22293 |
HEPG2 |
| 0.315863 |
4.983265e-24 |
975 |
CHEMBL2356693 |
LSM-6781 |
|
10uM |
6h |
LINCSCP_16796 |
LINCSCP_16796 |
HA1E |
| 0.315769 |
5.145753e-24 |
975 |
Zoxazolamine |
LSM-3476 |
|
10uM |
24h |
LINCSCP_243523 |
LINCSCP_243523 |
MCF7 |
| -0.315502 |
5.641232e-24 |
975 |
Pelitinib |
LSM-42796 |
EGFR |
10uM |
24h |
LINCSCP_136022 |
LINCSCP_136022 |
MCF7 |
| 0.315052 |
6.585430e-24 |
975 |
Alaproclate |
LSM-1333 |
SLC6A4 |
1.11uM |
24h |
LINCSCP_74484 |
LINCSCP_74484 |
A375 |
| 0.314964 |
6.788044e-24 |
975 |
FR-180204 |
LSM-42790 |
MAPK1|MAPK3 |
10uM |
24h |
LINCSCP_129637 |
LINCSCP_129637 |
JURKAT |
| 0.31452 |
7.903574e-24 |
975 |
7-Nitroindazole |
LSM-5222 |
|
10uM |
24h |
LINCSCP_31567 |
LINCSCP_31567 |
MCF7 |
| 0.314511 |
7.929067e-24 |
975 |
Cefaclor |
LSM-5368 |
|
10uM |
24h |
LINCSCP_31583 |
LINCSCP_31583 |
MCF7 |
| 0.314484 |
8.001798e-24 |
975 |
Sulfisoxazole |
LSM-3120 |
|
10uM |
24h |
LINCSCP_34294 |
LINCSCP_34294 |
MCF7 |
| -0.314467 |
8.048314e-24 |
975 |
Auranofin |
LSM-43136 |
|
10uM |
6h |
LINCSCP_45095 |
LINCSCP_45095 |
PC3 |
| 0.314418 |
8.184971e-24 |
975 |
Buspirone |
LSM-4105 |
HTR1A |
10uM |
24h |
LINCSCP_144095 |
LINCSCP_144095 |
MCF7 |
| 0.314306 |
8.504780e-24 |
975 |
Motesanib |
LSM-1042 |
FLT1|FLT4|KDR|KIT|PDGFRA|PDGFRB|RET |
0.5uM |
24h |
LINCSCP_39132 |
LINCSCP_39132 |
MDAMB231 |
| -0.314025 |
9.363561e-24 |
975 |
MK-5108 |
LSM-36812 |
AURKA|AURKB |
3.33uM |
24h |
LINCSCP_136873 |
LINCSCP_136873 |
MCF7 |
| 0.313838 |
9.981945e-24 |
975 |
PD-173074 |
LSM-1026 |
FGFR1|FGFR3 |
10uM |
6h |
LINCSCP_220165 |
LINCSCP_220165 |
HEPG2 |
| 0.313737 |
1.033274e-23 |
975 |
Emedastine |
LSM-5331 |
HRH1 |
0.12uM |
24h |
LINCSCP_74492 |
LINCSCP_74492 |
A375 |
| 0.313525 |
1.110956e-23 |
975 |
CHEMBL1868923 |
LSM-6103 |
|
10uM |
6h |
LINCSCP_211921 |
LINCSCP_211921 |
HA1E |
| 0.313484 |
1.126759e-23 |
975 |
Vitamin B12 |
LSM-46022 |
|
0.04uM |
24h |
LINCSCP_162775 |
LINCSCP_162775 |
PC3 |
| 0.313457 |
1.137052e-23 |
975 |
BRD-A73513677 |
LSM-45325 |
|
0.5uM |
24h |
LINCSCP_24120 |
LINCSCP_24120 |
HL60 |
| -0.313412 |
1.154516e-23 |
975 |
STK249718 |
LSM-6671 |
|
10uM |
6h |
LINCSCP_32752 |
LINCSCP_32752 |
MCF7 |
| -0.313329 |
1.187607e-23 |
975 |
BRD-K55149044 |
LSM-6839 |
|
10uM |
24h |
LINCSCP_35334 |
LINCSCP_35334 |
MCF7 |
| 0.312618 |
1.513425e-23 |
975 |
W 7 |
LSM-4021 |
|
10uM |
24h |
LINCSCP_33665 |
LINCSCP_33665 |
MCF7 |
| 0.312156 |
1.770755e-23 |
975 |
BRD-K67519589 |
LSM-40951 |
|
10uM |
6h |
LINCSCP_59375 |
LINCSCP_59375 |
VCAP |
| 0.311885 |
1.941698e-23 |
975 |
BRD-K57064803 |
LSM-6841 |
|
5uM |
6h |
LINCSCP_62558 |
LINCSCP_62558 |
VCAP |
| 0.311858 |
1.959007e-23 |
975 |
SR 33805 oxalate |
LSM-45933 |
|
1.11uM |
24h |
LINCSCP_75550 |
LINCSCP_75550 |
A375 |
| 0.311739 |
2.040247e-23 |
975 |
MK-8245 |
LSM-45756 |
|
0.12uM |
24h |
LINCSCP_101427 |
LINCSCP_101427 |
HELA |
| 0.311385 |
2.299713e-23 |
975 |
Iguratimod |
LSM-45469 |
|
10uM |
24h |
LINCSCP_74540 |
LINCSCP_74540 |
A375 |
| 0.311294 |
2.371966e-23 |
975 |
Gefitinib |
LSM-1098 |
EGFR |
0.37uM |
3h |
LINCSCP_145930 |
LINCSCP_145930 |
MDAMB231 |
| 0.311216 |
2.435104e-23 |
975 |
Dobutamine |
LSM-1807 |
ADRB1|ADRB2 |
10uM |
6h |
LINCSCP_14200 |
LINCSCP_14200 |
HA1E |
| 0.311183 |
2.462877e-23 |
975 |
Vecuronium |
LSM-5367 |
CHRNA1|CHRNA2|CHRNB1|CHRND|CHRNE|CHRNG |
10uM |
24h |
LINCSCP_31582 |
LINCSCP_31582 |
MCF7 |
| -0.311127 |
2.509870e-23 |
975 |
AZD-1775 |
LSM-1153 |
WEE1 |
10uM |
24h |
LINCSCP_30575 |
LINCSCP_30575 |
MCF7 |
| 0.311102 |
2.531608e-23 |
975 |
MLS002264440 |
LSM-42961 |
|
10uM |
6h |
LINCSCP_19746 |
LINCSCP_19746 |
HCC515 |
| 0.310872 |
2.736287e-23 |
975 |
Cholic acid |
LSM-5541 |
CES1|FECH|PLA2G1B |
0.04uM |
24h |
LINCSCP_75559 |
LINCSCP_75559 |
A375 |
| 0.310826 |
2.778871e-23 |
975 |
MLS002264514 |
LSM-42882 |
|
10uM |
24h |
LINCSCP_31130 |
LINCSCP_31130 |
MCF7 |
| -0.310421 |
3.185548e-23 |
975 |
Medroxyprogesterone Acetate |
LSM-5882 |
PGR |
10uM |
24h |
LINCSCP_47340 |
LINCSCP_47340 |
PC3 |
| -0.310231 |
3.396738e-23 |
975 |
Mebendazole |
LSM-3749 |
|
10uM |
24h |
LINCSCP_67594 |
LINCSCP_67594 |
MCF7 |
| 0.31017 |
3.467891e-23 |
975 |
Mafenide |
LSM-5445 |
CA6 |
10uM |
6h |
LINCSCP_57882 |
LINCSCP_57882 |
VCAP |
| -0.310166 |
3.472606e-23 |
975 |
Alisertib |
LSM-37184 |
AURKA |
3.33uM |
24h |
LINCSCP_109510 |
LINCSCP_109510 |
HELA |
| 0.310076 |
3.579064e-23 |
975 |
Celecoxib |
LSM-2032 |
PTGS2 |
10uM |
6h |
LINCSCP_57862 |
LINCSCP_57862 |
VCAP |
| -0.309816 |
3.906856e-23 |
975 |
Pimavanserin |
LSM-45960 |
HTR2A |
1.11uM |
24h |
LINCSCP_159550 |
LINCSCP_159550 |
PC3 |
| -0.309701 |
4.060263e-23 |
975 |
Withaferin A |
LSM-6685 |
IKBKB|NAMPT |
10uM |
6h |
LINCSCP_68007 |
LINCSCP_68007 |
PC3 |
| 0.309693 |
4.072028e-23 |
975 |
BRD-K02944060 |
LSM-8619 |
|
5uM |
24h |
LINCSCP_61542 |
LINCSCP_61542 |
VCAP |
| 0.309677 |
4.093382e-23 |
975 |
FR-180204 |
LSM-42790 |
MAPK1|MAPK3 |
10uM |
24h |
LINCSCP_251846 |
LINCSCP_251846 |
MCF7 |
| -0.309672 |
4.101205e-23 |
975 |
Tosedostat |
LSM-6286 |
ANPEP|C9orf3|DNPEP|ENPEP|ERAP1|ERAP2|LAP3|LNPEP|LVRN|METAP1|METAP1D|METAP2|NPEPL1|NPEPPS|RNPEP|RNPEPL1|XPNPEP1|XPNPEP2|XPNPEP3 |
3uM |
24h |
LINCSCP_38256 |
LINCSCP_38256 |
MCF7 |
| 0.309369 |
4.540024e-23 |
975 |
SCHEMBL1995782 |
LSM-36792 |
|
0.01uM |
24h |
LINCSCP_41926 |
LINCSCP_41926 |
NOMO1 |
| -0.309286 |
4.668385e-23 |
975 |
PD-0325901 |
LSM-1101 |
MAP2K1|MAP2K2 |
10uM |
24h |
LINCSCP_129805 |
LINCSCP_129805 |
LNCAP |
| 0.30905 |
5.054144e-23 |
975 |
BRD-K82071478 |
LSM-13442 |
|
5uM |
24h |
LINCSCP_61831 |
LINCSCP_61831 |
VCAP |
| 0.308932 |
5.258122e-23 |
975 |
noscapine |
|
|
0.12uM |
3h |
LINCSCP_130342 |
LINCSCP_130342 |
LNCAP |
| 0.308662 |
5.756783e-23 |
975 |
FPA1_000112 |
LSM-36718 |
|
10uM |
6h |
LINCSCP_20149 |
LINCSCP_20149 |
HCC515 |
| 0.308167 |
6.794557e-23 |
975 |
Cephalexin |
LSM-5957 |
|
10uM |
24h |
LINCSCP_34324 |
LINCSCP_34324 |
MCF7 |
| -0.30794 |
7.328386e-23 |
975 |
CHEMBL2361187 |
LSM-12338 |
|
1uM |
24h |
LINCSCP_66129 |
LINCSCP_66129 |
VCAP |
| 0.307816 |
7.640130e-23 |
975 |
BRD-K83155387 |
LSM-43611 |
|
10uM |
6h |
LINCSCP_279539 |
LINCSCP_279539 |
PC3 |
| 0.307345 |
8.941083e-23 |
975 |
pyrvinium-pamoate |
|
AR |
10uM |
6h |
LINCSCP_12886 |
LINCSCP_12886 |
DV90 |
| -0.307281 |
9.132088e-23 |
975 |
Temoporfin |
LSM-45995 |
|
10uM |
24h |
LINCSCP_120449 |
LINCSCP_120449 |
HT29 |
| 0.306972 |
1.012169e-22 |
975 |
Erlotinib |
LSM-1097 |
EGFR |
1.11uM |
3h |
LINCSCP_115370 |
LINCSCP_115370 |
HS578T |
| 0.306817 |
1.065899e-22 |
975 |
BRD-K24339152 |
LSM-9905 |
|
5uM |
24h |
LINCSCP_61966 |
LINCSCP_61966 |
VCAP |
| 0.306715 |
1.102662e-22 |
975 |
Remacemide |
LSM-1489 |
GRIN1 |
10uM |
24h |
LINCSCP_32827 |
LINCSCP_32827 |
MCF7 |
| -0.306694 |
1.110298e-22 |
975 |
Temoporfin |
LSM-45995 |
|
10uM |
24h |
LINCSCP_91846 |
LINCSCP_91846 |
HA1E |
| 0.306649 |
1.127281e-22 |
975 |
Swainsonine |
LSM-45602 |
|
1.28uM |
24h |
LINCSCP_74496 |
LINCSCP_74496 |
A375 |
| 0.30637 |
1.236677e-22 |
975 |
Hydroxyprogesterone Caproate |
LSM-4900 |
AR|ESR1|ESR2|NR1H4|NR1I2|NR3C1|PGR |
0.12uM |
24h |
LINCSCP_71311 |
LINCSCP_71311 |
A375 |
| 0.306353 |
1.243596e-22 |
975 |
BRD-K47128441 |
LSM-45358 |
|
10uM |
6h |
LINCSCP_310145 |
LINCSCP_310145 |
VCAP |
| 0.306227 |
1.296724e-22 |
975 |
Imatinib |
LSM-1023 |
ABL1|BCR|CSF1R|KIT|PDGFRA|PDGFRB |
0.04uM |
24h |
LINCSCP_130025 |
LINCSCP_130025 |
LNCAP |
| -0.305932 |
1.430009e-22 |
975 |
SB225002 |
LSM-3367 |
CXCR2 |
10uM |
24h |
LINCSCP_37926 |
LINCSCP_37926 |
MCF7 |
| 0.30551 |
1.644886e-22 |
975 |
Iguratimod |
LSM-45469 |
|
3.33uM |
24h |
LINCSCP_74541 |
LINCSCP_74541 |
A375 |
| 0.305415 |
1.697473e-22 |
975 |
BRD-K74163137 |
LSM-6150 |
|
10uM |
24h |
LINCSCP_242557 |
LINCSCP_242557 |
MCF7 |
| -0.305407 |
1.701575e-22 |
975 |
Infigratinib |
LSM-1184 |
FGFR1|FGFR2|FGFR3|FGFR4 |
10uM |
24h |
LINCSCP_146335 |
LINCSCP_146335 |
MNEU.E |
| -0.305087 |
1.891753e-22 |
975 |
Arecaidine Propargyl Ester |
LSM-2520 |
CHRM1 |
10uM |
24h |
LINCSCP_44018 |
LINCSCP_44018 |
PC3 |
| 0.304605 |
2.217809e-22 |
975 |
BRD-K64169482 |
LSM-12347 |
|
5uM |
24h |
LINCSCP_61484 |
LINCSCP_61484 |
VCAP |
| -0.304378 |
2.390237e-22 |
975 |
Hydroxyfasudil |
LSM-3744 |
ROCK1 |
10uM |
6h |
LINCSCP_30396 |
LINCSCP_30396 |
MCF7 |
| -0.304269 |
2.477878e-22 |
975 |
Balicatib |
LSM-45647 |
|
0.37uM |
24h |
LINCSCP_154143 |
LINCSCP_154143 |
PC3 |
| 0.304132 |
2.592515e-22 |
975 |
BRD-K35188965 |
LSM-10543 |
|
5uM |
24h |
LINCSCP_62277 |
LINCSCP_62277 |
VCAP |
| 0.303757 |
2.933016e-22 |
975 |
Tedizolid |
LSM-45778 |
|
0.12uM |
24h |
LINCSCP_123216 |
LINCSCP_123216 |
HT29 |
| -0.303722 |
2.966864e-22 |
975 |
CHEMBL2356547 |
LSM-8092 |
|
5uM |
24h |
LINCSCP_60102 |
LINCSCP_60102 |
VCAP |
| 0.303635 |
3.053279e-22 |
975 |
MDL 29951 |
LSM-3330 |
FBP1 |
10uM |
24h |
LINCSCP_32915 |
LINCSCP_32915 |
MCF7 |
| -0.303501 |
3.190072e-22 |
975 |
PD-173074 |
LSM-1026 |
FGFR1|FGFR3 |
1.11uM |
24h |
LINCSCP_151281 |
LINCSCP_151281 |
PC3 |
| -0.303216 |
3.502849e-22 |
975 |
Broad-Sai-560 |
LSM-45991 |
|
0.1uM |
6h |
LINCSCP_35583 |
LINCSCP_35583 |
MCF7 |
| 0.303161 |
3.567324e-22 |
975 |
BRD-K46448313 |
LSM-39840 |
|
5uM |
24h |
LINCSCP_309408 |
LINCSCP_309408 |
VCAP |
| 0.302977 |
3.788854e-22 |
975 |
Cholic acid |
LSM-5541 |
CES1|FECH|PLA2G1B |
3.33uM |
24h |
LINCSCP_105718 |
LINCSCP_105718 |
HELA |
| 0.302826 |
3.981523e-22 |
975 |
Aminoglutethimide |
LSM-1409 |
CYP11A1|CYP19A1 |
10uM |
6h |
LINCSCP_57846 |
LINCSCP_57846 |
VCAP |
| -0.302722 |
4.119213e-22 |
975 |
CHEMBL2357936 |
LSM-38158 |
|
10uM |
24h |
LINCSCP_35179 |
LINCSCP_35179 |
MCF7 |
| 0.302677 |
4.180564e-22 |
975 |
Gefitinib |
LSM-1098 |
EGFR |
0.37uM |
3h |
LINCSCP_130371 |
LINCSCP_130371 |
LNCAP |
| -0.302261 |
4.789623e-22 |
975 |
Lexibulin |
LSM-6232 |
TUBA1A|TUBA1B|TUBA1C|TUBA3E|TUBA4A|TUBB|TUBB1|TUBB2A|TUBB2B|TUBB3|TUBB4A|TUBB4B|TUBB6|TUBB8 |
10uM |
24h |
LINCSCP_135770 |
LINCSCP_135770 |
MCF7 |
| 0.302197 |
4.890121e-22 |
975 |
BRD-K96160456 |
LSM-14329 |
|
5uM |
24h |
LINCSCP_62069 |
LINCSCP_62069 |
VCAP |
| 0.302019 |
5.184532e-22 |
975 |
PF-04217903 |
LSM-1166 |
MET |
40uM |
6h |
LINCSCP_206560 |
LINCSCP_206560 |
DV90 |
| 0.30198 |
5.249707e-22 |
975 |
Sulfacetamide |
LSM-5374 |
|
10uM |
6h |
LINCSCP_212157 |
LINCSCP_212157 |
HA1E |
| 0.301909 |
5.373104e-22 |
975 |
CHEMBL2361312 |
LSM-12950 |
|
5uM |
24h |
LINCSCP_301291 |
LINCSCP_301291 |
VCAP |
| 0.301819 |
5.534313e-22 |
975 |
MLS003128719 |
LSM-39608 |
|
5uM |
24h |
LINCSCP_64285 |
LINCSCP_64285 |
VCAP |
| 0.301818 |
5.536190e-22 |
975 |
4-(Trans-4-butylcyclohexyl)benzoic acid |
LSM-4640 |
|
10uM |
6h |
LINCSCP_20117 |
LINCSCP_20117 |
HCC515 |
| -0.301703 |
5.746892e-22 |
975 |
Idebenone |
LSM-5505 |
|
10uM |
24h |
LINCSCP_46089 |
LINCSCP_46089 |
PC3 |
| 0.301438 |
6.265546e-22 |
975 |
BRD-K88058683 |
LSM-13835 |
|
5uM |
24h |
LINCSCP_63417 |
LINCSCP_63417 |
VCAP |
| 0.301302 |
6.550493e-22 |
975 |
BRD-K31774852 |
LSM-10354 |
|
5uM |
6h |
LINCSCP_62213 |
LINCSCP_62213 |
VCAP |
| 0.30124 |
6.682650e-22 |
975 |
Pyrazinamide |
LSM-5425 |
FASN |
3.33uM |
24h |
LINCSCP_89525 |
LINCSCP_89525 |
HA1E |
| 0.300798 |
7.715311e-22 |
975 |
Cdc |
LSM-42873 |
ALOX12 |
10uM |
24h |
LINCSCP_11406 |
LINCSCP_11406 |
ASC |
| 0.300782 |
7.756566e-22 |
975 |
BRD-K33676730 |
LSM-39115 |
|
10uM |
6h |
LINCSCP_16298 |
LINCSCP_16298 |
HA1E |
| 0.300576 |
8.294487e-22 |
975 |
(S)-(-)-BAY K 8644 |
LSM-4545 |
CACNA1C |
10uM |
6h |
LINCSCP_55456 |
LINCSCP_55456 |
U937 |
| 0.300523 |
8.436569e-22 |
975 |
ANISODAMINE HYDROBROMIDE |
LSM-45481 |
|
0.04uM |
24h |
LINCSCP_71300 |
LINCSCP_71300 |
A375 |
| -0.300281 |
9.125695e-22 |
975 |
Tacedinaline |
LSM-19036 |
HDAC1|HDAC10|HDAC11|HDAC2|HDAC3|HDAC4|HDAC5|HDAC6|HDAC7|HDAC8|HDAC9 |
0.1uM |
6h |
LINCSCP_279846 |
LINCSCP_279846 |
PC3 |
| 0.300234 |
9.265908e-22 |
975 |
BRD-A35207501 |
LSM-45361 |
|
0.5uM |
24h |
LINCSCP_55292 |
LINCSCP_55292 |
U937 |
| 0.300101 |
9.675984e-22 |
975 |
BRD-K46766834 |
LSM-6752 |
|
5uM |
24h |
LINCSCP_63085 |
LINCSCP_63085 |
VCAP |
| -0.299986 |
1.004170e-21 |
975 |
SA-90377 |
LSM-40102 |
|
10uM |
24h |
LINCSCP_186587 |
LINCSCP_186587 |
A375 |
| -0.299545 |
1.158312e-21 |
975 |
BRD-K65378566 |
LSM-12415 |
|
5uM |
24h |
LINCSCP_62025 |
LINCSCP_62025 |
VCAP |
| -0.29941 |
1.209963e-21 |
975 |
CDK4 Inhibitor III |
LSM-2121 |
CDK4 |
10uM |
6h |
LINCSCP_23581 |
LINCSCP_23581 |
HEPG2 |
| -0.299244 |
1.276636e-21 |
975 |
Cerulenin |
LSM-43210 |
FASN |
3uM |
24h |
LINCSCP_37924 |
LINCSCP_37924 |
MCF7 |
| -0.298999 |
1.381777e-21 |
975 |
CHEMBL3186688 |
LSM-3014 |
|
10uM |
6h |
LINCSCP_57671 |
LINCSCP_57671 |
VCAP |
| 0.298859 |
1.445649e-21 |
975 |
ALD1-H_001128 |
LSM-45103 |
|
10uM |
6h |
LINCSCP_20094 |
LINCSCP_20094 |
HCC515 |
| 0.298822 |
1.462974e-21 |
975 |
BRD-M85886474 |
LSM-45072 |
|
5uM |
24h |
LINCSCP_64051 |
LINCSCP_64051 |
VCAP |
| -0.298705 |
1.519421e-21 |
975 |
Palmidrol |
LSM-3518 |
CNR2|GPR119 |
0.04uM |
24h |
LINCSCP_142450 |
LINCSCP_142450 |
MCF7 |
| 0.29865 |
1.546617e-21 |
975 |
Vanoxerine |
LSM-2703 |
SLC6A3 |
10uM |
24h |
LINCSCP_11550 |
LINCSCP_11550 |
ASC |
| -0.298507 |
1.619537e-21 |
975 |
GNF-PF-2272 |
LSM-6669 |
|
10uM |
6h |
LINCSCP_32751 |
LINCSCP_32751 |
MCF7 |
| -0.29839 |
1.681664e-21 |
975 |
CHEMBL2362317 |
LSM-12520 |
|
10uM |
24h |
LINCSCP_35353 |
LINCSCP_35353 |
MCF7 |
| -0.298365 |
1.695161e-21 |
975 |
cortisone-acetate |
LSM-45387 |
TUBA1A|TUBA1B|TUBA1C|TUBA3E|TUBA4A|TUBB|TUBB1|TUBB2A|TUBB2B|TUBB3|TUBB4A|TUBB4B|TUBB6|TUBB8 |
0.37uM |
24h |
LINCSCP_143282 |
LINCSCP_143282 |
MCF7 |
| 0.2982 |
1.787538e-21 |
975 |
BRD-K04025047 |
LSM-8676 |
|
10uM |
24h |
LINCSCP_8992 |
LINCSCP_8992 |
A549 |
| 0.298191 |
1.793082e-21 |
975 |
BRD-M91876180 |
LSM-45082 |
|
5uM |
24h |
LINCSCP_64055 |
LINCSCP_64055 |
VCAP |
| 0.297923 |
1.954133e-21 |
975 |
Erlotinib |
LSM-1097 |
EGFR |
1.11uM |
3h |
LINCSCP_163411 |
LINCSCP_163411 |
SKBR3 |
| 0.297774 |
2.049962e-21 |
975 |
Cis-N,N-Dimethyl-9-(3-(1-Piperazinyl)Propylidene)Thioxanthene-2-Sulfonamide |
LSM-43212 |
HTR2A |
10uM |
6h |
LINCSCP_57897 |
LINCSCP_57897 |
VCAP |
| 0.297761 |
2.058665e-21 |
975 |
Moclobemide |
LSM-5247 |
MAOA |
10uM |
24h |
LINCSCP_74836 |
LINCSCP_74836 |
A375 |
| -0.297631 |
2.146455e-21 |
975 |
SA-102042 |
LSM-40575 |
|
3uM |
24h |
LINCSCP_38213 |
LINCSCP_38213 |
MCF7 |
| -0.297575 |
2.185631e-21 |
975 |
1-(5-Isoquinolinesulfonyl)piperazine |
LSM-3622 |
|
10uM |
24h |
LINCSCP_44411 |
LINCSCP_44411 |
PC3 |
| 0.297522 |
2.222964e-21 |
975 |
Danazol |
LSM-3073 |
AR|ESR1|GNRHR|PGR |
10uM |
6h |
LINCSCP_212188 |
LINCSCP_212188 |
HA1E |
| -0.29752 |
2.224044e-21 |
975 |
Withaferin A |
LSM-6685 |
IKBKB|NAMPT |
10uM |
24h |
LINCSCP_81502 |
LINCSCP_81502 |
A549 |
| 0.29744 |
2.281829e-21 |
975 |
BRD-K66586010 |
LSM-40898 |
|
5uM |
24h |
LINCSCP_64305 |
LINCSCP_64305 |
VCAP |
| 0.297434 |
2.286852e-21 |
975 |
Imatinib |
LSM-1023 |
ABL1|BCR|CSF1R|KIT|PDGFRA|PDGFRB |
0.12uM |
3h |
LINCSCP_164136 |
LINCSCP_164136 |
SKBR3 |
| 0.297412 |
2.302774e-21 |
975 |
Erastin |
LSM-4914 |
VDAC2 |
5uM |
6h |
LINCSCP_257044 |
LINCSCP_257044 |
NCIH2073 |
| 0.29741 |
2.304482e-21 |
975 |
BRD-K64099269 |
LSM-40768 |
|
10uM |
6h |
LINCSCP_295884 |
LINCSCP_295884 |
VCAP |
| -0.297337 |
2.358958e-21 |
975 |
Withaferin A |
LSM-6685 |
IKBKB|NAMPT |
0.1uM |
24h |
LINCSCP_245051 |
LINCSCP_245051 |
MCF7 |
| 0.297324 |
2.368610e-21 |
975 |
BRD-K33761091 |
LSM-10475 |
|
5uM |
24h |
LINCSCP_61980 |
LINCSCP_61980 |
VCAP |
| 0.297276 |
2.405658e-21 |
975 |
Imatinib |
LSM-1023 |
ABL1|BCR|CSF1R|KIT|PDGFRA|PDGFRB |
1.11uM |
3h |
LINCSCP_116094 |
LINCSCP_116094 |
HS578T |
| 0.297258 |
2.419345e-21 |
975 |
BRD-K39799535 |
LSM-10851 |
|
5uM |
24h |
LINCSCP_61776 |
LINCSCP_61776 |
VCAP |
| 0.297255 |
2.421583e-21 |
975 |
BRD-K61952473 |
LSM-12184 |
|
5uM |
24h |
LINCSCP_63509 |
LINCSCP_63509 |
VCAP |
| 0.296942 |
2.677391e-21 |
975 |
MLS000859112 |
LSM-6180 |
|
10uM |
6h |
LINCSCP_20165 |
LINCSCP_20165 |
HCC515 |
| 0.296924 |
2.692637e-21 |
975 |
Alpelisib |
LSM-4256 |
PIK3CA |
1.11uM |
3h |
LINCSCP_145217 |
LINCSCP_145217 |
MDAMB231 |
| -0.29691 |
2.704281e-21 |
975 |
EO 1428 |
LSM-1228 |
MAPK11|MAPK14 |
10uM |
6h |
LINCSCP_18413 |
LINCSCP_18413 |
HCC515 |
| -0.296834 |
2.771059e-21 |
975 |
Mebendazole |
LSM-3749 |
|
40uM |
24h |
LINCSCP_67633 |
LINCSCP_67633 |
MCF7 |
| -0.296385 |
3.198821e-21 |
975 |
Carbazole, 9-(4-methylbenzoyl)- |
LSM-3597 |
|
10uM |
24h |
LINCSCP_30997 |
LINCSCP_30997 |
MCF7 |
| 0.296341 |
3.244812e-21 |
975 |
BRD-K07642375 |
LSM-44682 |
|
10uM |
6h |
LINCSCP_49079 |
LINCSCP_49079 |
PC3 |
| 0.296053 |
3.556557e-21 |
975 |
BRD-K41763112 |
LSM-14821 |
|
5uM |
24h |
LINCSCP_64190 |
LINCSCP_64190 |
VCAP |
| -0.295988 |
3.631206e-21 |
975 |
KW-2449 |
LSM-42803 |
ABL1|AURKA|AURKB|FLT3 |
1.11uM |
24h |
LINCSCP_154022 |
LINCSCP_154022 |
PC3 |
| 0.295968 |
3.654510e-21 |
975 |
Tyrphostin AG 527 |
LSM-42874 |
EGFR |
10uM |
24h |
LINCSCP_23417 |
LINCSCP_23417 |
HEPG2 |
| 0.295814 |
3.838775e-21 |
975 |
Cholic acid |
LSM-5541 |
CES1|FECH|PLA2G1B |
10uM |
24h |
LINCSCP_105717 |
LINCSCP_105717 |
HELA |
| -0.295434 |
4.331581e-21 |
975 |
BRD-K65778880 |
LSM-12441 |
|
5uM |
24h |
LINCSCP_61637 |
LINCSCP_61637 |
VCAP |
| 0.295191 |
4.680668e-21 |
975 |
EX-8678 |
LSM-1147 |
|
0.37uM |
3h |
LINCSCP_164123 |
LINCSCP_164123 |
SKBR3 |
| -0.295179 |
4.698096e-21 |
975 |
D-64131 |
LSM-2592 |
TUBB |
0.5uM |
24h |
LINCSCP_37446 |
LINCSCP_37446 |
MCF7 |
| -0.294863 |
5.195096e-21 |
975 |
cortisone-acetate |
LSM-45387 |
TUBA1A|TUBA1B|TUBA1C|TUBA3E|TUBA4A|TUBB|TUBB1|TUBB2A|TUBB2B|TUBB3|TUBB4A|TUBB4B|TUBB6|TUBB8 |
1.11uM |
24h |
LINCSCP_143281 |
LINCSCP_143281 |
MCF7 |
| 0.294681 |
5.503750e-21 |
975 |
Nilotinib |
LSM-1099 |
ABL1|BCR|KIT |
0.12uM |
3h |
LINCSCP_145231 |
LINCSCP_145231 |
MDAMB231 |
| -0.294556 |
5.725127e-21 |
975 |
U 0126 |
LSM-42806 |
MAP2K1|MAP2K2 |
10uM |
24h |
LINCSCP_284925 |
LINCSCP_284925 |
SKB |
| -0.294282 |
6.244722e-21 |
975 |
306935-41-1 |
LSM-2331 |
HCAR3 |
10uM |
24h |
LINCSCP_52852 |
LINCSCP_52852 |
SKB |
| -0.294234 |
6.341803e-21 |
975 |
Lexibulin |
LSM-6232 |
TUBA1A|TUBA1B|TUBA1C|TUBA3E|TUBA4A|TUBB|TUBB1|TUBB2A|TUBB2B|TUBB3|TUBB4A|TUBB4B|TUBB6|TUBB8 |
10uM |
24h |
LINCSCP_90590 |
LINCSCP_90590 |
HA1E |
| 0.294093 |
6.630580e-21 |
975 |
BRD-K11517399 |
LSM-9131 |
|
5uM |
24h |
LINCSCP_61554 |
LINCSCP_61554 |
VCAP |
| 0.294059 |
6.701813e-21 |
975 |
SA-84902 |
LSM-42377 |
|
1uM |
24h |
LINCSCP_37497 |
LINCSCP_37497 |
MCF7 |
| -0.293975 |
6.882832e-21 |
975 |
Selamectin |
LSM-44969 |
|
10uM |
24h |
LINCSCP_139734 |
LINCSCP_139734 |
MCF7 |
| 0.29368 |
7.555645e-21 |
975 |
Nilotinib |
LSM-1099 |
ABL1|BCR|KIT |
0.12uM |
3h |
LINCSCP_163431 |
LINCSCP_163431 |
SKBR3 |
| -0.293433 |
8.169736e-21 |
975 |
BDBM82056 |
LSM-5188 |
CACNA1C|CACNA1D|CACNA1S |
10uM |
6h |
LINCSCP_46141 |
LINCSCP_46141 |
PC3 |
| -0.293377 |
8.313985e-21 |
975 |
Temoporfin |
LSM-45995 |
|
10uM |
24h |
LINCSCP_168835 |
LINCSCP_168835 |
YAPC |
| 0.29288 |
9.726849e-21 |
975 |
BRD-K32030161 |
LSM-10370 |
|
5uM |
24h |
LINCSCP_63990 |
LINCSCP_63990 |
VCAP |
| -0.292871 |
9.753506e-21 |
975 |
Mebendazole |
LSM-3749 |
|
20uM |
24h |
LINCSCP_67575 |
LINCSCP_67575 |
MCF7 |
| 0.292815 |
9.927567e-21 |
975 |
ANISODAMINE HYDROBROMIDE |
LSM-45481 |
|
0.37uM |
24h |
LINCSCP_71298 |
LINCSCP_71298 |
A375 |
| 0.292741 |
1.016282e-20 |
975 |
Veliparib |
LSM-1146 |
PARP1|PARP2 |
0.04uM |
24h |
LINCSCP_87532 |
LINCSCP_87532 |
CD34 |
| 0.292739 |
1.016622e-20 |
975 |
MLS002699918 |
LSM-2263 |
|
10uM |
24h |
LINCSCP_31877 |
LINCSCP_31877 |
MCF7 |
| -0.29261 |
1.058971e-20 |
975 |
TUL_XX087 |
LSM-36794 |
|
0.001uM |
6h |
LINCSCP_55137 |
LINCSCP_55137 |
THP1 |
| -0.292442 |
1.116375e-20 |
975 |
Mebendazole |
LSM-3749 |
|
20uM |
24h |
LINCSCP_67595 |
LINCSCP_67595 |
MCF7 |
| 0.292293 |
1.170069e-20 |
975 |
Tacedinaline |
LSM-19036 |
HDAC1|HDAC10|HDAC11|HDAC2|HDAC3|HDAC4|HDAC5|HDAC6|HDAC7|HDAC8|HDAC9 |
0.1uM |
24h |
LINCSCP_17111 |
LINCSCP_17111 |
HA1E |
| -0.292159 |
1.220382e-20 |
975 |
BRD-K09054764 |
LSM-37757 |
|
10uM |
24h |
LINCSCP_65572 |
LINCSCP_65572 |
VCAP |
| 0.292043 |
1.265473e-20 |
975 |
Acyclovir |
LSM-5459 |
|
10uM |
6h |
LINCSCP_57883 |
LINCSCP_57883 |
VCAP |
| 0.291978 |
1.291734e-20 |
975 |
ipratropium |
LSM-45809 |
|
0.12uM |
24h |
LINCSCP_123151 |
LINCSCP_123151 |
HT29 |
| 0.291723 |
1.399198e-20 |
975 |
ALD1-H_001009 |
LSM-45117 |
|
10uM |
6h |
LINCSCP_16386 |
LINCSCP_16386 |
HA1E |
| 0.291641 |
1.435536e-20 |
975 |
CP-724714 |
LSM-42777 |
ERBB2 |
0.04uM |
24h |
LINCSCP_99359 |
LINCSCP_99359 |
HCC515 |
| -0.291592 |
1.457696e-20 |
975 |
Momelotinib |
LSM-1141 |
JAK1|JAK2 |
0.5uM |
6h |
LINCSCP_39656 |
LINCSCP_39656 |
MDAMB231 |
| 0.291576 |
1.465345e-20 |
975 |
Hypericin |
LSM-2650 |
|
0.37uM |
24h |
LINCSCP_71286 |
LINCSCP_71286 |
A375 |
| -0.291483 |
1.508449e-20 |
975 |
DM-55-3 |
LSM-3831 |
|
10uM |
24h |
LINCSCP_1427 |
LINCSCP_1427 |
A375 |
| -0.291284 |
1.605360e-20 |
975 |
Cephalexin |
LSM-5957 |
|
10uM |
24h |
LINCSCP_293957 |
LINCSCP_293957 |
VCAP |
| 0.291253 |
1.621198e-20 |
975 |
Coumestrol |
LSM-4202 |
ESR1|ESR2 |
10uM |
6h |
LINCSCP_56200 |
LINCSCP_56200 |
VCAP |
| -0.291209 |
1.643896e-20 |
975 |
Propafenone |
LSM-1416 |
ADRB1|ADRB2|KCNH2|SCN10A|SCN11A|SCN1A|SCN2A|SCN3A|SCN4A|SCN5A|SCN7A|SCN8A|SCN9A |
10uM |
24h |
LINCSCP_47271 |
LINCSCP_47271 |
PC3 |
| 0.291044 |
1.730496e-20 |
975 |
Crizotinib |
LSM-1027 |
ALK|MET |
3.33uM |
24h |
LINCSCP_99367 |
LINCSCP_99367 |
HCC515 |
| -0.291036 |
1.734854e-20 |
975 |
Cyclophosphamide |
LSM-4961 |
CYP2A6|CYP2B6|CYP2C18|CYP2C19|CYP2C8|CYP2C9|CYP2D6|CYP3A4|CYP3A5|CYP3A7 |
10uM |
24h |
LINCSCP_47266 |
LINCSCP_47266 |
PC3 |
| 0.290949 |
1.782745e-20 |
975 |
BRD-K35669573 |
LSM-29348 |
|
0.001uM |
6h |
LINCSCP_55149 |
LINCSCP_55149 |
THP1 |
| -0.290842 |
1.843405e-20 |
975 |
Cnqx |
LSM-3184 |
|
10uM |
24h |
LINCSCP_72841 |
LINCSCP_72841 |
A375 |
| -0.290827 |
1.852482e-20 |
975 |
MLS003129663 |
LSM-7167 |
|
10uM |
24h |
LINCSCP_9009 |
LINCSCP_9009 |
A549 |
| 0.290333 |
2.161105e-20 |
975 |
Loperamide |
LSM-3365 |
OPRD1|OPRM1 |
0.04uM |
24h |
LINCSCP_139865 |
LINCSCP_139865 |
MCF7 |
| 0.290132 |
2.300944e-20 |
975 |
BRD-K00765103 |
LSM-8482 |
|
5uM |
24h |
LINCSCP_61396 |
LINCSCP_61396 |
VCAP |
| -0.290086 |
2.333722e-20 |
975 |
Ibrutinib (PCI-32765) |
LSM-45830 |
BTK |
0.04uM |
24h |
LINCSCP_97348 |
LINCSCP_97348 |
HA1E |
| -0.290035 |
2.371213e-20 |
975 |
KX2-391 |
LSM-45890 |
SRC |
0.12uM |
24h |
LINCSCP_137500 |
LINCSCP_137500 |
MCF7 |
| 0.289632 |
2.688440e-20 |
975 |
Pictilisib |
LSM-1047 |
PIK3CA|PIK3CB|PIK3CD|PIK3CG|PIK3R1|PIK3R2|PIK3R3|PIK3R5 |
3.33uM |
3h |
LINCSCP_145712 |
LINCSCP_145712 |
MDAMB231 |
| 0.289632 |
2.688601e-20 |
975 |
Alaproclate |
LSM-1333 |
SLC6A4 |
10uM |
24h |
LINCSCP_74482 |
LINCSCP_74482 |
A375 |
| 0.289552 |
2.755862e-20 |
975 |
ST092443 |
LSM-1481 |
ADORA1|ADORA2A|ADORA2B |
10uM |
24h |
LINCSCP_32825 |
LINCSCP_32825 |
MCF7 |
| -0.289476 |
2.822280e-20 |
975 |
Altretamine |
LSM-3492 |
|
10uM |
24h |
LINCSCP_272086 |
LINCSCP_272086 |
PC3 |
| -0.289456 |
2.839275e-20 |
975 |
cortisone-acetate |
LSM-45387 |
TUBA1A|TUBA1B|TUBA1C|TUBA3E|TUBA4A|TUBB|TUBB1|TUBB2A|TUBB2B|TUBB3|TUBB4A|TUBB4B|TUBB6|TUBB8 |
10uM |
24h |
LINCSCP_143279 |
LINCSCP_143279 |
MCF7 |
| 0.289426 |
2.866416e-20 |
975 |
YL-54 |
LSM-44651 |
|
10uM |
6h |
LINCSCP_217534 |
LINCSCP_217534 |
HCC515 |
| 0.289367 |
2.918890e-20 |
975 |
CHEMBL2360750 |
LSM-14345 |
|
5uM |
24h |
LINCSCP_61669 |
LINCSCP_61669 |
VCAP |
| 0.289358 |
2.927463e-20 |
975 |
Gimeracil |
LSM-45923 |
|
0.04uM |
24h |
LINCSCP_102153 |
LINCSCP_102153 |
HELA |
| 0.289241 |
3.035491e-20 |
975 |
Nimodipine |
LSM-1659 |
CACNA1C|CACNA1D|CACNA1F|CACNA1S|NR3C2 |
0.04uM |
24h |
LINCSCP_123104 |
LINCSCP_123104 |
HT29 |
| 0.289134 |
3.138339e-20 |
975 |
MLS001214919 |
LSM-6621 |
|
10uM |
6h |
LINCSCP_16857 |
LINCSCP_16857 |
HA1E |
| -0.288881 |
3.394389e-20 |
975 |
201038-74-6 |
LSM-2529 |
HTR7 |
10uM |
24h |
LINCSCP_33354 |
LINCSCP_33354 |
MCF7 |
| 0.28883 |
3.448262e-20 |
975 |
Protionamide |
LSM-4210 |
|
10uM |
6h |
LINCSCP_33036 |
LINCSCP_33036 |
MCF7 |
| -0.28877 |
3.513466e-20 |
975 |
AC1MVW5E |
LSM-4870 |
|
10uM |
24h |
LINCSCP_42264 |
LINCSCP_42264 |
NPC |
| 0.288489 |
3.832364e-20 |
975 |
Topiramate |
LSM-5435 |
CA2|CA4|GABRA1|GABRA2|GABRA3|GABRA4|GABRA5|GABRA6|GABRB1|GABRB2|GABRB3|GABRD|GABRE|GABRG1|GABRG2|GABRG3|GABRP|GABRQ|GRIA1|GRIA2|GRIA3|GRIA4|GRIK1|GRIK2|GRIK3|GRIK4|GRIK5|SCN10A|SCN11A|SCN1A|SCN2A|SCN3A|SCN4A|SCN5A|SCN7A|SCN8A|SCN9A |
0.12uM |
24h |
LINCSCP_71281 |
LINCSCP_71281 |
A375 |
| -0.288459 |
3.867931e-20 |
975 |
Mosapride |
LSM-5042 |
HTR4 |
10uM |
6h |
LINCSCP_46134 |
LINCSCP_46134 |
PC3 |
| -0.288426 |
3.908116e-20 |
975 |
Plinabulin |
LSM-43250 |
TUBA1A|TUBA1B|TUBA1C|TUBA3E|TUBA4A|TUBB|TUBB1|TUBB2A|TUBB2B|TUBB3|TUBB4A|TUBB4B|TUBB6|TUBB8 |
10uM |
24h |
LINCSCP_32579 |
LINCSCP_32579 |
MCF7 |
| -0.2884 |
3.940163e-20 |
975 |
BRD-A80960055-001-01-7 |
LSM-5162 |
|
10uM |
6h |
LINCSCP_22488 |
LINCSCP_22488 |
HEPG2 |
| -0.288355 |
3.994985e-20 |
975 |
BRD-K79102010 |
LSM-41589 |
|
10uM |
24h |
LINCSCP_3626 |
LINCSCP_3626 |
A375 |
| -0.288265 |
4.107242e-20 |
975 |
NSC 663284 |
LSM-2042 |
CDC25A|CDC25B |
10uM |
6h |
LINCSCP_30187 |
LINCSCP_30187 |
MCF7 |
| 0.288182 |
4.213979e-20 |
975 |
GW-5074 |
LSM-42779 |
RAF1 |
0.5uM |
24h |
LINCSCP_11645 |
LINCSCP_11645 |
BT20 |
| -0.288055 |
4.383720e-20 |
975 |
SA-102607 |
LSM-14734 |
|
3uM |
24h |
LINCSCP_38158 |
LINCSCP_38158 |
MCF7 |
| -0.288008 |
4.447407e-20 |
975 |
Temoporfin |
LSM-45995 |
|
10uM |
24h |
LINCSCP_73509 |
LINCSCP_73509 |
A375 |
| 0.287953 |
4.523938e-20 |
975 |
BRD-K05726929 |
LSM-8767 |
|
5uM |
24h |
LINCSCP_61935 |
LINCSCP_61935 |
VCAP |
| 0.287662 |
4.948245e-20 |
975 |
Alpelisib |
LSM-4256 |
PIK3CA |
1.11uM |
24h |
LINCSCP_144863 |
LINCSCP_144863 |
MDAMB231 |
| 0.287656 |
4.958416e-20 |
975 |
Scriptaid |
LSM-2499 |
HDAC1 |
0.001uM |
6h |
LINCSCP_36385 |
LINCSCP_36385 |
MCF7 |
| 0.287572 |
5.088123e-20 |
975 |
CARGLUMIC ACID |
LSM-45453 |
CPS1 |
10uM |
24h |
LINCSCP_139842 |
LINCSCP_139842 |
MCF7 |
| -0.287477 |
5.239491e-20 |
975 |
Cerulenin |
LSM-43210 |
FASN |
10uM |
24h |
LINCSCP_37922 |
LINCSCP_37922 |
MCF7 |
| 0.286973 |
6.118876e-20 |
975 |
Imatinib |
LSM-1023 |
ABL1|BCR|CSF1R|KIT|PDGFRA|PDGFRB |
0.04uM |
3h |
LINCSCP_86459 |
LINCSCP_86459 |
BT20 |
| 0.286912 |
6.234942e-20 |
975 |
CHEMBL2143694 |
LSM-6585 |
|
10uM |
6h |
LINCSCP_16821 |
LINCSCP_16821 |
HA1E |
| 0.286908 |
6.242954e-20 |
975 |
Alizapride |
LSM-4953 |
DRD2 |
1.11uM |
24h |
LINCSCP_75199 |
LINCSCP_75199 |
A375 |
| 0.286889 |
6.279099e-20 |
975 |
Tegobuvir |
LSM-45236 |
|
0.12uM |
24h |
LINCSCP_89439 |
LINCSCP_89439 |
HA1E |
| 0.286571 |
6.924526e-20 |
975 |
noscapine |
|
|
0.04uM |
3h |
LINCSCP_130343 |
LINCSCP_130343 |
LNCAP |
| 0.286309 |
7.503149e-20 |
975 |
Resveratrol |
LSM-42917 |
PTGS1|PTGS2|SIRT1 |
0.12uM |
24h |
LINCSCP_128940 |
LINCSCP_128940 |
HUVEC |
| 0.28628 |
7.570728e-20 |
975 |
BRD-K45735142 |
LSM-6782 |
|
10uM |
6h |
LINCSCP_59347 |
LINCSCP_59347 |
VCAP |
| 0.286254 |
7.631811e-20 |
975 |
Brivanib |
LSM-5421 |
FGFR1|FGFR2|FGFR3|FGFR4|FLT1|FLT4|KDR |
10uM |
6h |
LINCSCP_20432 |
LINCSCP_20432 |
HCC515 |
| -0.286251 |
7.637860e-20 |
975 |
cortisone-acetate |
LSM-45387 |
TUBA1A|TUBA1B|TUBA1C|TUBA3E|TUBA4A|TUBB|TUBB1|TUBB2A|TUBB2B|TUBB3|TUBB4A|TUBB4B|TUBB6|TUBB8 |
3.33uM |
24h |
LINCSCP_143280 |
LINCSCP_143280 |
MCF7 |
| 0.286247 |
7.648249e-20 |
975 |
2-(2-Bromo-4-methyl-phenylamino)-pyrido[3,2-e][1,3]thiazin-4-one |
LSM-45312 |
|
3uM |
24h |
LINCSCP_55313 |
LINCSCP_55313 |
U937 |
| -0.286182 |
7.801709e-20 |
975 |
SAR245409 |
LSM-1174 |
|
0.04uM |
24h |
LINCSCP_128045 |
LINCSCP_128045 |
HUES3 |
| 0.286096 |
8.010341e-20 |
975 |
Vorinostat |
LSM-3828 |
HDAC1|HDAC2|HDAC3|HDAC6|HDAC8 |
0.01uM |
24h |
LINCSCP_201493 |
LINCSCP_201493 |
A549 |
| 0.286086 |
8.036046e-20 |
975 |
AC1NXRFO |
LSM-43270 |
|
0.1uM |
24h |
LINCSCP_35659 |
LINCSCP_35659 |
MCF7 |
| 0.28585 |
8.636747e-20 |
975 |
BRD-K69218883 |
LSM-41036 |
|
10uM |
24h |
LINCSCP_3608 |
LINCSCP_3608 |
A375 |
| 0.285649 |
9.187520e-20 |
975 |
MLS000589843 |
LSM-43120 |
|
0.01uM |
24h |
LINCSCP_55115 |
LINCSCP_55115 |
THP1 |
| 0.285577 |
9.391962e-20 |
975 |
Acetazolamide |
LSM-5543 |
CA1|CA12|CA14|CA2|CA4|CA7 |
3.33uM |
24h |
LINCSCP_75561 |
LINCSCP_75561 |
A375 |
| -0.285415 |
9.867630e-20 |
975 |
BRD-A80960055-001-01-7 |
LSM-5162 |
|
10uM |
6h |
LINCSCP_20385 |
LINCSCP_20385 |
HCC515 |
| 0.285302 |
1.021539e-19 |
975 |
CHEMBL2356693 |
LSM-6781 |
|
10uM |
6h |
LINCSCP_59326 |
LINCSCP_59326 |
VCAP |
| -0.285118 |
1.080461e-19 |
975 |
AC1MD3YP |
LSM-1801 |
EIF2S1 |
10uM |
24h |
LINCSCP_15012 |
LINCSCP_15012 |
HA1E |
| 0.285086 |
1.091305e-19 |
975 |
Yohimbine |
LSM-2779 |
ADRA2A|ADRA2B|ADRA2C|HTR1A|HTR1B|HTR1D|HTR2B |
0.12uM |
24h |
LINCSCP_71997 |
LINCSCP_71997 |
A375 |
| 0.285056 |
1.101029e-19 |
975 |
CHEMBL1327417 |
LSM-4729 |
|
10uM |
6h |
LINCSCP_211471 |
LINCSCP_211471 |
HA1E |
| 0.28502 |
1.113337e-19 |
975 |
Alectinib |
LSM-1202 |
ALK|RET |
1.11uM |
24h |
LINCSCP_150407 |
LINCSCP_150407 |
NPC.TAK |
| -0.285002 |
1.119555e-19 |
975 |
Ibuprofen |
LSM-1354 |
PTGS1|PTGS2 |
10uM |
24h |
LINCSCP_47267 |
LINCSCP_47267 |
PC3 |
| 0.284976 |
1.128267e-19 |
975 |
BRD-K40478655 |
LSM-10898 |
|
5uM |
24h |
LINCSCP_62149 |
LINCSCP_62149 |
VCAP |
| -0.284908 |
1.152004e-19 |
975 |
Diazoxide |
LSM-3639 |
KCNJ11 |
10uM |
6h |
LINCSCP_46170 |
LINCSCP_46170 |
PC3 |
| 0.284746 |
1.210407e-19 |
975 |
BRD-K77326001 |
LSM-41491 |
|
5uM |
24h |
LINCSCP_64321 |
LINCSCP_64321 |
VCAP |
| 0.284733 |
1.215250e-19 |
975 |
BRD-K31856043 |
LSM-39013 |
|
10uM |
6h |
LINCSCP_20605 |
LINCSCP_20605 |
HCC515 |
| 0.284672 |
1.237956e-19 |
975 |
BRD-K41871066 |
LSM-39582 |
|
10uM |
24h |
LINCSCP_9030 |
LINCSCP_9030 |
A549 |
| -0.284558 |
1.281921e-19 |
975 |
Mebendazole |
LSM-3749 |
|
5uM |
24h |
LINCSCP_67613 |
LINCSCP_67613 |
MCF7 |
| -0.284481 |
1.312083e-19 |
975 |
naftidrofuryl |
LSM-45485 |
|
3.33uM |
24h |
LINCSCP_76386 |
LINCSCP_76386 |
A375 |
| 0.284424 |
1.335300e-19 |
975 |
BRD-K82004089 |
LSM-13434 |
|
5uM |
24h |
LINCSCP_62694 |
LINCSCP_62694 |
VCAP |
| 0.284323 |
1.376865e-19 |
975 |
4-(Trans-4-butylcyclohexyl)benzoic acid |
LSM-4640 |
|
10uM |
6h |
LINCSCP_16315 |
LINCSCP_16315 |
HA1E |
| 0.284241 |
1.411733e-19 |
975 |
BRD-K36910796 |
LSM-15073 |
|
0.5uM |
24h |
LINCSCP_37908 |
LINCSCP_37908 |
MCF7 |
| 0.284218 |
1.421700e-19 |
975 |
BMS-345541 |
LSM-1028 |
IKBKB |
0.5uM |
24h |
LINCSCP_11655 |
LINCSCP_11655 |
BT20 |
| 0.28419 |
1.433940e-19 |
975 |
BRD-M60886831 |
LSM-45052 |
|
5uM |
24h |
LINCSCP_64047 |
LINCSCP_64047 |
VCAP |
| -0.284042 |
1.499894e-19 |
975 |
BRD-K29396015 |
LSM-38869 |
|
10uM |
6h |
LINCSCP_49114 |
LINCSCP_49114 |
PC3 |
| 0.284016 |
1.511724e-19 |
975 |
Cholic acid |
LSM-5541 |
CES1|FECH|PLA2G1B |
1.11uM |
24h |
LINCSCP_75556 |
LINCSCP_75556 |
A375 |
| 0.283979 |
1.528744e-19 |
975 |
Dimethisoquin |
LSM-3647 |
|
10uM |
24h |
LINCSCP_241662 |
LINCSCP_241662 |
MCF7 |
| 0.283878 |
1.576514e-19 |
975 |
BRD-K71714567 |
LSM-41172 |
|
0.5uM |
6h |
LINCSCP_38085 |
LINCSCP_38085 |
MCF7 |
| 0.2837 |
1.664082e-19 |
975 |
GSK-1904529A |
LSM-1134 |
IGF1R|INSR |
10uM |
24h |
LINCSCP_24689 |
LINCSCP_24689 |
HS578T |
| -0.283692 |
1.668051e-19 |
975 |
Colchicine |
LSM-5199 |
TUBA1A|TUBA1B|TUBA1C|TUBA3E|TUBA4A|TUBB|TUBB1|TUBB2A|TUBB2B|TUBB3|TUBB4A|TUBB4B|TUBB6|TUBB8 |
10uM |
24h |
LINCSCP_34261 |
LINCSCP_34261 |
MCF7 |
| 0.283574 |
1.728801e-19 |
975 |
BRD-K31671785 |
LSM-10347 |
|
5uM |
24h |
LINCSCP_61761 |
LINCSCP_61761 |
VCAP |
| -0.283517 |
1.759108e-19 |
975 |
Trimethoprim |
LSM-5246 |
|
1.11uM |
24h |
LINCSCP_104988 |
LINCSCP_104988 |
HELA |
| 0.283513 |
1.761355e-19 |
975 |
SMR000178575 |
LSM-2708 |
|
10uM |
6h |
LINCSCP_20436 |
LINCSCP_20436 |
HCC515 |
| -0.28347 |
1.784544e-19 |
975 |
BMS-754807 |
LSM-6218 |
IGF1R|INSR |
10uM |
6h |
LINCSCP_40185 |
LINCSCP_40185 |
NCIH508 |
| 0.283404 |
1.820619e-19 |
975 |
Acetazolamide |
LSM-5543 |
CA1|CA12|CA14|CA2|CA4|CA7 |
10uM |
24h |
LINCSCP_75560 |
LINCSCP_75560 |
A375 |
| -0.283387 |
1.830053e-19 |
975 |
BRD-K74316684 |
LSM-41315 |
|
10uM |
24h |
LINCSCP_9073 |
LINCSCP_9073 |
A549 |
| 0.283346 |
1.852548e-19 |
975 |
Thiabendazole |
LSM-3741 |
|
10uM |
24h |
LINCSCP_32931 |
LINCSCP_32931 |
MCF7 |
| 0.283217 |
1.926567e-19 |
975 |
Wortmannin |
LSM-3947 |
PIK3CA|PIK3CG|PLK1 |
0.001uM |
24h |
LINCSCP_201090 |
LINCSCP_201090 |
A549 |
| -0.283186 |
1.944668e-19 |
975 |
BRD-K32593492 |
LSM-39065 |
|
10uM |
6h |
LINCSCP_49118 |
LINCSCP_49118 |
PC3 |
| -0.283146 |
1.968624e-19 |
975 |
Temoporfin |
LSM-45995 |
|
10uM |
24h |
LINCSCP_137028 |
LINCSCP_137028 |
MCF7 |
| -0.283108 |
1.991080e-19 |
975 |
RU-24969 |
LSM-1976 |
HTR1A|HTR1B|HTR6 |
10uM |
24h |
LINCSCP_52823 |
LINCSCP_52823 |
SKB |
| -0.283104 |
1.994041e-19 |
975 |
BRD-K38841486 |
LSM-39409 |
|
10uM |
6h |
LINCSCP_65819 |
LINCSCP_65819 |
VCAP |
| 0.282931 |
2.100694e-19 |
975 |
Gimeracil |
LSM-45923 |
|
0.04uM |
24h |
LINCSCP_72028 |
LINCSCP_72028 |
A375 |
| -0.282877 |
2.135656e-19 |
975 |
Rabusertib |
LSM-36359 |
CHEK1 |
3.33uM |
24h |
LINCSCP_149088 |
LINCSCP_149088 |
NPC |
| 0.282875 |
2.136748e-19 |
975 |
138402-11-6 |
LSM-3338 |
AGTR1 |
10uM |
24h |
LINCSCP_240697 |
LINCSCP_240697 |
MCF7 |
| -0.282872 |
2.138952e-19 |
975 |
Corvasal |
LSM-25617 |
|
0.04uM |
24h |
LINCSCP_107216 |
LINCSCP_107216 |
HELA |
| 0.282845 |
2.156405e-19 |
975 |
MLS003129264 |
LSM-7247 |
|
5uM |
24h |
LINCSCP_60535 |
LINCSCP_60535 |
VCAP |
| 0.282751 |
2.218432e-19 |
975 |
BRD-K54577741 |
LSM-40259 |
|
10uM |
6h |
LINCSCP_279492 |
LINCSCP_279492 |
PC3 |
| 0.282634 |
2.298512e-19 |
975 |
Yohimbine |
LSM-2779 |
ADRA2A|ADRA2B|ADRA2C|HTR1A|HTR1B|HTR1D|HTR2B |
0.37uM |
24h |
LINCSCP_102121 |
LINCSCP_102121 |
HELA |
| -0.282633 |
2.299042e-19 |
975 |
Withaferin A |
LSM-6685 |
IKBKB|NAMPT |
10uM |
24h |
LINCSCP_301315 |
LINCSCP_301315 |
VCAP |
| 0.282543 |
2.362320e-19 |
975 |
3-(4-Pyridyl)indole |
LSM-4569 |
ROCK1 |
0.37uM |
24h |
LINCSCP_140228 |
LINCSCP_140228 |
MCF7 |
| -0.282512 |
2.384603e-19 |
975 |
BRD-K47512679 |
LSM-39902 |
|
10uM |
24h |
LINCSCP_3579 |
LINCSCP_3579 |
A375 |
| 0.282329 |
2.520377e-19 |
975 |
BRD-K22787051 |
LSM-9813 |
|
5uM |
24h |
LINCSCP_48236 |
LINCSCP_48236 |
PC3 |
| 0.282206 |
2.615463e-19 |
975 |
BRD-K20310932 |
LSM-9669 |
|
5uM |
24h |
LINCSCP_61745 |
LINCSCP_61745 |
VCAP |
| 0.282201 |
2.620041e-19 |
975 |
Tedizolid |
LSM-45778 |
|
0.04uM |
24h |
LINCSCP_76259 |
LINCSCP_76259 |
A375 |
| 0.282171 |
2.643301e-19 |
975 |
SPECTRUM_001131 |
LSM-2307 |
|
10uM |
24h |
LINCSCP_240682 |
LINCSCP_240682 |
MCF7 |
| 0.282067 |
2.727611e-19 |
975 |
TPCA-1 |
LSM-1136 |
IKBKB |
0.1uM |
24h |
LINCSCP_251791 |
LINCSCP_251791 |
MCF7 |
| 0.281921 |
2.850906e-19 |
975 |
BRD-K19826330 |
LSM-9628 |
|
5uM |
24h |
LINCSCP_61569 |
LINCSCP_61569 |
VCAP |
| -0.28189 |
2.877634e-19 |
975 |
FK888 |
LSM-3876 |
TACR1 |
3.33uM |
24h |
LINCSCP_173160 |
LINCSCP_173160 |
YAPC |
| 0.281701 |
3.045779e-19 |
975 |
Lapatinib |
LSM-1051 |
EGFR|ERBB2 |
1.11uM |
24h |
LINCSCP_145564 |
LINCSCP_145564 |
MDAMB231 |
| -0.281669 |
3.075281e-19 |
975 |
CHEMBL2361787 |
LSM-13210 |
|
10uM |
24h |
LINCSCP_28298 |
LINCSCP_28298 |
HT29 |
| 0.281586 |
3.153271e-19 |
975 |
FK 866 |
LSM-43216 |
NAMPT |
0.1uM |
24h |
LINCSCP_30584 |
LINCSCP_30584 |
MCF7 |
| -0.281556 |
3.181621e-19 |
975 |
Temoporfin |
LSM-45995 |
|
10uM |
24h |
LINCSCP_103655 |
LINCSCP_103655 |
HELA |
| -0.281551 |
3.186110e-19 |
975 |
SCHEMBL618594 |
LSM-1070 |
|
10uM |
24h |
LINCSCP_240240 |
LINCSCP_240240 |
MCF7 |
| 0.281485 |
3.250334e-19 |
975 |
Zonisamide |
LSM-3062 |
CA1|CA12|CA7|SCN11A|SCN1A|SCN2A|SCN3A|SCN4A|SCN5A|SCN9A |
10uM |
6h |
LINCSCP_236437 |
LINCSCP_236437 |
MCF7 |
| 0.28142 |
3.315124e-19 |
975 |
NU-7441 |
LSM-1061 |
PRKDC |
0.1uM |
24h |
LINCSCP_38911 |
LINCSCP_38911 |
MDAMB231 |
| -0.281366 |
3.368791e-19 |
975 |
D-64131 |
LSM-2592 |
TUBB |
3uM |
24h |
LINCSCP_37449 |
LINCSCP_37449 |
MCF7 |
| 0.281189 |
3.553215e-19 |
975 |
BRD-K16811158 |
LSM-38156 |
|
5uM |
24h |
LINCSCP_64251 |
LINCSCP_64251 |
VCAP |
| -0.281152 |
3.592680e-19 |
975 |
423735-93-7 |
LSM-3308 |
|
10uM |
6h |
LINCSCP_13538 |
LINCSCP_13538 |
H1299 |
| -0.281081 |
3.670291e-19 |
975 |
AC1NS4S0 |
LSM-43073 |
ATP2A1 |
10uM |
6h |
LINCSCP_43712 |
LINCSCP_43712 |
OV7 |
| 0.281061 |
3.692795e-19 |
975 |
BRD-K13779607 |
LSM-9262 |
|
5uM |
24h |
LINCSCP_61944 |
LINCSCP_61944 |
VCAP |
| -0.281057 |
3.697362e-19 |
975 |
BRD-K18170480 |
LSM-38234 |
|
1uM |
24h |
LINCSCP_37879 |
LINCSCP_37879 |
MCF7 |
| -0.28091 |
3.863405e-19 |
975 |
TUL_XX087 |
LSM-36794 |
|
0.001uM |
24h |
LINCSCP_41935 |
LINCSCP_41935 |
NOMO1 |
| 0.280812 |
3.978583e-19 |
975 |
BRD-K83920942 |
LSM-13558 |
|
5uM |
24h |
LINCSCP_62325 |
LINCSCP_62325 |
VCAP |
| 0.280727 |
4.081980e-19 |
975 |
BRD-K36513323 |
LSM-10634 |
|
5uM |
24h |
LINCSCP_61985 |
LINCSCP_61985 |
VCAP |
| 0.28057 |
4.278454e-19 |
975 |
848193-68-0 |
LSM-6271 |
SIRT1 |
3.33uM |
24h |
LINCSCP_114108 |
LINCSCP_114108 |
HME1 |
| 0.280473 |
4.404683e-19 |
975 |
GSK-319347A |
LSM-1216 |
IKBKG |
5uM |
6h |
LINCSCP_55493 |
LINCSCP_55493 |
U937 |
| -0.280436 |
4.453995e-19 |
975 |
Marimastat |
LSM-45636 |
|
10uM |
24h |
LINCSCP_90513 |
LINCSCP_90513 |
HA1E |
| 0.280245 |
4.716057e-19 |
975 |
Alpelisib |
LSM-4256 |
PIK3CA |
0.04uM |
3h |
LINCSCP_163420 |
LINCSCP_163420 |
SKBR3 |
| 0.280197 |
4.784560e-19 |
975 |
SR 33805 oxalate |
LSM-45933 |
|
0.12uM |
24h |
LINCSCP_75552 |
LINCSCP_75552 |
A375 |
| 0.280146 |
4.857474e-19 |
975 |
Lapatinib |
LSM-1051 |
EGFR|ERBB2 |
0.12uM |
24h |
LINCSCP_130006 |
LINCSCP_130006 |
LNCAP |
| -0.279929 |
5.184115e-19 |
975 |
Tofacitinib (CP-690550) Citrate |
LSM-45505 |
|
10uM |
24h |
LINCSCP_102184 |
LINCSCP_102184 |
HELA |
| -0.279901 |
5.226730e-19 |
975 |
AB00540134 |
LSM-4868 |
|
10uM |
24h |
LINCSCP_261390 |
LINCSCP_261390 |
NPC |
| -0.27988 |
5.260655e-19 |
975 |
MLS002729050 |
LSM-1996 |
|
10uM |
24h |
LINCSCP_4894 |
LINCSCP_4894 |
A549 |
| 0.279861 |
5.290854e-19 |
975 |
Niacin |
LSM-4676 |
HCAR2|HCAR3 |
0.12uM |
24h |
LINCSCP_123239 |
LINCSCP_123239 |
HT29 |
| 0.279706 |
5.541549e-19 |
975 |
AC1MEEHF |
LSM-6366 |
|
10uM |
6h |
LINCSCP_16766 |
LINCSCP_16766 |
HA1E |
| 0.279624 |
5.677911e-19 |
975 |
Clonidine |
LSM-4223 |
ADRA2A|ADRA2B|ADRA2C |
10uM |
24h |
LINCSCP_18993 |
LINCSCP_18993 |
HCC515 |
| 0.279609 |
5.704158e-19 |
975 |
ZSTK 474 |
LSM-1053 |
PIK3CG |
0.04uM |
3h |
LINCSCP_145914 |
LINCSCP_145914 |
MDAMB231 |
| 0.279583 |
5.749291e-19 |
975 |
AMD-070 (hydrochloride) |
LSM-45591 |
|
0.04uM |
24h |
LINCSCP_75547 |
LINCSCP_75547 |
A375 |
| -0.279578 |
5.756440e-19 |
975 |
GSK-0660 |
LSM-6014 |
PPARD |
10uM |
24h |
LINCSCP_271221 |
LINCSCP_271221 |
PC3 |
| -0.279566 |
5.778245e-19 |
975 |
Simvastatin |
LSM-2492 |
HMGCR |
0.37uM |
24h |
LINCSCP_154047 |
LINCSCP_154047 |
PC3 |
| -0.279344 |
6.172741e-19 |
975 |
BRD-A24396574-001-01-5 |
LSM-5006 |
|
10uM |
3h |
LINCSCP_133031 |
LINCSCP_133031 |
MCF7 |
| 0.279336 |
6.188796e-19 |
975 |
BRD-K82794234 |
LSM-13485 |
|
5uM |
24h |
LINCSCP_62324 |
LINCSCP_62324 |
VCAP |
| 0.279285 |
6.283521e-19 |
975 |
BRD-K31931379 |
LSM-10366 |
|
5uM |
24h |
LINCSCP_302090 |
LINCSCP_302090 |
VCAP |
| 0.279222 |
6.402093e-19 |
975 |
Spironolactone |
LSM-4018 |
NR3C2 |
10uM |
6h |
LINCSCP_17020 |
LINCSCP_17020 |
HA1E |
| -0.279133 |
6.574617e-19 |
975 |
Withaferin A |
LSM-6685 |
IKBKB|NAMPT |
1uM |
6h |
LINCSCP_9874 |
LINCSCP_9874 |
A549 |
| 0.279093 |
6.653789e-19 |
975 |
MW-SHH-61 |
LSM-44611 |
|
0.5uM |
6h |
LINCSCP_9930 |
LINCSCP_9930 |
A549 |
| 0.279067 |
6.705694e-19 |
975 |
CP-724714 |
LSM-42777 |
ERBB2 |
0.37uM |
24h |
LINCSCP_68964 |
LINCSCP_68964 |
A375 |
| -0.278646 |
7.600285e-19 |
975 |
TUL_XX087 |
LSM-36794 |
|
0.001uM |
6h |
LINCSCP_42019 |
LINCSCP_42019 |
NOMO1 |
| -0.278542 |
7.839091e-19 |
975 |
Lexibulin |
LSM-6232 |
TUBA1A|TUBA1B|TUBA1C|TUBA3E|TUBA4A|TUBB|TUBB1|TUBB2A|TUBB2B|TUBB3|TUBB4A|TUBB4B|TUBB6|TUBB8 |
3.33uM |
24h |
LINCSCP_135771 |
LINCSCP_135771 |
MCF7 |
| 0.278436 |
8.089321e-19 |
975 |
Perhexiline |
LSM-4353 |
CPT1A|CPT2 |
0.001uM |
24h |
LINCSCP_250407 |
LINCSCP_250407 |
MCF7 |
| -0.278433 |
8.096118e-19 |
975 |
NMS-1286937 |
LSM-45818 |
|
0.12uM |
24h |
LINCSCP_141873 |
LINCSCP_141873 |
MCF7 |
| 0.278333 |
8.341069e-19 |
975 |
ZSTK 474 |
LSM-1053 |
PIK3CG |
0.12uM |
3h |
LINCSCP_86434 |
LINCSCP_86434 |
BT20 |
| -0.278272 |
8.494530e-19 |
975 |
MLS002264430 |
LSM-3594 |
|
10uM |
24h |
LINCSCP_177898 |
LINCSCP_177898 |
A375 |
| 0.278218 |
8.631405e-19 |
975 |
BRD-K70399291 |
LSM-12723 |
|
5uM |
24h |
LINCSCP_305884 |
LINCSCP_305884 |
VCAP |
| -0.278074 |
9.008867e-19 |
975 |
BRD-K80058284 |
LSM-41639 |
|
10uM |
24h |
LINCSCP_3632 |
LINCSCP_3632 |
A375 |
| 0.278029 |
9.128794e-19 |
975 |
Varenicline |
LSM-5358 |
CHRNA4 |
10uM |
6h |
LINCSCP_16271 |
LINCSCP_16271 |
HA1E |
| -0.277863 |
9.588608e-19 |
975 |
Norfloxacin |
LSM-5286 |
|
3.33uM |
24h |
LINCSCP_154465 |
LINCSCP_154465 |
PC3 |
| -0.277852 |
9.621214e-19 |
975 |
AZD-1775 |
LSM-1153 |
WEE1 |
10uM |
24h |
LINCSCP_140087 |
LINCSCP_140087 |
MCF7 |
| -0.277845 |
9.642419e-19 |
975 |
MLS002703099 |
LSM-2090 |
|
10uM |
24h |
LINCSCP_31568 |
LINCSCP_31568 |
MCF7 |
| 0.277823 |
9.704062e-19 |
975 |
Nilotinib |
LSM-1099 |
ABL1|BCR|KIT |
3.33uM |
3h |
LINCSCP_132493 |
LINCSCP_132493 |
MCF7 |
| -0.277802 |
9.765135e-19 |
975 |
Paricalcitol |
LSM-45519 |
VDR |
1.11uM |
24h |
LINCSCP_105971 |
LINCSCP_105971 |
HELA |
| 0.277708 |
1.004130e-18 |
975 |
Seliciclib |
LSM-1001 |
CDK1|CDK2|CDK5|CDK7|CDK9 |
0.37uM |
24h |
LINCSCP_130628 |
LINCSCP_130628 |
MCF10A |
| 0.277562 |
1.048426e-18 |
975 |
BRD-K97101742 |
LSM-14393 |
|
5uM |
24h |
LINCSCP_62333 |
LINCSCP_62333 |
VCAP |
| 0.277518 |
1.062211e-18 |
975 |
SCHEMBL1564574 |
LSM-1006 |
CHEK1|CHEK2 |
0.5uM |
24h |
LINCSCP_11704 |
LINCSCP_11704 |
BT20 |
| 0.277514 |
1.063538e-18 |
975 |
Naltrexone-HCl |
LSM-1850 |
OPRD1|OPRK1|OPRM1 |
10uM |
24h |
LINCSCP_44701 |
LINCSCP_44701 |
PC3 |
| 0.277484 |
1.072877e-18 |
975 |
MLS002264499 |
LSM-1853 |
|
10uM |
6h |
LINCSCP_57609 |
LINCSCP_57609 |
VCAP |
| 0.277413 |
1.095588e-18 |
975 |
Latanoprost |
LSM-43170 |
PTGFR |
3.33uM |
24h |
LINCSCP_102856 |
LINCSCP_102856 |
HELA |
| -0.277267 |
1.143988e-18 |
975 |
BRD-K53325797 |
LSM-45342 |
|
0.5uM |
24h |
LINCSCP_222167 |
LINCSCP_222167 |
HL60 |
| -0.277254 |
1.148507e-18 |
975 |
Afatinib |
LSM-43226 |
EGFR|ERBB2|ERBB4 |
10uM |
24h |
LINCSCP_140879 |
LINCSCP_140879 |
MCF7 |
| 0.277228 |
1.157467e-18 |
975 |
Ropinirole |
LSM-2351 |
DRD2|DRD3|DRD4 |
10uM |
6h |
LINCSCP_240875 |
LINCSCP_240875 |
MCF7 |
| -0.277178 |
1.174733e-18 |
975 |
BRD-A24396574-001-01-5 |
LSM-5006 |
|
3.33uM |
3h |
LINCSCP_113446 |
LINCSCP_113446 |
HME1 |
| 0.277023 |
1.229704e-18 |
975 |
Fenofibrate |
LSM-3107 |
PPARA |
10uM |
24h |
LINCSCP_243493 |
LINCSCP_243493 |
MCF7 |
| 0.277008 |
1.235188e-18 |
975 |
BRD-K64864583 |
LSM-12390 |
|
5uM |
24h |
LINCSCP_61806 |
LINCSCP_61806 |
VCAP |
| -0.276981 |
1.245178e-18 |
975 |
Erbstatin Analog |
LSM-43038 |
EGFR |
10uM |
24h |
LINCSCP_47309 |
LINCSCP_47309 |
PC3 |
| 0.276906 |
1.273042e-18 |
975 |
BRD-K90208654 |
LSM-13993 |
|
5uM |
24h |
LINCSCP_62062 |
LINCSCP_62062 |
VCAP |
| 0.27686 |
1.290178e-18 |
975 |
BRD-K69760878 |
LSM-41068 |
|
10uM |
24h |
LINCSCP_48567 |
LINCSCP_48567 |
PC3 |
| -0.276734 |
1.339083e-18 |
975 |
D-64406 |
LSM-2606 |
|
10uM |
24h |
LINCSCP_52742 |
LINCSCP_52742 |
SKB |
| -0.276602 |
1.392259e-18 |
975 |
KX2-391 |
LSM-45890 |
SRC |
0.37uM |
24h |
LINCSCP_137499 |
LINCSCP_137499 |
MCF7 |
| -0.276532 |
1.421622e-18 |
975 |
STK178014 |
LSM-43108 |
|
50uM |
6h |
LINCSCP_21269 |
LINCSCP_21269 |
HCT116 |
| 0.27646 |
1.451899e-18 |
975 |
CHEMBL3183285 |
LSM-10801 |
|
5uM |
24h |
LINCSCP_61987 |
LINCSCP_61987 |
VCAP |
| -0.276408 |
1.474548e-18 |
975 |
SCHEMBL2231351 |
LSM-36442 |
|
0.01uM |
24h |
LINCSCP_41943 |
LINCSCP_41943 |
NOMO1 |
| 0.276376 |
1.488381e-18 |
975 |
KW-2449 |
LSM-42803 |
ABL1|AURKA|AURKB|FLT3 |
10uM |
24h |
LINCSCP_129500 |
LINCSCP_129500 |
JURKAT |
| -0.276371 |
1.490569e-18 |
975 |
CHEMBL490083 |
LSM-2547 |
|
10uM |
24h |
LINCSCP_45295 |
LINCSCP_45295 |
PC3 |
| -0.276337 |
1.505749e-18 |
975 |
MLS002276510 |
LSM-3272 |
|
10uM |
24h |
LINCSCP_31626 |
LINCSCP_31626 |
MCF7 |
| -0.276294 |
1.524806e-18 |
975 |
Metergoline |
LSM-3265 |
HTR1A|HTR2A |
10uM |
24h |
LINCSCP_52761 |
LINCSCP_52761 |
SKB |
| 0.276257 |
1.541550e-18 |
975 |
Brinaldix |
LSM-5337 |
|
10uM |
24h |
LINCSCP_34273 |
LINCSCP_34273 |
MCF7 |
| 0.276164 |
1.584341e-18 |
975 |
GSK-1904529A |
LSM-1134 |
IGF1R|INSR |
0.04uM |
24h |
LINCSCP_151272 |
LINCSCP_151272 |
PC3 |
| 0.276144 |
1.593579e-18 |
975 |
BRD-K71611609 |
LSM-12812 |
|
5uM |
6h |
LINCSCP_62575 |
LINCSCP_62575 |
VCAP |
| 0.276032 |
1.646803e-18 |
975 |
BRD-K69747917 |
LSM-14908 |
|
5uM |
24h |
LINCSCP_64211 |
LINCSCP_64211 |
VCAP |
| -0.275999 |
1.663114e-18 |
975 |
PHA-767491 |
LSM-6304 |
|
3.33uM |
24h |
LINCSCP_133455 |
LINCSCP_133455 |
MCF7 |
| -0.275927 |
1.698602e-18 |
975 |
BRD-K73276569 |
LSM-41250 |
|
10uM |
24h |
LINCSCP_35357 |
LINCSCP_35357 |
MCF7 |
| -0.275898 |
1.713023e-18 |
975 |
BRD-K43579410 |
LSM-39667 |
|
1uM |
24h |
LINCSCP_312474 |
LINCSCP_312474 |
VCAP |
| 0.275851 |
1.737044e-18 |
975 |
Temefos |
LSM-3148 |
|
10uM |
24h |
LINCSCP_32909 |
LINCSCP_32909 |
MCF7 |
| 0.275806 |
1.760355e-18 |
975 |
Piperacillin |
LSM-5924 |
|
10uM |
6h |
LINCSCP_27343 |
LINCSCP_27343 |
HT29 |
| 0.275764 |
1.782061e-18 |
975 |
BRD-K56176052 |
LSM-11824 |
|
5uM |
24h |
LINCSCP_62299 |
LINCSCP_62299 |
VCAP |
| 0.275741 |
1.793938e-18 |
975 |
SAN1_004207 |
LSM-36734 |
|
10uM |
6h |
LINCSCP_16895 |
LINCSCP_16895 |
HA1E |
| -0.275703 |
1.814101e-18 |
975 |
BRD-K35638681 |
LSM-39222 |
|
10uM |
24h |
LINCSCP_46454 |
LINCSCP_46454 |
PC3 |
| 0.275599 |
1.870410e-18 |
975 |
SCHEMBL10028376 |
LSM-36648 |
|
10uM |
24h |
LINCSCP_10701 |
LINCSCP_10701 |
ASC |
| 0.275569 |
1.887015e-18 |
975 |
BRD-K95899688 |
LSM-14310 |
|
5uM |
24h |
LINCSCP_62706 |
LINCSCP_62706 |
VCAP |
| -0.275536 |
1.905437e-18 |
975 |
SPECTRUM_000281 |
LSM-4326 |
|
10uM |
24h |
LINCSCP_284828 |
LINCSCP_284828 |
SKB |
| 0.275525 |
1.911550e-18 |
975 |
Hypericin |
LSM-2650 |
|
0.12uM |
24h |
LINCSCP_71287 |
LINCSCP_71287 |
A375 |
| 0.27542 |
1.971567e-18 |
975 |
MLS-0435542.0001 |
LSM-1937 |
|
10uM |
6h |
LINCSCP_21807 |
LINCSCP_21807 |
HEPG2 |
| 0.275389 |
1.989630e-18 |
975 |
SUGA1_010064 |
LSM-36686 |
|
10uM |
6h |
LINCSCP_22365 |
LINCSCP_22365 |
HEPG2 |
| -0.275216 |
2.092851e-18 |
975 |
BRD-K39561907 |
LSM-39452 |
|
0.5uM |
24h |
LINCSCP_312463 |
LINCSCP_312463 |
VCAP |
| -0.275059 |
2.191468e-18 |
975 |
CHEMBL1394132 |
LSM-3090 |
|
10uM |
6h |
LINCSCP_267918 |
LINCSCP_267918 |
PC3 |
| -0.275002 |
2.228718e-18 |
975 |
Amuvatinib |
LSM-1118 |
FLT3|KIT|MET|PDGFRA |
10uM |
24h |
LINCSCP_39454 |
LINCSCP_39454 |
MDAMB231 |
| 0.274988 |
2.237949e-18 |
975 |
CHEMBL2131967 |
LSM-42358 |
|
10uM |
6h |
LINCSCP_22443 |
LINCSCP_22443 |
HEPG2 |
| 0.274914 |
2.286551e-18 |
975 |
Alpelisib |
LSM-4256 |
PIK3CA |
0.12uM |
3h |
LINCSCP_163419 |
LINCSCP_163419 |
SKBR3 |
| 0.274873 |
2.314832e-18 |
975 |
EX-8678 |
LSM-1147 |
|
0.12uM |
3h |
LINCSCP_164124 |
LINCSCP_164124 |
SKBR3 |
| 0.27477 |
2.385148e-18 |
975 |
NSC95397 |
LSM-3521 |
|
10uM |
6h |
LINCSCP_55522 |
LINCSCP_55522 |
U937 |
| 0.274714 |
2.424594e-18 |
975 |
CHEMBL2135770 |
LSM-38343 |
|
3uM |
6h |
LINCSCP_37775 |
LINCSCP_37775 |
MCF7 |
| 0.274412 |
2.648868e-18 |
975 |
Seliciclib |
LSM-1001 |
CDK1|CDK2|CDK5|CDK7|CDK9 |
1.11uM |
24h |
LINCSCP_130627 |
LINCSCP_130627 |
MCF10A |
| 0.274298 |
2.738569e-18 |
975 |
FPA1_000112 |
LSM-36718 |
|
10uM |
6h |
LINCSCP_211462 |
LINCSCP_211462 |
HA1E |
| -0.274066 |
2.930224e-18 |
975 |
CHEMBL1270605 |
LSM-3968 |
|
10uM |
6h |
LINCSCP_225507 |
LINCSCP_225507 |
HT29 |
| 0.273938 |
3.042203e-18 |
975 |
Indoprofen |
LSM-1564 |
PTGS1|PTGS2 |
0.12uM |
24h |
LINCSCP_122564 |
LINCSCP_122564 |
HT29 |
| -0.273916 |
3.061070e-18 |
975 |
Sulfisoxazole |
LSM-3120 |
|
10uM |
24h |
LINCSCP_47530 |
LINCSCP_47530 |
PC3 |
| -0.273893 |
3.081925e-18 |
975 |
13-Hydroxy-8,14,19-trimethoxy-4,10,12,16-tetramethyl-3,20,22-trioxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18-pentaen-9-yl carbamate |
LSM-42815 |
HSP90AA1 |
0.1uM |
24h |
LINCSCP_235583 |
LINCSCP_235583 |
MCF7 |
| 0.273845 |
3.125639e-18 |
975 |
AC1MG7IW |
LSM-4330 |
|
10uM |
6h |
LINCSCP_16219 |
LINCSCP_16219 |
HA1E |
| 0.27381 |
3.157452e-18 |
975 |
GAP-134 (Hydrochloride) |
LSM-45532 |
|
0.12uM |
24h |
LINCSCP_102146 |
LINCSCP_102146 |
HELA |
| 0.273808 |
3.159222e-18 |
975 |
BRD-M56188090 |
LSM-45048 |
|
5uM |
24h |
LINCSCP_64045 |
LINCSCP_64045 |
VCAP |
| -0.273711 |
3.249625e-18 |
975 |
BRD-K09068728 |
LSM-8979 |
|
10uM |
24h |
LINCSCP_3521 |
LINCSCP_3521 |
A375 |
| -0.273706 |
3.255132e-18 |
975 |
SMR000076922 |
LSM-3142 |
|
10uM |
6h |
LINCSCP_240127 |
LINCSCP_240127 |
MCF7 |
| -0.273644 |
3.313676e-18 |
975 |
Diflunisal |
LSM-2490 |
PTGS1|PTGS2 |
10uM |
24h |
LINCSCP_47302 |
LINCSCP_47302 |
PC3 |
| 0.273641 |
3.317396e-18 |
975 |
ST51005413 |
LSM-4948 |
|
10uM |
6h |
LINCSCP_51243 |
LINCSCP_51243 |
RMUGS |
| -0.273301 |
3.662525e-18 |
975 |
Cimetidine |
LSM-2404 |
HRH2 |
0.37uM |
24h |
LINCSCP_92520 |
LINCSCP_92520 |
HA1E |
| -0.273282 |
3.682573e-18 |
975 |
Withaferin A |
LSM-6685 |
IKBKB|NAMPT |
10uM |
24h |
LINCSCP_67406 |
LINCSCP_67406 |
MCF7 |
| 0.273252 |
3.714858e-18 |
975 |
CHEMBL565584 |
LSM-43004 |
|
10uM |
6h |
LINCSCP_20439 |
LINCSCP_20439 |
HCC515 |
| 0.273182 |
3.791408e-18 |
975 |
BRD-K98993678 |
LSM-14506 |
|
5uM |
24h |
LINCSCP_62337 |
LINCSCP_62337 |
VCAP |
| -0.273163 |
3.811963e-18 |
975 |
Nafcillin |
LSM-2402 |
CYP1A2|CYP3A4|SLC22A6 |
10uM |
24h |
LINCSCP_47299 |
LINCSCP_47299 |
PC3 |
| 0.273092 |
3.891900e-18 |
975 |
SCHEMBL3958507 |
LSM-5245 |
COQ8B|EGFR |
1.11uM |
24h |
LINCSCP_151113 |
LINCSCP_151113 |
PC3 |
| -0.272909 |
4.103895e-18 |
975 |
Methyl beta-carboline-3 carboxylate |
LSM-2630 |
|
10uM |
24h |
LINCSCP_52873 |
LINCSCP_52873 |
SKB |
| 0.272872 |
4.148572e-18 |
975 |
Imatinib |
LSM-1023 |
ABL1|BCR|CSF1R|KIT|PDGFRA|PDGFRB |
1.11uM |
3h |
LINCSCP_130376 |
LINCSCP_130376 |
LNCAP |
| 0.272862 |
4.160903e-18 |
975 |
BRD-K62951188 |
LSM-12255 |
|
5uM |
24h |
LINCSCP_61631 |
LINCSCP_61631 |
VCAP |
| -0.272606 |
4.481032e-18 |
975 |
BRD-K07569193 |
LSM-8880 |
|
1uM |
24h |
LINCSCP_41706 |
LINCSCP_41706 |
NKDBA |
| 0.272451 |
4.687033e-18 |
975 |
Emedastine |
LSM-5331 |
HRH1 |
10uM |
24h |
LINCSCP_74488 |
LINCSCP_74488 |
A375 |
| 0.272448 |
4.691709e-18 |
975 |
MLN 2480 |
LSM-45644 |
ARAF|BRAF|RAF1 |
0.04uM |
24h |
LINCSCP_75583 |
LINCSCP_75583 |
A375 |
| 0.272287 |
4.915211e-18 |
975 |
SC_I_004 |
LSM-45332 |
|
10uM |
6h |
LINCSCP_16291 |
LINCSCP_16291 |
HA1E |
| -0.272281 |
4.923998e-18 |
975 |
Fludrocortisone |
LSM-1510 |
NR3C2 |
10uM |
24h |
LINCSCP_243377 |
LINCSCP_243377 |
MCF7 |
| 0.272258 |
4.956787e-18 |
975 |
BRD-K14614387-001-01-8 |
LSM-38030 |
|
0.5uM |
24h |
LINCSCP_37431 |
LINCSCP_37431 |
MCF7 |
| 0.272255 |
4.961750e-18 |
975 |
Tioconazole |
LSM-5028 |
|
3.33uM |
24h |
LINCSCP_74143 |
LINCSCP_74143 |
A375 |
| 0.272176 |
5.076778e-18 |
975 |
BRD-K19677752 |
LSM-9619 |
|
5uM |
24h |
LINCSCP_61743 |
LINCSCP_61743 |
VCAP |
| -0.272125 |
5.151367e-18 |
975 |
OTSSP167 |
LSM-6340 |
|
1.11uM |
24h |
LINCSCP_146307 |
LINCSCP_146307 |
MNEU.E |
| -0.272052 |
5.262273e-18 |
975 |
Mpep |
LSM-4678 |
GRM5 |
10uM |
24h |
LINCSCP_52910 |
LINCSCP_52910 |
SKB |
| -0.271865 |
5.554194e-18 |
975 |
BRD-A24396574-001-01-5 |
LSM-5006 |
|
10uM |
3h |
LINCSCP_163964 |
LINCSCP_163964 |
SKBR3 |
| 0.271859 |
5.563747e-18 |
975 |
BG-51 |
LSM-45301 |
HDAC3 |
0.5uM |
6h |
LINCSCP_279838 |
LINCSCP_279838 |
PC3 |
| -0.271631 |
5.943984e-18 |
975 |
BRD-A41986761 |
LSM-45957 |
|
0.12uM |
24h |
LINCSCP_101828 |
LINCSCP_101828 |
HELA |
| 0.271573 |
6.043305e-18 |
975 |
3-(4-Pyridyl)indole |
LSM-4569 |
ROCK1 |
1.11uM |
24h |
LINCSCP_140227 |
LINCSCP_140227 |
MCF7 |
| -0.271399 |
6.354448e-18 |
975 |
CL-976 |
LSM-6282 |
ACAT1 |
80uM |
6h |
LINCSCP_218597 |
LINCSCP_218597 |
HCT116 |
| 0.271381 |
6.387443e-18 |
975 |
BRD-K22912836 |
LSM-38513 |
|
5uM |
6h |
LINCSCP_64376 |
LINCSCP_64376 |
VCAP |
| 0.271337 |
6.470206e-18 |
975 |
BRD-K36360168 |
LSM-10624 |
|
5uM |
24h |
LINCSCP_62449 |
LINCSCP_62449 |
VCAP |
| -0.271321 |
6.500606e-18 |
975 |
Dalcetrapib |
LSM-6227 |
CETP |
80uM |
6h |
LINCSCP_289030 |
LINCSCP_289030 |
U937 |
| -0.271315 |
6.511002e-18 |
975 |
BRD-K15935695 |
LSM-9381 |
|
10uM |
24h |
LINCSCP_186518 |
LINCSCP_186518 |
A375 |
| -0.271292 |
6.555275e-18 |
975 |
Famciclovir |
LSM-2990 |
|
0.37uM |
24h |
LINCSCP_172804 |
LINCSCP_172804 |
YAPC |
| 0.27117 |
6.789670e-18 |
975 |
CHEMBL1616521 |
LSM-1793 |
OPRD1 |
10uM |
24h |
LINCSCP_30249 |
LINCSCP_30249 |
MCF7 |
| -0.271151 |
6.826596e-18 |
975 |
OTSSP167 |
LSM-6340 |
|
0.37uM |
24h |
LINCSCP_146308 |
LINCSCP_146308 |
MNEU.E |
| 0.270953 |
7.228425e-18 |
975 |
BRD-K46920162 |
LSM-11288 |
|
5uM |
24h |
LINCSCP_62657 |
LINCSCP_62657 |
VCAP |
| 0.270937 |
7.260893e-18 |
975 |
Crizotinib |
LSM-1027 |
ALK|MET |
0.37uM |
24h |
LINCSCP_68976 |
LINCSCP_68976 |
A375 |
| 0.270924 |
7.287754e-18 |
975 |
Acetazolamide |
LSM-5543 |
CA1|CA12|CA14|CA2|CA4|CA7 |
1.11uM |
24h |
LINCSCP_75562 |
LINCSCP_75562 |
A375 |
| -0.270884 |
7.373158e-18 |
975 |
SA-97378 |
LSM-41563 |
|
3uM |
24h |
LINCSCP_252332 |
LINCSCP_252332 |
MCF7 |
| -0.270859 |
7.424925e-18 |
975 |
Albendazole |
LSM-3782 |
|
1.11uM |
24h |
LINCSCP_126888 |
LINCSCP_126888 |
HT29 |
| 0.270839 |
7.467783e-18 |
975 |
GSK-1904529A |
LSM-1134 |
IGF1R|INSR |
0.5uM |
24h |
LINCSCP_39351 |
LINCSCP_39351 |
MDAMB231 |
| -0.270832 |
7.484363e-18 |
975 |
AC1NCVYC |
LSM-2836 |
|
10uM |
24h |
LINCSCP_45916 |
LINCSCP_45916 |
PC3 |
| -0.270804 |
7.544378e-18 |
975 |
BRD-K71614913 |
LSM-15157 |
|
10uM |
24h |
LINCSCP_278876 |
LINCSCP_278876 |
PC3 |
| 0.270743 |
7.678349e-18 |
975 |
BRD-K98168679 |
LSM-14463 |
|
5uM |
24h |
LINCSCP_61519 |
LINCSCP_61519 |
VCAP |
| -0.2707 |
7.774397e-18 |
975 |
Auranofin |
LSM-43136 |
|
10uM |
6h |
LINCSCP_36347 |
LINCSCP_36347 |
MCF7 |
| 0.270632 |
7.928033e-18 |
975 |
MLS000859112 |
LSM-6180 |
|
10uM |
6h |
LINCSCP_16377 |
LINCSCP_16377 |
HA1E |
| 0.270607 |
7.984133e-18 |
975 |
Megestrol Acetate |
LSM-2441 |
PGR |
10uM |
24h |
LINCSCP_44711 |
LINCSCP_44711 |
PC3 |
| 0.270378 |
8.528285e-18 |
975 |
BRD-K85822033 |
LSM-45305 |
|
1uM |
24h |
LINCSCP_205504 |
LINCSCP_205504 |
CD34 |
| -0.270329 |
8.648492e-18 |
975 |
CHEMBL2361187 |
LSM-12338 |
|
0.5uM |
24h |
LINCSCP_312496 |
LINCSCP_312496 |
VCAP |
| 0.270324 |
8.661925e-18 |
975 |
SCHEMBL16980224 |
LSM-1092 |
AURKA |
0.1uM |
24h |
LINCSCP_251885 |
LINCSCP_251885 |
MCF7 |
| 0.270307 |
8.704379e-18 |
975 |
Tadalafil |
LSM-4109 |
PDE11A|PDE5A |
10uM |
24h |
LINCSCP_32939 |
LINCSCP_32939 |
MCF7 |
| -0.270235 |
8.886492e-18 |
975 |
Pimavanserin |
LSM-45960 |
HTR2A |
1.11uM |
24h |
LINCSCP_173143 |
LINCSCP_173143 |
YAPC |
| 0.270228 |
8.904882e-18 |
975 |
AC1O9B20 |
LSM-4696 |
|
10uM |
6h |
LINCSCP_16344 |
LINCSCP_16344 |
HA1E |
| 0.270168 |
9.059238e-18 |
975 |
BRD-K75969390 |
LSM-41413 |
|
10uM |
6h |
LINCSCP_49176 |
LINCSCP_49176 |
PC3 |
| -0.270051 |
9.367611e-18 |
975 |
Isoliquiritigenin |
LSM-43093 |
GABBR1 |
10uM |
24h |
LINCSCP_30537 |
LINCSCP_30537 |
MCF7 |
| 0.269977 |
9.569504e-18 |
975 |
CHEMBL1965318 |
LSM-6612 |
|
10uM |
6h |
LINCSCP_16849 |
LINCSCP_16849 |
HA1E |
| 0.269817 |
1.001815e-17 |
975 |
EX-8678 |
LSM-1147 |
|
0.12uM |
3h |
LINCSCP_133191 |
LINCSCP_133191 |
MCF7 |
| 0.269689 |
1.039260e-17 |
975 |
Iguratimod |
LSM-45469 |
|
0.37uM |
24h |
LINCSCP_138069 |
LINCSCP_138069 |
MCF7 |
| 0.269603 |
1.065210e-17 |
975 |
BRD-K11883928 |
LSM-37878 |
|
10uM |
24h |
LINCSCP_31876 |
LINCSCP_31876 |
MCF7 |
| 0.269509 |
1.094393e-17 |
975 |
HG6-64-1 |
LSM-43248 |
|
0.5uM |
24h |
LINCSCP_11851 |
LINCSCP_11851 |
BT20 |
| 0.269448 |
1.113405e-17 |
975 |
AC1O9CRC |
LSM-4712 |
|
10uM |
24h |
LINCSCP_239492 |
LINCSCP_239492 |
MCF7 |
| -0.269384 |
1.134265e-17 |
975 |
5-Bromo-n-(6-butyl-1,3-benzothiazol-2-yl)furan-2-carboxamide |
LSM-2765 |
|
10uM |
24h |
LINCSCP_177817 |
LINCSCP_177817 |
A375 |
| -0.269072 |
1.240078e-17 |
975 |
BH3I-1′ |
LSM-42832 |
BCL2L1 |
10uM |
6h |
LINCSCP_452 |
LINCSCP_452 |
A375 |
| 0.268989 |
1.269658e-17 |
975 |
BRD-K51825814 |
LSM-11599 |
|
5uM |
6h |
LINCSCP_62550 |
LINCSCP_62550 |
VCAP |
| 0.26898 |
1.272928e-17 |
975 |
PIK-93 |
LSM-1191 |
|
0.04uM |
24h |
LINCSCP_144806 |
LINCSCP_144806 |
MDAMB231 |
| 0.268902 |
1.301704e-17 |
975 |
BRD-K03795299 |
LSM-6910 |
|
5uM |
24h |
LINCSCP_298712 |
LINCSCP_298712 |
VCAP |
| -0.268871 |
1.313226e-17 |
975 |
Wortmannin |
LSM-3947 |
PIK3CA|PIK3CG|PLK1 |
3uM |
24h |
LINCSCP_66690 |
LINCSCP_66690 |
A549 |
| -0.268821 |
1.332242e-17 |
975 |
Fluspirilene |
LSM-3748 |
DRD2|HTR2A |
5uM |
6h |
LINCSCP_51215 |
LINCSCP_51215 |
RMUGS |
| -0.268812 |
1.335565e-17 |
975 |
Lexibulin |
LSM-6232 |
TUBA1A|TUBA1B|TUBA1C|TUBA3E|TUBA4A|TUBB|TUBB1|TUBB2A|TUBB2B|TUBB3|TUBB4A|TUBB4B|TUBB6|TUBB8 |
10uM |
24h |
LINCSCP_153978 |
LINCSCP_153978 |
PC3 |
| -0.268794 |
1.342676e-17 |
975 |
Mebendazole |
LSM-3749 |
|
5uM |
24h |
LINCSCP_67634 |
LINCSCP_67634 |
MCF7 |
| 0.268757 |
1.356623e-17 |
975 |
Gemfibrozil |
LSM-2227 |
CYP2C8|LPL|PPARA |
0.12uM |
24h |
LINCSCP_72726 |
LINCSCP_72726 |
A375 |
| -0.268723 |
1.369930e-17 |
975 |
2-Chloro-7-methoxy-10H-phenothiazine |
LSM-3405 |
|
10uM |
24h |
LINCSCP_1417 |
LINCSCP_1417 |
A375 |
| -0.268617 |
1.412005e-17 |
975 |
Cisatracurium Besylate |
LSM-45935 |
CHRNA1|CHRNB1|CHRND|CHRNE|CHRNG |
10uM |
24h |
LINCSCP_71576 |
LINCSCP_71576 |
A375 |
| -0.268605 |
1.417124e-17 |
975 |
Afatinib |
LSM-43226 |
EGFR|ERBB2|ERBB4 |
10uM |
24h |
LINCSCP_46493 |
LINCSCP_46493 |
PC3 |
| -0.268517 |
1.452870e-17 |
975 |
CHEMBL3185651 |
LSM-3257 |
|
10uM |
24h |
LINCSCP_45515 |
LINCSCP_45515 |
PC3 |
| 0.268483 |
1.467092e-17 |
975 |
BRD-K07700224 |
LSM-8893 |
|
5uM |
24h |
LINCSCP_62853 |
LINCSCP_62853 |
VCAP |
| -0.268473 |
1.471345e-17 |
975 |
CHEMBL2143415 |
LSM-6085 |
|
1uM |
6h |
LINCSCP_37081 |
LINCSCP_37081 |
MCF7 |
| -0.268411 |
1.497733e-17 |
975 |
TP7 |
LSM-46015 |
|
10uM |
6h |
LINCSCP_49771 |
LINCSCP_49771 |
PC3 |
| -0.268353 |
1.522472e-17 |
975 |
R547 |
LSM-45812 |
|
0.37uM |
24h |
LINCSCP_106606 |
LINCSCP_106606 |
HELA |
| 0.268326 |
1.534295e-17 |
975 |
BRD-K69936629 |
LSM-12696 |
|
5uM |
24h |
LINCSCP_63109 |
LINCSCP_63109 |
VCAP |
| -0.2683 |
1.545600e-17 |
975 |
Wortmannin |
LSM-3947 |
PIK3CA|PIK3CG|PLK1 |
10uM |
24h |
LINCSCP_30110 |
LINCSCP_30110 |
MCF7 |
| -0.268269 |
1.559565e-17 |
975 |
SCHEMBL3954849 |
LSM-5982 |
|
0.12uM |
3h |
LINCSCP_163149 |
LINCSCP_163149 |
SKBR3 |
| 0.268203 |
1.589190e-17 |
975 |
Anandamide |
LSM-43816 |
CNR1|CNR2|TRPV1 |
10uM |
24h |
LINCSCP_43444 |
LINCSCP_43444 |
NPC |
| -0.267997 |
1.684829e-17 |
975 |
TL_HRAS26 |
LSM-2013 |
|
10uM |
24h |
LINCSCP_44867 |
LINCSCP_44867 |
PC3 |
| -0.267993 |
1.686860e-17 |
975 |
Diltiazem |
LSM-2523 |
CACNA1C|CACNA1D|CACNA1F|CACNA1S |
10uM |
6h |
LINCSCP_16953 |
LINCSCP_16953 |
HA1E |
| -0.267972 |
1.697050e-17 |
975 |
BRD-A41986761 |
LSM-45957 |
|
10uM |
24h |
LINCSCP_101824 |
LINCSCP_101824 |
HELA |
| -0.267927 |
1.718944e-17 |
975 |
CHEMBL2142684 |
LSM-40126 |
|
10uM |
6h |
LINCSCP_32053 |
LINCSCP_32053 |
MCF7 |
| 0.267871 |
1.746470e-17 |
975 |
Zaprinast |
LSM-2259 |
PDE5A |
3.33uM |
24h |
LINCSCP_153182 |
LINCSCP_153182 |
PC3 |
| 0.267865 |
1.749318e-17 |
975 |
CHEMBL3183436 |
LSM-15092 |
|
0.01uM |
6h |
LINCSCP_9327 |
LINCSCP_9327 |
A549 |
| -0.26785 |
1.756666e-17 |
975 |
Cobalt (Ii) Chloride |
LSM-5958 |
HIF1A |
10uM |
24h |
LINCSCP_272134 |
LINCSCP_272134 |
PC3 |
| 0.267774 |
1.795532e-17 |
975 |
Ingenol 3,20-dibenzoate |
LSM-4445 |
PRKCD|PRKCE |
0.01uM |
6h |
LINCSCP_9295 |
LINCSCP_9295 |
A549 |
| -0.267685 |
1.841284e-17 |
975 |
BRD-K18170480 |
LSM-38234 |
|
3uM |
24h |
LINCSCP_37880 |
LINCSCP_37880 |
MCF7 |
| 0.267675 |
1.846449e-17 |
975 |
MK-2206 |
LSM-1057 |
AKT1|AKT2|AKT3 |
0.04uM |
3h |
LINCSCP_145746 |
LINCSCP_145746 |
MDAMB231 |
| 0.267426 |
1.981959e-17 |
975 |
Dacarbazine |
LSM-5487 |
|
0.12uM |
24h |
LINCSCP_102140 |
LINCSCP_102140 |
HELA |
| 0.267327 |
2.038423e-17 |
975 |
Lapatinib |
LSM-1051 |
EGFR|ERBB2 |
3.33uM |
3h |
LINCSCP_145916 |
LINCSCP_145916 |
MDAMB231 |
| 0.26727 |
2.071300e-17 |
975 |
NSC403917 |
LSM-4816 |
|
10uM |
24h |
LINCSCP_31984 |
LINCSCP_31984 |
MCF7 |
| -0.267256 |
2.079984e-17 |
975 |
Parbendazole |
LSM-4893 |
TUBB |
3uM |
24h |
LINCSCP_37426 |
LINCSCP_37426 |
MCF7 |
| 0.267221 |
2.100519e-17 |
975 |
BRD-K44777226 |
LSM-11152 |
|
5uM |
6h |
LINCSCP_62544 |
LINCSCP_62544 |
VCAP |
| -0.266996 |
2.238929e-17 |
975 |
NU1025 |
LSM-4643 |
PARP1 |
10uM |
6h |
LINCSCP_12545 |
LINCSCP_12545 |
CL34 |
| -0.266953 |
2.266241e-17 |
975 |
BRD-K22937431 |
LSM-38515 |
|
5uM |
24h |
LINCSCP_64258 |
LINCSCP_64258 |
VCAP |
| -0.266903 |
2.298632e-17 |
975 |
NCGC00018102-06 |
LSM-2250 |
CACNA1G|CACNA1H |
10uM |
24h |
LINCSCP_55634 |
LINCSCP_55634 |
VCAP |
| -0.266899 |
2.301143e-17 |
975 |
CI-1040 |
LSM-1048 |
MAP2K1|MAP2K2 |
0.12uM |
24h |
LINCSCP_138184 |
LINCSCP_138184 |
MCF7 |
| -0.266884 |
2.311397e-17 |
975 |
17-DMAG (Alvespimycin) HCl |
LSM-46133 |
|
0.04uM |
24h |
LINCSCP_153443 |
LINCSCP_153443 |
PC3 |
| 0.266852 |
2.332213e-17 |
975 |
CAY-10415 |
LSM-5100 |
INS |
10uM |
24h |
LINCSCP_239374 |
LINCSCP_239374 |
MCF7 |
| -0.266823 |
2.351222e-17 |
975 |
BRD-A73558769 |
LSM-45352 |
|
1uM |
24h |
LINCSCP_24121 |
LINCSCP_24121 |
HL60 |
| 0.266701 |
2.434069e-17 |
975 |
BRD-K28184645 |
LSM-38807 |
|
10uM |
6h |
LINCSCP_279446 |
LINCSCP_279446 |
PC3 |
| 0.266594 |
2.509172e-17 |
975 |
BRD-K39504007 |
LSM-10828 |
|
5uM |
6h |
LINCSCP_62374 |
LINCSCP_62374 |
VCAP |
| 0.266575 |
2.522084e-17 |
975 |
BRD-A74382794 |
LSM-45339 |
|
3uM |
24h |
LINCSCP_55295 |
LINCSCP_55295 |
U937 |
| 0.266564 |
2.530303e-17 |
975 |
Carbinoxamine |
LSM-1435 |
HRH1 |
10uM |
6h |
LINCSCP_16926 |
LINCSCP_16926 |
HA1E |
| 0.266543 |
2.545447e-17 |
975 |
Clorgiline |
LSM-5808 |
MAOA |
10uM |
24h |
LINCSCP_243543 |
LINCSCP_243543 |
MCF7 |
| 0.266478 |
2.592300e-17 |
975 |
BRD-K65541951 |
LSM-12428 |
|
5uM |
24h |
LINCSCP_64015 |
LINCSCP_64015 |
VCAP |
| -0.266474 |
2.595237e-17 |
975 |
NINDS_000152 |
LSM-4661 |
CYCS |
10uM |
6h |
LINCSCP_16325 |
LINCSCP_16325 |
HA1E |
| -0.26646 |
2.605494e-17 |
975 |
BRD-K47728674 |
LSM-7461 |
|
5uM |
24h |
LINCSCP_60383 |
LINCSCP_60383 |
VCAP |
| -0.266457 |
2.607854e-17 |
975 |
MK-2206 |
LSM-1057 |
AKT1|AKT2|AKT3 |
0.04uM |
24h |
LINCSCP_142432 |
LINCSCP_142432 |
MCF7 |
| -0.266457 |
2.607937e-17 |
975 |
AC1O9BZM |
LSM-4580 |
|
10uM |
6h |
LINCSCP_16287 |
LINCSCP_16287 |
HA1E |
| -0.266373 |
2.670662e-17 |
975 |
Phensuximide |
LSM-1359 |
CACNA1G|CACNA1H|CACNA1I |
1.11uM |
24h |
LINCSCP_153350 |
LINCSCP_153350 |
PC3 |
| 0.266306 |
2.721330e-17 |
975 |
Emedastine |
LSM-5331 |
HRH1 |
0.12uM |
24h |
LINCSCP_156221 |
LINCSCP_156221 |
PC3 |
| 0.266296 |
2.729713e-17 |
975 |
BSPBIO_001542 |
LSM-42823 |
PPP1CA|PPP2CA |
10uM |
24h |
LINCSCP_4155 |
LINCSCP_4155 |
A549 |
| 0.266281 |
2.741056e-17 |
975 |
BRD-K37014875 |
LSM-10668 |
|
5uM |
6h |
LINCSCP_62973 |
LINCSCP_62973 |
VCAP |
| -0.266213 |
2.794413e-17 |
975 |
CHIR-99021 |
LSM-1181 |
|
0.12uM |
3h |
LINCSCP_145979 |
LINCSCP_145979 |
MDAMB231 |
| 0.2661 |
2.884523e-17 |
975 |
Infigratinib |
LSM-1184 |
FGFR1|FGFR2|FGFR3|FGFR4 |
0.12uM |
24h |
LINCSCP_84380 |
LINCSCP_84380 |
ASC |
| -0.266065 |
2.913011e-17 |
975 |
Mebendazole |
LSM-3749 |
|
40uM |
24h |
LINCSCP_67576 |
LINCSCP_67576 |
MCF7 |
| -0.266019 |
2.951244e-17 |
975 |
BRD-K79758054 |
LSM-41623 |
|
10uM |
24h |
LINCSCP_3629 |
LINCSCP_3629 |
A375 |
| 0.265936 |
3.021351e-17 |
975 |
BRD-K19275171 |
LSM-9587 |
|
5uM |
24h |
LINCSCP_61567 |
LINCSCP_61567 |
VCAP |
| -0.265893 |
3.058137e-17 |
975 |
CHEMBL34095 |
LSM-3355 |
|
10uM |
24h |
LINCSCP_52766 |
LINCSCP_52766 |
SKB |
| 0.265811 |
3.129422e-17 |
975 |
amcinonide |
|
|
0.12uM |
24h |
LINCSCP_117601 |
LINCSCP_117601 |
HT29 |
| -0.265776 |
3.160776e-17 |
975 |
Apafant |
LSM-2613 |
PTAFR |
1.11uM |
24h |
LINCSCP_120973 |
LINCSCP_120973 |
HT29 |
| -0.265753 |
3.181281e-17 |
975 |
Podofilox |
LSM-3055 |
|
0.37uM |
24h |
LINCSCP_141626 |
LINCSCP_141626 |
MCF7 |
| 0.265728 |
3.204021e-17 |
975 |
Aurora A Inhibitor I |
LSM-1065 |
AURKA |
10uM |
24h |
LINCSCP_166067 |
LINCSCP_166067 |
SKL |
| 0.265641 |
3.283183e-17 |
975 |
CHEMBL1877309 |
LSM-3358 |
PKM |
10uM |
24h |
LINCSCP_31631 |
LINCSCP_31631 |
MCF7 |
| -0.26561 |
3.311903e-17 |
975 |
Clozapine |
LSM-2823 |
ADRA1A|ADRA1B|CHRM1|CHRM2|CHRM3|CHRM4|DRD1|DRD2|DRD3|DRD4|HRH1|HRH4|HTR1A|HTR1B|HTR1D|HTR1E|HTR2A|HTR2C|HTR6|HTR7 |
1.11uM |
24h |
LINCSCP_122238 |
LINCSCP_122238 |
HT29 |
| 0.2655 |
3.416058e-17 |
975 |
Hydroxyprogesterone Caproate |
LSM-4900 |
AR|ESR1|ESR2|NR1H4|NR1I2|NR3C1|PGR |
1.11uM |
24h |
LINCSCP_153009 |
LINCSCP_153009 |
PC3 |
| -0.265419 |
3.494699e-17 |
975 |
BRD-K55149044 |
LSM-6839 |
|
10uM |
24h |
LINCSCP_28367 |
LINCSCP_28367 |
HT29 |
| 0.265383 |
3.531245e-17 |
975 |
AC1LDBAO |
LSM-4032 |
|
20uM |
6h |
LINCSCP_10655 |
LINCSCP_10655 |
AGS |
| 0.265381 |
3.532651e-17 |
975 |
BRD-K71225733 |
LSM-12779 |
|
5uM |
24h |
LINCSCP_63110 |
LINCSCP_63110 |
VCAP |
| 0.265359 |
3.554844e-17 |
975 |
AKT Inhibitor VIII |
LSM-1035 |
AKT1|AKT2 |
1.11uM |
24h |
LINCSCP_68993 |
LINCSCP_68993 |
A375 |
| -0.265355 |
3.558660e-17 |
975 |
NCGC00238427-01 |
LSM-1511 |
RORC |
10uM |
24h |
LINCSCP_177728 |
LINCSCP_177728 |
A375 |
| 0.265298 |
3.616203e-17 |
975 |
Erlotinib |
LSM-1097 |
EGFR |
1.11uM |
24h |
LINCSCP_85376 |
LINCSCP_85376 |
BT20 |
| -0.265279 |
3.635547e-17 |
975 |
MLS001065861 |
LSM-2986 |
|
10uM |
24h |
LINCSCP_4957 |
LINCSCP_4957 |
A549 |
| -0.265058 |
3.868921e-17 |
975 |
KUC103898N |
LSM-2754 |
|
10uM |
24h |
LINCSCP_31596 |
LINCSCP_31596 |
MCF7 |
| 0.264995 |
3.937485e-17 |
975 |
Selumetinib |
LSM-1056 |
MAP2K1|MAP2K2 |
0.12uM |
3h |
LINCSCP_130348 |
LINCSCP_130348 |
LNCAP |
| -0.26496 |
3.976282e-17 |
975 |
BAS 05532738 |
LSM-4550 |
RPS6KA1|RPS6KA2|RPS6KA3 |
10uM |
6h |
LINCSCP_32306 |
LINCSCP_32306 |
MCF7 |
| -0.264904 |
4.040069e-17 |
975 |
Tocainide |
LSM-1909 |
SCN10A|SCN11A|SCN1A|SCN2A|SCN3A|SCN4A|SCN5A|SCN7A|SCN8A|SCN9A |
10uM |
6h |
LINCSCP_4328 |
LINCSCP_4328 |
A549 |
| 0.264693 |
4.286644e-17 |
975 |
Rifampicin |
LSM-43162 |
NR1I2 |
10uM |
6h |
LINCSCP_217434 |
LINCSCP_217434 |
HCC515 |
| 0.26466 |
4.326221e-17 |
975 |
BRD-K47102646 |
LSM-11305 |
|
5uM |
24h |
LINCSCP_62289 |
LINCSCP_62289 |
VCAP |
| -0.264562 |
4.446235e-17 |
975 |
Colchicine |
LSM-5199 |
TUBA1A|TUBA1B|TUBA1C|TUBA3E|TUBA4A|TUBB|TUBB1|TUBB2A|TUBB2B|TUBB3|TUBB4A|TUBB4B|TUBB6|TUBB8 |
3uM |
24h |
LINCSCP_37619 |
LINCSCP_37619 |
MCF7 |
| -0.264555 |
4.455579e-17 |
975 |
Tolazamide |
LSM-2699 |
ABCC8|KCNJ11 |
10uM |
24h |
LINCSCP_272023 |
LINCSCP_272023 |
PC3 |
| -0.264535 |
4.480208e-17 |
975 |
Pfmrk inhibitor, wr 216174 |
LSM-42921 |
|
10uM |
24h |
LINCSCP_44023 |
LINCSCP_44023 |
PC3 |
| 0.264404 |
4.648465e-17 |
975 |
KUC103885 |
LSM-2794 |
|
10uM |
6h |
LINCSCP_292576 |
LINCSCP_292576 |
VCAP |
| 0.264324 |
4.753282e-17 |
975 |
CHEMBL2355314 |
LSM-9253 |
|
5uM |
24h |
LINCSCP_62256 |
LINCSCP_62256 |
VCAP |
| 0.264284 |
4.807460e-17 |
975 |
ST021200 |
LSM-4601 |
|
10uM |
6h |
LINCSCP_12822 |
LINCSCP_12822 |
DV90 |
| -0.264229 |
4.882000e-17 |
975 |
BCB03_000082 |
LSM-36632 |
|
10uM |
6h |
LINCSCP_16602 |
LINCSCP_16602 |
HA1E |
| -0.264128 |
5.021618e-17 |
975 |
AZD-1775 |
LSM-1153 |
WEE1 |
10uM |
6h |
LINCSCP_4779 |
LINCSCP_4779 |
A549 |
| 0.264126 |
5.024258e-17 |
975 |
BSPBIO_001530 |
LSM-1549 |
|
10uM |
24h |
LINCSCP_14979 |
LINCSCP_14979 |
HA1E |
| 0.264058 |
5.121527e-17 |
975 |
BRD-K37991633 |
LSM-10729 |
|
5uM |
24h |
LINCSCP_62649 |
LINCSCP_62649 |
VCAP |
| -0.263926 |
5.313323e-17 |
975 |
BRD-K37650321 |
LSM-39345 |
|
10uM |
24h |
LINCSCP_3565 |
LINCSCP_3565 |
A375 |
| 0.263907 |
5.341739e-17 |
975 |
Tyrphostin B7 |
LSM-42938 |
PDGFRB |
10uM |
24h |
LINCSCP_33618 |
LINCSCP_33618 |
MCF7 |
| -0.263892 |
5.365132e-17 |
975 |
BRD-A28746609 |
LSM-1102 |
NR1I2|TUBB |
0.04uM |
24h |
LINCSCP_137549 |
LINCSCP_137549 |
MCF7 |
| 0.263874 |
5.391345e-17 |
975 |
Gimeracil |
LSM-45923 |
|
3.33uM |
24h |
LINCSCP_72024 |
LINCSCP_72024 |
A375 |
| 0.263874 |
5.391806e-17 |
975 |
MK-2206 |
LSM-1057 |
AKT1|AKT2|AKT3 |
1.11uM |
24h |
LINCSCP_113071 |
LINCSCP_113071 |
HME1 |
| 0.263779 |
5.536985e-17 |
975 |
BRD-K50149017 |
LSM-11478 |
|
5uM |
6h |
LINCSCP_62216 |
LINCSCP_62216 |
VCAP |
| -0.263745 |
5.589633e-17 |
975 |
Dapivirine (TMC120) |
LSM-45463 |
|
10uM |
24h |
LINCSCP_104447 |
LINCSCP_104447 |
HELA |
| -0.263717 |
5.634000e-17 |
975 |
Atrasentan (hydrochloride) |
LSM-45787 |
EDNRA |
0.37uM |
24h |
LINCSCP_153148 |
LINCSCP_153148 |
PC3 |
| 0.263646 |
5.746938e-17 |
975 |
CHEMBL2362220 |
LSM-39025 |
|
5uM |
24h |
LINCSCP_64274 |
LINCSCP_64274 |
VCAP |
| -0.263638 |
5.759018e-17 |
975 |
MLS003153121 |
LSM-2123 |
|
10uM |
24h |
LINCSCP_1367 |
LINCSCP_1367 |
A375 |
| -0.26354 |
5.919639e-17 |
975 |
20554-84-1 |
LSM-43090 |
|
10uM |
24h |
LINCSCP_32158 |
LINCSCP_32158 |
MCF7 |
| -0.26344 |
6.085988e-17 |
975 |
HG-9-91-01 |
LSM-6343 |
|
0.37uM |
24h |
LINCSCP_129604 |
LINCSCP_129604 |
JURKAT |
| -0.263366 |
6.214562e-17 |
975 |
TAK-285 |
LSM-45987 |
EGFR|ERBB2 |
10uM |
24h |
LINCSCP_141701 |
LINCSCP_141701 |
MCF7 |
| 0.263319 |
6.295938e-17 |
975 |
Alpelisib |
LSM-4256 |
PIK3CA |
1.11uM |
3h |
LINCSCP_132482 |
LINCSCP_132482 |
MCF7 |
| -0.2633 |
6.328729e-17 |
975 |
BRD-K91600270 |
LSM-4050 |
|
10uM |
24h |
LINCSCP_1442 |
LINCSCP_1442 |
A375 |
| 0.26323 |
6.454930e-17 |
975 |
CHEMBL2143784 |
LSM-6141 |
|
10uM |
24h |
LINCSCP_7887 |
LINCSCP_7887 |
A549 |
| 0.263153 |
6.593752e-17 |
975 |
BRD-K74656908 |
LSM-13003 |
|
5uM |
24h |
LINCSCP_63112 |
LINCSCP_63112 |
VCAP |
| -0.263113 |
6.667890e-17 |
975 |
Sappanone A Trimethyl Ether |
LSM-42843 |
|
10uM |
24h |
LINCSCP_32865 |
LINCSCP_32865 |
MCF7 |
| -0.263098 |
6.695927e-17 |
975 |
SMR000206938 |
LSM-1663 |
|
10uM |
24h |
LINCSCP_30908 |
LINCSCP_30908 |
MCF7 |
| -0.263091 |
6.709726e-17 |
975 |
CHEMBL3186554 |
LSM-41075 |
|
10uM |
24h |
LINCSCP_43038 |
LINCSCP_43038 |
NPC |
| 0.263083 |
6.724063e-17 |
975 |
BRD-K44229115 |
LSM-11128 |
|
5uM |
24h |
LINCSCP_61997 |
LINCSCP_61997 |
VCAP |
| 0.263016 |
6.850243e-17 |
975 |
BRD-K25290948 |
LSM-43380 |
|
5uM |
24h |
LINCSCP_60016 |
LINCSCP_60016 |
VCAP |
| -0.262957 |
6.964704e-17 |
975 |
LY-294002 |
LSM-2597 |
MTOR|PIK3CA|PIK3CB|PIK3CD|PIK3CG|PLK1|PRKDC |
10uM |
24h |
LINCSCP_68557 |
LINCSCP_68557 |
VCAP |
| -0.262665 |
7.553504e-17 |
975 |
Prosteride |
LSM-1842 |
SRD5A1|SRD5A2 |
0.04uM |
24h |
LINCSCP_173140 |
LINCSCP_173140 |
YAPC |
| 0.262628 |
7.632956e-17 |
975 |
AC1O9CBL |
LSM-4596 |
|
0.5uM |
24h |
LINCSCP_253913 |
LINCSCP_253913 |
MCF7 |
| 0.262579 |
7.738043e-17 |
975 |
HMS3264J07 |
LSM-1485 |
|
10uM |
6h |
LINCSCP_32965 |
LINCSCP_32965 |
MCF7 |
| -0.262562 |
7.773930e-17 |
975 |
BRD-A28746609 |
LSM-1102 |
NR1I2|TUBB |
1.11uM |
24h |
LINCSCP_137546 |
LINCSCP_137546 |
MCF7 |
| -0.262526 |
7.852645e-17 |
975 |
Diethylpropion |
LSM-5038 |
SLC6A2|SLC6A3 |
10uM |
24h |
LINCSCP_243360 |
LINCSCP_243360 |
MCF7 |
| 0.262468 |
7.979187e-17 |
975 |
Gallocatechin Gallate |
LSM-6228 |
BACE1|FASN |
90uM |
6h |
LINCSCP_12804 |
LINCSCP_12804 |
DV90 |
| 0.262435 |
8.052006e-17 |
975 |
BRD-K85498716 |
LSM-13655 |
|
5uM |
24h |
LINCSCP_304600 |
LINCSCP_304600 |
VCAP |
| 0.262315 |
8.325278e-17 |
975 |
BRD-K75418563 |
LSM-6850 |
|
3uM |
6h |
LINCSCP_23721 |
LINCSCP_23721 |
HEPG2 |
| -0.262296 |
8.369058e-17 |
975 |
altrenogest |
LSM-45498 |
|
0.04uM |
24h |
LINCSCP_139859 |
LINCSCP_139859 |
MCF7 |
| 0.26225 |
8.477841e-17 |
975 |
BRD-K75693278 |
LSM-13056 |
|
5uM |
24h |
LINCSCP_63526 |
LINCSCP_63526 |
VCAP |
| -0.26224 |
8.501807e-17 |
975 |
CHEMBL2143415 |
LSM-6085 |
|
10uM |
6h |
LINCSCP_37080 |
LINCSCP_37080 |
MCF7 |
| -0.262224 |
8.539512e-17 |
975 |
MLS000925170 |
LSM-4856 |
|
10uM |
24h |
LINCSCP_34147 |
LINCSCP_34147 |
MCF7 |
| 0.262217 |
8.556358e-17 |
975 |
BRD-K42357106 |
LSM-7386 |
|
5uM |
24h |
LINCSCP_60186 |
LINCSCP_60186 |
VCAP |
| 0.26218 |
8.644785e-17 |
975 |
BRD-K18396390 |
LSM-38254 |
|
5uM |
24h |
LINCSCP_64253 |
LINCSCP_64253 |
VCAP |
| 0.261994 |
9.101293e-17 |
975 |
BRD-K14636731 |
LSM-6084 |
|
10uM |
6h |
LINCSCP_33983 |
LINCSCP_33983 |
MCF7 |
| 0.261988 |
9.116221e-17 |
975 |
BRD-K14471942 |
LSM-9305 |
|
5uM |
24h |
LINCSCP_61738 |
LINCSCP_61738 |
VCAP |
| -0.261909 |
9.318717e-17 |
975 |
BRD-K48508383 |
LSM-39964 |
|
10uM |
24h |
LINCSCP_278844 |
LINCSCP_278844 |
PC3 |
| 0.261823 |
9.544439e-17 |
975 |
BRD-K80301668 |
LSM-13335 |
|
5uM |
24h |
LINCSCP_62691 |
LINCSCP_62691 |
VCAP |
| 0.261769 |
9.688000e-17 |
975 |
MLN 2238 |
LSM-4944 |
PSMB1 |
10uM |
6h |
LINCSCP_55536 |
LINCSCP_55536 |
U937 |
| -0.261731 |
9.791571e-17 |
975 |
Cyclohexanecarboxamide, 4-(1-aminoethyl)-n-4-pyridinyl-, trans- |
LSM-1177 |
ROCK1|ROCK2 |
0.04uM |
24h |
LINCSCP_76641 |
LINCSCP_76641 |
A375 |
| 0.261679 |
9.931791e-17 |
975 |
IAA-94 |
LSM-3913 |
|
10uM |
6h |
LINCSCP_14309 |
LINCSCP_14309 |
HA1E |
| 0.261664 |
9.975229e-17 |
975 |
BRD4770 |
LSM-42692 |
EHMT2 |
10uM |
24h |
LINCSCP_270325 |
LINCSCP_270325 |
PC3 |
| 0.261589 |
1.018380e-16 |
975 |
Tranylcypromine |
LSM-5578 |
KDM1A|MAOA|MAOB |
0.12uM |
24h |
LINCSCP_128970 |
LINCSCP_128970 |
HUVEC |
| -0.261581 |
1.020568e-16 |
975 |
Ergothioneine |
LSM-45829 |
|
0.04uM |
24h |
LINCSCP_154127 |
LINCSCP_154127 |
PC3 |
| -0.261485 |
1.048059e-16 |
975 |
MLS003370613 |
LSM-1679 |
TSHR |
10uM |
24h |
LINCSCP_177732 |
LINCSCP_177732 |
A375 |
| -0.261469 |
1.052826e-16 |
975 |
BAY 61-3606 |
LSM-1167 |
SYK |
10uM |
24h |
LINCSCP_134115 |
LINCSCP_134115 |
MCF7 |
| 0.261467 |
1.053268e-16 |
975 |
BRD-K27839561 |
LSM-10110 |
|
5uM |
24h |
LINCSCP_62636 |
LINCSCP_62636 |
VCAP |
| -0.261435 |
1.062705e-16 |
975 |
BRD-A28746609 |
LSM-1102 |
NR1I2|TUBB |
0.12uM |
24h |
LINCSCP_137548 |
LINCSCP_137548 |
MCF7 |
| -0.261413 |
1.069298e-16 |
975 |
MLS000038113 |
LSM-4839 |
|
3uM |
24h |
LINCSCP_260462 |
LINCSCP_260462 |
NKDBA |
| -0.261411 |
1.069729e-16 |
975 |
Lexibulin |
LSM-6232 |
TUBA1A|TUBA1B|TUBA1C|TUBA3E|TUBA4A|TUBB|TUBB1|TUBB2A|TUBB2B|TUBB3|TUBB4A|TUBB4B|TUBB6|TUBB8 |
1.11uM |
24h |
LINCSCP_135772 |
LINCSCP_135772 |
MCF7 |
| 0.261346 |
1.089328e-16 |
975 |
Rhapontin |
LSM-42872 |
|
10uM |
6h |
LINCSCP_475 |
LINCSCP_475 |
A375 |
| -0.261306 |
1.101385e-16 |
975 |
Alimta |
LSM-6253 |
DHFR|GART|TYMS |
90uM |
6h |
LINCSCP_51159 |
LINCSCP_51159 |
RMUGS |
| 0.26129 |
1.106223e-16 |
975 |
Enzalutamide |
LSM-6254 |
AR |
0.1uM |
24h |
LINCSCP_30581 |
LINCSCP_30581 |
MCF7 |
| 0.261248 |
1.119236e-16 |
975 |
ANISODAMINE HYDROBROMIDE |
LSM-45481 |
|
1.11uM |
24h |
LINCSCP_71297 |
LINCSCP_71297 |
A375 |
| 0.261102 |
1.165138e-16 |
975 |
BRD-K79131144 |
LSM-14937 |
|
5uM |
24h |
LINCSCP_64219 |
LINCSCP_64219 |
VCAP |
| 0.261073 |
1.174557e-16 |
975 |
Tivantinib |
LSM-1131 |
MET |
0.1uM |
24h |
LINCSCP_39384 |
LINCSCP_39384 |
MDAMB231 |
| 0.260945 |
1.216978e-16 |
975 |
SA-246522 |
LSM-38089 |
|
0.5uM |
24h |
LINCSCP_37647 |
LINCSCP_37647 |
MCF7 |
| -0.260875 |
1.240537e-16 |
975 |
Clarithromycin |
LSM-5606 |
|
0.12uM |
24h |
LINCSCP_153227 |
LINCSCP_153227 |
PC3 |
| -0.260863 |
1.244674e-16 |
975 |
TENOVIN-1 |
LSM-5238 |
SIRT1 |
10uM |
24h |
LINCSCP_46715 |
LINCSCP_46715 |
PC3 |
| -0.260861 |
1.245553e-16 |
975 |
GR 159897 |
LSM-3158 |
TAC1|TACR2 |
10uM |
24h |
LINCSCP_284734 |
LINCSCP_284734 |
SKB |
| -0.26084 |
1.252531e-16 |
975 |
GSK-1070916 |
LSM-1062 |
AURKB|AURKC |
10uM |
24h |
LINCSCP_164581 |
LINCSCP_164581 |
SKL.C |
| -0.260818 |
1.260283e-16 |
975 |
Withaferin A |
LSM-6685 |
IKBKB|NAMPT |
10uM |
3h |
LINCSCP_85584 |
LINCSCP_85584 |
BT20 |
| -0.260801 |
1.266339e-16 |
975 |
Mebendazole |
LSM-3749 |
|
10uM |
24h |
LINCSCP_67574 |
LINCSCP_67574 |
MCF7 |
| -0.260714 |
1.296845e-16 |
975 |
MLS003448149 |
LSM-3003 |
|
10uM |
6h |
LINCSCP_40210 |
LINCSCP_40210 |
NCIH508 |
| -0.260711 |
1.298215e-16 |
975 |
Albendazole |
LSM-3782 |
|
1.11uM |
24h |
LINCSCP_110086 |
LINCSCP_110086 |
HELA |
| -0.260622 |
1.330366e-16 |
975 |
GSK 525762A |
LSM-6334 |
|
10uM |
24h |
LINCSCP_164718 |
LINCSCP_164718 |
SKL.C |
| 0.260585 |
1.344109e-16 |
975 |
Tetrahydrozoline |
LSM-1430 |
ADRA1A|ADRA1B|ADRA1D|ADRA2A|ADRA2B|ADRA2C |
10uM |
24h |
LINCSCP_34438 |
LINCSCP_34438 |
MCF7 |
| 0.260542 |
1.360177e-16 |
975 |
SCHEMBL13991002 |
LSM-6278 |
|
40uM |
6h |
LINCSCP_29402 |
LINCSCP_29402 |
LOVO |
| -0.260488 |
1.380354e-16 |
975 |
LY-294002 |
LSM-2597 |
MTOR|PIK3CA|PIK3CB|PIK3CD|PIK3CG|PLK1|PRKDC |
10uM |
24h |
LINCSCP_310791 |
LINCSCP_310791 |
VCAP |
| 0.260486 |
1.381000e-16 |
975 |
BRD-K91701366 |
LSM-42265 |
|
10uM |
24h |
LINCSCP_8974 |
LINCSCP_8974 |
A549 |
| 0.260421 |
1.405948e-16 |
975 |
Lapatinib |
LSM-1051 |
EGFR|ERBB2 |
0.04uM |
24h |
LINCSCP_145567 |
LINCSCP_145567 |
MDAMB231 |
| 0.260401 |
1.413778e-16 |
975 |
ethyl 6-(2,3-dihydro-1H-indol-1-ylmethyl)-4-(3-nitrophenyl)-2-oxo-1,2,3,4-tetrahydro-5-pyrimidinecarboxylate |
LSM-45350 |
|
0.5uM |
24h |
LINCSCP_12364 |
LINCSCP_12364 |
CD34 |
| -0.260391 |
1.417730e-16 |
975 |
Dextromethorphan |
LSM-2726 |
GRIN2A|SIGMAR1|SLC6A4 |
1.11uM |
24h |
LINCSCP_153560 |
LINCSCP_153560 |
PC3 |
| 0.260291 |
1.457464e-16 |
975 |
LY2886721 |
LSM-45433 |
|
3.33uM |
24h |
LINCSCP_71666 |
LINCSCP_71666 |
A375 |
| 0.260246 |
1.475634e-16 |
975 |
AC1NWAJL |
LSM-1643 |
|
10uM |
6h |
LINCSCP_30173 |
LINCSCP_30173 |
MCF7 |
| 0.260149 |
1.515381e-16 |
975 |
BRD-K47690943 |
LSM-39919 |
|
10uM |
6h |
LINCSCP_16837 |
LINCSCP_16837 |
HA1E |
| -0.26001 |
1.574376e-16 |
975 |
Dictamnine |
LSM-2642 |
|
10uM |
24h |
LINCSCP_44027 |
LINCSCP_44027 |
PC3 |
| -0.259982 |
1.586815e-16 |
975 |
BRD-K86671899 |
LSM-13737 |
|
10uM |
24h |
LINCSCP_3640 |
LINCSCP_3640 |
A375 |
| -0.259961 |
1.595970e-16 |
975 |
BRD-K33676730 |
LSM-39115 |
|
10uM |
24h |
LINCSCP_10736 |
LINCSCP_10736 |
ASC |
| -0.259939 |
1.605428e-16 |
975 |
Motesanib |
LSM-1042 |
FLT1|FLT4|KDR|KIT|PDGFRA|PDGFRB|RET |
10uM |
24h |
LINCSCP_239992 |
LINCSCP_239992 |
MCF7 |
| 0.259932 |
1.608872e-16 |
975 |
Latanoprost |
LSM-43170 |
PTGFR |
0.37uM |
24h |
LINCSCP_72731 |
LINCSCP_72731 |
A375 |
| 0.259924 |
1.612471e-16 |
975 |
BRD-K10894258 |
LSM-9095 |
|
5uM |
24h |
LINCSCP_62255 |
LINCSCP_62255 |
VCAP |
| -0.25991 |
1.618545e-16 |
975 |
BRD-K41593073 |
LSM-39569 |
|
10uM |
24h |
LINCSCP_278835 |
LINCSCP_278835 |
PC3 |
| 0.2599 |
1.622902e-16 |
975 |
BRD-K02117849 |
LSM-8563 |
|
10uM |
24h |
LINCSCP_8987 |
LINCSCP_8987 |
A549 |
| -0.259883 |
1.630655e-16 |
975 |
GR-55562 |
LSM-3026 |
HTR1B |
10uM |
24h |
LINCSCP_42642 |
LINCSCP_42642 |
NPC |
| 0.259876 |
1.633759e-16 |
975 |
MLS004683634 |
LSM-6156 |
|
10uM |
6h |
LINCSCP_20667 |
LINCSCP_20667 |
HCC515 |
| 0.259861 |
1.640422e-16 |
975 |
CHEMBL2137336 |
LSM-37457 |
|
10uM |
6h |
LINCSCP_16780 |
LINCSCP_16780 |
HA1E |
| 0.259825 |
1.656560e-16 |
975 |
BRD-K73434853 |
LSM-41258 |
|
10uM |
6h |
LINCSCP_64800 |
LINCSCP_64800 |
VCAP |
| 0.259776 |
1.679425e-16 |
975 |
BRD-K00381581 |
LSM-8449 |
|
10uM |
24h |
LINCSCP_3509 |
LINCSCP_3509 |
A375 |
| -0.259741 |
1.695214e-16 |
975 |
13-Hydroxy-8,14,19-trimethoxy-4,10,12,16-tetramethyl-3,20,22-trioxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18-pentaen-9-yl carbamate |
LSM-42815 |
HSP90AA1 |
10uM |
6h |
LINCSCP_264450 |
LINCSCP_264450 |
PC3 |
| 0.25967 |
1.728794e-16 |
975 |
AC1O7M2R |
LSM-3745 |
ADCY2 |
10uM |
6h |
LINCSCP_21559 |
LINCSCP_21559 |
HEPG2 |
| 0.259632 |
1.746900e-16 |
975 |
Latanoprost |
LSM-43170 |
PTGFR |
3.33uM |
24h |
LINCSCP_72729 |
LINCSCP_72729 |
A375 |
| 0.2596 |
1.762305e-16 |
975 |
BRD-K21629388 |
LSM-9743 |
|
5uM |
24h |
LINCSCP_62633 |
LINCSCP_62633 |
VCAP |
| 0.259591 |
1.766670e-16 |
975 |
Benfluorex |
LSM-4365 |
HMGCR |
10uM |
24h |
LINCSCP_252545 |
LINCSCP_252545 |
MCF7 |
| -0.259554 |
1.784911e-16 |
975 |
Nemonapride |
LSM-45497 |
|
1.11uM |
24h |
LINCSCP_96482 |
LINCSCP_96482 |
HA1E |
| -0.259485 |
1.818866e-16 |
975 |
MLS002699341 |
LSM-3152 |
|
10uM |
24h |
LINCSCP_267654 |
LINCSCP_267654 |
PC3 |
| 0.259422 |
1.850413e-16 |
975 |
BRD-K30934390 |
LSM-14787 |
|
5uM |
24h |
LINCSCP_309140 |
LINCSCP_309140 |
VCAP |
| 0.259308 |
1.909184e-16 |
975 |
DG-041 |
LSM-43279 |
PTGER3 |
40uM |
6h |
LINCSCP_257359 |
LINCSCP_257359 |
NCIH508 |
| -0.259305 |
1.910778e-16 |
975 |
MLS003568137 |
LSM-1980 |
|
10uM |
24h |
LINCSCP_1361 |
LINCSCP_1361 |
A375 |
| 0.259291 |
1.918420e-16 |
975 |
Taurocholate |
LSM-5866 |
CEL |
10uM |
24h |
LINCSCP_32548 |
LINCSCP_32548 |
MCF7 |
| -0.259261 |
1.934384e-16 |
975 |
Tosedostat |
LSM-6286 |
ANPEP|C9orf3|DNPEP|ENPEP|ERAP1|ERAP2|LAP3|LNPEP|LVRN|METAP1|METAP1D|METAP2|NPEPL1|NPEPPS|RNPEP|RNPEPL1|XPNPEP1|XPNPEP2|XPNPEP3 |
10uM |
24h |
LINCSCP_38254 |
LINCSCP_38254 |
MCF7 |
| -0.25926 |
1.934654e-16 |
975 |
nifedipine |
LSM-4176 |
CACNA1C|CACNA1D|CACNA1F|CACNA1S|CACNA2D1 |
10uM |
6h |
LINCSCP_26319 |
LINCSCP_26319 |
HT29 |
| -0.259239 |
1.945923e-16 |
975 |
STK178014 |
LSM-43108 |
|
50uM |
6h |
LINCSCP_286650 |
LINCSCP_286650 |
SNGM |
| -0.259229 |
1.951028e-16 |
975 |
Isoniazid |
LSM-46042 |
CYP1A2|CYP2C19|CYP2C8|CYP2E1|CYP3A4 |
0.37uM |
24h |
LINCSCP_103904 |
LINCSCP_103904 |
HELA |
| -0.259214 |
1.959101e-16 |
975 |
Albendazole |
LSM-3782 |
|
1uM |
24h |
LINCSCP_37947 |
LINCSCP_37947 |
MCF7 |
| -0.259092 |
2.025694e-16 |
975 |
Withaferin A |
LSM-6685 |
IKBKB|NAMPT |
10uM |
24h |
LINCSCP_69099 |
LINCSCP_69099 |
A375 |
| -0.258935 |
2.114899e-16 |
975 |
Linagliptin |
LSM-45916 |
DPP4 |
1.11uM |
24h |
LINCSCP_135436 |
LINCSCP_135436 |
MCF7 |
| -0.258827 |
2.178506e-16 |
975 |
BRD-K22052171 |
LSM-9763 |
|
10uM |
24h |
LINCSCP_9006 |
LINCSCP_9006 |
A549 |
| -0.258802 |
2.193364e-16 |
975 |
Benzylpenicillin |
LSM-3229 |
|
0.12uM |
24h |
LINCSCP_76616 |
LINCSCP_76616 |
A375 |
| -0.25879 |
2.200462e-16 |
975 |
BSPBIO_000981 |
LSM-43126 |
ACTA1 |
10uM |
6h |
LINCSCP_20244 |
LINCSCP_20244 |
HCC515 |
| 0.258778 |
2.207553e-16 |
975 |
Lapatinib |
LSM-1051 |
EGFR|ERBB2 |
0.04uM |
24h |
LINCSCP_130007 |
LINCSCP_130007 |
LNCAP |
| 0.258743 |
2.228954e-16 |
975 |
Tropicamide |
LSM-1814 |
CHRM3|CHRM4 |
10uM |
24h |
LINCSCP_236089 |
LINCSCP_236089 |
MCF7 |
| -0.258737 |
2.232443e-16 |
975 |
Senicapoc |
LSM-45645 |
KCNN4 |
1.11uM |
24h |
LINCSCP_72204 |
LINCSCP_72204 |
A375 |
| 0.258718 |
2.244094e-16 |
975 |
BRD-K57732441 |
LSM-40434 |
|
10uM |
6h |
LINCSCP_295865 |
LINCSCP_295865 |
VCAP |
| 0.258684 |
2.265089e-16 |
975 |
BRD-K76454674 |
LSM-13105 |
|
5uM |
24h |
LINCSCP_61820 |
LINCSCP_61820 |
VCAP |
| 0.258676 |
2.270046e-16 |
975 |
EX-8678 |
LSM-1147 |
|
0.04uM |
3h |
LINCSCP_86447 |
LINCSCP_86447 |
BT20 |
| -0.258672 |
2.272524e-16 |
975 |
AZD-1152-HQPA |
LSM-1067 |
AURKA|AURKB |
0.1uM |
24h |
LINCSCP_11762 |
LINCSCP_11762 |
BT20 |
| 0.258625 |
2.301835e-16 |
975 |
GSK-1904529A |
LSM-1134 |
IGF1R|INSR |
0.1uM |
24h |
LINCSCP_205005 |
LINCSCP_205005 |
BT20 |
| 0.25861 |
2.311573e-16 |
975 |
Alfadolone |
LSM-5265 |
|
10uM |
6h |
LINCSCP_47893 |
LINCSCP_47893 |
PC3 |
| -0.258597 |
2.319596e-16 |
975 |
PK04PUR_000067 |
LSM-36645 |
|
10uM |
24h |
LINCSCP_32121 |
LINCSCP_32121 |
MCF7 |
| 0.258564 |
2.340529e-16 |
975 |
MLS002699811 |
LSM-3541 |
|
10uM |
6h |
LINCSCP_219542 |
LINCSCP_219542 |
HEPG2 |
| 0.258523 |
2.367239e-16 |
975 |
CHEMBL2361177 |
LSM-37819 |
|
10uM |
6h |
LINCSCP_16787 |
LINCSCP_16787 |
HA1E |
| -0.258517 |
2.371292e-16 |
975 |
CHEMBL2141850 |
LSM-6136 |
|
10uM |
24h |
LINCSCP_46488 |
LINCSCP_46488 |
PC3 |
| 0.258482 |
2.393800e-16 |
975 |
Rifampicin |
LSM-43162 |
NR1I2 |
10uM |
6h |
LINCSCP_194060 |
LINCSCP_194060 |
A549 |
| -0.258467 |
2.403484e-16 |
975 |
BRD-K84450674 |
LSM-41883 |
|
10uM |
6h |
LINCSCP_16896 |
LINCSCP_16896 |
HA1E |
| -0.258452 |
2.413887e-16 |
975 |
Mepireserpate |
LSM-1758 |
SLC18A1|SLC18A2 |
10uM |
24h |
LINCSCP_245 |
LINCSCP_245 |
A375 |
| 0.258358 |
2.476162e-16 |
975 |
BMS-345541 |
LSM-1028 |
IKBKB |
0.5uM |
24h |
LINCSCP_38945 |
LINCSCP_38945 |
MDAMB231 |
| -0.258333 |
2.493470e-16 |
975 |
Triciribine |
LSM-3810 |
AKT1|AKT2|AKT3 |
10uM |
24h |
LINCSCP_42927 |
LINCSCP_42927 |
NPC |
| -0.258218 |
2.572841e-16 |
975 |
MLS002264466 |
LSM-3995 |
|
10uM |
24h |
LINCSCP_5440 |
LINCSCP_5440 |
A549 |
| -0.25811 |
2.649778e-16 |
975 |
Albendazole |
LSM-3782 |
|
10uM |
6h |
LINCSCP_228015 |
LINCSCP_228015 |
HT29 |
| -0.258107 |
2.652246e-16 |
975 |
HMN-214 |
LSM-42802 |
CSF1R|FLT1|FLT3|FLT4|KDR|KIT|PDGFRB|RET |
10uM |
24h |
LINCSCP_134181 |
LINCSCP_134181 |
MCF7 |
| -0.258094 |
2.661125e-16 |
975 |
BRD-K79793579 |
LSM-41625 |
|
10uM |
24h |
LINCSCP_201007 |
LINCSCP_201007 |
A549 |
| 0.25798 |
2.745502e-16 |
975 |
BRD-K35769695 |
LSM-10575 |
|
5uM |
24h |
LINCSCP_63370 |
LINCSCP_63370 |
VCAP |
| 0.257938 |
2.776763e-16 |
975 |
BRD-M77293869 |
LSM-45066 |
|
5uM |
24h |
LINCSCP_64050 |
LINCSCP_64050 |
VCAP |
| -0.257742 |
2.929730e-16 |
975 |
Auranofin |
LSM-43136 |
|
10uM |
6h |
LINCSCP_894 |
LINCSCP_894 |
A375 |
| -0.257651 |
3.002897e-16 |
975 |
PS-1145 |
LSM-5975 |
IKBKB |
5uM |
6h |
LINCSCP_257472 |
LINCSCP_257472 |
NCIH508 |
| -0.257649 |
3.004857e-16 |
975 |
ZM-241385 |
LSM-2444 |
ADORA1|ADORA2A|ADORA2B |
10uM |
24h |
LINCSCP_52863 |
LINCSCP_52863 |
SKB |
| 0.257636 |
3.015494e-16 |
975 |
BRD-K74294292 |
LSM-12978 |
|
5uM |
24h |
LINCSCP_61280 |
LINCSCP_61280 |
VCAP |
| -0.257604 |
3.041634e-16 |
975 |
BRD-K84976438 |
LSM-13619 |
|
3uM |
24h |
LINCSCP_252760 |
LINCSCP_252760 |
MCF7 |
| 0.25754 |
3.095353e-16 |
975 |
Bumetanide |
LSM-2848 |
SLC12A1|SLC12A2 |
3.33uM |
24h |
LINCSCP_171251 |
LINCSCP_171251 |
YAPC |
| -0.257536 |
3.098360e-16 |
975 |
10-DEBC |
LSM-4710 |
PIM1 |
20uM |
24h |
LINCSCP_45004 |
LINCSCP_45004 |
PC3 |
| 0.25747 |
3.154872e-16 |
975 |
COT Inhibitor-2 |
LSM-1154 |
|
0.12uM |
24h |
LINCSCP_128152 |
LINCSCP_128152 |
HUES3 |
| -0.257377 |
3.235799e-16 |
975 |
CHEMBL2361739 |
LSM-8809 |
|
5uM |
24h |
LINCSCP_63333 |
LINCSCP_63333 |
VCAP |
| 0.257324 |
3.282350e-16 |
975 |
BRD-K07039703 |
LSM-14704 |
|
5uM |
24h |
LINCSCP_64153 |
LINCSCP_64153 |
VCAP |
| -0.257313 |
3.291869e-16 |
975 |
Buparlisib |
LSM-1148 |
PIK3CA|PIK3CB|PIK3CD|PIK3CG|PIK3R1|PIK3R2|PIK3R3|PIK3R5 |
10uM |
24h |
LINCSCP_136776 |
LINCSCP_136776 |
MCF7 |
| -0.257262 |
3.337744e-16 |
975 |
BRD-K44070326 |
LSM-7405 |
|
10uM |
24h |
LINCSCP_312013 |
LINCSCP_312013 |
VCAP |
| -0.257228 |
3.369608e-16 |
975 |
Coumestrol |
LSM-4202 |
ESR1|ESR2 |
10uM |
24h |
LINCSCP_284556 |
LINCSCP_284556 |
SKB |
| -0.257225 |
3.371537e-16 |
975 |
GW843682X |
LSM-1014 |
PLK1|PLK3 |
10uM |
24h |
LINCSCP_38251 |
LINCSCP_38251 |
MCF7 |
| -0.257214 |
3.381660e-16 |
975 |
CHEMBL2137726 |
LSM-2429 |
|
10uM |
24h |
LINCSCP_57527 |
LINCSCP_57527 |
VCAP |
| -0.25716 |
3.431592e-16 |
975 |
Isocarboxazid |
LSM-4101 |
MAOA|MAOB |
10uM |
24h |
LINCSCP_47675 |
LINCSCP_47675 |
PC3 |
| -0.257067 |
3.519945e-16 |
975 |
BRD-K13688115-001-01-2 |
LSM-5315 |
NR3C1 |
10uM |
24h |
LINCSCP_243940 |
LINCSCP_243940 |
MCF7 |
| -0.25705 |
3.536061e-16 |
975 |
BRD-A72596465 |
LSM-1765 |
PPARA |
10uM |
6h |
LINCSCP_290268 |
LINCSCP_290268 |
VCAP |
| 0.257046 |
3.539492e-16 |
975 |
Disopyramide |
LSM-1439 |
SCN10A|SCN11A|SCN1A|SCN2A|SCN3A|SCN4A|SCN5A|SCN7A|SCN8A|SCN9A |
0.37uM |
24h |
LINCSCP_71292 |
LINCSCP_71292 |
A375 |
| 0.257045 |
3.541074e-16 |
975 |
SCHEMBL3958507 |
LSM-5245 |
COQ8B|EGFR |
0.37uM |
3h |
LINCSCP_131499 |
LINCSCP_131499 |
MCF10A |
| 0.257031 |
3.554253e-16 |
975 |
BRD-K38865695 |
LSM-10782 |
|
5uM |
24h |
LINCSCP_61596 |
LINCSCP_61596 |
VCAP |
| -0.256947 |
3.636369e-16 |
975 |
WHI-P154 |
|
EGFR|JAK3 |
10uM |
24h |
LINCSCP_52756 |
LINCSCP_52756 |
SKB |
| -0.25684 |
3.743613e-16 |
975 |
Pimavanserin |
LSM-45960 |
HTR2A |
0.12uM |
24h |
LINCSCP_173145 |
LINCSCP_173145 |
YAPC |
| -0.256817 |
3.767033e-16 |
975 |
Balicatib |
LSM-45647 |
|
1.11uM |
24h |
LINCSCP_154142 |
LINCSCP_154142 |
PC3 |
| -0.256807 |
3.777687e-16 |
975 |
L-694247 |
LSM-2416 |
HTR1D |
10uM |
6h |
LINCSCP_56133 |
LINCSCP_56133 |
VCAP |
| -0.256792 |
3.792559e-16 |
975 |
MLS002473640 |
LSM-3067 |
|
10uM |
24h |
LINCSCP_177851 |
LINCSCP_177851 |
A375 |
| 0.256752 |
3.833721e-16 |
975 |
BRD-K34431359 |
LSM-10507 |
|
5uM |
24h |
LINCSCP_61765 |
LINCSCP_61765 |
VCAP |
| 0.256716 |
3.871474e-16 |
975 |
SB-431542 |
LSM-3498 |
ACVR1C|TGFBR1 |
10uM |
24h |
LINCSCP_33404 |
LINCSCP_33404 |
MCF7 |
| 0.256707 |
3.881076e-16 |
975 |
Nicardipine |
LSM-1418 |
CACNA1C|CACNA1D|CACNA1F|CACNA1S |
10uM |
6h |
LINCSCP_55408 |
LINCSCP_55408 |
U937 |
| -0.256658 |
3.932917e-16 |
975 |
AC1MSUFC |
LSM-6191 |
HMGCR |
40uM |
6h |
LINCSCP_51060 |
LINCSCP_51060 |
RMUGS |
| -0.256619 |
3.975059e-16 |
975 |
CHEMBL2136735 |
LSM-1152 |
FGFR1|FGFR3|FLT1|FLT4|KDR|PDGFRA|PDGFRB |
0.37uM |
24h |
LINCSCP_151252 |
LINCSCP_151252 |
PC3 |
| 0.256598 |
3.997072e-16 |
975 |
ZSTK 474 |
LSM-1053 |
PIK3CG |
0.04uM |
3h |
LINCSCP_130355 |
LINCSCP_130355 |
LNCAP |
| 0.256534 |
4.067711e-16 |
975 |
CHEMBL2135537 |
LSM-6149 |
|
10uM |
6h |
LINCSCP_59386 |
LINCSCP_59386 |
VCAP |
| 0.256486 |
4.120802e-16 |
975 |
Penitrem A |
LSM-2058 |
KCNMA1 |
0.01uM |
24h |
LINCSCP_134859 |
LINCSCP_134859 |
MCF7 |
| -0.256453 |
4.157622e-16 |
975 |
BRD-K06170455 |
LSM-37608 |
|
5uM |
6h |
LINCSCP_4100 |
LINCSCP_4100 |
A375 |
| 0.256444 |
4.167382e-16 |
975 |
Homatropine |
LSM-1299 |
CHRM1 |
10uM |
6h |
LINCSCP_4262 |
LINCSCP_4262 |
A549 |
| -0.256271 |
4.368237e-16 |
975 |
NMS-1286937 |
LSM-45818 |
|
1.11uM |
24h |
LINCSCP_141871 |
LINCSCP_141871 |
MCF7 |
| -0.256264 |
4.375593e-16 |
975 |
Temozolomide |
LSM-4590 |
MGMT |
10uM |
6h |
LINCSCP_29132 |
LINCSCP_29132 |
JHUEM2 |
| -0.256233 |
4.412977e-16 |
975 |
Lexibulin |
LSM-6232 |
TUBA1A|TUBA1B|TUBA1C|TUBA3E|TUBA4A|TUBB|TUBB1|TUBB2A|TUBB2B|TUBB3|TUBB4A|TUBB4B|TUBB6|TUBB8 |
0.12uM |
24h |
LINCSCP_135774 |
LINCSCP_135774 |
MCF7 |
| -0.256159 |
4.502337e-16 |
975 |
BRD-K02575886 |
LSM-37417 |
|
10uM |
24h |
LINCSCP_311954 |
LINCSCP_311954 |
VCAP |
| -0.25615 |
4.513080e-16 |
975 |
Colchicine |
LSM-5199 |
TUBA1A|TUBA1B|TUBA1C|TUBA3E|TUBA4A|TUBB|TUBB1|TUBB2A|TUBB2B|TUBB3|TUBB4A|TUBB4B|TUBB6|TUBB8 |
10uM |
24h |
LINCSCP_37617 |
LINCSCP_37617 |
MCF7 |
| -0.2561 |
4.574354e-16 |
975 |
BRD-K03641022 |
LSM-37474 |
|
10uM |
24h |
LINCSCP_3514 |
LINCSCP_3514 |
A375 |
| 0.256079 |
4.600430e-16 |
975 |
BRD-K52904986 |
LSM-11657 |
|
5uM |
24h |
LINCSCP_62011 |
LINCSCP_62011 |
VCAP |
| -0.256012 |
4.684270e-16 |
975 |
PD-0325901 |
LSM-1101 |
MAP2K1|MAP2K2 |
10uM |
6h |
LINCSCP_46605 |
LINCSCP_46605 |
PC3 |
| 0.255837 |
4.911136e-16 |
975 |
BRD-K48877010 |
LSM-11404 |
|
5uM |
24h |
LINCSCP_61464 |
LINCSCP_61464 |
VCAP |
| 0.255734 |
5.050406e-16 |
975 |
Vorinostat |
LSM-3828 |
HDAC1|HDAC2|HDAC3|HDAC6|HDAC8 |
0.1uM |
24h |
LINCSCP_68901 |
LINCSCP_68901 |
VCAP |
| 0.255645 |
5.172347e-16 |
975 |
Ondansetron |
LSM-1375 |
HTR3A |
0.04uM |
24h |
LINCSCP_72136 |
LINCSCP_72136 |
A375 |
| 0.25561 |
5.222625e-16 |
975 |
BRD-K16331350 |
LSM-9411 |
|
5uM |
24h |
LINCSCP_62861 |
LINCSCP_62861 |
VCAP |
| 0.255566 |
5.284598e-16 |
975 |
EX-8678 |
LSM-1147 |
|
1.11uM |
3h |
LINCSCP_164122 |
LINCSCP_164122 |
SKBR3 |
| 0.255512 |
5.361995e-16 |
975 |
BRD-K52225919 |
LSM-11625 |
|
5uM |
24h |
LINCSCP_62891 |
LINCSCP_62891 |
VCAP |
| -0.255474 |
5.417587e-16 |
975 |
SA-89068 |
LSM-42386 |
|
3uM |
6h |
LINCSCP_252531 |
LINCSCP_252531 |
MCF7 |
| 0.255466 |
5.428964e-16 |
975 |
Kinetin Riboside |
LSM-6292 |
|
10uM |
6h |
LINCSCP_15688 |
LINCSCP_15688 |
HA1E |
| -0.255456 |
5.444187e-16 |
975 |
SB 239063 |
LSM-44951 |
MAPK11|MAPK14 |
10uM |
6h |
LINCSCP_51721 |
LINCSCP_51721 |
SKBR3 |
| 0.255412 |
5.507841e-16 |
975 |
Indigo Red |
LSM-42899 |
CDK1|CDK5|GSK3A |
1.11uM |
24h |
LINCSCP_71637 |
LINCSCP_71637 |
A375 |
| 0.255343 |
5.611464e-16 |
975 |
CHEMBL1986318 |
LSM-6610 |
|
10uM |
6h |
LINCSCP_34037 |
LINCSCP_34037 |
MCF7 |
| 0.255325 |
5.639252e-16 |
975 |
RASAGILINE |
LSM-45548 |
MAOB |
0.04uM |
24h |
LINCSCP_123128 |
LINCSCP_123128 |
HT29 |
| 0.255309 |
5.663165e-16 |
975 |
BRD-K78528600 |
LSM-13229 |
|
5uM |
24h |
LINCSCP_61827 |
LINCSCP_61827 |
VCAP |
| -0.255237 |
5.774962e-16 |
975 |
N-(1,3-Benzothiazol-2-yl)thiophene-2-carboxamide |
LSM-3900 |
|
10uM |
24h |
LINCSCP_1430 |
LINCSCP_1430 |
A375 |
| 0.255221 |
5.799180e-16 |
975 |
Lapatinib |
LSM-1051 |
EGFR|ERBB2 |
10uM |
3h |
LINCSCP_133181 |
LINCSCP_133181 |
MCF7 |
| 0.255207 |
5.822224e-16 |
975 |
CYTO7H11 |
LSM-4351 |
BAX |
1uM |
6h |
LINCSCP_201831 |
LINCSCP_201831 |
A549 |
| 0.255167 |
5.883818e-16 |
975 |
BRD-K71915010 |
LSM-6148 |
|
10uM |
6h |
LINCSCP_217317 |
LINCSCP_217317 |
HCC515 |
| 0.255099 |
5.993114e-16 |
975 |
LY456236 |
LSM-3955 |
GRM1 |
10uM |
24h |
LINCSCP_33127 |
LINCSCP_33127 |
MCF7 |
| 0.254869 |
6.375526e-16 |
975 |
CID755673 |
LSM-2050 |
|
10uM |
24h |
LINCSCP_45282 |
LINCSCP_45282 |
PC3 |
| -0.254816 |
6.468103e-16 |
975 |
MLS003337115 |
LSM-3510 |
|
10uM |
24h |
LINCSCP_45730 |
LINCSCP_45730 |
PC3 |
| -0.254793 |
6.508534e-16 |
975 |
LY-294002 |
LSM-2597 |
MTOR|PIK3CA|PIK3CB|PIK3CD|PIK3CG|PLK1|PRKDC |
10uM |
24h |
LINCSCP_200925 |
LINCSCP_200925 |
A549 |
| 0.254785 |
6.522201e-16 |
975 |
BRD-K80789291 |
LSM-13369 |
|
5uM |
24h |
LINCSCP_62320 |
LINCSCP_62320 |
VCAP |
| 0.254759 |
6.567767e-16 |
975 |
Carbacyclin |
LSM-42923 |
PPARD|PTGIR |
10uM |
24h |
LINCSCP_55311 |
LINCSCP_55311 |
U937 |
| -0.254737 |
6.606168e-16 |
975 |
CHEMBL1433941 |
LSM-3587 |
|
10uM |
24h |
LINCSCP_31645 |
LINCSCP_31645 |
MCF7 |
| -0.254634 |
6.791868e-16 |
975 |
Auranofin |
LSM-43136 |
|
10uM |
6h |
LINCSCP_30721 |
LINCSCP_30721 |
MCF7 |
| 0.254505 |
7.031107e-16 |
975 |
AKT Inhibitor VIII |
LSM-1035 |
AKT1|AKT2 |
10uM |
6h |
LINCSCP_12784 |
LINCSCP_12784 |
DV90 |
| 0.254456 |
7.125281e-16 |
975 |
BRD-K66413861 |
LSM-12475 |
|
5uM |
24h |
LINCSCP_62676 |
LINCSCP_62676 |
VCAP |
| 0.254442 |
7.151459e-16 |
975 |
Dibenzoylmethane |
LSM-2003 |
|
10uM |
6h |
LINCSCP_4331 |
LINCSCP_4331 |
A549 |
| 0.254388 |
7.256797e-16 |
975 |
BRD-K72381041 |
LSM-41194 |
|
10uM |
6h |
LINCSCP_22412 |
LINCSCP_22412 |
HEPG2 |
| 0.254384 |
7.263440e-16 |
975 |
Chlorprothixene |
LSM-42990 |
DRD2|DRD3|HTR2A|HTR2C |
10uM |
24h |
LINCSCP_34315 |
LINCSCP_34315 |
MCF7 |
| -0.254362 |
7.306836e-16 |
975 |
AZD-5438 |
LSM-1159 |
CDK1|CDK10|CDK11B|CDK12|CDK13|CDK14|CDK15|CDK16|CDK17|CDK18|CDK19|CDK2|CDK20|CDK3|CDK4|CDK5|CDK6|CDK7|CDK8|CDK9 |
0.04uM |
24h |
LINCSCP_151302 |
LINCSCP_151302 |
PC3 |
| 0.254331 |
7.367704e-16 |
975 |
BRD-K67766243 |
LSM-12557 |
|
5uM |
24h |
LINCSCP_61487 |
LINCSCP_61487 |
VCAP |
| -0.254306 |
7.416600e-16 |
975 |
MLS001065837 |
LSM-2605 |
|
10uM |
24h |
LINCSCP_1138 |
LINCSCP_1138 |
A375 |
| -0.254264 |
7.501300e-16 |
975 |
Mitotane |
LSM-1451 |
CYP11A1|CYP11B1 |
10uM |
24h |
LINCSCP_32819 |
LINCSCP_32819 |
MCF7 |
| 0.254131 |
7.774754e-16 |
975 |
BRD-K69498175 |
LSM-12668 |
|
5uM |
24h |
LINCSCP_61813 |
LINCSCP_61813 |
VCAP |
| -0.254127 |
7.782253e-16 |
975 |
Maprotiline |
LSM-2043 |
SLC6A2 |
10uM |
24h |
LINCSCP_46081 |
LINCSCP_46081 |
PC3 |
| -0.254116 |
7.806072e-16 |
975 |
2-(4-Nitro-phenylamino)-benzoic acid |
LSM-45307 |
|
1uM |
24h |
LINCSCP_222191 |
LINCSCP_222191 |
HL60 |
| 0.254066 |
7.911072e-16 |
975 |
BRD-K26684619 |
LSM-45323 |
|
1uM |
24h |
LINCSCP_205456 |
LINCSCP_205456 |
CD34 |
| 0.254049 |
7.946169e-16 |
975 |
XMD 8-92 |
LSM-1094 |
MAPK7 |
3.33uM |
24h |
LINCSCP_87217 |
LINCSCP_87217 |
CD34 |
| -0.254029 |
7.990309e-16 |
975 |
MK-5108 |
LSM-36812 |
AURKA|AURKB |
10uM |
24h |
LINCSCP_38688 |
LINCSCP_38688 |
MCF7 |
| 0.254021 |
8.007669e-16 |
975 |
BRD-K10600561 |
LSM-9066 |
|
5uM |
24h |
LINCSCP_63970 |
LINCSCP_63970 |
VCAP |
| 0.253948 |
8.165157e-16 |
975 |
GSK429286A |
LSM-1012 |
ROCK1 |
0.04uM |
24h |
LINCSCP_87227 |
LINCSCP_87227 |
CD34 |
| 0.253907 |
8.256038e-16 |
975 |
BRD-K51083659 |
LSM-40089 |
|
10uM |
6h |
LINCSCP_16848 |
LINCSCP_16848 |
HA1E |
| -0.253836 |
8.414439e-16 |
975 |
Nocodazole |
LSM-2260 |
|
3uM |
24h |
LINCSCP_37646 |
LINCSCP_37646 |
MCF7 |
| 0.253815 |
8.461066e-16 |
975 |
CHEMBL552425 |
LSM-1003 |
DDR1 |
0.12uM |
24h |
LINCSCP_133278 |
LINCSCP_133278 |
MCF7 |
| -0.253791 |
8.515198e-16 |
975 |
Vitinoin |
LSM-2135 |
RARA|RARB|RARG|RORB |
10uM |
24h |
LINCSCP_253452 |
LINCSCP_253452 |
MCF7 |
| -0.253767 |
8.569477e-16 |
975 |
PLX-4720 |
LSM-1049 |
BRAF |
0.1uM |
6h |
LINCSCP_36 |
LINCSCP_36 |
A375 |
| -0.253735 |
8.645072e-16 |
975 |
Leu-Enkephalin |
LSM-1461 |
OPRD1|OPRM1 |
10uM |
6h |
LINCSCP_4278 |
LINCSCP_4278 |
A549 |
| -0.253713 |
8.694984e-16 |
975 |
NMS-1286937 |
LSM-45818 |
|
10uM |
24h |
LINCSCP_141869 |
LINCSCP_141869 |
MCF7 |
| 0.253612 |
8.934253e-16 |
975 |
BRD-K92758184 |
LSM-14113 |
|
5uM |
24h |
LINCSCP_61851 |
LINCSCP_61851 |
VCAP |
| -0.253591 |
8.984668e-16 |
975 |
Clofibric acid |
LSM-2427 |
PPARA |
10uM |
24h |
LINCSCP_108323 |
LINCSCP_108323 |
HELA |
| 0.253437 |
9.360477e-16 |
975 |
TIE2 Kinase Inhibitor |
LSM-1194 |
|
0.04uM |
24h |
LINCSCP_87544 |
LINCSCP_87544 |
CD34 |
| -0.253359 |
9.559844e-16 |
975 |
MLS-0208612.0001 |
LSM-3196 |
|
10uM |
24h |
LINCSCP_31621 |
LINCSCP_31621 |
MCF7 |
| 0.253341 |
9.604341e-16 |
975 |
BRD-K38481268 |
LSM-10756 |
|
5uM |
24h |
LINCSCP_62148 |
LINCSCP_62148 |
VCAP |
| 0.253334 |
9.621913e-16 |
975 |
SCHEMBL618594 |
LSM-1070 |
|
10uM |
24h |
LINCSCP_52331 |
LINCSCP_52331 |
SKB |
| 0.253271 |
9.785418e-16 |
975 |
BRD-K59176197 |
LSM-12003 |
|
5uM |
24h |
LINCSCP_62302 |
LINCSCP_62302 |
VCAP |
| -0.25325 |
9.842213e-16 |
975 |
Cnqx |
LSM-3184 |
|
1.11uM |
24h |
LINCSCP_72843 |
LINCSCP_72843 |
A375 |
| 0.253163 |
1.007192e-15 |
975 |
4-Iodo-6-phenylpyrimidine |
LSM-6233 |
MIF |
40uM |
6h |
LINCSCP_40196 |
LINCSCP_40196 |
NCIH508 |
| -0.253163 |
1.007375e-15 |
975 |
PCL2_000154 |
LSM-36683 |
|
10uM |
6h |
LINCSCP_32333 |
LINCSCP_32333 |
MCF7 |
| -0.253162 |
1.007637e-15 |
975 |
Triazine Scaffold, 31 |
LSM-2261 |
|
10uM |
6h |
LINCSCP_31053 |
LINCSCP_31053 |
MCF7 |
| 0.253138 |
1.013912e-15 |
975 |
BRD-K11088254 |
LSM-9105 |
|
5uM |
24h |
LINCSCP_62431 |
LINCSCP_62431 |
VCAP |
| -0.253128 |
1.016581e-15 |
975 |
Methylergonovine |
LSM-2758 |
DRD1|HTR2B |
10uM |
6h |
LINCSCP_4359 |
LINCSCP_4359 |
A549 |
| 0.253113 |
1.020772e-15 |
975 |
BRD-K83541009 |
LSM-41836 |
|
5uM |
24h |
LINCSCP_64331 |
LINCSCP_64331 |
VCAP |
| -0.253078 |
1.030463e-15 |
975 |
Dasatinib |
LSM-1020 |
ABL1|BCR|BLK|EPHA2|FGR|FRK|FYN|HCK|KIT|LCK|LYN|PDGFRB|SRC|SRMS|YES1 |
1.11uM |
24h |
LINCSCP_69023 |
LINCSCP_69023 |
A375 |
| 0.253058 |
1.035803e-15 |
975 |
NSC95397 |
LSM-3521 |
|
10uM |
6h |
LINCSCP_6982 |
LINCSCP_6982 |
A549 |
| -0.252999 |
1.052381e-15 |
975 |
SA-84869 |
LSM-41398 |
|
10uM |
24h |
LINCSCP_260399 |
LINCSCP_260399 |
NKDBA |
| 0.252886 |
1.084601e-15 |
975 |
Tozasertib |
LSM-1021 |
ABL1|AURKA|AURKB|AURKC|BCR|FLT3|JAK2 |
1.11uM |
24h |
LINCSCP_76250 |
LINCSCP_76250 |
A375 |
| -0.252875 |
1.087792e-15 |
975 |
BRD-K48193278 |
LSM-39946 |
|
5uM |
24h |
LINCSCP_249256 |
LINCSCP_249256 |
MCF7 |
| 0.252812 |
1.106250e-15 |
975 |
Ricolinostat |
LSM-6324 |
|
0.12uM |
24h |
LINCSCP_164656 |
LINCSCP_164656 |
SKL.C |
| -0.252749 |
1.124770e-15 |
975 |
Tangeretin |
LSM-2548 |
|
10uM |
24h |
LINCSCP_52867 |
LINCSCP_52867 |
SKB |
| -0.252669 |
1.149086e-15 |
975 |
BRD-K81646882 |
LSM-41730 |
|
10uM |
6h |
LINCSCP_279534 |
LINCSCP_279534 |
PC3 |
| 0.252655 |
1.153366e-15 |
975 |
AC1NWAOC |
LSM-21624 |
|
0.37uM |
24h |
LINCSCP_123298 |
LINCSCP_123298 |
HT29 |
| -0.252655 |
1.153451e-15 |
975 |
Levobunolol |
LSM-6578 |
ADRB1|ADRB2 |
0.37uM |
24h |
LINCSCP_101899 |
LINCSCP_101899 |
HELA |
| -0.252649 |
1.155270e-15 |
975 |
Podofilox |
LSM-3055 |
|
0.04uM |
24h |
LINCSCP_141628 |
LINCSCP_141628 |
MCF7 |
| 0.252597 |
1.171511e-15 |
975 |
BRD-K96257627 |
LSM-14334 |
|
5uM |
24h |
LINCSCP_61515 |
LINCSCP_61515 |
VCAP |
| -0.252484 |
1.207298e-15 |
975 |
CAY10603 |
LSM-4941 |
HDAC6 |
10uM |
6h |
LINCSCP_218567 |
LINCSCP_218567 |
HCT116 |
| 0.252481 |
1.208246e-15 |
975 |
EX-8678 |
LSM-1147 |
|
0.37uM |
3h |
LINCSCP_133190 |
LINCSCP_133190 |
MCF7 |
| 0.252477 |
1.209260e-15 |
975 |
Gefitinib |
LSM-1098 |
EGFR |
10uM |
24h |
LINCSCP_130014 |
LINCSCP_130014 |
LNCAP |
| -0.252421 |
1.227589e-15 |
975 |
Thioguanosine |
LSM-5832 |
|
3.33uM |
24h |
LINCSCP_143346 |
LINCSCP_143346 |
MCF7 |
| -0.252393 |
1.236739e-15 |
975 |
Metyrapone |
LSM-3035 |
CYP11B1 |
10uM |
6h |
LINCSCP_30372 |
LINCSCP_30372 |
MCF7 |
| -0.252368 |
1.245129e-15 |
975 |
Colchicine |
LSM-5199 |
TUBA1A|TUBA1B|TUBA1C|TUBA3E|TUBA4A|TUBB|TUBB1|TUBB2A|TUBB2B|TUBB3|TUBB4A|TUBB4B|TUBB6|TUBB8 |
1uM |
24h |
LINCSCP_37618 |
LINCSCP_37618 |
MCF7 |
| -0.252336 |
1.255753e-15 |
975 |
BRD-K53640012 |
LSM-40218 |
|
1uM |
24h |
LINCSCP_66117 |
LINCSCP_66117 |
VCAP |
| -0.25233 |
1.257537e-15 |
975 |
PNU-74654 |
LSM-44945 |
CTNNB1|TCF4 |
80uM |
6h |
LINCSCP_25750 |
LINCSCP_25750 |
HT29 |
| -0.252238 |
1.288678e-15 |
975 |
KX2-391 |
LSM-45890 |
SRC |
3.33uM |
24h |
LINCSCP_137497 |
LINCSCP_137497 |
MCF7 |
| -0.252113 |
1.332457e-15 |
975 |
BRD-K84976438 |
LSM-13619 |
|
10uM |
24h |
LINCSCP_252758 |
LINCSCP_252758 |
MCF7 |
| -0.252109 |
1.333852e-15 |
975 |
Mosapride |
LSM-5042 |
HTR4 |
10uM |
6h |
LINCSCP_5811 |
LINCSCP_5811 |
A549 |
| -0.252089 |
1.340993e-15 |
975 |
Tropicamide |
LSM-1814 |
CHRM3|CHRM4 |
10uM |
24h |
LINCSCP_271966 |
LINCSCP_271966 |
PC3 |
| -0.252083 |
1.343123e-15 |
975 |
Mozavaptan |
LSM-45912 |
|
10uM |
24h |
LINCSCP_137568 |
LINCSCP_137568 |
MCF7 |
| 0.25201 |
1.369521e-15 |
975 |
BRD-K46359800 |
LSM-11257 |
|
5uM |
24h |
LINCSCP_60886 |
LINCSCP_60886 |
VCAP |
| 0.252003 |
1.371955e-15 |
975 |
AC1MEVG9 |
LSM-3935 |
PTPN1 |
10uM |
6h |
LINCSCP_40249 |
LINCSCP_40249 |
NCIH508 |
| -0.251961 |
1.387325e-15 |
975 |
Procaterol |
LSM-1391 |
ADRB2 |
10uM |
24h |
LINCSCP_37848 |
LINCSCP_37848 |
MCF7 |
| -0.25192 |
1.402647e-15 |
975 |
altrenogest |
LSM-45498 |
|
0.12uM |
24h |
LINCSCP_139858 |
LINCSCP_139858 |
MCF7 |
| 0.251845 |
1.430718e-15 |
975 |
BRD-K62957477 |
LSM-12256 |
|
5uM |
24h |
LINCSCP_63105 |
LINCSCP_63105 |
VCAP |
| 0.251695 |
1.488664e-15 |
975 |
Cholic acid |
LSM-5541 |
CES1|FECH|PLA2G1B |
3.33uM |
24h |
LINCSCP_122513 |
LINCSCP_122513 |
HT29 |
| -0.251678 |
1.495706e-15 |
975 |
MLS001207806 |
LSM-43094 |
|
10uM |
24h |
LINCSCP_37912 |
LINCSCP_37912 |
MCF7 |
| -0.251675 |
1.496771e-15 |
975 |
CHEMBL1165368 |
LSM-42920 |
CHRNA7 |
10uM |
24h |
LINCSCP_44022 |
LINCSCP_44022 |
PC3 |
| 0.251634 |
1.513049e-15 |
975 |
Bifonazole |
LSM-5184 |
|
1.11uM |
24h |
LINCSCP_162166 |
LINCSCP_162166 |
PC3 |
| -0.251615 |
1.520681e-15 |
975 |
Dorzolamide HCL |
LSM-45672 |
|
10uM |
24h |
LINCSCP_142643 |
LINCSCP_142643 |
MCF7 |
| -0.251583 |
1.533828e-15 |
975 |
MLS003221389 |
LSM-4220 |
|
10uM |
24h |
LINCSCP_177960 |
LINCSCP_177960 |
A375 |
| 0.251566 |
1.540495e-15 |
975 |
BRD-K24192521 |
LSM-9892 |
|
5uM |
24h |
LINCSCP_63356 |
LINCSCP_63356 |
VCAP |
| 0.251548 |
1.548026e-15 |
975 |
Emedastine |
LSM-5331 |
HRH1 |
0.04uM |
24h |
LINCSCP_74493 |
LINCSCP_74493 |
A375 |
| 0.251545 |
1.549060e-15 |
975 |
BRD-K28105726 |
LSM-10132 |
|
5uM |
24h |
LINCSCP_62639 |
LINCSCP_62639 |
VCAP |
| -0.251528 |
1.556117e-15 |
975 |
Cidoxepin |
LSM-42948 |
HRH1|HRH2|SLC6A2|SLC6A4 |
10uM |
24h |
LINCSCP_284715 |
LINCSCP_284715 |
SKB |
| 0.251505 |
1.565796e-15 |
975 |
BRD-K66205522 |
LSM-12467 |
|
5uM |
6h |
LINCSCP_62569 |
LINCSCP_62569 |
VCAP |
| 0.251473 |
1.579069e-15 |
975 |
BRD-K56943062 |
LSM-11873 |
|
5uM |
6h |
LINCSCP_62220 |
LINCSCP_62220 |
VCAP |
| 0.25147 |
1.580187e-15 |
975 |
Niacin |
LSM-4676 |
HCAR2|HCAR3 |
10uM |
24h |
LINCSCP_28825 |
LINCSCP_28825 |
HUH7 |
| -0.251466 |
1.582184e-15 |
975 |
Dactolisib |
LSM-4255 |
MTOR|PIK3CA|PIK3CB|PIK3CD|PIK3CG|PIK3R1|PIK3R2|PIK3R3|PIK3R5 |
0.5uM |
24h |
LINCSCP_4488 |
LINCSCP_4488 |
A549 |
| -0.251449 |
1.589181e-15 |
975 |
Linoleic acid |
LSM-42867 |
|
10uM |
6h |
LINCSCP_472 |
LINCSCP_472 |
A375 |
| -0.251397 |
1.611113e-15 |
975 |
ENMD-2076 |
LSM-45335 |
AURKA|AURKB|CSF1R|FGFR3|FLT3|KDR|KIT|PDGFRA|SRC |
3.33uM |
24h |
LINCSCP_97098 |
LINCSCP_97098 |
HA1E |
| 0.251377 |
1.619939e-15 |
975 |
BRD-K74711637 |
LSM-6151 |
|
10uM |
6h |
LINCSCP_16361 |
LINCSCP_16361 |
HA1E |
| -0.251302 |
1.652224e-15 |
975 |
Rifapentine |
LSM-46028 |
CYP2C8|CYP2C9|CYP3A4 |
10uM |
24h |
LINCSCP_237850 |
LINCSCP_237850 |
MCF7 |
| 0.251229 |
1.684731e-15 |
975 |
BS-181 |
LSM-6305 |
|
0.04uM |
24h |
LINCSCP_86837 |
LINCSCP_86837 |
CD34 |
| -0.251076 |
1.754152e-15 |
975 |
U0126 |
LSM-1220 |
|
10uM |
24h |
LINCSCP_42898 |
LINCSCP_42898 |
NPC |
| 0.251074 |
1.754974e-15 |
975 |
Dacinostat |
LSM-43097 |
HDAC1 |
10uM |
24h |
LINCSCP_203706 |
LINCSCP_203706 |
ASC |
| 0.251019 |
1.780933e-15 |
975 |
SCHEMBL3958507 |
LSM-5245 |
COQ8B|EGFR |
1.11uM |
24h |
LINCSCP_116513 |
LINCSCP_116513 |
HT29 |
| -0.25099 |
1.794415e-15 |
975 |
Oxandrolone |
LSM-5544 |
AR |
10uM |
6h |
LINCSCP_243739 |
LINCSCP_243739 |
MCF7 |
| -0.25097 |
1.803826e-15 |
975 |
NMS-1286937 |
LSM-45818 |
|
3.33uM |
24h |
LINCSCP_141870 |
LINCSCP_141870 |
MCF7 |
| 0.250965 |
1.806385e-15 |
975 |
Trichostatin |
LSM-43005 |
HDAC1|HDAC10|HDAC3|HDAC4|HDAC6|HDAC7|HDAC8 |
0.01uM |
24h |
LINCSCP_35992 |
LINCSCP_35992 |
MCF7 |
| -0.250944 |
1.816329e-15 |
975 |
13-Methyl-7-[9-(4,4,5,5,5-pentafluoropentylsulfinyl)nonyl]-6,7,8,9,11,12,14,15,16,17-decahydrocyclopenta[a]phenanthrene-3,17-diol |
LSM-1895 |
ESR1 |
10uM |
6h |
LINCSCP_279389 |
LINCSCP_279389 |
PC3 |
| 0.25094 |
1.818329e-15 |
975 |
Dexniguldipine |
LSM-15285 |
|
0.37uM |
24h |
LINCSCP_105774 |
LINCSCP_105774 |
HELA |
| -0.250936 |
1.820479e-15 |
975 |
MLS001116189 |
LSM-6172 |
|
10uM |
24h |
LINCSCP_31868 |
LINCSCP_31868 |
MCF7 |
| 0.250903 |
1.836145e-15 |
975 |
Cobalt (Ii) Chloride |
LSM-5958 |
HIF1A |
10uM |
6h |
LINCSCP_228037 |
LINCSCP_228037 |
HT29 |
| -0.250878 |
1.848374e-15 |
975 |
BRD-K40397365 |
LSM-39496 |
|
1uM |
24h |
LINCSCP_312467 |
LINCSCP_312467 |
VCAP |
| 0.250823 |
1.875596e-15 |
975 |
CHEMBL2136735 |
LSM-1152 |
FGFR1|FGFR3|FLT1|FLT4|KDR|PDGFRA|PDGFRB |
1.11uM |
24h |
LINCSCP_131286 |
LINCSCP_131286 |
MCF10A |
| -0.25081 |
1.881910e-15 |
975 |
BRD-A08662020 |
LSM-45607 |
|
1.11uM |
24h |
LINCSCP_76500 |
LINCSCP_76500 |
A375 |
| -0.250789 |
1.892187e-15 |
975 |
Carbamazepine |
LSM-3610 |
SCN10A|SCN11A|SCN1A|SCN2A|SCN3A|SCN4A|SCN5A|SCN7A|SCN8A|SCN9A |
10uM |
24h |
LINCSCP_263892 |
LINCSCP_263892 |
NPC |
| 0.250781 |
1.896511e-15 |
975 |
Imatinib |
LSM-1023 |
ABL1|BCR|CSF1R|KIT|PDGFRA|PDGFRB |
0.04uM |
3h |
LINCSCP_116097 |
LINCSCP_116097 |
HS578T |
| 0.250767 |
1.903507e-15 |
975 |
Promazine |
LSM-2137 |
CHRM5|DRD2|DRD3|DRD4|HTR2A |
10uM |
24h |
LINCSCP_243934 |
LINCSCP_243934 |
MCF7 |
| -0.250746 |
1.914177e-15 |
975 |
GSK-1070916 |
LSM-1062 |
AURKB|AURKC |
1.11uM |
24h |
LINCSCP_147758 |
LINCSCP_147758 |
NPC.CAS9 |
| 0.250743 |
1.915460e-15 |
975 |
Torsemide |
LSM-2662 |
SLC12A1 |
10uM |
6h |
LINCSCP_4355 |
LINCSCP_4355 |
A549 |
| 0.250726 |
1.924408e-15 |
975 |
Lapatinib |
LSM-1051 |
EGFR|ERBB2 |
0.5uM |
24h |
LINCSCP_11667 |
LINCSCP_11667 |
BT20 |
| -0.250667 |
1.954296e-15 |
975 |
BRD-K34174785 |
LSM-39137 |
|
10uM |
6h |
LINCSCP_311844 |
LINCSCP_311844 |
VCAP |
| -0.250625 |
1.976273e-15 |
975 |
galantamine |
|
|
10uM |
24h |
LINCSCP_150323 |
LINCSCP_150323 |
NPC.TAK |
| 0.250606 |
1.986353e-15 |
975 |
TWS 119 |
LSM-1111 |
GSK3B |
0.04uM |
3h |
LINCSCP_145196 |
LINCSCP_145196 |
MDAMB231 |
| 0.250554 |
2.013406e-15 |
975 |
SCHEMBL3092652 |
LSM-6193 |
DPP4 |
10uM |
6h |
LINCSCP_51062 |
LINCSCP_51062 |
RMUGS |
| -0.2505 |
2.042606e-15 |
975 |
Dolastatin 10 |
LSM-45943 |
|
0.12uM |
24h |
LINCSCP_143055 |
LINCSCP_143055 |
MCF7 |
| 0.250459 |
2.064584e-15 |
975 |
Nilotinib |
LSM-1099 |
ABL1|BCR|KIT |
0.12uM |
3h |
LINCSCP_132496 |
LINCSCP_132496 |
MCF7 |
| 0.250419 |
2.086694e-15 |
975 |
Tadalafil |
LSM-4109 |
PDE11A|PDE5A |
10uM |
6h |
LINCSCP_240999 |
LINCSCP_240999 |
MCF7 |
| -0.250363 |
2.117436e-15 |
975 |
AMG-517 |
LSM-45865 |
TRPV1 |
10uM |
24h |
LINCSCP_121133 |
LINCSCP_121133 |
HT29 |
| -0.250317 |
2.143449e-15 |
975 |
TGX-115 |
LSM-6262 |
|
100uM |
6h |
LINCSCP_51186 |
LINCSCP_51186 |
RMUGS |
| 0.250313 |
2.145818e-15 |
975 |
BRD-K46555627 |
LSM-39850 |
|
10uM |
24h |
LINCSCP_193596 |
LINCSCP_193596 |
A549 |
| 0.250307 |
2.149177e-15 |
975 |
BRD-K10689551 |
LSM-9074 |
|
5uM |
6h |
LINCSCP_63923 |
LINCSCP_63923 |
VCAP |
| -0.250302 |
2.152258e-15 |
975 |
estriol |
LSM-2368 |
ESR1|ESR2 |
10uM |
24h |
LINCSCP_101705 |
LINCSCP_101705 |
HELA |
| -0.250298 |
2.154109e-15 |
975 |
GSK 1059615 |
LSM-42799 |
PIK3CA|PIK3CB|PIK3CD|PIK3CG |
3.33uM |
24h |
LINCSCP_116230 |
LINCSCP_116230 |
HT29 |
| -0.250291 |
2.158135e-15 |
975 |
Pimavanserin |
LSM-45960 |
HTR2A |
0.04uM |
24h |
LINCSCP_107968 |
LINCSCP_107968 |
HELA |
| 0.25027 |
2.170130e-15 |
975 |
CHEMBL2132289 |
LSM-1044 |
RPS6KA3 |
10uM |
24h |
LINCSCP_38965 |
LINCSCP_38965 |
MDAMB231 |
| -0.250217 |
2.200730e-15 |
975 |
BRD-K69406317-001-01-8 |
LSM-41049 |
|
10uM |
24h |
LINCSCP_31960 |
LINCSCP_31960 |
MCF7 |
| -0.250148 |
2.241010e-15 |
975 |
CHEMBL1394132 |
LSM-3090 |
|
10uM |
24h |
LINCSCP_25933 |
LINCSCP_25933 |
HT29 |
| -0.250108 |
2.265223e-15 |
975 |
Volasertib (BI 6727) |
LSM-45277 |
PLK1 |
0.04uM |
24h |
LINCSCP_142576 |
LINCSCP_142576 |
MCF7 |
| 0.249996 |
2.333036e-15 |
975 |
BRD-M04224464 |
LSM-45000 |
|
5uM |
6h |
LINCSCP_308584 |
LINCSCP_308584 |
VCAP |
| 0.249954 |
2.358840e-15 |
975 |
AC1MG5Y0 |
LSM-4794 |
|
10uM |
6h |
LINCSCP_16222 |
LINCSCP_16222 |
HA1E |
| -0.249943 |
2.365715e-15 |
975 |
BRD-K58191509 |
LSM-40452 |
|
10uM |
6h |
LINCSCP_34049 |
LINCSCP_34049 |
MCF7 |
| -0.249904 |
2.390205e-15 |
975 |
SB225002 |
LSM-3367 |
CXCR2 |
10uM |
24h |
LINCSCP_30591 |
LINCSCP_30591 |
MCF7 |
| 0.249859 |
2.418437e-15 |
975 |
SB-216763 |
LSM-1161 |
GSK3B |
1.11uM |
24h |
LINCSCP_165294 |
LINCSCP_165294 |
SKL |
| -0.249854 |
2.421885e-15 |
975 |
MW-STK33-97 |
LSM-44613 |
|
0.001uM |
24h |
LINCSCP_288133 |
LINCSCP_288133 |
THP1 |
| -0.249823 |
2.441752e-15 |
975 |
Phensuximide |
LSM-1359 |
CACNA1G|CACNA1H|CACNA1I |
10uM |
6h |
LINCSCP_4269 |
LINCSCP_4269 |
A549 |
| -0.249814 |
2.447529e-15 |
975 |
Bindarit |
LSM-45435 |
|
1.11uM |
24h |
LINCSCP_153752 |
LINCSCP_153752 |
PC3 |
| 0.249749 |
2.489307e-15 |
975 |
Mitoxantrone |
LSM-2481 |
TOP2A |
0.37uM |
3h |
LINCSCP_145690 |
LINCSCP_145690 |
MDAMB231 |
| 0.249729 |
2.502383e-15 |
975 |
BRD-K16512302 |
LSM-9428 |
|
5uM |
24h |
LINCSCP_63978 |
LINCSCP_63978 |
VCAP |
| -0.249728 |
2.503281e-15 |
975 |
IC 261 |
LSM-42870 |
|
10uM |
6h |
LINCSCP_37770 |
LINCSCP_37770 |
MCF7 |
| 0.249725 |
2.505009e-15 |
975 |
MGCD-265 |
LSM-1124 |
AXL|FLT1|FLT4|KDR|MET|MST1R|TEK |
1.11uM |
24h |
LINCSCP_134249 |
LINCSCP_134249 |
MCF7 |
| 0.249686 |
2.530988e-15 |
975 |
FPA1_000311 |
LSM-36744 |
|
10uM |
6h |
LINCSCP_20527 |
LINCSCP_20527 |
HCC515 |
| -0.249685 |
2.531994e-15 |
975 |
BRD-K42182933 |
LSM-10990 |
|
5uM |
24h |
LINCSCP_61994 |
LINCSCP_61994 |
VCAP |
| 0.249668 |
2.542748e-15 |
975 |
ZSTK 474 |
LSM-1053 |
PIK3CG |
10uM |
3h |
LINCSCP_145909 |
LINCSCP_145909 |
MDAMB231 |
| -0.249637 |
2.564199e-15 |
975 |
PX 12 |
LSM-4918 |
TXN|TXNRD1 |
30uM |
6h |
LINCSCP_883 |
LINCSCP_883 |
A375 |
| 0.24963 |
2.568301e-15 |
975 |
XAV 939 |
LSM-5303 |
TNKS|TNKS2 |
10uM |
6h |
LINCSCP_257326 |
LINCSCP_257326 |
NCIH508 |
| 0.249616 |
2.578204e-15 |
975 |
Dovitinib |
LSM-1127 |
EGFR|FGFR1|FGFR2|FGFR3|FLT1|FLT3|FLT4|KDR|KIT|PDGFRA|PDGFRB |
3.33uM |
3h |
LINCSCP_145030 |
LINCSCP_145030 |
MDAMB231 |
| -0.249603 |
2.587185e-15 |
975 |
Cilengitide |
LSM-45233 |
|
3.33uM |
24h |
LINCSCP_139225 |
LINCSCP_139225 |
MCF7 |
| 0.249584 |
2.599602e-15 |
975 |
BRD-K60857329 |
LSM-12112 |
|
5uM |
24h |
LINCSCP_61801 |
LINCSCP_61801 |
VCAP |
| -0.249562 |
2.614676e-15 |
975 |
Blebbistatin |
LSM-6195 |
MYH2 |
40uM |
6h |
LINCSCP_218458 |
LINCSCP_218458 |
HCT116 |
| -0.249548 |
2.624525e-15 |
975 |
SCHEMBL16980224 |
LSM-1092 |
AURKA |
1.11uM |
24h |
LINCSCP_150259 |
LINCSCP_150259 |
NPC.TAK |
| -0.249443 |
2.697944e-15 |
975 |
Selegiline |
LSM-5920 |
MAOA|MAOB |
10uM |
24h |
LINCSCP_47345 |
LINCSCP_47345 |
PC3 |
| 0.249377 |
2.745123e-15 |
975 |
Cyclacillin |
LSM-3987 |
|
10uM |
24h |
LINCSCP_42671 |
LINCSCP_42671 |
NPC |
| 0.249361 |
2.756679e-15 |
975 |
Erlotinib |
LSM-1097 |
EGFR |
0.12uM |
3h |
LINCSCP_132478 |
LINCSCP_132478 |
MCF7 |
| 0.249336 |
2.774883e-15 |
975 |
SCHEMBL6468298 |
LSM-6130 |
|
10uM |
6h |
LINCSCP_216723 |
LINCSCP_216723 |
HCC515 |
| 0.249322 |
2.785432e-15 |
975 |
Anandamide |
LSM-43816 |
CNR1|CNR2|TRPV1 |
0.37uM |
24h |
LINCSCP_122467 |
LINCSCP_122467 |
HT29 |
| 0.249318 |
2.788120e-15 |
975 |
84215-10-1 |
LSM-3529 |
CALM2 |
10uM |
24h |
LINCSCP_44054 |
LINCSCP_44054 |
PC3 |
| 0.249304 |
2.798532e-15 |
975 |
AZD-1152-HQPA |
LSM-1067 |
AURKA|AURKB |
1.11uM |
24h |
LINCSCP_150813 |
LINCSCP_150813 |
PC3 |
| -0.24929 |
2.808937e-15 |
975 |
7,2'-Dihydroxyflavone |
LSM-4674 |
|
10uM |
24h |
LINCSCP_52909 |
LINCSCP_52909 |
SKB |
| -0.249289 |
2.809487e-15 |
975 |
BRD-K84559549 |
LSM-41887 |
|
10uM |
6h |
LINCSCP_49184 |
LINCSCP_49184 |
PC3 |
| -0.249257 |
2.833314e-15 |
975 |
BRD-A41986761 |
LSM-45957 |
|
3.33uM |
24h |
LINCSCP_101825 |
LINCSCP_101825 |
HELA |
| -0.249237 |
2.848003e-15 |
975 |
MAZ51 |
LSM-43044 |
FLT4 |
10uM |
24h |
LINCSCP_30305 |
LINCSCP_30305 |
MCF7 |
| 0.24915 |
2.913766e-15 |
975 |
ST51005413 |
LSM-4948 |
|
10uM |
6h |
LINCSCP_310201 |
LINCSCP_310201 |
VCAP |
| 0.249149 |
2.914665e-15 |
975 |
BRD-K05395601 |
LSM-37560 |
|
5uM |
6h |
LINCSCP_59730 |
LINCSCP_59730 |
VCAP |
| 0.249145 |
2.917548e-15 |
975 |
CHEMBL2133926 |
LSM-6788 |
|
10uM |
6h |
LINCSCP_20713 |
LINCSCP_20713 |
HCC515 |
| 0.249136 |
2.924819e-15 |
975 |
BRD-K02117849 |
LSM-8563 |
|
5uM |
6h |
LINCSCP_61859 |
LINCSCP_61859 |
VCAP |
| 0.249001 |
3.030202e-15 |
975 |
Salsolidine |
LSM-5140 |
|
10uM |
24h |
LINCSCP_34456 |
LINCSCP_34456 |
MCF7 |
| -0.248994 |
3.035038e-15 |
975 |
Parbendazole |
LSM-4893 |
TUBB |
10uM |
24h |
LINCSCP_37424 |
LINCSCP_37424 |
MCF7 |
| -0.248939 |
3.079637e-15 |
975 |
17-DMAG (Alvespimycin) HCl |
LSM-46133 |
|
0.04uM |
24h |
LINCSCP_101865 |
LINCSCP_101865 |
HELA |
| 0.248935 |
3.082770e-15 |
975 |
Ipidacrine |
LSM-37163 |
ACHE |
10uM |
6h |
LINCSCP_46167 |
LINCSCP_46167 |
PC3 |
| -0.248911 |
3.102437e-15 |
975 |
QX-222 |
LSM-2905 |
|
10uM |
6h |
LINCSCP_4365 |
LINCSCP_4365 |
A549 |
| 0.248907 |
3.105120e-15 |
975 |
Lovastatin |
LSM-2189 |
HMGCR |
10uM |
6h |
LINCSCP_57866 |
LINCSCP_57866 |
VCAP |
| 0.248906 |
3.106387e-15 |
975 |
Emtricitabine |
LSM-45730 |
|
1.11uM |
24h |
LINCSCP_139868 |
LINCSCP_139868 |
MCF7 |
| -0.24889 |
3.119687e-15 |
975 |
Withaferin A |
LSM-6685 |
IKBKB|NAMPT |
10uM |
24h |
LINCSCP_151237 |
LINCSCP_151237 |
PC3 |
| 0.248855 |
3.148234e-15 |
975 |
MLS002276524 |
LSM-3088 |
|
10uM |
6h |
LINCSCP_5123 |
LINCSCP_5123 |
A549 |
| 0.248854 |
3.148707e-15 |
975 |
Imatinib |
LSM-1023 |
ABL1|BCR|CSF1R|KIT|PDGFRA|PDGFRB |
10uM |
3h |
LINCSCP_131784 |
LINCSCP_131784 |
MCF10A |
| 0.248842 |
3.159129e-15 |
975 |
BRD-K58719691 |
LSM-11976 |
|
5uM |
24h |
LINCSCP_61479 |
LINCSCP_61479 |
VCAP |
| 0.248837 |
3.162724e-15 |
975 |
BRD-M11500571 |
LSM-45004 |
|
5uM |
24h |
LINCSCP_63912 |
LINCSCP_63912 |
VCAP |
| -0.248821 |
3.176027e-15 |
975 |
MLS002703104 |
LSM-1920 |
|
10uM |
6h |
LINCSCP_15837 |
LINCSCP_15837 |
HA1E |
| -0.24881 |
3.185051e-15 |
975 |
MLS000583956 |
LSM-1515 |
|
10uM |
24h |
LINCSCP_30903 |
LINCSCP_30903 |
MCF7 |
| -0.248803 |
3.190938e-15 |
975 |
Ivacaftor (VX-770) |
LSM-45975 |
CFTR |
1.11uM |
24h |
LINCSCP_76476 |
LINCSCP_76476 |
A375 |
| 0.248774 |
3.215691e-15 |
975 |
JZL-184 |
LSM-6246 |
|
10uM |
6h |
LINCSCP_285891 |
LINCSCP_285891 |
SKM1 |
| 0.24874 |
3.244625e-15 |
975 |
Adapalene |
LSM-37048 |
RARA|RARB|RARG |
1.11uM |
24h |
LINCSCP_74150 |
LINCSCP_74150 |
A375 |
| -0.24874 |
3.244656e-15 |
975 |
IN1128 |
LSM-2557 |
PTGS1|PTGS2|SIRT1 |
10uM |
24h |
LINCSCP_44019 |
LINCSCP_44019 |
PC3 |
| 0.248656 |
3.316713e-15 |
975 |
BRD-K21037590 |
LSM-9709 |
|
5uM |
24h |
LINCSCP_61422 |
LINCSCP_61422 |
VCAP |
| 0.248625 |
3.343213e-15 |
975 |
BRD-K81646882 |
LSM-41730 |
|
5uM |
24h |
LINCSCP_64329 |
LINCSCP_64329 |
VCAP |
| -0.248522 |
3.434902e-15 |
975 |
BRD-K48222931 |
LSM-7469 |
|
10uM |
24h |
LINCSCP_3581 |
LINCSCP_3581 |
A375 |
| -0.248433 |
3.515329e-15 |
975 |
BRD-K88008216 |
LSM-42071 |
|
10uM |
6h |
LINCSCP_20675 |
LINCSCP_20675 |
HCC515 |
| -0.248397 |
3.548684e-15 |
975 |
MLS002232305 |
LSM-4515 |
|
10uM |
24h |
LINCSCP_32119 |
LINCSCP_32119 |
MCF7 |
| -0.248396 |
3.550203e-15 |
975 |
CCG-208038 |
LSM-36933 |
|
10uM |
24h |
LINCSCP_43389 |
LINCSCP_43389 |
NPC |
| -0.248389 |
3.556060e-15 |
975 |
ML239 |
LSM-3882 |
|
10uM |
24h |
LINCSCP_1429 |
LINCSCP_1429 |
A375 |
| -0.248271 |
3.667397e-15 |
975 |
MW-STK33-97 |
LSM-44613 |
|
0.001uM |
24h |
LINCSCP_41963 |
LINCSCP_41963 |
NOMO1 |
| 0.248234 |
3.703620e-15 |
975 |
BRD-K83509924 |
LSM-41833 |
|
10uM |
6h |
LINCSCP_59398 |
LINCSCP_59398 |
VCAP |
| 0.248186 |
3.749943e-15 |
975 |
AZD-1152-HQPA |
LSM-1067 |
AURKA|AURKB |
10uM |
6h |
LINCSCP_16679 |
LINCSCP_16679 |
HA1E |
| -0.24801 |
3.926068e-15 |
975 |
AC1MDRA3 |
LSM-4493 |
|
10uM |
24h |
LINCSCP_6336 |
LINCSCP_6336 |
A549 |
| 0.248003 |
3.933742e-15 |
975 |
522-11-2 |
LSM-3052 |
|
10uM |
6h |
LINCSCP_14268 |
LINCSCP_14268 |
HA1E |
| -0.247979 |
3.958832e-15 |
975 |
Quizartinib |
LSM-1037 |
CSF1R|FLT3|KIT|PDGFRA|PDGFRB|RET |
10uM |
24h |
LINCSCP_32570 |
LINCSCP_32570 |
MCF7 |
| 0.247975 |
3.962747e-15 |
975 |
Hydroxyprogesterone Caproate |
LSM-4900 |
AR|ESR1|ESR2|NR1H4|NR1I2|NR3C1|PGR |
3.33uM |
24h |
LINCSCP_71308 |
LINCSCP_71308 |
A375 |
| 0.247936 |
4.003609e-15 |
975 |
BRD-K41042536 |
LSM-39539 |
|
0.5uM |
24h |
LINCSCP_312469 |
LINCSCP_312469 |
VCAP |
| -0.247901 |
4.039682e-15 |
975 |
BAY 61-3606 |
LSM-1167 |
SYK |
10uM |
24h |
LINCSCP_114529 |
LINCSCP_114529 |
HME1 |
| 0.247829 |
4.116227e-15 |
975 |
BRD-K04986062 |
LSM-45341 |
|
1uM |
24h |
LINCSCP_288793 |
LINCSCP_288793 |
U937 |
| 0.247814 |
4.132816e-15 |
975 |
Imiloxan |
LSM-1308 |
ADRA2A|ADRA2B |
0.12uM |
24h |
LINCSCP_72708 |
LINCSCP_72708 |
A375 |
| 0.247772 |
4.178502e-15 |
975 |
SCHEMBL17052537 |
LSM-5803 |
BTK|JAK3|MKNK2|MTOR|PRKDC |
0.04uM |
24h |
LINCSCP_151224 |
LINCSCP_151224 |
PC3 |
| 0.247739 |
4.214254e-15 |
975 |
Actarit |
LSM-5475 |
|
3.33uM |
24h |
LINCSCP_137653 |
LINCSCP_137653 |
MCF7 |
| 0.24768 |
4.280076e-15 |
975 |
ABT-888,VELIPARIB |
LSM-5067 |
PARP1|PARP2 |
0.1uM |
6h |
LINCSCP_24858 |
LINCSCP_24858 |
HS578T |
| 0.247657 |
4.305533e-15 |
975 |
BRD-K37088230 |
LSM-10671 |
|
10uM |
24h |
LINCSCP_8910 |
LINCSCP_8910 |
A549 |
| 0.247643 |
4.321255e-15 |
975 |
Lapatinib |
LSM-1051 |
EGFR|ERBB2 |
0.12uM |
24h |
LINCSCP_113245 |
LINCSCP_113245 |
HME1 |
| 0.247587 |
4.383976e-15 |
975 |
SAN1_004207 |
LSM-36734 |
|
10uM |
6h |
LINCSCP_59399 |
LINCSCP_59399 |
VCAP |
| 0.247554 |
4.422091e-15 |
975 |
Phensuximide |
LSM-1359 |
CACNA1G|CACNA1H|CACNA1I |
0.12uM |
24h |
LINCSCP_71651 |
LINCSCP_71651 |
A375 |
| -0.247512 |
4.471399e-15 |
975 |
Cinaciguat |
LSM-45801 |
|
0.04uM |
24h |
LINCSCP_126909 |
LINCSCP_126909 |
HT29 |
| 0.247406 |
4.596731e-15 |
975 |
Imatinib |
LSM-1023 |
ABL1|BCR|CSF1R|KIT|PDGFRA|PDGFRB |
3.33uM |
3h |
LINCSCP_116093 |
LINCSCP_116093 |
HS578T |
| 0.247397 |
4.606683e-15 |
975 |
CHEMBL2359916 |
LSM-8908 |
|
5uM |
6h |
LINCSCP_62496 |
LINCSCP_62496 |
VCAP |
| 0.247312 |
4.709547e-15 |
975 |
Linoleoylethanolamide |
LSM-43037 |
CNR1|CNR2|TRPV1 |
10uM |
24h |
LINCSCP_33128 |
LINCSCP_33128 |
MCF7 |
| 0.247289 |
4.738672e-15 |
975 |
CHEMBL3186032 |
LSM-40660 |
|
10uM |
6h |
LINCSCP_20640 |
LINCSCP_20640 |
HCC515 |
| 0.247239 |
4.800386e-15 |
975 |
FPA1_000301 |
LSM-36736 |
|
10uM |
6h |
LINCSCP_22431 |
LINCSCP_22431 |
HEPG2 |
| -0.247121 |
4.949563e-15 |
975 |
UNII-EE9FJW53Z2 |
LSM-3437 |
|
10uM |
24h |
LINCSCP_52770 |
LINCSCP_52770 |
SKB |
| 0.247093 |
4.986209e-15 |
975 |
Emtricitabine |
LSM-45730 |
|
0.12uM |
24h |
LINCSCP_123287 |
LINCSCP_123287 |
HT29 |
| -0.24706 |
5.029405e-15 |
975 |
BRD-K40358966 |
LSM-10889 |
|
5uM |
6h |
LINCSCP_63795 |
LINCSCP_63795 |
VCAP |
| 0.247026 |
5.073041e-15 |
975 |
PF-04217903 |
LSM-1166 |
MET |
0.37uM |
24h |
LINCSCP_125701 |
LINCSCP_125701 |
HT29 |
| 0.247016 |
5.087304e-15 |
975 |
SR-142948 |
LSM-4038 |
|
10uM |
6h |
LINCSCP_220823 |
LINCSCP_220823 |
HEPG2 |
| -0.246955 |
5.168557e-15 |
975 |
BRD-A95504714 |
LSM-45336 |
|
0.5uM |
24h |
LINCSCP_24124 |
LINCSCP_24124 |
HL60 |
| -0.246808 |
5.368939e-15 |
975 |
Tizanidine |
LSM-5242 |
ADRA2A|ADRA2B|ADRA2C |
10uM |
24h |
LINCSCP_47291 |
LINCSCP_47291 |
PC3 |
| -0.246748 |
5.453345e-15 |
975 |
PCA-4248 |
LSM-1433 |
PTAFR |
0.12uM |
24h |
LINCSCP_71239 |
LINCSCP_71239 |
A375 |
| 0.246745 |
5.457117e-15 |
975 |
CHEMBL2426181 |
LSM-3160 |
|
10uM |
24h |
LINCSCP_31384 |
LINCSCP_31384 |
MCF7 |
| 0.246714 |
5.502237e-15 |
975 |
AB00540134 |
LSM-4868 |
|
10uM |
6h |
LINCSCP_16264 |
LINCSCP_16264 |
HA1E |
| 0.246676 |
5.556344e-15 |
975 |
OSI-930 |
LSM-1179 |
FLT1|FLT4|KDR|KIT |
0.12uM |
24h |
LINCSCP_113765 |
LINCSCP_113765 |
HME1 |
| 0.246654 |
5.587980e-15 |
975 |
BRD-K83816656 |
LSM-41851 |
|
10uM |
6h |
LINCSCP_295918 |
LINCSCP_295918 |
VCAP |
| -0.246629 |
5.624384e-15 |
975 |
CHEMBL1712678 |
LSM-2319 |
|
10uM |
24h |
LINCSCP_1378 |
LINCSCP_1378 |
A375 |
| -0.246613 |
5.647352e-15 |
975 |
BRD-K37184875 |
LSM-39311 |
|
5uM |
24h |
LINCSCP_35021 |
LINCSCP_35021 |
MCF7 |
| 0.24659 |
5.682170e-15 |
975 |
Citalopram |
LSM-1585 |
SLC6A4 |
10uM |
6h |
LINCSCP_189079 |
LINCSCP_189079 |
A549 |
| -0.246574 |
5.704821e-15 |
975 |
PD-0325901 |
LSM-1101 |
MAP2K1|MAP2K2 |
10uM |
24h |
LINCSCP_165910 |
LINCSCP_165910 |
SKL |
| -0.246551 |
5.739104e-15 |
975 |
2-(4-chlorophenyl)-3-(2-methoxyphenyl)hexahydro-1H-pyrrolo[1,2-c]imidazol-1-one |
LSM-45309 |
|
1uM |
24h |
LINCSCP_222086 |
LINCSCP_222086 |
HL60 |
| -0.246508 |
5.804472e-15 |
975 |
Alisertib |
LSM-37184 |
AURKA |
10uM |
24h |
LINCSCP_126310 |
LINCSCP_126310 |
HT29 |
| 0.246506 |
5.806844e-15 |
975 |
BRD-K98634983 |
LSM-45119 |
|
10uM |
24h |
LINCSCP_10960 |
LINCSCP_10960 |
ASC |
| -0.246448 |
5.894368e-15 |
975 |
Tacedinaline |
LSM-19036 |
HDAC1|HDAC10|HDAC11|HDAC2|HDAC3|HDAC4|HDAC5|HDAC6|HDAC7|HDAC8|HDAC9 |
0.5uM |
24h |
LINCSCP_49313 |
LINCSCP_49313 |
PC3 |
| 0.246403 |
5.964508e-15 |
975 |
CHEMBL2381520 |
LSM-36786 |
|
0.1uM |
24h |
LINCSCP_250109 |
LINCSCP_250109 |
MCF7 |
| -0.246317 |
6.099169e-15 |
975 |
CGS-15943 |
LSM-3076 |
ADORA1|ADORA2A|ADORA2B |
10uM |
24h |
LINCSCP_44728 |
LINCSCP_44728 |
PC3 |
| -0.246294 |
6.134462e-15 |
975 |
BRD-K28184645 |
LSM-38807 |
|
10uM |
24h |
LINCSCP_311993 |
LINCSCP_311993 |
VCAP |
| -0.246218 |
6.256376e-15 |
975 |
BRD-A80960055-001-01-7 |
LSM-5162 |
|
10uM |
6h |
LINCSCP_6561 |
LINCSCP_6561 |
A549 |
| 0.246187 |
6.306621e-15 |
975 |
ZINC77024257 |
LSM-1171 |
MDM2 |
1.11uM |
24h |
LINCSCP_129343 |
LINCSCP_129343 |
HUVEC |
| 0.246151 |
6.366625e-15 |
975 |
BRD-K32864614 |
LSM-10423 |
|
5uM |
24h |
LINCSCP_61589 |
LINCSCP_61589 |
VCAP |
| -0.246056 |
6.524188e-15 |
975 |
BRD-K04476933 |
LSM-37520 |
|
10uM |
6h |
LINCSCP_49076 |
LINCSCP_49076 |
PC3 |
| 0.246033 |
6.564235e-15 |
975 |
STK383264 |
LSM-44978 |
|
10uM |
6h |
LINCSCP_57855 |
LINCSCP_57855 |
VCAP |
| 0.246015 |
6.594147e-15 |
975 |
Phenelzine |
LSM-5928 |
AOC3|MAOA|MAOB |
10uM |
6h |
LINCSCP_1942 |
LINCSCP_1942 |
A375 |
| -0.245982 |
6.651488e-15 |
975 |
KCl |
LSM-46006 |
|
0.1uM |
24h |
LINCSCP_263922 |
LINCSCP_263922 |
NPC |
| -0.24596 |
6.689799e-15 |
975 |
SA-1938820 |
LSM-38649 |
|
3uM |
6h |
LINCSCP_37099 |
LINCSCP_37099 |
MCF7 |
| 0.245857 |
6.869249e-15 |
975 |
Gefitinib |
LSM-1098 |
EGFR |
1.11uM |
3h |
LINCSCP_145929 |
LINCSCP_145929 |
MDAMB231 |
| -0.245855 |
6.872787e-15 |
975 |
CHEMBL1271011 |
LSM-3631 |
|
10uM |
6h |
LINCSCP_5546 |
LINCSCP_5546 |
A549 |
| -0.245851 |
6.879693e-15 |
975 |
SU 11274 |
LSM-42792 |
MET |
10uM |
3h |
LINCSCP_115290 |
LINCSCP_115290 |
HS578T |
| -0.245826 |
6.924857e-15 |
975 |
BRD-K30150248 |
LSM-38916 |
|
1uM |
24h |
LINCSCP_66100 |
LINCSCP_66100 |
VCAP |
| -0.245819 |
6.936995e-15 |
975 |
Ganetespib (STA-9090) |
LSM-45281 |
HSP90AA1|HSP90AB1 |
3.33uM |
24h |
LINCSCP_120175 |
LINCSCP_120175 |
HT29 |
| -0.245798 |
6.975743e-15 |
975 |
BMS-299897 |
LSM-6207 |
|
10uM |
6h |
LINCSCP_289014 |
LINCSCP_289014 |
U937 |
| -0.245767 |
7.031532e-15 |
975 |
Dalcetrapib |
LSM-6227 |
CETP |
80uM |
6h |
LINCSCP_54187 |
LINCSCP_54187 |
SW620 |
| 0.245716 |
7.125198e-15 |
975 |
Resveratrol |
LSM-42917 |
PTGS1|PTGS2|SIRT1 |
10uM |
24h |
LINCSCP_236585 |
LINCSCP_236585 |
MCF7 |
| 0.24569 |
7.172133e-15 |
975 |
Famciclovir |
LSM-2990 |
|
10uM |
6h |
LINCSCP_239232 |
LINCSCP_239232 |
MCF7 |
| 0.245681 |
7.189430e-15 |
975 |
Benoxinate |
LSM-2069 |
SCN10A|SCN11A|SCN1A|SCN2A|SCN3A|SCN4A|SCN5A|SCN7A|SCN8A|SCN9A |
10uM |
24h |
LINCSCP_243406 |
LINCSCP_243406 |
MCF7 |
| -0.245612 |
7.317911e-15 |
975 |
AMG-517 |
LSM-45865 |
TRPV1 |
0.12uM |
24h |
LINCSCP_121137 |
LINCSCP_121137 |
HT29 |
| -0.245574 |
7.390566e-15 |
975 |
Simvastatin |
LSM-2492 |
HMGCR |
0.04uM |
24h |
LINCSCP_72344 |
LINCSCP_72344 |
A375 |
| 0.24553 |
7.475567e-15 |
975 |
BRD-K76662562 |
LSM-13119 |
|
5uM |
24h |
LINCSCP_62318 |
LINCSCP_62318 |
VCAP |
| 0.245527 |
7.480891e-15 |
975 |
Mitoxantrone |
LSM-2481 |
TOP2A |
0.37uM |
3h |
LINCSCP_115849 |
LINCSCP_115849 |
HS578T |
| 0.245525 |
7.485479e-15 |
975 |
AC1O9CBL |
LSM-4596 |
|
1uM |
24h |
LINCSCP_253914 |
LINCSCP_253914 |
MCF7 |
| 0.245524 |
7.485918e-15 |
975 |
BRD-K92810472 |
LSM-14119 |
|
5uM |
24h |
LINCSCP_62064 |
LINCSCP_62064 |
VCAP |
| 0.245524 |
7.486622e-15 |
975 |
SB525334 |
LSM-1121 |
TGFBR1 |
10uM |
24h |
LINCSCP_129613 |
LINCSCP_129613 |
JURKAT |
| -0.245511 |
7.512771e-15 |
975 |
GNF-PF-2272 |
LSM-6669 |
|
10uM |
6h |
LINCSCP_22600 |
LINCSCP_22600 |
HEPG2 |
| -0.24551 |
7.513512e-15 |
975 |
SA-1925246 |
LSM-41762 |
|
3uM |
24h |
LINCSCP_252344 |
LINCSCP_252344 |
MCF7 |
| 0.245499 |
7.535966e-15 |
975 |
BRD-K28582709 |
LSM-10159 |
|
5uM |
24h |
LINCSCP_63360 |
LINCSCP_63360 |
VCAP |
| -0.245402 |
7.726529e-15 |
975 |
Mebendazole |
LSM-3749 |
|
3.33uM |
24h |
LINCSCP_139711 |
LINCSCP_139711 |
MCF7 |
| -0.245348 |
7.835566e-15 |
975 |
Withaferin A |
LSM-6685 |
IKBKB|NAMPT |
10uM |
6h |
LINCSCP_68638 |
LINCSCP_68638 |
VCAP |
| -0.245311 |
7.908848e-15 |
975 |
Pravastatin |
LSM-3347 |
HMGCR |
10uM |
24h |
LINCSCP_293922 |
LINCSCP_293922 |
VCAP |
| -0.245295 |
7.941901e-15 |
975 |
Isoxsuprine |
LSM-1778 |
ADRB2 |
10uM |
24h |
LINCSCP_284619 |
LINCSCP_284619 |
SKB |
| -0.245197 |
8.144902e-15 |
975 |
CHEMBL2136735 |
LSM-1152 |
FGFR1|FGFR3|FLT1|FLT4|KDR|PDGFRA|PDGFRB |
0.12uM |
24h |
LINCSCP_151253 |
LINCSCP_151253 |
PC3 |
| -0.245193 |
8.153254e-15 |
975 |
GSK 1059615 |
LSM-42799 |
PIK3CA|PIK3CB|PIK3CD|PIK3CG |
0.1uM |
24h |
LINCSCP_222609 |
LINCSCP_222609 |
HS578T |
| 0.24517 |
8.202721e-15 |
975 |
AZD-1152-HQPA |
LSM-1067 |
AURKA|AURKB |
3.33uM |
24h |
LINCSCP_130495 |
LINCSCP_130495 |
MCF10A |
| -0.245166 |
8.212057e-15 |
975 |
Tropisetron HCl |
LSM-46040 |
HTR3A |
10uM |
6h |
LINCSCP_46159 |
LINCSCP_46159 |
PC3 |
| -0.245154 |
8.236131e-15 |
975 |
PLX-4720 |
LSM-1049 |
BRAF |
0.12uM |
24h |
LINCSCP_144793 |
LINCSCP_144793 |
MDAMB231 |
| 0.245146 |
8.253767e-15 |
975 |
WH-4-023 |
LSM-5613 |
ABL1|SRC |
0.5uM |
24h |
LINCSCP_29537 |
LINCSCP_29537 |
MCF10A |
| -0.245134 |
8.278929e-15 |
975 |
CHEMBL2361787 |
LSM-13210 |
|
10uM |
24h |
LINCSCP_48463 |
LINCSCP_48463 |
PC3 |
| 0.245112 |
8.327056e-15 |
975 |
C21H27N7O3 |
LSM-1128 |
AKT1|AKT2|AKT3|PRKCQ |
3.33uM |
3h |
LINCSCP_130902 |
LINCSCP_130902 |
MCF10A |
| -0.245097 |
8.358414e-15 |
975 |
BRD-K77760488 |
LSM-41512 |
|
10uM |
6h |
LINCSCP_49180 |
LINCSCP_49180 |
PC3 |
| 0.24509 |
8.373703e-15 |
975 |
Resveratrol |
LSM-42917 |
PTGS1|PTGS2|SIRT1 |
10uM |
24h |
LINCSCP_72746 |
LINCSCP_72746 |
A375 |
| 0.245035 |
8.493476e-15 |
975 |
KUC104545N |
LSM-2814 |
|
10uM |
24h |
LINCSCP_31153 |
LINCSCP_31153 |
MCF7 |
| 0.245001 |
8.568069e-15 |
975 |
Benzohydroxamate |
LSM-36789 |
|
0.1uM |
24h |
LINCSCP_279589 |
LINCSCP_279589 |
PC3 |
| -0.244997 |
8.575671e-15 |
975 |
Vindesine |
LSM-5693 |
|
10uM |
24h |
LINCSCP_46104 |
LINCSCP_46104 |
PC3 |
| -0.244994 |
8.583813e-15 |
975 |
ZINC03978011 |
LSM-5441 |
NR3C1 |
10uM |
6h |
LINCSCP_243716 |
LINCSCP_243716 |
MCF7 |
| -0.244958 |
8.662534e-15 |
975 |
JX401 |
LSM-2097 |
MAPK14 |
10uM |
6h |
LINCSCP_44113 |
LINCSCP_44113 |
PC3 |
| -0.244834 |
8.944059e-15 |
975 |
Withaferin A |
LSM-6685 |
IKBKB|NAMPT |
10uM |
3h |
LINCSCP_86292 |
LINCSCP_86292 |
BT20 |
| -0.244801 |
9.020843e-15 |
975 |
BRD-K64930281 |
LSM-7714 |
|
5uM |
24h |
LINCSCP_60064 |
LINCSCP_60064 |
VCAP |
| -0.24478 |
9.070343e-15 |
975 |
Exifone |
LSM-37157 |
TYR |
10uM |
24h |
LINCSCP_263883 |
LINCSCP_263883 |
NPC |
| 0.244774 |
9.082513e-15 |
975 |
AGK 2 |
LSM-43196 |
SIRT2 |
1.11uM |
24h |
LINCSCP_83426 |
LINCSCP_83426 |
ASC.C |
| -0.244769 |
9.095947e-15 |
975 |
Amylocaine |
LSM-1292 |
|
10uM |
24h |
LINCSCP_14960 |
LINCSCP_14960 |
HA1E |
| -0.244726 |
9.195933e-15 |
975 |
Flutamide |
LSM-2621 |
AR |
10uM |
24h |
LINCSCP_272491 |
LINCSCP_272491 |
PC3 |
| -0.244713 |
9.226261e-15 |
975 |
Amuvatinib |
LSM-1118 |
FLT3|KIT|MET|PDGFRA |
0.5uM |
6h |
LINCSCP_39618 |
LINCSCP_39618 |
MDAMB231 |
| -0.244713 |
9.227586e-15 |
975 |
Buparlisib |
LSM-1148 |
PIK3CA|PIK3CB|PIK3CD|PIK3CG|PIK3R1|PIK3R2|PIK3R3|PIK3R5 |
3.33uM |
24h |
LINCSCP_69112 |
LINCSCP_69112 |
A375 |
| 0.24466 |
9.352675e-15 |
975 |
BRD-K61779668 |
LSM-40651 |
|
10uM |
6h |
LINCSCP_64788 |
LINCSCP_64788 |
VCAP |
| 0.244656 |
9.362843e-15 |
975 |
CHEMBL2355513 |
LSM-39806 |
|
0.5uM |
24h |
LINCSCP_252239 |
LINCSCP_252239 |
MCF7 |
| -0.244635 |
9.414318e-15 |
975 |
BRD-K63157607 |
LSM-15152 |
|
10uM |
24h |
LINCSCP_48807 |
LINCSCP_48807 |
PC3 |
| -0.244625 |
9.438413e-15 |
975 |
Dolastatin 10 |
LSM-45943 |
|
10uM |
24h |
LINCSCP_143051 |
LINCSCP_143051 |
MCF7 |
| -0.244576 |
9.556969e-15 |
975 |
BRD-K42125900-001-01-9 |
LSM-5535 |
TUBB |
10uM |
24h |
LINCSCP_6169 |
LINCSCP_6169 |
A549 |
| -0.244572 |
9.568694e-15 |
975 |
BRD-A28746609 |
LSM-1102 |
NR1I2|TUBB |
0.37uM |
24h |
LINCSCP_137547 |
LINCSCP_137547 |
MCF7 |
| 0.244524 |
9.687035e-15 |
975 |
BRD-K37168393 |
LSM-7324 |
|
5uM |
24h |
LINCSCP_60176 |
LINCSCP_60176 |
VCAP |
| 0.24452 |
9.696765e-15 |
975 |
amcinonide |
|
|
0.04uM |
24h |
LINCSCP_87245 |
LINCSCP_87245 |
CD34 |
| -0.244504 |
9.737437e-15 |
975 |
GSK 1059615 |
LSM-42799 |
PIK3CA|PIK3CB|PIK3CD|PIK3CG |
0.1uM |
24h |
LINCSCP_39344 |
LINCSCP_39344 |
MDAMB231 |
| 0.244492 |
9.767119e-15 |
975 |
Cilomilast |
LSM-5719 |
PDE4A|PDE4B|PDE4D |
10uM |
6h |
LINCSCP_22390 |
LINCSCP_22390 |
HEPG2 |
| -0.244474 |
9.810775e-15 |
975 |
galantamine |
|
|
10uM |
24h |
LINCSCP_149199 |
LINCSCP_149199 |
NPC |
| -0.244443 |
9.890038e-15 |
975 |
SC-514 |
LSM-2579 |
IKBKB |
10uM |
6h |
LINCSCP_56334 |
LINCSCP_56334 |
VCAP |
| -0.244398 |
1.000387e-14 |
975 |
Withaferin A |
LSM-6685 |
IKBKB|NAMPT |
1uM |
24h |
LINCSCP_67405 |
LINCSCP_67405 |
MCF7 |
| -0.244333 |
1.017317e-14 |
975 |
Withaferin A |
LSM-6685 |
IKBKB|NAMPT |
10uM |
24h |
LINCSCP_81148 |
LINCSCP_81148 |
A549 |
| 0.24431 |
1.023481e-14 |
975 |
SA-1458026 |
LSM-40479 |
|
3uM |
6h |
LINCSCP_253343 |
LINCSCP_253343 |
MCF7 |
| 0.2443 |
1.025995e-14 |
975 |
Orphenadrine |
LSM-1630 |
GRIN1|GRIN2A|GRIN2B|GRIN2C|GRIN2D|GRIN3A|GRIN3B|HRH1|SCN10A|SCN11A|SCN1A|SCN2A|SCN3A|SCN4A|SCN5A|SCN7A|SCN8A|SCN9A|SLC6A2 |
10uM |
24h |
LINCSCP_284851 |
LINCSCP_284851 |
SKB |
| -0.244256 |
1.037687e-14 |
975 |
Bardoxolone Methyl |
LSM-45471 |
IKBKB|KEAP1|NFE2L2|PPARG |
0.04uM |
24h |
LINCSCP_153953 |
LINCSCP_153953 |
PC3 |
| 0.244208 |
1.050450e-14 |
975 |
NCGC00346967-01 |
LSM-6297 |
EPHB3 |
0.04uM |
24h |
LINCSCP_87215 |
LINCSCP_87215 |
CD34 |
| 0.244192 |
1.054751e-14 |
975 |
SPECTRUM_000051 |
LSM-1749 |
OPRD1|OPRK1|OPRM1 |
10uM |
6h |
LINCSCP_56114 |
LINCSCP_56114 |
VCAP |
| 0.244183 |
1.057233e-14 |
975 |
C24H25CLFN5O3 |
LSM-42794 |
EGFR|ERBB2|ERBB4 |
0.5uM |
24h |
LINCSCP_12093 |
LINCSCP_12093 |
BT20 |
| 0.24414 |
1.069022e-14 |
975 |
Hyoscine N-Oxide |
LSM-1606 |
CHRM1|CHRM2|CHRM3|CHRM4 |
10uM |
24h |
LINCSCP_241519 |
LINCSCP_241519 |
MCF7 |
| -0.244135 |
1.070341e-14 |
975 |
Tyrphostin B7 |
LSM-42938 |
PDGFRB |
10uM |
6h |
LINCSCP_14241 |
LINCSCP_14241 |
HA1E |
| -0.244036 |
1.097951e-14 |
975 |
MLS002264477 |
LSM-4186 |
|
10uM |
24h |
LINCSCP_1448 |
LINCSCP_1448 |
A375 |
| -0.244014 |
1.104070e-14 |
975 |
BMS-536924 |
LSM-1210 |
IGF1R |
10uM |
6h |
LINCSCP_40205 |
LINCSCP_40205 |
NCIH508 |
| -0.243992 |
1.110240e-14 |
975 |
BRD-K42466986 |
LSM-7389 |
|
5uM |
24h |
LINCSCP_60554 |
LINCSCP_60554 |
VCAP |
| -0.243984 |
1.112582e-14 |
975 |
BRD-A00474148 |
LSM-45242 |
|
1.11uM |
24h |
LINCSCP_135958 |
LINCSCP_135958 |
MCF7 |
| -0.243931 |
1.127746e-14 |
975 |
BRD-K69406317-001-01-8 |
LSM-41049 |
|
10uM |
24h |
LINCSCP_283572 |
LINCSCP_283572 |
SKB |
| 0.243918 |
1.131511e-14 |
975 |
XMD-132 |
LSM-42742 |
|
10uM |
6h |
LINCSCP_6733 |
LINCSCP_6733 |
A549 |
| 0.243875 |
1.144226e-14 |
975 |
STK222600 |
LSM-3535 |
|
10uM |
6h |
LINCSCP_20136 |
LINCSCP_20136 |
HCC515 |
| 0.243849 |
1.151922e-14 |
975 |
BRD-K75416754 |
LSM-13045 |
|
5uM |
24h |
LINCSCP_48250 |
LINCSCP_48250 |
PC3 |
| -0.243818 |
1.161076e-14 |
975 |
MK-5108 |
LSM-36812 |
AURKA|AURKB |
10uM |
24h |
LINCSCP_136872 |
LINCSCP_136872 |
MCF7 |
| -0.243761 |
1.177952e-14 |
975 |
MLS002607703 |
LSM-3242 |
|
10uM |
24h |
LINCSCP_31390 |
LINCSCP_31390 |
MCF7 |
| 0.243743 |
1.183467e-14 |
975 |
BRD-K84239628 |
LSM-13579 |
|
5uM |
6h |
LINCSCP_62588 |
LINCSCP_62588 |
VCAP |
| 0.243706 |
1.194724e-14 |
975 |
CHEMBL2136735 |
LSM-1152 |
FGFR1|FGFR3|FLT1|FLT4|KDR|PDGFRA|PDGFRB |
3.33uM |
24h |
LINCSCP_77669 |
LINCSCP_77669 |
A375 |
| 0.243691 |
1.199545e-14 |
975 |
BRD-K52309792 |
LSM-11627 |
|
5uM |
24h |
LINCSCP_62294 |
LINCSCP_62294 |
VCAP |
| -0.24369 |
1.199740e-14 |
975 |
KX2-391 |
LSM-45890 |
SRC |
10uM |
24h |
LINCSCP_137496 |
LINCSCP_137496 |
MCF7 |
| -0.243672 |
1.205140e-14 |
975 |
SPECTRUM_001095 |
LSM-1280 |
NR3C1 |
10uM |
6h |
LINCSCP_398 |
LINCSCP_398 |
A375 |
| 0.243585 |
1.232292e-14 |
975 |
BRD-K62473229 |
LSM-12224 |
|
10uM |
24h |
LINCSCP_9061 |
LINCSCP_9061 |
A549 |
| -0.243579 |
1.234348e-14 |
975 |
BI-2536 |
LSM-1041 |
PLK1 |
0.12uM |
24h |
LINCSCP_140811 |
LINCSCP_140811 |
MCF7 |
| 0.243567 |
1.237986e-14 |
975 |
TGX 221 |
LSM-1172 |
PIK3CB |
3.33uM |
24h |
LINCSCP_116314 |
LINCSCP_116314 |
HT29 |
| 0.243551 |
1.243105e-14 |
975 |
Idelalisib |
LSM-1205 |
PIK3CD|PIK3CG |
10uM |
24h |
LINCSCP_86838 |
LINCSCP_86838 |
CD34 |
| -0.243531 |
1.249516e-14 |
975 |
BSPBIO_000981 |
LSM-43126 |
ACTA1 |
10uM |
24h |
LINCSCP_6160 |
LINCSCP_6160 |
A549 |
| 0.243428 |
1.283051e-14 |
975 |
SCHEMBL570779 |
LSM-1149 |
|
0.12uM |
24h |
LINCSCP_144709 |
LINCSCP_144709 |
MDAMB231 |
| 0.243371 |
1.301786e-14 |
975 |
GSK-J1 |
LSM-44939 |
|
0.37uM |
24h |
LINCSCP_164638 |
LINCSCP_164638 |
SKL.C |
| 0.243366 |
1.303557e-14 |
975 |
BRD-K09186736-001-01-2 |
LSM-37761 |
|
10uM |
6h |
LINCSCP_47392 |
LINCSCP_47392 |
PC3 |
| -0.243309 |
1.322430e-14 |
975 |
BRD-K94498396 |
LSM-36822 |
|
10uM |
6h |
LINCSCP_38113 |
LINCSCP_38113 |
MCF7 |
| -0.24325 |
1.342682e-14 |
975 |
BRD-K98062050 |
LSM-42582 |
|
10uM |
24h |
LINCSCP_186667 |
LINCSCP_186667 |
A375 |
| 0.243249 |
1.342872e-14 |
975 |
MLS000703473 |
LSM-6571 |
|
10uM |
6h |
LINCSCP_59330 |
LINCSCP_59330 |
VCAP |
| -0.24319 |
1.363333e-14 |
975 |
GSK 1059615 |
LSM-42799 |
PIK3CA|PIK3CB|PIK3CD|PIK3CG |
3.33uM |
24h |
LINCSCP_150436 |
LINCSCP_150436 |
NPC.TAK |
| -0.24317 |
1.370526e-14 |
975 |
BRD-K45232279 |
LSM-39776 |
|
10uM |
24h |
LINCSCP_33861 |
LINCSCP_33861 |
MCF7 |
| 0.243164 |
1.372360e-14 |
975 |
Darinaparsin |
LSM-4924 |
|
10uM |
6h |
LINCSCP_286560 |
LINCSCP_286560 |
SNGM |
| -0.243148 |
1.378057e-14 |
975 |
PF-04217903 |
LSM-1166 |
MET |
0.001uM |
6h |
LINCSCP_201950 |
LINCSCP_201950 |
A549 |
| -0.243124 |
1.386687e-14 |
975 |
Wortmannin |
LSM-3947 |
PIK3CA|PIK3CG|PLK1 |
10uM |
24h |
LINCSCP_55297 |
LINCSCP_55297 |
U937 |
| 0.243117 |
1.388993e-14 |
975 |
ALD1-H_001009 |
LSM-45117 |
|
10uM |
6h |
LINCSCP_20172 |
LINCSCP_20172 |
HCC515 |
| -0.24308 |
1.402366e-14 |
975 |
D-64131 |
LSM-2592 |
TUBB |
10uM |
24h |
LINCSCP_37447 |
LINCSCP_37447 |
MCF7 |
| 0.243063 |
1.408413e-14 |
975 |
AC1O8PZP |
LSM-1327 |
|
10uM |
24h |
LINCSCP_32805 |
LINCSCP_32805 |
MCF7 |
| 0.243042 |
1.415736e-14 |
975 |
BRD-K08371414 |
LSM-8932 |
|
5uM |
6h |
LINCSCP_63775 |
LINCSCP_63775 |
VCAP |
| -0.243036 |
1.418045e-14 |
975 |
CHEMBL1965318 |
LSM-6612 |
|
10uM |
24h |
LINCSCP_295629 |
LINCSCP_295629 |
VCAP |
| 0.242986 |
1.436292e-14 |
975 |
Nebivolol |
LSM-45235 |
|
3.33uM |
24h |
LINCSCP_104796 |
LINCSCP_104796 |
HELA |
| -0.242819 |
1.498720e-14 |
975 |
vinorelbine |
|
TUBB |
10uM |
24h |
LINCSCP_284061 |
LINCSCP_284061 |
SKB |
| 0.242791 |
1.509670e-14 |
975 |
BRD-K03016409 |
LSM-8621 |
|
5uM |
24h |
LINCSCP_62752 |
LINCSCP_62752 |
VCAP |
| -0.242764 |
1.519778e-14 |
975 |
BRD-K95090559 |
LSM-42424 |
|
10uM |
6h |
LINCSCP_49197 |
LINCSCP_49197 |
PC3 |
| 0.242756 |
1.523180e-14 |
975 |
Loxoprofen |
LSM-5054 |
|
0.12uM |
24h |
LINCSCP_75576 |
LINCSCP_75576 |
A375 |
| -0.242741 |
1.528860e-14 |
975 |
BSPBIO_001530 |
LSM-1549 |
|
10uM |
24h |
LINCSCP_44675 |
LINCSCP_44675 |
PC3 |
| -0.2427 |
1.545096e-14 |
975 |
Mebendazole |
LSM-3749 |
|
5uM |
24h |
LINCSCP_67547 |
LINCSCP_67547 |
MCF7 |
| 0.242683 |
1.551758e-14 |
975 |
CHEMBL2143681 |
LSM-6163 |
|
10uM |
6h |
LINCSCP_16727 |
LINCSCP_16727 |
HA1E |
| -0.242653 |
1.563495e-14 |
975 |
TAK-285 |
LSM-45987 |
EGFR|ERBB2 |
3.33uM |
24h |
LINCSCP_141702 |
LINCSCP_141702 |
MCF7 |
| 0.242625 |
1.574605e-14 |
975 |
JNK-IN-2 |
LSM-43288 |
IRAK1 |
0.5uM |
6h |
LINCSCP_39612 |
LINCSCP_39612 |
MDAMB231 |
| 0.242621 |
1.576238e-14 |
975 |
Disulfiram |
LSM-5467 |
ALDH2 |
0.04uM |
24h |
LINCSCP_118747 |
LINCSCP_118747 |
HT29 |
| -0.242581 |
1.592394e-14 |
975 |
TORIN-2 |
LSM-1080 |
MTOR |
10uM |
24h |
LINCSCP_29584 |
LINCSCP_29584 |
MCF10A |
| 0.24258 |
1.593037e-14 |
975 |
AC1MSUFC |
LSM-6191 |
HMGCR |
40uM |
6h |
LINCSCP_12766 |
LINCSCP_12766 |
DV90 |
| -0.242579 |
1.593326e-14 |
975 |
ZINC06431970 |
LSM-43103 |
|
10uM |
6h |
LINCSCP_22408 |
LINCSCP_22408 |
HEPG2 |
| -0.242577 |
1.594184e-14 |
975 |
Butyrolactone 3 |
LSM-37169 |
|
10uM |
24h |
LINCSCP_43483 |
LINCSCP_43483 |
NPC |
| -0.24257 |
1.597046e-14 |
975 |
TAE-684 |
LSM-1024 |
ALK |
0.12uM |
24h |
LINCSCP_99940 |
LINCSCP_99940 |
HCC515 |
| -0.242524 |
1.615770e-14 |
975 |
Aminosalicylic acid |
LSM-5862 |
PTGS1|PTGS2 |
0.12uM |
24h |
LINCSCP_141717 |
LINCSCP_141717 |
MCF7 |
| -0.242459 |
1.642761e-14 |
975 |
331771-20-1 |
LSM-1096 |
AURKA|AURKB |
1.11uM |
24h |
LINCSCP_150479 |
LINCSCP_150479 |
NPC.TAK |
| 0.242405 |
1.665514e-14 |
975 |
BRD-K68201904 |
LSM-12586 |
|
5uM |
24h |
LINCSCP_62029 |
LINCSCP_62029 |
VCAP |
| -0.242395 |
1.669587e-14 |
975 |
Rotenone |
LSM-5260 |
MT-ND1 |
0.5uM |
24h |
LINCSCP_30481 |
LINCSCP_30481 |
MCF7 |
| -0.242381 |
1.675588e-14 |
975 |
AZD-5438 |
LSM-1159 |
CDK1|CDK10|CDK11B|CDK12|CDK13|CDK14|CDK15|CDK16|CDK17|CDK18|CDK19|CDK2|CDK20|CDK3|CDK4|CDK5|CDK6|CDK7|CDK8|CDK9 |
3.33uM |
24h |
LINCSCP_111740 |
LINCSCP_111740 |
HEPG2 |
| -0.242381 |
1.675876e-14 |
975 |
SB225002 |
LSM-3367 |
CXCR2 |
10uM |
6h |
LINCSCP_257404 |
LINCSCP_257404 |
NCIH508 |
| 0.242376 |
1.677966e-14 |
975 |
BRD-K89699317 |
LSM-13965 |
|
5uM |
24h |
LINCSCP_61840 |
LINCSCP_61840 |
VCAP |
| -0.242337 |
1.694531e-14 |
975 |
Dephostatin |
LSM-3344 |
PTPN1|PTPN6 |
10uM |
6h |
LINCSCP_235901 |
LINCSCP_235901 |
MCF7 |
| 0.24233 |
1.697450e-14 |
975 |
Lintitript |
LSM-2780 |
CCKAR |
10uM |
24h |
LINCSCP_71999 |
LINCSCP_71999 |
A375 |
| -0.242319 |
1.702320e-14 |
975 |
Mitoxantrone |
LSM-2481 |
TOP2A |
1uM |
24h |
LINCSCP_250780 |
LINCSCP_250780 |
MCF7 |
| 0.242296 |
1.712301e-14 |
975 |
CHEMBL2362357 |
LSM-13661 |
|
10uM |
24h |
LINCSCP_9085 |
LINCSCP_9085 |
A549 |
| -0.242289 |
1.715461e-14 |
975 |
BRD-K01121544 |
LSM-6873 |
|
5uM |
24h |
LINCSCP_60494 |
LINCSCP_60494 |
VCAP |
| -0.24225 |
1.732649e-14 |
975 |
Graveoline |
LSM-4078 |
|
10uM |
24h |
LINCSCP_262443 |
LINCSCP_262443 |
NPC |
| 0.242215 |
1.748258e-14 |
975 |
Bemegride |
LSM-2325 |
GABRA1 |
0.12uM |
24h |
LINCSCP_74510 |
LINCSCP_74510 |
A375 |
| -0.242212 |
1.749477e-14 |
975 |
MLS002264379 |
LSM-2753 |
|
10uM |
6h |
LINCSCP_31477 |
LINCSCP_31477 |
MCF7 |
| 0.242189 |
1.759876e-14 |
975 |
BRD-K75809222 |
LSM-13064 |
|
5uM |
6h |
LINCSCP_62226 |
LINCSCP_62226 |
VCAP |
| -0.242179 |
1.764302e-14 |
975 |
vincristine |
|
TUBB |
0.5uM |
24h |
LINCSCP_37612 |
LINCSCP_37612 |
MCF7 |
| 0.242162 |
1.771719e-14 |
975 |
Mesoridazine |
LSM-1329 |
DRD2|HTR2A |
10uM |
6h |
LINCSCP_4648 |
LINCSCP_4648 |
A549 |
| -0.242159 |
1.773163e-14 |
975 |
PF-03758309 |
LSM-4254 |
PAK4 |
1.11uM |
24h |
LINCSCP_149153 |
LINCSCP_149153 |
NPC |
| 0.242155 |
1.774747e-14 |
975 |
BRD-K82794234 |
LSM-13485 |
|
5uM |
6h |
LINCSCP_303409 |
LINCSCP_303409 |
VCAP |
| -0.242131 |
1.785946e-14 |
975 |
KX2-391 |
LSM-45890 |
SRC |
0.04uM |
24h |
LINCSCP_137501 |
LINCSCP_137501 |
MCF7 |
| -0.24212 |
1.790737e-14 |
975 |
GSK 1059615 |
LSM-42799 |
PIK3CA|PIK3CB|PIK3CD|PIK3CG |
10uM |
24h |
LINCSCP_150829 |
LINCSCP_150829 |
PC3 |
| -0.24209 |
1.804701e-14 |
975 |
BRD-K02589376-001-01-9 |
LSM-6780 |
|
10uM |
24h |
LINCSCP_33811 |
LINCSCP_33811 |
MCF7 |
| -0.242055 |
1.820629e-14 |
975 |
Y-27632 |
LSM-44936 |
ROCK1|ROCK2 |
10uM |
6h |
LINCSCP_501 |
LINCSCP_501 |
A375 |
| -0.242051 |
1.822509e-14 |
975 |
Tivantinib |
LSM-1131 |
MET |
10uM |
24h |
LINCSCP_135380 |
LINCSCP_135380 |
MCF7 |
| -0.242027 |
1.833474e-14 |
975 |
GSK 1059615 |
LSM-42799 |
PIK3CA|PIK3CB|PIK3CD|PIK3CG |
10uM |
24h |
LINCSCP_69045 |
LINCSCP_69045 |
A375 |
| -0.242015 |
1.839018e-14 |
975 |
AKT Inhibitor VIII |
LSM-1035 |
AKT1|AKT2 |
10uM |
6h |
LINCSCP_40042 |
LINCSCP_40042 |
NCIH2073 |
| 0.242 |
1.846444e-14 |
975 |
CHEMBL179288 |
LSM-3648 |
|
1.11uM |
24h |
LINCSCP_73417 |
LINCSCP_73417 |
A375 |
| 0.241909 |
1.889286e-14 |
975 |
Tyrphostin 1 |
LSM-2933 |
|
10uM |
24h |
LINCSCP_209946 |
LINCSCP_209946 |
HA1E |
| -0.241857 |
1.914351e-14 |
975 |
Broad-Sai-560 |
LSM-45991 |
|
3uM |
24h |
LINCSCP_250254 |
LINCSCP_250254 |
MCF7 |
| 0.241807 |
1.939151e-14 |
975 |
Triacsin C |
LSM-43284 |
ACSL1 |
10uM |
6h |
LINCSCP_40243 |
LINCSCP_40243 |
NCIH508 |
| -0.241781 |
1.951682e-14 |
975 |
vinorelbine |
|
TUBB |
10uM |
24h |
LINCSCP_32583 |
LINCSCP_32583 |
MCF7 |
| 0.241705 |
1.989939e-14 |
975 |
BRD-K09031632 |
LSM-37755 |
|
10uM |
6h |
LINCSCP_49084 |
LINCSCP_49084 |
PC3 |
| 0.241694 |
1.995501e-14 |
975 |
SCHEMBL3958507 |
LSM-5245 |
COQ8B|EGFR |
0.37uM |
24h |
LINCSCP_99723 |
LINCSCP_99723 |
HCC515 |
| 0.241622 |
2.032337e-14 |
975 |
GW843682X |
LSM-1014 |
PLK1|PLK3 |
0.12uM |
24h |
LINCSCP_69342 |
LINCSCP_69342 |
A375 |
| 0.241554 |
2.067425e-14 |
975 |
Motesanib |
LSM-1042 |
FLT1|FLT4|KDR|KIT|PDGFRA|PDGFRB|RET |
1.11uM |
24h |
LINCSCP_129645 |
LINCSCP_129645 |
JURKAT |
| -0.241497 |
2.097624e-14 |
975 |
MLS002264449 |
LSM-3136 |
|
10uM |
6h |
LINCSCP_5523 |
LINCSCP_5523 |
A549 |
| 0.241427 |
2.135357e-14 |
975 |
Bromopyruvate |
LSM-6288 |
HK2 |
100uM |
24h |
LINCSCP_25647 |
LINCSCP_25647 |
HT29 |
| -0.241397 |
2.151778e-14 |
975 |
Rebastinib |
LSM-6708 |
ABL1 |
3.33uM |
24h |
LINCSCP_146182 |
LINCSCP_146182 |
MNEU.E |
| -0.24139 |
2.155429e-14 |
975 |
MLS002264363 |
LSM-2417 |
|
10uM |
6h |
LINCSCP_31461 |
LINCSCP_31461 |
MCF7 |
| -0.241365 |
2.169304e-14 |
975 |
Olaparib |
LSM-1145 |
PARP1|PARP2|PARP3 |
40uM |
6h |
LINCSCP_50559 |
LINCSCP_50559 |
PL21 |
| -0.241324 |
2.191558e-14 |
975 |
Brompheniramine |
LSM-1736 |
HRH1 |
10uM |
24h |
LINCSCP_11139 |
LINCSCP_11139 |
ASC |
| 0.241298 |
2.206362e-14 |
975 |
Tranilast |
LSM-42898 |
|
0.12uM |
24h |
LINCSCP_71633 |
LINCSCP_71633 |
A375 |
| -0.241271 |
2.221400e-14 |
975 |
HMN-214 |
LSM-42802 |
CSF1R|FLT1|FLT3|FLT4|KDR|KIT|PDGFRB|RET |
3.33uM |
24h |
LINCSCP_142602 |
LINCSCP_142602 |
MCF7 |
| -0.241261 |
2.227020e-14 |
975 |
Cerulenin |
LSM-43210 |
FASN |
0.5uM |
24h |
LINCSCP_37921 |
LINCSCP_37921 |
MCF7 |
| -0.241252 |
2.231877e-14 |
975 |
Mebendazole |
LSM-3749 |
|
40uM |
24h |
LINCSCP_67546 |
LINCSCP_67546 |
MCF7 |
| -0.241232 |
2.243364e-14 |
975 |
Azasetron |
LSM-1565 |
HTR3A |
10uM |
24h |
LINCSCP_52708 |
LINCSCP_52708 |
SKB |
| 0.241207 |
2.257622e-14 |
975 |
6,10,10B-Trihydroxy-3,4a,7,7,10a-pentamethyl-1-oxo-3-vinyldodecahydro-1H-benzo[f]chromen-5-yl acetate |
LSM-4467 |
ADCY2 |
10uM |
6h |
LINCSCP_53534 |
LINCSCP_53534 |
SNGM |
| -0.241191 |
2.266606e-14 |
975 |
Iodipamide |
LSM-3496 |
|
10uM |
24h |
LINCSCP_284776 |
LINCSCP_284776 |
SKB |
| -0.241152 |
2.289245e-14 |
975 |
SA-85377 |
LSM-39088 |
|
3uM |
24h |
LINCSCP_37237 |
LINCSCP_37237 |
MCF7 |
| 0.241143 |
2.294740e-14 |
975 |
BRD-K58070753 |
LSM-40447 |
|
10uM |
6h |
LINCSCP_16328 |
LINCSCP_16328 |
HA1E |
| 0.24114 |
2.296281e-14 |
975 |
AG 14361 |
LSM-1988 |
PARP1 |
0.001uM |
6h |
LINCSCP_250838 |
LINCSCP_250838 |
MCF7 |
| -0.241136 |
2.298591e-14 |
975 |
Famciclovir |
LSM-2990 |
|
0.04uM |
24h |
LINCSCP_141010 |
LINCSCP_141010 |
MCF7 |
| 0.241091 |
2.324627e-14 |
975 |
Emedastine |
LSM-5331 |
HRH1 |
0.12uM |
24h |
LINCSCP_169822 |
LINCSCP_169822 |
YAPC |
| -0.241088 |
2.326441e-14 |
975 |
TORIN1 |
LSM-1079 |
MTOR |
0.1uM |
6h |
LINCSCP_39196 |
LINCSCP_39196 |
MDAMB231 |
| 0.241076 |
2.333891e-14 |
975 |
BMN 673 |
LSM-45245 |
|
3.33uM |
24h |
LINCSCP_162597 |
LINCSCP_162597 |
PC3 |
| -0.24106 |
2.343136e-14 |
975 |
CHEMBL2141850 |
LSM-6136 |
|
10uM |
24h |
LINCSCP_32211 |
LINCSCP_32211 |
MCF7 |
| -0.241026 |
2.363243e-14 |
975 |
SPECTRUM1505012 |
LSM-1773 |
CYP19A1 |
0.37uM |
24h |
LINCSCP_79240 |
LINCSCP_79240 |
A375 |
| 0.241016 |
2.369176e-14 |
975 |
BMS-345541 |
LSM-1028 |
IKBKB |
3.33uM |
24h |
LINCSCP_81425 |
LINCSCP_81425 |
A549 |
| 0.240981 |
2.390510e-14 |
975 |
Rebamipide |
LSM-4343 |
|
0.04uM |
24h |
LINCSCP_118298 |
LINCSCP_118298 |
HT29 |
| 0.240971 |
2.396602e-14 |
975 |
SA-1925610 |
LSM-38660 |
|
0.5uM |
6h |
LINCSCP_37100 |
LINCSCP_37100 |
MCF7 |
| -0.240959 |
2.403935e-14 |
975 |
BRD-A28746609 |
LSM-1102 |
NR1I2|TUBB |
0.12uM |
24h |
LINCSCP_169354 |
LINCSCP_169354 |
YAPC |
| -0.24095 |
2.409176e-14 |
975 |
Piperacillin |
LSM-5924 |
|
10uM |
24h |
LINCSCP_272126 |
LINCSCP_272126 |
PC3 |
| 0.240948 |
2.410264e-14 |
975 |
BRD-A82197375 |
LSM-45476 |
|
0.37uM |
24h |
LINCSCP_121034 |
LINCSCP_121034 |
HT29 |
| -0.240908 |
2.434914e-14 |
975 |
BAY 61-3606 |
LSM-1167 |
SYK |
10uM |
24h |
LINCSCP_82578 |
LINCSCP_82578 |
A549 |
| 0.240847 |
2.473150e-14 |
975 |
BRD-K58788895 |
LSM-11982 |
|
5uM |
24h |
LINCSCP_63392 |
LINCSCP_63392 |
VCAP |
| -0.24083 |
2.483556e-14 |
975 |
HMN-214 |
LSM-42802 |
CSF1R|FLT1|FLT3|FLT4|KDR|KIT|PDGFRB|RET |
10uM |
24h |
LINCSCP_142601 |
LINCSCP_142601 |
MCF7 |
| 0.240785 |
2.512052e-14 |
975 |
Dubinidine |
LSM-1971 |
|
10uM |
24h |
LINCSCP_266800 |
LINCSCP_266800 |
PC3 |
| 0.240781 |
2.514277e-14 |
975 |
BRD-K50149017 |
LSM-11478 |
|
5uM |
24h |
LINCSCP_62157 |
LINCSCP_62157 |
VCAP |
| 0.24072 |
2.553570e-14 |
975 |
Niacin |
LSM-4676 |
HCAR2|HCAR3 |
0.12uM |
24h |
LINCSCP_139822 |
LINCSCP_139822 |
MCF7 |
| -0.240697 |
2.568312e-14 |
975 |
Vorinostat |
LSM-3828 |
HDAC1|HDAC2|HDAC3|HDAC6|HDAC8 |
1uM |
24h |
LINCSCP_38236 |
LINCSCP_38236 |
MCF7 |
| -0.24069 |
2.573252e-14 |
975 |
Lexibulin |
LSM-6232 |
TUBA1A|TUBA1B|TUBA1C|TUBA3E|TUBA4A|TUBB|TUBB1|TUBB2A|TUBB2B|TUBB3|TUBB4A|TUBB4B|TUBB6|TUBB8 |
0.37uM |
24h |
LINCSCP_135773 |
LINCSCP_135773 |
MCF7 |
| 0.240625 |
2.615866e-14 |
975 |
BRD-K75418563 |
LSM-6850 |
|
10uM |
6h |
LINCSCP_23720 |
LINCSCP_23720 |
HEPG2 |
| 0.24062 |
2.619111e-14 |
975 |
NCGC00011940 |
LSM-2623 |
|
10uM |
24h |
LINCSCP_4936 |
LINCSCP_4936 |
A549 |
| 0.240593 |
2.636640e-14 |
975 |
Lenalidomide |
LSM-6187 |
CRBN|CUL4A|DDB1|RBX1|TNF |
0.04uM |
24h |
LINCSCP_71658 |
LINCSCP_71658 |
A375 |
| -0.240589 |
2.639188e-14 |
975 |
SCHEMBL2231351 |
LSM-36442 |
|
0.001uM |
6h |
LINCSCP_55139 |
LINCSCP_55139 |
THP1 |
| 0.240571 |
2.651235e-14 |
975 |
BMS-345541 |
LSM-1028 |
IKBKB |
1uM |
24h |
LINCSCP_24259 |
LINCSCP_24259 |
HS578T |
| -0.240484 |
2.710260e-14 |
975 |
4,11-Diethyl-4,9-dihydroxy-1H-pyrano[3',4':6,7]indolizino[1,2-b]quinoline-3,14(4H,12H)-dione |
LSM-6189 |
TOP1 |
3uM |
24h |
LINCSCP_35637 |
LINCSCP_35637 |
MCF7 |
| 0.240481 |
2.712211e-14 |
975 |
BRD-K47029744 |
LSM-11298 |
|
5uM |
24h |
LINCSCP_63086 |
LINCSCP_63086 |
VCAP |
| -0.240473 |
2.718125e-14 |
975 |
BRD-K36959991 |
LSM-8215 |
|
3uM |
6h |
LINCSCP_37122 |
LINCSCP_37122 |
MCF7 |
| 0.240438 |
2.742137e-14 |
975 |
SCHEMBL618594 |
LSM-1070 |
|
0.37uM |
24h |
LINCSCP_86873 |
LINCSCP_86873 |
CD34 |
| -0.240373 |
2.787028e-14 |
975 |
Nitrendipine |
LSM-1246 |
CACNA1C|CACNA1D|CACNA2D1 |
10uM |
24h |
LINCSCP_153930 |
LINCSCP_153930 |
PC3 |
| -0.240368 |
2.790538e-14 |
975 |
BRD-K48296029 |
LSM-11366 |
|
10uM |
24h |
LINCSCP_9045 |
LINCSCP_9045 |
A549 |
| -0.240365 |
2.793310e-14 |
975 |
TAK-715 |
LSM-1060 |
MAPK14 |
10uM |
6h |
LINCSCP_16661 |
LINCSCP_16661 |
HA1E |
| -0.240357 |
2.798268e-14 |
975 |
BRD-K23217353 |
LSM-38534 |
|
5uM |
24h |
LINCSCP_249192 |
LINCSCP_249192 |
MCF7 |
| -0.240342 |
2.809325e-14 |
975 |
SCHEMBL16226068 |
LSM-43297 |
HSP90AA1 |
20uM |
6h |
LINCSCP_64548 |
LINCSCP_64548 |
VCAP |
| 0.240332 |
2.816360e-14 |
975 |
BCB03_000082 |
LSM-36632 |
|
10uM |
6h |
LINCSCP_32632 |
LINCSCP_32632 |
MCF7 |
| 0.240192 |
2.917558e-14 |
975 |
Splitomicin |
LSM-2607 |
|
10uM |
6h |
LINCSCP_4354 |
LINCSCP_4354 |
A549 |
| 0.240181 |
2.925577e-14 |
975 |
BRD-K95367721 |
LSM-14275 |
|
5uM |
24h |
LINCSCP_62949 |
LINCSCP_62949 |
VCAP |
| -0.240123 |
2.968850e-14 |
975 |
MLS000526305 |
LSM-4036 |
|
10uM |
6h |
LINCSCP_45859 |
LINCSCP_45859 |
PC3 |
| 0.24011 |
2.978326e-14 |
975 |
Hydroflumethiazide |
LSM-5497 |
SLC12A1|SLC12A3 |
1.11uM |
24h |
LINCSCP_103705 |
LINCSCP_103705 |
HELA |
| -0.240098 |
2.987180e-14 |
975 |
VU0420363-1 |
LSM-3326 |
|
10uM |
24h |
LINCSCP_1412 |
LINCSCP_1412 |
A375 |
| -0.240083 |
2.998956e-14 |
975 |
BI-2536 |
LSM-1041 |
PLK1 |
0.04uM |
24h |
LINCSCP_140812 |
LINCSCP_140812 |
MCF7 |
| 0.240046 |
3.026555e-14 |
975 |
BRD-K67519589 |
LSM-40951 |
|
10uM |
6h |
LINCSCP_20650 |
LINCSCP_20650 |
HCC515 |
| 0.239996 |
3.064846e-14 |
975 |
BRD-K36490574 |
LSM-39267 |
|
10uM |
24h |
LINCSCP_33852 |
LINCSCP_33852 |
MCF7 |
| -0.239961 |
3.091936e-14 |
975 |
Cabazitaxel |
LSM-46002 |
|
1.11uM |
24h |
LINCSCP_138308 |
LINCSCP_138308 |
MCF7 |
| 0.239933 |
3.114121e-14 |
975 |
Prostoglandin A1 |
LSM-42846 |
|
1uM |
24h |
LINCSCP_25456 |
LINCSCP_25456 |
HT29 |
| -0.239923 |
3.122139e-14 |
975 |
Acivicin |
LSM-45583 |
|
0.14uM |
24h |
LINCSCP_169648 |
LINCSCP_169648 |
YAPC |
| 0.239906 |
3.135335e-14 |
975 |
4-Fluoro-n-(pyridin-3-yl)benzamide |
LSM-3702 |
CYP11B2 |
10uM |
24h |
LINCSCP_5006 |
LINCSCP_5006 |
A549 |
| -0.239889 |
3.148962e-14 |
975 |
Broad-Sai-370 |
LSM-45321 |
|
10uM |
24h |
LINCSCP_43506 |
LINCSCP_43506 |
NPC |
| -0.239883 |
3.153294e-14 |
975 |
BRD-K06303559 |
LSM-37610 |
|
5uM |
24h |
LINCSCP_28063 |
LINCSCP_28063 |
HT29 |
| 0.239855 |
3.175889e-14 |
975 |
apicidin |
LSM-45760 |
|
0.04uM |
24h |
LINCSCP_139565 |
LINCSCP_139565 |
MCF7 |
| 0.239838 |
3.189725e-14 |
975 |
BS-181 |
LSM-6305 |
|
0.12uM |
24h |
LINCSCP_149846 |
LINCSCP_149846 |
NPC.TAK |
| -0.239801 |
3.219596e-14 |
975 |
GSK-2334470 |
LSM-1222 |
PDK1|PDPK1 |
1.11uM |
24h |
LINCSCP_150455 |
LINCSCP_150455 |
NPC.TAK |
| -0.239767 |
3.247404e-14 |
975 |
Volasertib (BI 6727) |
LSM-45277 |
PLK1 |
0.12uM |
24h |
LINCSCP_160776 |
LINCSCP_160776 |
PC3 |
| -0.239759 |
3.253783e-14 |
975 |
Proglumide |
LSM-4439 |
CCKAR|CCKBR |
0.37uM |
24h |
LINCSCP_140996 |
LINCSCP_140996 |
MCF7 |
| -0.239747 |
3.263040e-14 |
975 |
Methyldopa |
LSM-5596 |
ADRA2A|ADRA2B|ADRA2C|DDC |
10uM |
24h |
LINCSCP_47526 |
LINCSCP_47526 |
PC3 |
| -0.239709 |
3.294637e-14 |
975 |
ABT-751 |
LSM-6285 |
|
10uM |
6h |
LINCSCP_12737 |
LINCSCP_12737 |
COV644 |
| 0.23969 |
3.310834e-14 |
975 |
Tropisetron |
LSM-5617 |
HTR3A |
10uM |
24h |
LINCSCP_34457 |
LINCSCP_34457 |
MCF7 |
| 0.239664 |
3.331886e-14 |
975 |
BRD-K49553303-001-01-8 |
LSM-40022 |
|
10uM |
6h |
LINCSCP_295846 |
LINCSCP_295846 |
VCAP |
| 0.239623 |
3.367027e-14 |
975 |
Lenalidomide |
LSM-6187 |
CRBN|CUL4A|DDB1|RBX1|TNF |
1.11uM |
24h |
LINCSCP_71655 |
LINCSCP_71655 |
A375 |
| -0.239615 |
3.373904e-14 |
975 |
Bosentan |
LSM-5825 |
EDNRA|EDNRB |
10uM |
6h |
LINCSCP_16998 |
LINCSCP_16998 |
HA1E |
| 0.239603 |
3.383479e-14 |
975 |
ipratropium |
LSM-45809 |
|
0.12uM |
24h |
LINCSCP_139732 |
LINCSCP_139732 |
MCF7 |
| 0.23953 |
3.446479e-14 |
975 |
LY2886721 |
LSM-45433 |
|
0.37uM |
24h |
LINCSCP_101791 |
LINCSCP_101791 |
HELA |
| 0.239499 |
3.473419e-14 |
975 |
CHEMBL2361430 |
LSM-39835 |
|
10uM |
6h |
LINCSCP_16834 |
LINCSCP_16834 |
HA1E |
| -0.239488 |
3.482752e-14 |
975 |
BRD-K36864553 |
LSM-39288 |
|
5uM |
24h |
LINCSCP_27446 |
LINCSCP_27446 |
HT29 |
| 0.239438 |
3.526744e-14 |
975 |
QL47 |
LSM-6019 |
BMX|BTK |
0.12uM |
24h |
LINCSCP_100036 |
LINCSCP_100036 |
HCC515 |
| 0.239423 |
3.540580e-14 |
975 |
GRANISETRON HYDROCHLORIDE |
LSM-45509 |
HTR3A |
0.37uM |
24h |
LINCSCP_72713 |
LINCSCP_72713 |
A375 |
| 0.239394 |
3.566248e-14 |
975 |
SR 33805 oxalate |
LSM-45933 |
|
0.12uM |
24h |
LINCSCP_105715 |
LINCSCP_105715 |
HELA |
| -0.239382 |
3.577026e-14 |
975 |
Idelalisib |
LSM-1205 |
PIK3CD|PIK3CG |
1.11uM |
24h |
LINCSCP_165580 |
LINCSCP_165580 |
SKL |
| -0.239376 |
3.582373e-14 |
975 |
Flunisolide |
LSM-3089 |
NR3C1 |
10uM |
24h |
LINCSCP_31380 |
LINCSCP_31380 |
MCF7 |
| 0.239364 |
3.593091e-14 |
975 |
Fusaric acid |
LSM-3944 |
DBH |
10uM |
24h |
LINCSCP_33125 |
LINCSCP_33125 |
MCF7 |
| -0.23932 |
3.633397e-14 |
975 |
Albendazole |
LSM-3782 |
|
3.33uM |
24h |
LINCSCP_126887 |
LINCSCP_126887 |
HT29 |
| -0.23929 |
3.660411e-14 |
975 |
CHEMBL2362635 |
LSM-10581 |
|
5uM |
24h |
LINCSCP_34979 |
LINCSCP_34979 |
MCF7 |
| -0.239274 |
3.675099e-14 |
975 |
COT Inhibitor-2 |
LSM-1154 |
|
10uM |
6h |
LINCSCP_39581 |
LINCSCP_39581 |
MDAMB231 |
| 0.23921 |
3.735192e-14 |
975 |
1166227-08-2 |
LSM-1204 |
|
0.37uM |
24h |
LINCSCP_69705 |
LINCSCP_69705 |
A375 |
| 0.239094 |
3.844916e-14 |
975 |
BRD-K37552925 |
LSM-10699 |
|
5uM |
24h |
LINCSCP_61770 |
LINCSCP_61770 |
VCAP |
| -0.239027 |
3.909869e-14 |
975 |
Setiptiline |
LSM-45982 |
|
0.04uM |
24h |
LINCSCP_153785 |
LINCSCP_153785 |
PC3 |
| -0.23902 |
3.916954e-14 |
975 |
Methyltestosterone |
LSM-5902 |
AR |
10uM |
24h |
LINCSCP_31775 |
LINCSCP_31775 |
MCF7 |
| -0.239007 |
3.930177e-14 |
975 |
Minaprine |
LSM-2037 |
HTR2B|SLC6A4 |
0.12uM |
24h |
LINCSCP_138694 |
LINCSCP_138694 |
MCF7 |
| 0.238996 |
3.940751e-14 |
975 |
Tenofovir |
LSM-5340 |
|
10uM |
6h |
LINCSCP_16623 |
LINCSCP_16623 |
HA1E |
| -0.238981 |
3.955385e-14 |
975 |
BSPBIO_000981 |
LSM-43126 |
ACTA1 |
10uM |
24h |
LINCSCP_10876 |
LINCSCP_10876 |
ASC |
| 0.238954 |
3.982594e-14 |
975 |
2-Chloroadenosine |
LSM-37201 |
|
10uM |
6h |
LINCSCP_46172 |
LINCSCP_46172 |
PC3 |
| -0.238937 |
3.999874e-14 |
975 |
GSK 1059615 |
LSM-42799 |
PIK3CA|PIK3CB|PIK3CD|PIK3CG |
10uM |
24h |
LINCSCP_150435 |
LINCSCP_150435 |
NPC.TAK |
| 0.238915 |
4.021577e-14 |
975 |
BRD-K24621485 |
LSM-9922 |
|
1uM |
24h |
LINCSCP_253060 |
LINCSCP_253060 |
MCF7 |
| -0.238913 |
4.023198e-14 |
975 |
IN1092 |
LSM-1739 |
|
10uM |
24h |
LINCSCP_43977 |
LINCSCP_43977 |
PC3 |
| -0.238771 |
4.168879e-14 |
975 |
PD-0325901 |
LSM-1101 |
MAP2K1|MAP2K2 |
10uM |
24h |
LINCSCP_68997 |
LINCSCP_68997 |
A375 |
| -0.238757 |
4.183839e-14 |
975 |
cortisone-acetate |
LSM-45387 |
TUBA1A|TUBA1B|TUBA1C|TUBA3E|TUBA4A|TUBB|TUBB1|TUBB2A|TUBB2B|TUBB3|TUBB4A|TUBB4B|TUBB6|TUBB8 |
0.12uM |
24h |
LINCSCP_143283 |
LINCSCP_143283 |
MCF7 |
| -0.238754 |
4.187132e-14 |
975 |
BRD-K13077924 |
LSM-45363 |
|
10uM |
24h |
LINCSCP_55303 |
LINCSCP_55303 |
U937 |
| 0.238723 |
4.219448e-14 |
975 |
BRD-K38797319 |
LSM-10780 |
|
5uM |
24h |
LINCSCP_48240 |
LINCSCP_48240 |
PC3 |
| -0.238718 |
4.225373e-14 |
975 |
CHEMBL585951 |
LSM-36386 |
MAPK8 |
1.11uM |
24h |
LINCSCP_131368 |
LINCSCP_131368 |
MCF10A |
| 0.238704 |
4.239389e-14 |
975 |
Gemcitabine |
LSM-5333 |
POLA1|POLD1|POLE|RRM1|RRM2|RRM2B |
0.1uM |
6h |
LINCSCP_55458 |
LINCSCP_55458 |
U937 |
| -0.238698 |
4.245767e-14 |
975 |
BRD-A28746609 |
LSM-1102 |
NR1I2|TUBB |
3.33uM |
24h |
LINCSCP_137545 |
LINCSCP_137545 |
MCF7 |
| -0.238624 |
4.325514e-14 |
975 |
GSK-1070916 |
LSM-1062 |
AURKB|AURKC |
3.33uM |
24h |
LINCSCP_83359 |
LINCSCP_83359 |
ASC.C |
| 0.238614 |
4.336423e-14 |
975 |
Cholic acid |
LSM-5541 |
CES1|FECH|PLA2G1B |
0.12uM |
24h |
LINCSCP_75558 |
LINCSCP_75558 |
A375 |
| 0.238592 |
4.359871e-14 |
975 |
Gemifloxacin |
LSM-44972 |
|
10uM |
24h |
LINCSCP_93780 |
LINCSCP_93780 |
HA1E |
| -0.238591 |
4.361053e-14 |
975 |
GSK-923295 |
LSM-45692 |
|
10uM |
24h |
LINCSCP_137220 |
LINCSCP_137220 |
MCF7 |
| -0.238557 |
4.398525e-14 |
975 |
CHEMBL2355890 |
LSM-6823 |
|
3uM |
24h |
LINCSCP_23360 |
LINCSCP_23360 |
HEPG2 |
| -0.238489 |
4.473850e-14 |
975 |
WHI-P97 |
LSM-1033 |
JAK3 |
10uM |
6h |
LINCSCP_20490 |
LINCSCP_20490 |
HCC515 |
| -0.238473 |
4.491665e-14 |
975 |
Verapamil |
LSM-1298 |
CACNA1C|CACNA1D|CACNA1F|CACNA1G|CACNA1S |
10uM |
24h |
LINCSCP_52793 |
LINCSCP_52793 |
SKB |
| -0.238397 |
4.578209e-14 |
975 |
PD-0325901 |
LSM-1101 |
MAP2K1|MAP2K2 |
3.33uM |
24h |
LINCSCP_150782 |
LINCSCP_150782 |
PC3 |
| 0.238375 |
4.603917e-14 |
975 |
Gefitinib |
LSM-1098 |
EGFR |
0.04uM |
24h |
LINCSCP_130019 |
LINCSCP_130019 |
LNCAP |
| -0.238347 |
4.635917e-14 |
975 |
SPECTRUM_001092 |
LSM-1337 |
NR3C1 |
10uM |
6h |
LINCSCP_266952 |
LINCSCP_266952 |
PC3 |
| 0.238324 |
4.663051e-14 |
975 |
Lapatinib |
LSM-1051 |
EGFR|ERBB2 |
0.37uM |
3h |
LINCSCP_133184 |
LINCSCP_133184 |
MCF7 |
| -0.238293 |
4.699241e-14 |
975 |
PJ34 |
LSM-4937 |
|
10uM |
6h |
LINCSCP_43737 |
LINCSCP_43737 |
OV7 |
| -0.238252 |
4.746790e-14 |
975 |
2-(4-Nitro-phenylamino)-benzoic acid |
LSM-45307 |
|
10uM |
6h |
LINCSCP_24202 |
LINCSCP_24202 |
HL60 |
| 0.238238 |
4.763448e-14 |
975 |
BRD-K67319066 |
LSM-12525 |
|
5uM |
24h |
LINCSCP_61809 |
LINCSCP_61809 |
VCAP |
| -0.238227 |
4.776528e-14 |
975 |
N6022 |
LSM-45697 |
|
0.12uM |
24h |
LINCSCP_159540 |
LINCSCP_159540 |
PC3 |
| 0.238212 |
4.795252e-14 |
975 |
CHEMBL1617726 |
LSM-6255 |
|
80uM |
6h |
LINCSCP_19561 |
LINCSCP_19561 |
HCC515 |
| -0.238198 |
4.811585e-14 |
975 |
GSK-461364 |
LSM-1013 |
PLK1 |
0.12uM |
24h |
LINCSCP_144237 |
LINCSCP_144237 |
MCF7 |
| 0.238077 |
4.958836e-14 |
975 |
Azacitidine |
LSM-5218 |
DNMT1|DNMT3A |
0.04uM |
24h |
LINCSCP_87011 |
LINCSCP_87011 |
CD34 |
| 0.238073 |
4.964076e-14 |
975 |
AZD-1775 |
LSM-1153 |
WEE1 |
0.04uM |
24h |
LINCSCP_86881 |
LINCSCP_86881 |
CD34 |
| -0.238061 |
4.978823e-14 |
975 |
SA-1459975 |
LSM-40000 |
|
3uM |
24h |
LINCSCP_37242 |
LINCSCP_37242 |
MCF7 |
| 0.23802 |
5.030453e-14 |
975 |
CHEMBL2204241 |
LSM-36798 |
|
0.5uM |
24h |
LINCSCP_55109 |
LINCSCP_55109 |
THP1 |
| -0.237979 |
5.081874e-14 |
975 |
GW843682X |
LSM-1014 |
PLK1|PLK3 |
10uM |
24h |
LINCSCP_25640 |
LINCSCP_25640 |
HT29 |
| 0.237978 |
5.082860e-14 |
975 |
Cholic acid |
LSM-5541 |
CES1|FECH|PLA2G1B |
0.12uM |
24h |
LINCSCP_122516 |
LINCSCP_122516 |
HT29 |
| -0.2379 |
5.182518e-14 |
975 |
Buparlisib |
LSM-1148 |
PIK3CA|PIK3CB|PIK3CD|PIK3CG|PIK3R1|PIK3R2|PIK3R3|PIK3R5 |
3.33uM |
24h |
LINCSCP_81161 |
LINCSCP_81161 |
A549 |
| -0.237838 |
5.263578e-14 |
975 |
Medrysone |
LSM-3259 |
NR3C1 |
10uM |
24h |
LINCSCP_272069 |
LINCSCP_272069 |
PC3 |
| 0.237814 |
5.295597e-14 |
975 |
Pfmrk inhibitor, wr 216174 |
LSM-42921 |
|
10uM |
24h |
LINCSCP_33357 |
LINCSCP_33357 |
MCF7 |
| -0.237777 |
5.344557e-14 |
975 |
BRD-K72343629 |
LSM-41191 |
|
10uM |
24h |
LINCSCP_3614 |
LINCSCP_3614 |
A375 |
| -0.2377 |
5.448050e-14 |
975 |
Procaterol |
LSM-1391 |
ADRB2 |
3uM |
24h |
LINCSCP_37849 |
LINCSCP_37849 |
MCF7 |
| -0.237622 |
5.555426e-14 |
975 |
Vorinostat |
LSM-3828 |
HDAC1|HDAC2|HDAC3|HDAC6|HDAC8 |
0.5uM |
6h |
LINCSCP_49377 |
LINCSCP_49377 |
PC3 |
| 0.237592 |
5.596386e-14 |
975 |
BRD-K47423282 |
LSM-11322 |
|
5uM |
24h |
LINCSCP_64001 |
LINCSCP_64001 |
VCAP |
| 0.237582 |
5.610404e-14 |
975 |
MLS002264443 |
LSM-3540 |
|
10uM |
6h |
LINCSCP_31507 |
LINCSCP_31507 |
MCF7 |
| -0.237535 |
5.676070e-14 |
975 |
Lexibulin |
LSM-6232 |
TUBA1A|TUBA1B|TUBA1C|TUBA3E|TUBA4A|TUBB|TUBB1|TUBB2A|TUBB2B|TUBB3|TUBB4A|TUBB4B|TUBB6|TUBB8 |
1.11uM |
24h |
LINCSCP_153980 |
LINCSCP_153980 |
PC3 |
| 0.237521 |
5.696498e-14 |
975 |
MEGXM0_000032 |
LSM-4453 |
|
10uM |
6h |
LINCSCP_20055 |
LINCSCP_20055 |
HCC515 |
| -0.237516 |
5.703838e-14 |
975 |
MLS001060847 |
LSM-1427 |
|
10uM |
24h |
LINCSCP_4872 |
LINCSCP_4872 |
A549 |
| -0.237498 |
5.729854e-14 |
975 |
SCHEMBL17857056 |
LSM-5545 |
|
10uM |
24h |
LINCSCP_29512 |
LINCSCP_29512 |
MCF10A |
| -0.237469 |
5.770679e-14 |
975 |
CHEMBL3182990 |
LSM-2587 |
|
10uM |
6h |
LINCSCP_19711 |
LINCSCP_19711 |
HCC515 |
| 0.237434 |
5.821576e-14 |
975 |
BRD-K51894281 |
LSM-11604 |
|
5uM |
24h |
LINCSCP_62462 |
LINCSCP_62462 |
VCAP |
| -0.23742 |
5.841113e-14 |
975 |
SA-97110 |
LSM-37431 |
|
10uM |
6h |
LINCSCP_37068 |
LINCSCP_37068 |
MCF7 |
| 0.237415 |
5.849433e-14 |
975 |
Glycopyrrolate |
LSM-5163 |
CHRM1|CHRM2|CHRM3 |
10uM |
24h |
LINCSCP_5360 |
LINCSCP_5360 |
A549 |
| -0.237343 |
5.954725e-14 |
975 |
MLS003128818 |
LSM-11790 |
|
5uM |
24h |
LINCSCP_64295 |
LINCSCP_64295 |
VCAP |
| -0.237227 |
6.128570e-14 |
975 |
NCGC00166323-01 |
LSM-6478 |
|
10uM |
24h |
LINCSCP_140429 |
LINCSCP_140429 |
MCF7 |
| 0.237175 |
6.209400e-14 |
975 |
2-(2-Bromo-4-methyl-phenylamino)-pyrido[3,2-e][1,3]thiazin-4-one |
LSM-45312 |
|
0.5uM |
24h |
LINCSCP_12377 |
LINCSCP_12377 |
CD34 |
| 0.23716 |
6.231751e-14 |
975 |
Gemfibrozil |
LSM-2227 |
CYP2C8|LPL|PPARA |
10uM |
24h |
LINCSCP_72722 |
LINCSCP_72722 |
A375 |
| 0.237117 |
6.298679e-14 |
975 |
Midodrine |
LSM-1815 |
ADRA1A|ADRA1B|ADRA1D |
0.37uM |
24h |
LINCSCP_143456 |
LINCSCP_143456 |
MCF7 |
| -0.237115 |
6.302280e-14 |
975 |
ST50851843 |
LSM-4704 |
|
10uM |
24h |
LINCSCP_31961 |
LINCSCP_31961 |
MCF7 |
| -0.237101 |
6.324303e-14 |
975 |
BRD-K65517548 |
LSM-12427 |
|
5uM |
6h |
LINCSCP_61365 |
LINCSCP_61365 |
VCAP |
| 0.237097 |
6.329695e-14 |
975 |
Flunisolide |
LSM-3089 |
NR3C1 |
10uM |
6h |
LINCSCP_57892 |
LINCSCP_57892 |
VCAP |
| -0.237092 |
6.338105e-14 |
975 |
Procaine |
LSM-5396 |
HTR3A|SCN10A|SCN11A|SCN1A|SCN2A|SCN3A|SCN4A|SCN5A|SCN7A|SCN8A|SCN9A |
10uM |
24h |
LINCSCP_34277 |
LINCSCP_34277 |
MCF7 |
| 0.237074 |
6.367096e-14 |
975 |
Imatinib |
LSM-1023 |
ABL1|BCR|CSF1R|KIT|PDGFRA|PDGFRB |
0.37uM |
24h |
LINCSCP_130023 |
LINCSCP_130023 |
LNCAP |
| -0.237065 |
6.379934e-14 |
975 |
BL003-049-HDAC3 |
LSM-36785 |
|
10uM |
24h |
LINCSCP_43453 |
LINCSCP_43453 |
NPC |
| -0.237047 |
6.409115e-14 |
975 |
Isonicotinamide |
LSM-37066 |
|
10uM |
24h |
LINCSCP_263849 |
LINCSCP_263849 |
NPC |
| 0.237018 |
6.455765e-14 |
975 |
BRD-K35210537 |
LSM-39201 |
|
10uM |
6h |
LINCSCP_49124 |
LINCSCP_49124 |
PC3 |
| -0.236996 |
6.490411e-14 |
975 |
Lurasidone |
LSM-45843 |
DRD2|HTR2A |
1.11uM |
24h |
LINCSCP_171706 |
LINCSCP_171706 |
YAPC |
| 0.236942 |
6.579448e-14 |
975 |
Iloprost |
LSM-43147 |
PTGER1|PTGER2|PTGIR |
10uM |
24h |
LINCSCP_288767 |
LINCSCP_288767 |
U937 |
| 0.236933 |
6.593038e-14 |
975 |
BRD-K76352008 |
LSM-41440 |
|
5uM |
24h |
LINCSCP_64319 |
LINCSCP_64319 |
VCAP |
| 0.236928 |
6.601473e-14 |
975 |
SA-1939915 |
LSM-41811 |
|
1uM |
24h |
LINCSCP_38240 |
LINCSCP_38240 |
MCF7 |
| -0.236889 |
6.666635e-14 |
975 |
NMS-1286937 |
LSM-45818 |
|
0.37uM |
24h |
LINCSCP_141872 |
LINCSCP_141872 |
MCF7 |
| 0.236881 |
6.679817e-14 |
975 |
BRD-K93406156 |
LSM-14990 |
|
5uM |
24h |
LINCSCP_64236 |
LINCSCP_64236 |
VCAP |
| 0.23683 |
6.764295e-14 |
975 |
BRD-K16813995 |
LSM-9448 |
|
5uM |
24h |
LINCSCP_62863 |
LINCSCP_62863 |
VCAP |
| -0.236767 |
6.871345e-14 |
975 |
BRD-K76103428 |
LSM-41424 |
|
10uM |
24h |
LINCSCP_48825 |
LINCSCP_48825 |
PC3 |
| 0.236765 |
6.873976e-14 |
975 |
Estradiol |
LSM-2421 |
ESR1|ESR2|NR1I2 |
0.5uM |
24h |
LINCSCP_253472 |
LINCSCP_253472 |
MCF7 |
| 0.23672 |
6.951009e-14 |
975 |
CID 75060947 |
LSM-36700 |
|
10uM |
6h |
LINCSCP_216732 |
LINCSCP_216732 |
HCC515 |
| -0.236711 |
6.967104e-14 |
975 |
Tivozanib |
LSM-1005 |
FLT1|FLT4|KDR|KIT|PDGFRA|PDGFRB |
10uM |
24h |
LINCSCP_113707 |
LINCSCP_113707 |
HME1 |
| -0.236697 |
6.991862e-14 |
975 |
CEP-701 |
LSM-45844 |
|
10uM |
24h |
LINCSCP_71133 |
LINCSCP_71133 |
A375 |
| 0.236693 |
6.997290e-14 |
975 |
BRD-K25991572 |
LSM-14772 |
|
5uM |
24h |
LINCSCP_64179 |
LINCSCP_64179 |
VCAP |
| -0.23663 |
7.108634e-14 |
975 |
Olmesartan Medoxomil |
LSM-3767 |
AGTR1 |
0.04uM |
24h |
LINCSCP_143050 |
LINCSCP_143050 |
MCF7 |
| -0.236627 |
7.113535e-14 |
975 |
Dasatinib |
LSM-1020 |
ABL1|BCR|BLK|EPHA2|FGR|FRK|FYN|HCK|KIT|LCK|LYN|PDGFRB|SRC|SRMS|YES1 |
10uM |
24h |
LINCSCP_69021 |
LINCSCP_69021 |
A375 |
| -0.236623 |
7.119779e-14 |
975 |
BRD-K36959991 |
LSM-8215 |
|
0.5uM |
6h |
LINCSCP_37119 |
LINCSCP_37119 |
MCF7 |
| -0.236615 |
7.134562e-14 |
975 |
CGP 60474 |
LSM-1025 |
CDK1 |
10uM |
24h |
LINCSCP_42318 |
LINCSCP_42318 |
NPC |
| -0.23661 |
7.143300e-14 |
975 |
N-(3-Cyano-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)-2-{[3-cyano-6-(thiophen-2-yl)pyridin-2-yl]sulfanyl}acetamide |
LSM-4755 |
|
10uM |
6h |
LINCSCP_16385 |
LINCSCP_16385 |
HA1E |
| 0.236553 |
7.246019e-14 |
975 |
GRANISETRON HYDROCHLORIDE |
LSM-45509 |
HTR3A |
0.12uM |
24h |
LINCSCP_102841 |
LINCSCP_102841 |
HELA |
| 0.236536 |
7.275447e-14 |
975 |
MK-8245 |
LSM-45756 |
|
1.11uM |
24h |
LINCSCP_71303 |
LINCSCP_71303 |
A375 |
| 0.236536 |
7.276286e-14 |
975 |
BSPBIO_001542 |
LSM-42823 |
PPP1CA|PPP2CA |
10uM |
24h |
LINCSCP_210 |
LINCSCP_210 |
A375 |
| -0.236516 |
7.312139e-14 |
975 |
Beta-Narcotine |
LSM-4043 |
SIGMAR1 |
10uM |
24h |
LINCSCP_285024 |
LINCSCP_285024 |
SKB |
| 0.236483 |
7.372584e-14 |
975 |
BRD-K03707297 |
LSM-14688 |
|
5uM |
24h |
LINCSCP_64149 |
LINCSCP_64149 |
VCAP |
| -0.23643 |
7.470395e-14 |
975 |
Infigratinib |
LSM-1184 |
FGFR1|FGFR2|FGFR3|FGFR4 |
10uM |
24h |
LINCSCP_24739 |
LINCSCP_24739 |
HS578T |
| -0.23634 |
7.638760e-14 |
975 |
CHEMBL2355554 |
LSM-6843 |
|
5uM |
24h |
LINCSCP_34986 |
LINCSCP_34986 |
MCF7 |
| -0.236338 |
7.640885e-14 |
975 |
Podofilox |
LSM-3055 |
|
3.33uM |
24h |
LINCSCP_141624 |
LINCSCP_141624 |
MCF7 |
| 0.236332 |
7.653949e-14 |
975 |
Taranabant |
LSM-45803 |
CNR1 |
3.33uM |
24h |
LINCSCP_74208 |
LINCSCP_74208 |
A375 |
| -0.236331 |
7.655349e-14 |
975 |
GSK 1059615 |
LSM-42799 |
PIK3CA|PIK3CB|PIK3CD|PIK3CG |
3.33uM |
24h |
LINCSCP_69351 |
LINCSCP_69351 |
A375 |
| -0.236248 |
7.813296e-14 |
975 |
BRD-K69040870-001-01-4 |
LSM-41026 |
|
10uM |
24h |
LINCSCP_35355 |
LINCSCP_35355 |
MCF7 |
| 0.236246 |
7.818574e-14 |
975 |
SU 11274 |
LSM-42792 |
MET |
0.37uM |
24h |
LINCSCP_85299 |
LINCSCP_85299 |
BT20 |
| 0.236215 |
7.877749e-14 |
975 |
Rilmenidine |
LSM-4253 |
ADRA2A|NISCH |
10uM |
6h |
LINCSCP_15520 |
LINCSCP_15520 |
HA1E |
| -0.236195 |
7.917446e-14 |
975 |
Cyclohexanecarboxamide, 4-(1-aminoethyl)-n-4-pyridinyl-, trans- |
LSM-1177 |
ROCK1|ROCK2 |
0.04uM |
24h |
LINCSCP_158384 |
LINCSCP_158384 |
PC3 |
| 0.236164 |
7.978122e-14 |
975 |
SPOX1_000139 |
LSM-4762 |
|
10uM |
6h |
LINCSCP_6123 |
LINCSCP_6123 |
A549 |
| 0.236136 |
8.034247e-14 |
975 |
BRD-K50280607 |
LSM-40057 |
|
10uM |
6h |
LINCSCP_59354 |
LINCSCP_59354 |
VCAP |
| -0.236108 |
8.088627e-14 |
975 |
Motesanib |
LSM-1042 |
FLT1|FLT4|KDR|KIT|PDGFRA|PDGFRB|RET |
10uM |
24h |
LINCSCP_52459 |
LINCSCP_52459 |
SKB |
| -0.23608 |
8.145782e-14 |
975 |
CID 91122153 |
LSM-44934 |
|
10uM |
6h |
LINCSCP_19152 |
LINCSCP_19152 |
HCC515 |
| -0.236031 |
8.245482e-14 |
975 |
7-Hydroxyflavone |
LSM-4663 |
|
10uM |
24h |
LINCSCP_7609 |
LINCSCP_7609 |
A549 |
| 0.236028 |
8.251201e-14 |
975 |
Fluspirilene |
LSM-3748 |
DRD2|HTR2A |
5uM |
6h |
LINCSCP_29390 |
LINCSCP_29390 |
LOVO |
| 0.236014 |
8.278873e-14 |
975 |
AKT Inhibitor VIII |
LSM-1035 |
AKT1|AKT2 |
10uM |
6h |
LINCSCP_29299 |
LINCSCP_29299 |
LOVO |
| 0.236013 |
8.282454e-14 |
975 |
Imatinib |
LSM-1023 |
ABL1|BCR|CSF1R|KIT|PDGFRA|PDGFRB |
10uM |
3h |
LINCSCP_116092 |
LINCSCP_116092 |
HS578T |
| 0.236002 |
8.304408e-14 |
975 |
20554-84-1 |
LSM-43090 |
|
10uM |
6h |
LINCSCP_22342 |
LINCSCP_22342 |
HEPG2 |
| -0.235998 |
8.311617e-14 |
975 |
Tamatinib |
LSM-1040 |
SYK |
10uM |
24h |
LINCSCP_90477 |
LINCSCP_90477 |
HA1E |
| 0.235987 |
8.334711e-14 |
975 |
Testosterone Propionate |
LSM-4025 |
AR |
10uM |
6h |
LINCSCP_56188 |
LINCSCP_56188 |
VCAP |
| 0.23597 |
8.371080e-14 |
975 |
Pazopanib |
LSM-1114 |
CSF1R|FGFR1|FGFR3|FLT1|FLT4|ITK|KDR|KIT|LCK|PDGFRA|PDGFRB |
0.1uM |
6h |
LINCSCP_39642 |
LINCSCP_39642 |
MDAMB231 |
| 0.235885 |
8.547017e-14 |
975 |
Alpelisib |
LSM-4256 |
PIK3CA |
0.12uM |
24h |
LINCSCP_144865 |
LINCSCP_144865 |
MDAMB231 |
| -0.235871 |
8.577927e-14 |
975 |
GSK 1059615 |
LSM-42799 |
PIK3CA|PIK3CB|PIK3CD|PIK3CG |
10uM |
24h |
LINCSCP_116229 |
LINCSCP_116229 |
HT29 |
| -0.23587 |
8.578858e-14 |
975 |
BRD-8899 |
LSM-29350 |
|
0.001uM |
24h |
LINCSCP_41948 |
LINCSCP_41948 |
NOMO1 |
| 0.235866 |
8.589023e-14 |
975 |
TWS 119 |
LSM-1111 |
GSK3B |
0.5uM |
6h |
LINCSCP_39664 |
LINCSCP_39664 |
MDAMB231 |
| 0.235829 |
8.667314e-14 |
975 |
Tivozanib |
LSM-1005 |
FLT1|FLT4|KDR|KIT|PDGFRA|PDGFRB |
10uM |
24h |
LINCSCP_129417 |
LINCSCP_129417 |
JURKAT |
| 0.235828 |
8.668235e-14 |
975 |
Wortmannin |
LSM-3947 |
PIK3CA|PIK3CG|PLK1 |
0.001uM |
24h |
LINCSCP_201089 |
LINCSCP_201089 |
A549 |
| 0.235803 |
8.722572e-14 |
975 |
MLS000094380 |
LSM-3180 |
|
10uM |
6h |
LINCSCP_20007 |
LINCSCP_20007 |
HCC515 |
| -0.235796 |
8.738508e-14 |
975 |
Neratinib |
LSM-42778 |
EGFR|ERBB2|ERBB4 |
3.33uM |
3h |
LINCSCP_115093 |
LINCSCP_115093 |
HS578T |
| -0.235792 |
8.746897e-14 |
975 |
AZ628 |
LSM-1050 |
BRAF|RAF1 |
3.33uM |
24h |
LINCSCP_128083 |
LINCSCP_128083 |
HUES3 |
| 0.235763 |
8.810161e-14 |
975 |
Gefitinib |
LSM-1098 |
EGFR |
0.04uM |
24h |
LINCSCP_131431 |
LINCSCP_131431 |
MCF10A |
| 0.235759 |
8.818146e-14 |
975 |
BRD-K66052559 |
LSM-12458 |
|
5uM |
24h |
LINCSCP_62675 |
LINCSCP_62675 |
VCAP |
| 0.23575 |
8.838857e-14 |
975 |
Mesulergine |
LSM-4045 |
HTR2A|HTR2C|HTR7 |
10uM |
6h |
LINCSCP_547 |
LINCSCP_547 |
A375 |
| -0.235728 |
8.885489e-14 |
975 |
Hyperoside |
LSM-5907 |
|
10uM |
6h |
LINCSCP_5903 |
LINCSCP_5903 |
A549 |
| -0.235703 |
8.940510e-14 |
975 |
AC1MDKLV |
LSM-1956 |
|
10uM |
24h |
LINCSCP_188242 |
LINCSCP_188242 |
A549 |
| 0.235685 |
8.981770e-14 |
975 |
BI-2536 |
LSM-1041 |
PLK1 |
0.04uM |
3h |
LINCSCP_113390 |
LINCSCP_113390 |
HME1 |
| -0.235682 |
8.986825e-14 |
975 |
MLS003448162 |
LSM-3552 |
|
10uM |
24h |
LINCSCP_177893 |
LINCSCP_177893 |
A375 |
| 0.235581 |
9.215399e-14 |
975 |
BRD-K10856568 |
LSM-9092 |
|
5uM |
24h |
LINCSCP_62622 |
LINCSCP_62622 |
VCAP |
| 0.235459 |
9.496515e-14 |
975 |
Piperacillin |
LSM-5924 |
|
10uM |
6h |
LINCSCP_17015 |
LINCSCP_17015 |
HA1E |
| 0.235446 |
9.526840e-14 |
975 |
BRD-K54674054 |
LSM-40265 |
|
10uM |
24h |
LINCSCP_33880 |
LINCSCP_33880 |
MCF7 |
| 0.23539 |
9.657945e-14 |
975 |
Erismodegib |
LSM-4938 |
SMO |
10uM |
6h |
LINCSCP_13488 |
LINCSCP_13488 |
H1299 |
| -0.235372 |
9.701234e-14 |
975 |
BAS 09531330 |
LSM-32192 |
|
0.5uM |
24h |
LINCSCP_222160 |
LINCSCP_222160 |
HL60 |
| 0.235322 |
9.823292e-14 |
975 |
Tretinoin |
LSM-42854 |
RARA|RARB|RARG|RORB |
0.5uM |
24h |
LINCSCP_24143 |
LINCSCP_24143 |
HL60 |
| -0.235302 |
9.871947e-14 |
975 |
BRD-K77793090 |
LSM-13185 |
|
10uM |
24h |
LINCSCP_9080 |
LINCSCP_9080 |
A549 |
| 0.235298 |
9.879692e-14 |
975 |
BRD-K46666779 |
LSM-15075 |
|
3uM |
24h |
LINCSCP_253946 |
LINCSCP_253946 |
MCF7 |
| -0.235281 |
9.922191e-14 |
975 |
AZD-5438 |
LSM-1159 |
CDK1|CDK10|CDK11B|CDK12|CDK13|CDK14|CDK15|CDK16|CDK17|CDK18|CDK19|CDK2|CDK20|CDK3|CDK4|CDK5|CDK6|CDK7|CDK8|CDK9 |
1.11uM |
24h |
LINCSCP_111741 |
LINCSCP_111741 |
HEPG2 |
| -0.235246 |
1.000744e-13 |
975 |
1-(2,6-Dichlorobenzylideneamino)guanidine |
LSM-3266 |
|
10uM |
24h |
LINCSCP_42914 |
LINCSCP_42914 |
NPC |
| 0.235212 |
1.009205e-13 |
975 |
ML179 |
LSM-3734 |
|
10uM |
24h |
LINCSCP_57572 |
LINCSCP_57572 |
VCAP |
| -0.235189 |
1.014981e-13 |
975 |
Disulfiram |
LSM-5467 |
ALDH2 |
0.37uM |
24h |
LINCSCP_71828 |
LINCSCP_71828 |
A375 |
| -0.235158 |
1.022646e-13 |
975 |
Ciglitazone |
LSM-1911 |
PPARG |
10uM |
24h |
LINCSCP_42817 |
LINCSCP_42817 |
NPC |
| 0.235146 |
1.025630e-13 |
975 |
BRD-K03515977 |
LSM-8651 |
|
5uM |
24h |
LINCSCP_63964 |
LINCSCP_63964 |
VCAP |
| -0.235145 |
1.026015e-13 |
975 |
BI-2536 |
LSM-1041 |
PLK1 |
0.12uM |
24h |
LINCSCP_81440 |
LINCSCP_81440 |
A549 |
| 0.235121 |
1.032069e-13 |
975 |
CHEMBL1619263 |
LSM-4840 |
|
10uM |
6h |
LINCSCP_16236 |
LINCSCP_16236 |
HA1E |
| 0.235096 |
1.038430e-13 |
975 |
ZINC00164494 |
LSM-4660 |
|
10uM |
6h |
LINCSCP_16324 |
LINCSCP_16324 |
HA1E |
| -0.235077 |
1.043350e-13 |
975 |
BAY 61-3606 |
LSM-1167 |
SYK |
1.11uM |
24h |
LINCSCP_82580 |
LINCSCP_82580 |
A549 |
| -0.235065 |
1.046301e-13 |
975 |
BRD-K42125900-001-01-9 |
LSM-5535 |
TUBB |
10uM |
6h |
LINCSCP_32332 |
LINCSCP_32332 |
MCF7 |
| 0.23506 |
1.047628e-13 |
975 |
Imatinib |
LSM-1023 |
ABL1|BCR|CSF1R|KIT|PDGFRA|PDGFRB |
1.11uM |
24h |
LINCSCP_113261 |
LINCSCP_113261 |
HME1 |
| -0.235051 |
1.050083e-13 |
975 |
Promazine |
LSM-2137 |
CHRM5|DRD2|DRD3|DRD4|HTR2A |
10uM |
24h |
LINCSCP_52841 |
LINCSCP_52841 |
SKB |
| -0.235019 |
1.058325e-13 |
975 |
JLK-6 |
LSM-2489 |
PSEN1 |
10uM |
24h |
LINCSCP_44209 |
LINCSCP_44209 |
PC3 |
| 0.235017 |
1.058776e-13 |
975 |
ST021200 |
LSM-4601 |
|
10uM |
6h |
LINCSCP_4755 |
LINCSCP_4755 |
A549 |
| 0.235011 |
1.060490e-13 |
975 |
BAS 00631343 |
LSM-6284 |
|
10uM |
6h |
LINCSCP_51245 |
LINCSCP_51245 |
RMUGS |
| 0.235009 |
1.061036e-13 |
975 |
Tezampanel |
LSM-45407 |
|
0.12uM |
24h |
LINCSCP_74199 |
LINCSCP_74199 |
A375 |
| 0.234946 |
1.077618e-13 |
975 |
BRD-K21528100 |
LSM-9734 |
|
5uM |
24h |
LINCSCP_61747 |
LINCSCP_61747 |
VCAP |
| 0.234943 |
1.078383e-13 |
975 |
Alaproclate |
LSM-1333 |
SLC6A4 |
0.37uM |
24h |
LINCSCP_74485 |
LINCSCP_74485 |
A375 |
| -0.234939 |
1.079272e-13 |
975 |
CHEMBL1270811 |
LSM-2573 |
|
10uM |
6h |
LINCSCP_178205 |
LINCSCP_178205 |
A375 |
| 0.23493 |
1.081765e-13 |
975 |
Nilotinib |
LSM-1099 |
ABL1|BCR|KIT |
0.04uM |
24h |
LINCSCP_81315 |
LINCSCP_81315 |
A549 |
| -0.234905 |
1.088433e-13 |
975 |
BRN 1549781 |
LSM-4461 |
|
10uM |
24h |
LINCSCP_33805 |
LINCSCP_33805 |
MCF7 |
| -0.234782 |
1.121997e-13 |
975 |
NSC 663284 |
LSM-2042 |
CDC25A|CDC25B |
10uM |
6h |
LINCSCP_221504 |
LINCSCP_221504 |
HEPG2 |
| -0.234772 |
1.124677e-13 |
975 |
PNU-74654 |
LSM-44945 |
CTNNB1|TCF4 |
80uM |
24h |
LINCSCP_30530 |
LINCSCP_30530 |
MCF7 |
| 0.234769 |
1.125470e-13 |
975 |
Karakoline |
LSM-1556 |
|
10uM |
24h |
LINCSCP_25227 |
LINCSCP_25227 |
HT29 |
| -0.234752 |
1.130274e-13 |
975 |
Dolastatin 10 |
LSM-45943 |
|
3.33uM |
24h |
LINCSCP_143052 |
LINCSCP_143052 |
MCF7 |
| -0.234743 |
1.132710e-13 |
975 |
KW-2449 |
LSM-42803 |
ABL1|AURKA|AURKB|FLT3 |
10uM |
24h |
LINCSCP_116983 |
LINCSCP_116983 |
HT29 |
| 0.234735 |
1.134906e-13 |
975 |
BRD-K76904146 |
LSM-13136 |
|
5uM |
24h |
LINCSCP_62319 |
LINCSCP_62319 |
VCAP |
| -0.234733 |
1.135360e-13 |
975 |
SB-216763 |
LSM-1161 |
GSK3B |
10uM |
6h |
LINCSCP_13539 |
LINCSCP_13539 |
H1299 |
| -0.234704 |
1.143506e-13 |
975 |
GSK-923295 |
LSM-45692 |
|
3.33uM |
24h |
LINCSCP_137221 |
LINCSCP_137221 |
MCF7 |
| -0.234641 |
1.161453e-13 |
975 |
Triazine Scaffold, 51 |
LSM-3296 |
|
10uM |
6h |
LINCSCP_20012 |
LINCSCP_20012 |
HCC515 |
| 0.234612 |
1.169710e-13 |
975 |
Crizotinib |
LSM-1027 |
ALK|MET |
0.37uM |
24h |
LINCSCP_81026 |
LINCSCP_81026 |
A549 |
| -0.234603 |
1.172225e-13 |
975 |
AKT Inhibitor VIII |
LSM-1035 |
AKT1|AKT2 |
10uM |
24h |
LINCSCP_51289 |
LINCSCP_51289 |
SKBR3 |
| 0.234586 |
1.177150e-13 |
975 |
6,2'-Dimethoxyflavone |
LSM-4621 |
|
10uM |
6h |
LINCSCP_33765 |
LINCSCP_33765 |
MCF7 |
| 0.234571 |
1.181532e-13 |
975 |
BRD-K44681861 |
LSM-11145 |
|
5uM |
24h |
LINCSCP_61457 |
LINCSCP_61457 |
VCAP |
| -0.234562 |
1.184197e-13 |
975 |
BRD-K70697816 |
LSM-41120 |
|
10uM |
24h |
LINCSCP_186615 |
LINCSCP_186615 |
A375 |
| -0.234544 |
1.189328e-13 |
975 |
SPECTRUM_000011 |
LSM-1767 |
|
3.33uM |
24h |
LINCSCP_126167 |
LINCSCP_126167 |
HT29 |
| -0.234535 |
1.191995e-13 |
975 |
CHEMBL1472453 |
LSM-2683 |
|
10uM |
6h |
LINCSCP_225377 |
LINCSCP_225377 |
HT29 |
| 0.234519 |
1.196685e-13 |
975 |
CHEMBL552425 |
LSM-1003 |
DDR1 |
0.04uM |
24h |
LINCSCP_133279 |
LINCSCP_133279 |
MCF7 |
| -0.234511 |
1.199038e-13 |
975 |
MLS002264363 |
LSM-2417 |
|
10uM |
24h |
LINCSCP_45679 |
LINCSCP_45679 |
PC3 |
| -0.234501 |
1.201963e-13 |
975 |
Alprenolol |
LSM-1238 |
ADRB1|ADRB2 |
10uM |
24h |
LINCSCP_47442 |
LINCSCP_47442 |
PC3 |
| 0.234429 |
1.223637e-13 |
975 |
AC1N92C7 |
LSM-1822 |
EDNRA |
10uM |
24h |
LINCSCP_241042 |
LINCSCP_241042 |
MCF7 |
| -0.234413 |
1.228229e-13 |
975 |
CHEMBL585951 |
LSM-36386 |
MAPK8 |
0.04uM |
3h |
LINCSCP_86393 |
LINCSCP_86393 |
BT20 |
| -0.234404 |
1.230903e-13 |
975 |
Colchicine |
LSM-5199 |
TUBA1A|TUBA1B|TUBA1C|TUBA3E|TUBA4A|TUBB|TUBB1|TUBB2A|TUBB2B|TUBB3|TUBB4A|TUBB4B|TUBB6|TUBB8 |
0.5uM |
24h |
LINCSCP_37616 |
LINCSCP_37616 |
MCF7 |
| 0.234362 |
1.243665e-13 |
975 |
Voglibose |
LSM-45566 |
|
10uM |
24h |
LINCSCP_76242 |
LINCSCP_76242 |
A375 |
| -0.234355 |
1.246049e-13 |
975 |
BAY 87-2243 |
LSM-45786 |
|
0.04uM |
24h |
LINCSCP_96994 |
LINCSCP_96994 |
HA1E |
| -0.234328 |
1.254177e-13 |
975 |
BRD-K22673215 |
LSM-7143 |
|
5uM |
24h |
LINCSCP_60148 |
LINCSCP_60148 |
VCAP |
| 0.234327 |
1.254509e-13 |
975 |
BRD-K36701739 |
LSM-10648 |
|
5uM |
24h |
LINCSCP_63993 |
LINCSCP_63993 |
VCAP |
| -0.234305 |
1.261305e-13 |
975 |
Ethacrynic acid |
LSM-3420 |
SLC12A1 |
10uM |
6h |
LINCSCP_4402 |
LINCSCP_4402 |
A549 |
| 0.23424 |
1.281656e-13 |
975 |
MLS001030493 |
LSM-43128 |
|
10uM |
6h |
LINCSCP_20672 |
LINCSCP_20672 |
HCC515 |
| -0.234237 |
1.282568e-13 |
975 |
Ginsenoside RC |
LSM-1713 |
|
10uM |
24h |
LINCSCP_264542 |
LINCSCP_264542 |
PC3 |
| -0.234228 |
1.285506e-13 |
975 |
Skiii |
LSM-2462 |
SPHK1 |
40uM |
6h |
LINCSCP_51118 |
LINCSCP_51118 |
RMUGS |
| 0.234198 |
1.294852e-13 |
975 |
Dactolisib |
LSM-4255 |
MTOR|PIK3CA|PIK3CB|PIK3CD|PIK3CG|PIK3R1|PIK3R2|PIK3R3|PIK3R5 |
0.12uM |
3h |
LINCSCP_132472 |
LINCSCP_132472 |
MCF7 |
| -0.234165 |
1.305356e-13 |
975 |
UNII-884KT10YB7 |
LSM-2298 |
HRH2 |
10uM |
24h |
LINCSCP_243452 |
LINCSCP_243452 |
MCF7 |
| -0.234133 |
1.315757e-13 |
975 |
Ipratropium |
LSM-1497 |
CHRM1|CHRM2|CHRM3|CHRM4 |
10uM |
6h |
LINCSCP_420 |
LINCSCP_420 |
A375 |
| -0.234132 |
1.315833e-13 |
975 |
BRD-K93158953 |
LSM-42330 |
|
5uM |
24h |
LINCSCP_64338 |
LINCSCP_64338 |
VCAP |
| 0.234107 |
1.324055e-13 |
975 |
SR 33805 oxalate |
LSM-45933 |
|
0.04uM |
24h |
LINCSCP_75553 |
LINCSCP_75553 |
A375 |
| 0.234051 |
1.342222e-13 |
975 |
Imatinib |
LSM-1023 |
ABL1|BCR|CSF1R|KIT|PDGFRA|PDGFRB |
0.04uM |
24h |
LINCSCP_88210 |
LINCSCP_88210 |
HA1E |
| 0.234044 |
1.344520e-13 |
975 |
Emtricitabine |
LSM-45730 |
|
0.12uM |
24h |
LINCSCP_139870 |
LINCSCP_139870 |
MCF7 |
| 0.233917 |
1.387239e-13 |
975 |
MLS000589843 |
LSM-43120 |
|
0.001uM |
6h |
LINCSCP_42083 |
LINCSCP_42083 |
NOMO1 |
| 0.233894 |
1.394944e-13 |
975 |
BRD-K58191509 |
LSM-40452 |
|
10uM |
24h |
LINCSCP_7864 |
LINCSCP_7864 |
A549 |
| 0.233882 |
1.398953e-13 |
975 |
CHEMBL3186940 |
LSM-15140 |
|
10uM |
6h |
LINCSCP_49140 |
LINCSCP_49140 |
PC3 |
| 0.233857 |
1.407617e-13 |
975 |
Levocabastine |
LSM-2731 |
HRH1|NTSR2 |
10uM |
24h |
LINCSCP_241103 |
LINCSCP_241103 |
MCF7 |
| -0.233802 |
1.426938e-13 |
975 |
5-Bromo-n-(6-butyl-1,3-benzothiazol-2-yl)furan-2-carboxamide |
LSM-2765 |
|
10uM |
6h |
LINCSCP_26083 |
LINCSCP_26083 |
HT29 |
| -0.233775 |
1.436140e-13 |
975 |
Treprostinil |
LSM-5119 |
PTGIR |
10uM |
24h |
LINCSCP_239376 |
LINCSCP_239376 |
MCF7 |
| -0.233748 |
1.445605e-13 |
975 |
BMS-536924 |
LSM-1210 |
IGF1R |
10uM |
6h |
LINCSCP_9599 |
LINCSCP_9599 |
A549 |
| -0.233704 |
1.461378e-13 |
975 |
KW-2449 |
LSM-42803 |
ABL1|AURKA|AURKB|FLT3 |
10uM |
24h |
LINCSCP_90632 |
LINCSCP_90632 |
HA1E |
| 0.233691 |
1.466157e-13 |
975 |
BRD-K38493271 |
LSM-10757 |
|
5uM |
6h |
LINCSCP_61337 |
LINCSCP_61337 |
VCAP |
| 0.233688 |
1.466981e-13 |
975 |
CHEMBL1327417 |
LSM-4729 |
|
10uM |
24h |
LINCSCP_270341 |
LINCSCP_270341 |
PC3 |
| 0.233664 |
1.475961e-13 |
975 |
CHEMBL2133926 |
LSM-6788 |
|
0.5uM |
24h |
LINCSCP_37866 |
LINCSCP_37866 |
MCF7 |
| -0.233642 |
1.483880e-13 |
975 |
NaCl |
LSM-46007 |
|
0.1uM |
24h |
LINCSCP_263923 |
LINCSCP_263923 |
NPC |
| -0.233621 |
1.491556e-13 |
975 |
Lenvatinib (E7080) |
LSM-45581 |
FLT1|FLT4|KDR |
1.11uM |
24h |
LINCSCP_93740 |
LINCSCP_93740 |
HA1E |
| -0.233617 |
1.492908e-13 |
975 |
AS-605240 |
LSM-42784 |
PIK3CG |
10uM |
24h |
LINCSCP_24298 |
LINCSCP_24298 |
HS578T |
| -0.233601 |
1.498672e-13 |
975 |
Purmorphamine |
LSM-3649 |
SMO |
10uM |
24h |
LINCSCP_44057 |
LINCSCP_44057 |
PC3 |
| -0.233592 |
1.502153e-13 |
975 |
4-(3-Ethyl[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl)aniline |
LSM-4945 |
|
10uM |
6h |
LINCSCP_51219 |
LINCSCP_51219 |
RMUGS |
| -0.233509 |
1.532631e-13 |
975 |
Dacomitinib |
LSM-42808 |
EGFR|ERBB2|ERBB3|ERBB4 |
10uM |
24h |
LINCSCP_133388 |
LINCSCP_133388 |
MCF7 |
| -0.233416 |
1.568175e-13 |
975 |
MLS002264514 |
LSM-42882 |
|
10uM |
24h |
LINCSCP_57521 |
LINCSCP_57521 |
VCAP |
| 0.233388 |
1.578799e-13 |
975 |
Gemfibrozil |
LSM-2227 |
CYP2C8|LPL|PPARA |
3.33uM |
24h |
LINCSCP_72723 |
LINCSCP_72723 |
A375 |
| 0.233388 |
1.578876e-13 |
975 |
Felbamate |
LSM-4232 |
GRIN1|GRIN2A|GRIN2B|GRIN2C|GRIN2D|GRIN3A|GRIN3B |
10uM |
24h |
LINCSCP_73515 |
LINCSCP_73515 |
A375 |
| -0.23338 |
1.581853e-13 |
975 |
AT-7519 |
LSM-1004 |
CDK1|CDK10|CDK11B|CDK12|CDK13|CDK14|CDK15|CDK16|CDK17|CDK18|CDK19|CDK2|CDK20|CDK3|CDK4|CDK5|CDK6|CDK7|CDK8|CDK9 |
3.33uM |
24h |
LINCSCP_137905 |
LINCSCP_137905 |
MCF7 |
| 0.233365 |
1.587523e-13 |
975 |
Cobalt (Ii) Chloride |
LSM-5958 |
HIF1A |
10uM |
6h |
LINCSCP_59615 |
LINCSCP_59615 |
VCAP |
| -0.233361 |
1.589262e-13 |
975 |
Wortmannin |
LSM-3947 |
PIK3CA|PIK3CG|PLK1 |
10uM |
24h |
LINCSCP_68199 |
LINCSCP_68199 |
SKB |
| 0.233206 |
1.650354e-13 |
975 |
THZ-2-98-01 |
LSM-44946 |
|
0.12uM |
24h |
LINCSCP_88168 |
LINCSCP_88168 |
HA1E |
| -0.233167 |
1.666463e-13 |
975 |
Fluphenazine |
LSM-3226 |
DRD1|DRD2 |
10uM |
24h |
LINCSCP_349 |
LINCSCP_349 |
A375 |
| 0.233093 |
1.696586e-13 |
975 |
Cyclohexanecarboxamide, 4-(1-aminoethyl)-n-4-pyridinyl-, trans- |
LSM-1177 |
ROCK1|ROCK2 |
0.37uM |
24h |
LINCSCP_82333 |
LINCSCP_82333 |
A549 |
| -0.233085 |
1.700036e-13 |
975 |
BRD-K84023371 |
LSM-15058 |
|
0.01uM |
6h |
LINCSCP_65189 |
LINCSCP_65189 |
VCAP |
| -0.233069 |
1.706492e-13 |
975 |
PF-03758309 |
LSM-4254 |
PAK4 |
10uM |
24h |
LINCSCP_139404 |
LINCSCP_139404 |
MCF7 |
| 0.233061 |
1.709950e-13 |
975 |
BRD-K31812348 |
LSM-10357 |
|
5uM |
24h |
LINCSCP_61762 |
LINCSCP_61762 |
VCAP |
| -0.233037 |
1.719902e-13 |
975 |
4449-51-8 |
LSM-4304 |
SMO |
10uM |
24h |
LINCSCP_46397 |
LINCSCP_46397 |
PC3 |
| 0.233029 |
1.723208e-13 |
975 |
Tosufloxacin |
LSM-5050 |
|
10uM |
6h |
LINCSCP_46135 |
LINCSCP_46135 |
PC3 |
| 0.232993 |
1.738753e-13 |
975 |
BS-181 |
LSM-6305 |
|
0.04uM |
24h |
LINCSCP_84357 |
LINCSCP_84357 |
ASC |
| 0.232987 |
1.741201e-13 |
975 |
(3-Isopropoxyphenyl)(1-((5-methyl-1-propyl-1H-pyrazol-4-yl)methyl)piperidin-3-yl)methanone |
LSM-1323 |
|
10uM |
6h |
LINCSCP_17547 |
LINCSCP_17547 |
HCC15 |
| -0.232968 |
1.749076e-13 |
975 |
Seliciclib |
LSM-1001 |
CDK1|CDK2|CDK5|CDK7|CDK9 |
10uM |
6h |
LINCSCP_39162 |
LINCSCP_39162 |
MDAMB231 |
| -0.232968 |
1.749398e-13 |
975 |
INOSITOL |
LSM-45237 |
|
3.33uM |
24h |
LINCSCP_106852 |
LINCSCP_106852 |
HELA |
| -0.232914 |
1.772486e-13 |
975 |
Bardoxolone Methyl |
LSM-45471 |
IKBKB|KEAP1|NFE2L2|PPARG |
10uM |
24h |
LINCSCP_72243 |
LINCSCP_72243 |
A375 |
| 0.232819 |
1.813712e-13 |
975 |
SPECTRUM_001645 |
LSM-1721 |
OPRD1|OPRK1|OPRM1 |
3uM |
24h |
LINCSCP_37212 |
LINCSCP_37212 |
MCF7 |
| -0.232793 |
1.825400e-13 |
975 |
Zardaverine |
LSM-2833 |
PDE4D |
10uM |
24h |
LINCSCP_46090 |
LINCSCP_46090 |
PC3 |
| -0.232786 |
1.828466e-13 |
975 |
Alvespimycin |
LSM-43241 |
HSP90AA1 |
10uM |
24h |
LINCSCP_32556 |
LINCSCP_32556 |
MCF7 |
| 0.232782 |
1.830353e-13 |
975 |
BRD-K20876879 |
LSM-9701 |
|
5uM |
6h |
LINCSCP_63569 |
LINCSCP_63569 |
VCAP |
| -0.232777 |
1.832542e-13 |
975 |
IN1152 |
LSM-2575 |
|
10uM |
24h |
LINCSCP_50196 |
LINCSCP_50196 |
PHH |
| 0.232754 |
1.842953e-13 |
975 |
BRD-K51556300-001-01-9 |
LSM-40116 |
|
0.1uM |
24h |
LINCSCP_261249 |
LINCSCP_261249 |
NOMO1 |
| 0.232734 |
1.852082e-13 |
975 |
rifampicin |
|
|
0.37uM |
3h |
LINCSCP_131835 |
LINCSCP_131835 |
MCF10A |
| 0.232714 |
1.860836e-13 |
975 |
rifampicin |
|
|
1.11uM |
3h |
LINCSCP_130424 |
LINCSCP_130424 |
LNCAP |
| -0.232663 |
1.884252e-13 |
975 |
K784-3187 |
LSM-45465 |
ESR2 |
1.11uM |
24h |
LINCSCP_78180 |
LINCSCP_78180 |
A375 |
| 0.232652 |
1.889113e-13 |
975 |
Hydroxyprogesterone Caproate |
LSM-4900 |
AR|ESR1|ESR2|NR1H4|NR1I2|NR3C1|PGR |
0.37uM |
24h |
LINCSCP_71310 |
LINCSCP_71310 |
A375 |
| 0.232644 |
1.893005e-13 |
975 |
BRD-K18351060 |
LSM-9533 |
|
5uM |
24h |
LINCSCP_63670 |
LINCSCP_63670 |
VCAP |
| -0.232624 |
1.901955e-13 |
975 |
KW-2449 |
LSM-42803 |
ABL1|AURKA|AURKB|FLT3 |
10uM |
24h |
LINCSCP_113797 |
LINCSCP_113797 |
HME1 |
| -0.232564 |
1.930040e-13 |
975 |
1-(4-Amino-1,2,5-oxadiazol-3-yl)-5-(azepan-1-ylmethyl)-n-[(2-ethoxyphenyl)methylideneamino]triazole-4-carboxamide |
LSM-6604 |
|
10uM |
24h |
LINCSCP_33868 |
LINCSCP_33868 |
MCF7 |
| -0.232494 |
1.963058e-13 |
975 |
GNF-PF-5186 |
LSM-4449 |
|
10uM |
24h |
LINCSCP_52194 |
LINCSCP_52194 |
SKB |
| 0.232484 |
1.967905e-13 |
975 |
ST50885743 |
LSM-4113 |
|
10uM |
24h |
LINCSCP_267761 |
LINCSCP_267761 |
PC3 |
| -0.232469 |
1.975060e-13 |
975 |
Dolastatin 10 |
LSM-45943 |
|
0.37uM |
24h |
LINCSCP_143054 |
LINCSCP_143054 |
MCF7 |
| 0.232466 |
1.976765e-13 |
975 |
N-(3-Fluoro-4-((7-methoxyquinolin-4-yl)oxy)phenyl)-1-(2-hydroxy-2-methylpropyl)-5-methyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazole-4-carboxamide |
LSM-1113 |
|
10uM |
6h |
LINCSCP_256193 |
LINCSCP_256193 |
MDAMB231 |
| -0.232449 |
1.984669e-13 |
975 |
Chlormezanone |
LSM-4356 |
GABRA1 |
10uM |
24h |
LINCSCP_47449 |
LINCSCP_47449 |
PC3 |
| -0.232444 |
1.987325e-13 |
975 |
ZINC03977910 |
LSM-5391 |
NR3C1 |
10uM |
6h |
LINCSCP_34368 |
LINCSCP_34368 |
MCF7 |
| 0.232424 |
1.997069e-13 |
975 |
BRD-K00196194 |
LSM-8435 |
|
5uM |
24h |
LINCSCP_60830 |
LINCSCP_60830 |
VCAP |
| 0.232403 |
2.007124e-13 |
975 |
Hydroxyprogesterone Caproate |
LSM-4900 |
AR|ESR1|ESR2|NR1H4|NR1I2|NR3C1|PGR |
1.11uM |
24h |
LINCSCP_71309 |
LINCSCP_71309 |
A375 |
| -0.232403 |
2.007168e-13 |
975 |
Zopiclone |
LSM-4408 |
GABRA1 |
10uM |
24h |
LINCSCP_243878 |
LINCSCP_243878 |
MCF7 |
| -0.232352 |
2.032498e-13 |
975 |
BRD-K22912836 |
LSM-38513 |
|
10uM |
24h |
LINCSCP_249954 |
LINCSCP_249954 |
MCF7 |
| -0.232338 |
2.039235e-13 |
975 |
Fenbendazole |
LSM-3134 |
TUBB |
10uM |
24h |
LINCSCP_38199 |
LINCSCP_38199 |
MCF7 |
| -0.232281 |
2.067773e-13 |
975 |
Ambelline |
LSM-1309 |
|
10uM |
6h |
LINCSCP_404 |
LINCSCP_404 |
A375 |
| -0.23218 |
2.118826e-13 |
975 |
SCHEMBL10015911 |
LSM-43159 |
PTGFR |
10uM |
24h |
LINCSCP_271974 |
LINCSCP_271974 |
PC3 |
| -0.232179 |
2.119491e-13 |
975 |
BRD-A41986761 |
LSM-45957 |
|
3.33uM |
24h |
LINCSCP_135195 |
LINCSCP_135195 |
MCF7 |
| -0.232107 |
2.156774e-13 |
975 |
ON-01910 |
LSM-43198 |
CDK1|FLT1|FYN|PDGFRA|PLK1|PLK2|SRC |
10uM |
24h |
LINCSCP_32168 |
LINCSCP_32168 |
MCF7 |
| -0.232099 |
2.161344e-13 |
975 |
MLS002264455 |
LSM-3236 |
|
10uM |
24h |
LINCSCP_31178 |
LINCSCP_31178 |
MCF7 |
| -0.232073 |
2.175024e-13 |
975 |
BRD-K65968856 |
LSM-12452 |
|
10uM |
24h |
LINCSCP_3606 |
LINCSCP_3606 |
A375 |
| -0.232052 |
2.186146e-13 |
975 |
ZINC00399124 |
LSM-5611 |
|
10uM |
24h |
LINCSCP_272053 |
LINCSCP_272053 |
PC3 |
| -0.232047 |
2.188580e-13 |
975 |
Thioguanosine |
LSM-5832 |
|
0.37uM |
24h |
LINCSCP_161549 |
LINCSCP_161549 |
PC3 |
| 0.232044 |
2.190336e-13 |
975 |
ZINC00969081 |
LSM-3555 |
|
10uM |
6h |
LINCSCP_220128 |
LINCSCP_220128 |
HEPG2 |
| -0.232016 |
2.205218e-13 |
975 |
MLS-0435526.0001 |
LSM-4881 |
|
10uM |
24h |
LINCSCP_32523 |
LINCSCP_32523 |
MCF7 |
| -0.231996 |
2.215940e-13 |
975 |
Batimastat |
LSM-6276 |
|
1.11uM |
24h |
LINCSCP_71021 |
LINCSCP_71021 |
A375 |
| -0.231971 |
2.229550e-13 |
975 |
Quinoxaline1 |
LSM-2675 |
CDK1|CDK5|GSK3A |
10uM |
24h |
LINCSCP_44030 |
LINCSCP_44030 |
PC3 |
| 0.231963 |
2.233629e-13 |
975 |
SB-366791 |
LSM-3316 |
TRPV1 |
10uM |
24h |
LINCSCP_33102 |
LINCSCP_33102 |
MCF7 |
| -0.231958 |
2.236642e-13 |
975 |
altrenogest |
LSM-45498 |
|
10uM |
24h |
LINCSCP_139854 |
LINCSCP_139854 |
MCF7 |
| 0.231954 |
2.238306e-13 |
975 |
Maprotiline |
LSM-2043 |
SLC6A2 |
0.37uM |
24h |
LINCSCP_72390 |
LINCSCP_72390 |
A375 |
| 0.231927 |
2.253405e-13 |
975 |
KO143 |
LSM-6260 |
ABCG2 |
40uM |
6h |
LINCSCP_13548 |
LINCSCP_13548 |
H1299 |
| 0.231919 |
2.257745e-13 |
975 |
Bambuterol |
LSM-4346 |
ADRB2 |
10uM |
6h |
LINCSCP_34331 |
LINCSCP_34331 |
MCF7 |
| -0.231883 |
2.277596e-13 |
975 |
KX2-391 |
LSM-45890 |
SRC |
1.11uM |
24h |
LINCSCP_137498 |
LINCSCP_137498 |
MCF7 |
| 0.231861 |
2.289682e-13 |
975 |
Gefitinib |
LSM-1098 |
EGFR |
0.37uM |
24h |
LINCSCP_145577 |
LINCSCP_145577 |
MDAMB231 |
| 0.23186 |
2.290004e-13 |
975 |
BRD-K63828515 |
LSM-14887 |
|
5uM |
24h |
LINCSCP_64206 |
LINCSCP_64206 |
VCAP |
| -0.231848 |
2.296859e-13 |
975 |
BRD-K68690198 |
LSM-41003 |
|
10uM |
24h |
LINCSCP_59258 |
LINCSCP_59258 |
VCAP |
| -0.231839 |
2.301835e-13 |
975 |
Valpropylhydroxamic acid |
LSM-37248 |
|
10uM |
24h |
LINCSCP_263916 |
LINCSCP_263916 |
NPC |
| -0.23182 |
2.312365e-13 |
975 |
BSPBIO_000981 |
LSM-43126 |
ACTA1 |
10uM |
6h |
LINCSCP_32323 |
LINCSCP_32323 |
MCF7 |
| -0.231805 |
2.321076e-13 |
975 |
Quizartinib |
LSM-1037 |
CSF1R|FLT3|KIT|PDGFRA|PDGFRB|RET |
0.04uM |
24h |
LINCSCP_146276 |
LINCSCP_146276 |
MNEU.E |
| 0.231786 |
2.331464e-13 |
975 |
Ziprasidone |
LSM-5433 |
DRD2|HRH1|HTR1A|HTR1B|HTR1D|HTR1E|HTR2A|HTR2C|HTR7 |
0.37uM |
24h |
LINCSCP_71274 |
LINCSCP_71274 |
A375 |
| -0.231754 |
2.349604e-13 |
975 |
Dequalinium |
LSM-5846 |
|
0.37uM |
24h |
LINCSCP_79848 |
LINCSCP_79848 |
A375 |
| -0.231726 |
2.365774e-13 |
975 |
Hexylresorcinol |
LSM-4250 |
|
10uM |
24h |
LINCSCP_266935 |
LINCSCP_266935 |
PC3 |
| 0.231722 |
2.368427e-13 |
975 |
CHEMBL2361406 |
LSM-41857 |
|
1uM |
24h |
LINCSCP_38242 |
LINCSCP_38242 |
MCF7 |
| -0.231699 |
2.381519e-13 |
975 |
GW843682X |
LSM-1014 |
PLK1|PLK3 |
10uM |
24h |
LINCSCP_30660 |
LINCSCP_30660 |
MCF7 |
| -0.231692 |
2.385227e-13 |
975 |
T-0156 |
LSM-3414 |
PDE5A |
1uM |
24h |
LINCSCP_38216 |
LINCSCP_38216 |
MCF7 |
| -0.231655 |
2.407184e-13 |
975 |
KUC105208 KUC105208N |
LSM-45316 |
|
1uM |
24h |
LINCSCP_222179 |
LINCSCP_222179 |
HL60 |
| 0.23163 |
2.421572e-13 |
975 |
NSC119236 |
LSM-4575 |
|
20uM |
6h |
LINCSCP_57103 |
LINCSCP_57103 |
VCAP |
| -0.23161 |
2.433087e-13 |
975 |
Cycloserine |
LSM-5932 |
|
10uM |
24h |
LINCSCP_272127 |
LINCSCP_272127 |
PC3 |
| 0.231605 |
2.436253e-13 |
975 |
6-Methoxy-harmalan |
LSM-3224 |
|
10uM |
24h |
LINCSCP_33099 |
LINCSCP_33099 |
MCF7 |
| 0.231603 |
2.437270e-13 |
975 |
BRD-K53467073 |
LSM-11689 |
|
5uM |
24h |
LINCSCP_61619 |
LINCSCP_61619 |
VCAP |
| -0.231599 |
2.440067e-13 |
975 |
N-(6-Butyl-1,3-benzothiazol-2-yl)thiophene-2-carboxamide |
LSM-4011 |
|
10uM |
24h |
LINCSCP_1439 |
LINCSCP_1439 |
A375 |
| 0.231591 |
2.444582e-13 |
975 |
Meclofenamic acid |
LSM-3108 |
ALOX5|PTGS1|PTGS2 |
10uM |
24h |
LINCSCP_141311 |
LINCSCP_141311 |
MCF7 |
| 0.231551 |
2.468609e-13 |
975 |
SA-1456625 |
LSM-41910 |
|
1uM |
6h |
LINCSCP_254552 |
LINCSCP_254552 |
MCF7 |
| -0.231518 |
2.488207e-13 |
975 |
Podofilox |
LSM-3055 |
|
0.12uM |
24h |
LINCSCP_141627 |
LINCSCP_141627 |
MCF7 |
| -0.231469 |
2.518032e-13 |
975 |
AZD 1480 |
LSM-1140 |
JAK1|JAK2 |
10uM |
24h |
LINCSCP_24656 |
LINCSCP_24656 |
HS578T |
| 0.231463 |
2.521572e-13 |
975 |
GW-5074 |
LSM-42779 |
RAF1 |
1uM |
24h |
LINCSCP_38938 |
LINCSCP_38938 |
MDAMB231 |
| -0.231443 |
2.533980e-13 |
975 |
CHEMDIV3_007370 |
LSM-4399 |
|
10uM |
24h |
LINCSCP_42224 |
LINCSCP_42224 |
NPC |
| 0.231424 |
2.545305e-13 |
975 |
BX 912 |
LSM-1055 |
PDK1|PDPK1 |
0.12uM |
3h |
LINCSCP_163389 |
LINCSCP_163389 |
SKBR3 |
| -0.23138 |
2.572933e-13 |
975 |
Immepip |
LSM-2567 |
HRH3 |
10uM |
24h |
LINCSCP_52869 |
LINCSCP_52869 |
SKB |
| 0.231367 |
2.580888e-13 |
975 |
SMR000200744 |
LSM-2679 |
|
10uM |
6h |
LINCSCP_5500 |
LINCSCP_5500 |
A549 |
| -0.231333 |
2.601883e-13 |
975 |
Capsazepine |
LSM-2983 |
TRPV1 |
10uM |
24h |
LINCSCP_284973 |
LINCSCP_284973 |
SKB |
| -0.231326 |
2.606294e-13 |
975 |
BRD-K63827443 |
LSM-12316 |
|
10uM |
24h |
LINCSCP_35348 |
LINCSCP_35348 |
MCF7 |
| 0.231268 |
2.643142e-13 |
975 |
CHEMBL566722 |
LSM-4073 |
|
10uM |
6h |
LINCSCP_45426 |
LINCSCP_45426 |
PC3 |
| -0.231258 |
2.649814e-13 |
975 |
BRD-K88008216 |
LSM-42071 |
|
10uM |
24h |
LINCSCP_33936 |
LINCSCP_33936 |
MCF7 |
| 0.231239 |
2.661715e-13 |
975 |
SCHEMBL3954849 |
LSM-5982 |
|
0.12uM |
24h |
LINCSCP_116167 |
LINCSCP_116167 |
HT29 |
| 0.231211 |
2.680282e-13 |
975 |
Sirolimus |
LSM-42783 |
FKBP1A|MTOR |
1uM |
24h |
LINCSCP_250731 |
LINCSCP_250731 |
MCF7 |
| 0.231185 |
2.697156e-13 |
975 |
Cinacalcet |
LSM-5815 |
CASR |
10uM |
6h |
LINCSCP_211817 |
LINCSCP_211817 |
HA1E |
| -0.231163 |
2.711518e-13 |
975 |
vincristine |
|
TUBB |
3uM |
24h |
LINCSCP_37615 |
LINCSCP_37615 |
MCF7 |
| 0.231147 |
2.721917e-13 |
975 |
BRL-15,572 |
LSM-1618 |
HTR1D |
10uM |
24h |
LINCSCP_262529 |
LINCSCP_262529 |
NPC |
| 0.231135 |
2.729566e-13 |
975 |
WHI-P97 |
LSM-1033 |
JAK3 |
10uM |
24h |
LINCSCP_87533 |
LINCSCP_87533 |
CD34 |
| -0.231108 |
2.747404e-13 |
975 |
CEP-701 |
LSM-45844 |
|
3.33uM |
24h |
LINCSCP_89447 |
LINCSCP_89447 |
HA1E |
| -0.231071 |
2.772177e-13 |
975 |
LY-294002 |
LSM-2597 |
MTOR|PIK3CA|PIK3CB|PIK3CD|PIK3CG|PLK1|PRKDC |
10uM |
24h |
LINCSCP_67506 |
LINCSCP_67506 |
MCF7 |
| -0.231065 |
2.776175e-13 |
975 |
CBDIVE_003036 |
LSM-4324 |
|
10uM |
24h |
LINCSCP_42217 |
LINCSCP_42217 |
NPC |
| -0.231044 |
2.790352e-13 |
975 |
BRD-K99692850 |
LSM-15174 |
|
10uM |
6h |
LINCSCP_65550 |
LINCSCP_65550 |
VCAP |
| -0.23104 |
2.793213e-13 |
975 |
Econazole |
LSM-1617 |
|
0.04uM |
24h |
LINCSCP_171775 |
LINCSCP_171775 |
YAPC |
| 0.230981 |
2.833436e-13 |
975 |
Benzbromarone |
LSM-2239 |
|
0.04uM |
24h |
LINCSCP_119719 |
LINCSCP_119719 |
HT29 |
| -0.230977 |
2.836144e-13 |
975 |
MLS003448162 |
LSM-3552 |
|
10uM |
24h |
LINCSCP_268206 |
LINCSCP_268206 |
PC3 |
| -0.230973 |
2.839066e-13 |
975 |
TWS 119 |
LSM-1111 |
GSK3B |
3.33uM |
24h |
LINCSCP_69226 |
LINCSCP_69226 |
A375 |
| 0.230971 |
2.839917e-13 |
975 |
BRD-K49907578 |
LSM-11460 |
|
5uM |
24h |
LINCSCP_62007 |
LINCSCP_62007 |
VCAP |
| -0.230926 |
2.871274e-13 |
975 |
Gliclazide |
LSM-5096 |
ABCC8 |
1.11uM |
24h |
LINCSCP_106498 |
LINCSCP_106498 |
HELA |
| -0.230914 |
2.879569e-13 |
975 |
CHEMBL3400874 |
LSM-42482 |
|
10uM |
6h |
LINCSCP_252540 |
LINCSCP_252540 |
MCF7 |
| -0.230882 |
2.901809e-13 |
975 |
Tetraidofluorescein |
LSM-2320 |
|
10uM |
6h |
LINCSCP_44632 |
LINCSCP_44632 |
PC3 |
| 0.230869 |
2.910929e-13 |
975 |
MAYBRIDGE4_003950 |
LSM-4735 |
|
10uM |
6h |
LINCSCP_17012 |
LINCSCP_17012 |
HA1E |
| 0.230832 |
2.937244e-13 |
975 |
Erlotinib |
LSM-1097 |
EGFR |
1.11uM |
3h |
LINCSCP_145211 |
LINCSCP_145211 |
MDAMB231 |
| -0.23083 |
2.938479e-13 |
975 |
CHEMBL2135649 |
LSM-42661 |
|
10uM |
6h |
LINCSCP_227811 |
LINCSCP_227811 |
HT29 |
| 0.230816 |
2.948453e-13 |
975 |
BRD-K78467731 |
LSM-13226 |
|
5uM |
24h |
LINCSCP_62041 |
LINCSCP_62041 |
VCAP |
| -0.230773 |
2.979370e-13 |
975 |
CGS-15943 |
LSM-3076 |
ADORA1|ADORA2A|ADORA2B |
10uM |
6h |
LINCSCP_67580 |
LINCSCP_67580 |
MCF7 |
| -0.230771 |
2.980338e-13 |
975 |
Morin |
LSM-36988 |
|
20uM |
24h |
LINCSCP_34743 |
LINCSCP_34743 |
MCF7 |
| 0.230771 |
2.980711e-13 |
975 |
TPCA-1 |
LSM-1136 |
IKBKB |
0.1uM |
24h |
LINCSCP_205067 |
LINCSCP_205067 |
BT20 |
| -0.230748 |
2.997538e-13 |
975 |
BRD-K17139610 |
LSM-9464 |
|
10uM |
24h |
LINCSCP_249729 |
LINCSCP_249729 |
MCF7 |
| -0.230727 |
3.012668e-13 |
975 |
Broad-Sai-560 |
LSM-45991 |
|
10uM |
24h |
LINCSCP_35538 |
LINCSCP_35538 |
MCF7 |
| -0.230712 |
3.023457e-13 |
975 |
Fenbendazole |
LSM-3134 |
TUBB |
0.5uM |
24h |
LINCSCP_38198 |
LINCSCP_38198 |
MCF7 |
| 0.230698 |
3.033858e-13 |
975 |
NU1025 |
LSM-4643 |
PARP1 |
10uM |
24h |
LINCSCP_30558 |
LINCSCP_30558 |
MCF7 |
| -0.230669 |
3.055239e-13 |
975 |
XAV 939 |
LSM-5303 |
TNKS|TNKS2 |
10uM |
6h |
LINCSCP_53439 |
LINCSCP_53439 |
SKMEL28 |
| -0.230584 |
3.118296e-13 |
975 |
Lexibulin |
LSM-6232 |
TUBA1A|TUBA1B|TUBA1C|TUBA3E|TUBA4A|TUBB|TUBB1|TUBB2A|TUBB2B|TUBB3|TUBB4A|TUBB4B|TUBB6|TUBB8 |
1uM |
24h |
LINCSCP_30515 |
LINCSCP_30515 |
MCF7 |
| 0.230582 |
3.120020e-13 |
975 |
L-690488 |
LSM-4703 |
IMPA1 |
10uM |
6h |
LINCSCP_261152 |
LINCSCP_261152 |
NOMO1 |
| -0.230581 |
3.120167e-13 |
975 |
13-Hydroxy-8,14,19-trimethoxy-4,10,12,16-tetramethyl-3,20,22-trioxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18-pentaen-9-yl carbamate |
LSM-42815 |
HSP90AA1 |
10uM |
6h |
LINCSCP_68439 |
LINCSCP_68439 |
VCAP |
| 0.23053 |
3.158831e-13 |
975 |
BRD-K12738359 |
LSM-9183 |
|
5uM |
24h |
LINCSCP_63341 |
LINCSCP_63341 |
VCAP |
| -0.23052 |
3.166440e-13 |
975 |
Sirolimus |
LSM-42783 |
FKBP1A|MTOR |
20uM |
48h |
LINCSCP_64527 |
LINCSCP_64527 |
VCAP |
| -0.230489 |
3.190760e-13 |
975 |
Eplerenone |
LSM-42771 |
NR3C2 |
10uM |
24h |
LINCSCP_154614 |
LINCSCP_154614 |
PC3 |
| -0.230476 |
3.200454e-13 |
975 |
Chelidonine |
LSM-2715 |
|
10uM |
24h |
LINCSCP_37680 |
LINCSCP_37680 |
MCF7 |
| 0.230471 |
3.204289e-13 |
975 |
Vorinostat |
LSM-3828 |
HDAC1|HDAC2|HDAC3|HDAC6|HDAC8 |
0.12uM |
24h |
LINCSCP_164680 |
LINCSCP_164680 |
SKL.C |
| 0.230469 |
3.205972e-13 |
975 |
Gefitinib |
LSM-1098 |
EGFR |
10uM |
3h |
LINCSCP_130368 |
LINCSCP_130368 |
LNCAP |
| -0.230448 |
3.222284e-13 |
975 |
Azacitidine |
LSM-5218 |
DNMT1|DNMT3A |
3.33uM |
24h |
LINCSCP_140148 |
LINCSCP_140148 |
MCF7 |
| 0.23043 |
3.235911e-13 |
975 |
Fcodpguefhccia-Uhfffaoysa-N |
LSM-42689 |
CASP3 |
10uM |
24h |
LINCSCP_30528 |
LINCSCP_30528 |
MCF7 |
| -0.230385 |
3.271485e-13 |
975 |
Tivozanib |
LSM-1005 |
FLT1|FLT4|KDR|KIT|PDGFRA|PDGFRB |
10uM |
24h |
LINCSCP_81757 |
LINCSCP_81757 |
A549 |
| -0.230372 |
3.281398e-13 |
975 |
ARG-TCRUZI2-9 |
LSM-6161 |
|
10uM |
6h |
LINCSCP_16898 |
LINCSCP_16898 |
HA1E |
| 0.230319 |
3.324081e-13 |
975 |
Niacin |
LSM-4676 |
HCAR2|HCAR3 |
3uM |
24h |
LINCSCP_28826 |
LINCSCP_28826 |
HUH7 |
| -0.230299 |
3.339588e-13 |
975 |
HDACi1,2+3_mix |
|
|
0.5uM |
24h |
LINCSCP_250169 |
LINCSCP_250169 |
MCF7 |
| 0.230291 |
3.346251e-13 |
975 |
ST51005413 |
LSM-4948 |
|
10uM |
6h |
LINCSCP_289133 |
LINCSCP_289133 |
U937 |
| 0.230288 |
3.348626e-13 |
975 |
Infigratinib |
LSM-1184 |
FGFR1|FGFR2|FGFR3|FGFR4 |
0.04uM |
24h |
LINCSCP_86861 |
LINCSCP_86861 |
CD34 |
| -0.23024 |
3.387603e-13 |
975 |
2-Chloro-7-methoxy-10H-phenothiazine |
LSM-3405 |
|
10uM |
24h |
LINCSCP_268186 |
LINCSCP_268186 |
PC3 |
| -0.230227 |
3.398638e-13 |
975 |
SB-431542 |
LSM-3498 |
ACVR1C|TGFBR1 |
10uM |
6h |
LINCSCP_44322 |
LINCSCP_44322 |
PC3 |
| -0.230217 |
3.406610e-13 |
975 |
Sufentanil |
LSM-45544 |
OPRM1 |
3.33uM |
24h |
LINCSCP_72970 |
LINCSCP_72970 |
A375 |
| -0.230198 |
3.422201e-13 |
975 |
Enzastaurin |
LSM-1069 |
PRKCB |
1.11uM |
24h |
LINCSCP_161314 |
LINCSCP_161314 |
PC3 |
| -0.230185 |
3.433088e-13 |
975 |
KU-C104137 |
LSM-2101 |
|
10uM |
6h |
LINCSCP_19685 |
LINCSCP_19685 |
HCC515 |
| 0.230159 |
3.454297e-13 |
975 |
MLS003672589 |
LSM-36804 |
|
10uM |
6h |
LINCSCP_29359 |
LINCSCP_29359 |
LOVO |
| 0.230139 |
3.470702e-13 |
975 |
BMS-299897 |
LSM-6207 |
|
10uM |
6h |
LINCSCP_282746 |
LINCSCP_282746 |
PL21 |
| -0.230138 |
3.471585e-13 |
975 |
Racephedrine |
LSM-1633 |
ADRA1A|ADRA2A |
10uM |
6h |
LINCSCP_56736 |
LINCSCP_56736 |
VCAP |
| -0.23013 |
3.478614e-13 |
975 |
CHEMBL2131985 |
LSM-39083 |
|
10uM |
6h |
LINCSCP_16815 |
LINCSCP_16815 |
HA1E |
| -0.23012 |
3.486618e-13 |
975 |
CHEMBL2140880 |
LSM-39548 |
|
10uM |
24h |
LINCSCP_37914 |
LINCSCP_37914 |
MCF7 |
| 0.230113 |
3.492545e-13 |
975 |
Ziprasidone |
LSM-5433 |
DRD2|HRH1|HTR1A|HTR1B|HTR1D|HTR1E|HTR2A|HTR2C|HTR7 |
0.12uM |
24h |
LINCSCP_71275 |
LINCSCP_71275 |
A375 |
| -0.230103 |
3.501499e-13 |
975 |
BRD-K26484692 |
LSM-10032 |
|
10uM |
24h |
LINCSCP_42976 |
LINCSCP_42976 |
NPC |
| -0.2301 |
3.503647e-13 |
975 |
BRD-K36296949 |
LSM-10621 |
|
5uM |
24h |
LINCSCP_61222 |
LINCSCP_61222 |
VCAP |
| -0.230088 |
3.513669e-13 |
975 |
Sulfisoxazole |
LSM-3120 |
|
10uM |
24h |
LINCSCP_42899 |
LINCSCP_42899 |
NPC |
| 0.230084 |
3.517336e-13 |
975 |
BRD-K96707310 |
LSM-14368 |
|
5uM |
6h |
LINCSCP_63856 |
LINCSCP_63856 |
VCAP |
| 0.230071 |
3.528413e-13 |
975 |
PRL-3InhibitorI |
LSM-43277 |
PTP4A3 |
40uM |
6h |
LINCSCP_40182 |
LINCSCP_40182 |
NCIH508 |
| -0.230068 |
3.531115e-13 |
975 |
SCHEMBL16980224 |
LSM-1092 |
AURKA |
1.11uM |
24h |
LINCSCP_82468 |
LINCSCP_82468 |
A549 |
| -0.230033 |
3.560722e-13 |
975 |
MLS000063258 |
LSM-2808 |
|
10uM |
24h |
LINCSCP_31599 |
LINCSCP_31599 |
MCF7 |
| 0.230012 |
3.578822e-13 |
975 |
BRD-K38524184 |
LSM-10762 |
|
5uM |
24h |
LINCSCP_62650 |
LINCSCP_62650 |
VCAP |
| 0.229999 |
3.589743e-13 |
975 |
GSK-319347A |
LSM-1216 |
IKBKG |
5uM |
6h |
LINCSCP_40215 |
LINCSCP_40215 |
NCIH508 |
| 0.22998 |
3.606386e-13 |
975 |
Pioglitazone |
LSM-1592 |
PPARG |
0.12uM |
24h |
LINCSCP_172131 |
LINCSCP_172131 |
YAPC |
| -0.229975 |
3.610793e-13 |
975 |
SCHEMBL2231351 |
LSM-36442 |
|
0.001uM |
6h |
LINCSCP_42026 |
LINCSCP_42026 |
NOMO1 |
| -0.229973 |
3.612654e-13 |
975 |
Cabazitaxel |
LSM-46002 |
|
10uM |
24h |
LINCSCP_138306 |
LINCSCP_138306 |
MCF7 |
| 0.229971 |
3.614395e-13 |
975 |
PCI-32765 |
LSM-1129 |
BTK |
3.33uM |
24h |
LINCSCP_83123 |
LINCSCP_83123 |
ASC.C |
| -0.229963 |
3.621441e-13 |
975 |
Momelotinib |
LSM-1141 |
JAK1|JAK2 |
1.11uM |
3h |
LINCSCP_115424 |
LINCSCP_115424 |
HS578T |
| -0.229925 |
3.654289e-13 |
975 |
MLS002703107 |
LSM-3603 |
|
10uM |
24h |
LINCSCP_31646 |
LINCSCP_31646 |
MCF7 |
| -0.229919 |
3.659463e-13 |
975 |
ST50591990 |
LSM-42844 |
|
10uM |
24h |
LINCSCP_1364 |
LINCSCP_1364 |
A375 |
| -0.229828 |
3.740206e-13 |
975 |
Ivacaftor (VX-770) |
LSM-45975 |
CFTR |
0.12uM |
24h |
LINCSCP_76478 |
LINCSCP_76478 |
A375 |
| -0.229824 |
3.744368e-13 |
975 |
BRD-K37299375 |
LSM-10679 |
|
1uM |
24h |
LINCSCP_312310 |
LINCSCP_312310 |
VCAP |
| -0.229805 |
3.760946e-13 |
975 |
Acitretin |
LSM-43217 |
RARA|RARB|RARG|RXRA|RXRB|RXRG |
10uM |
6h |
LINCSCP_26680 |
LINCSCP_26680 |
HT29 |
| -0.229785 |
3.779480e-13 |
975 |
BRD-K05114711 |
LSM-35178 |
|
10uM |
24h |
LINCSCP_42118 |
LINCSCP_42118 |
NPC |
| -0.229771 |
3.792150e-13 |
975 |
HLI-373 |
LSM-6225 |
MDM2 |
10uM |
24h |
LINCSCP_44907 |
LINCSCP_44907 |
PC3 |
| 0.229757 |
3.804977e-13 |
975 |
Retapamulin |
LSM-45949 |
|
3.33uM |
24h |
LINCSCP_71660 |
LINCSCP_71660 |
A375 |
| -0.229748 |
3.812780e-13 |
975 |
AKT Inhibitor VIII |
LSM-1035 |
AKT1|AKT2 |
10uM |
6h |
LINCSCP_51086 |
LINCSCP_51086 |
RMUGS |
| -0.229743 |
3.818171e-13 |
975 |
BI-2536 |
LSM-1041 |
PLK1 |
0.04uM |
24h |
LINCSCP_124228 |
LINCSCP_124228 |
HT29 |
| -0.229691 |
3.865633e-13 |
975 |
SR-02000000246 |
LSM-4247 |
|
10uM |
6h |
LINCSCP_15909 |
LINCSCP_15909 |
HA1E |
| 0.229688 |
3.868312e-13 |
975 |
Bisacodyl |
LSM-2883 |
|
10uM |
6h |
LINCSCP_14909 |
LINCSCP_14909 |
HA1E |
| 0.229677 |
3.878395e-13 |
975 |
XMD 8-92 |
LSM-1094 |
MAPK7 |
0.5uM |
6h |
LINCSCP_39588 |
LINCSCP_39588 |
MDAMB231 |
| -0.229656 |
3.898001e-13 |
975 |
AC1NX97Q |
LSM-45125 |
|
20uM |
24h |
LINCSCP_34745 |
LINCSCP_34745 |
MCF7 |
| 0.229655 |
3.899240e-13 |
975 |
TR-14035 |
LSM-45616 |
|
0.12uM |
24h |
LINCSCP_102487 |
LINCSCP_102487 |
HELA |
| -0.229649 |
3.904851e-13 |
975 |
DOCETAXEL |
LSM-45649 |
|
3.33uM |
24h |
LINCSCP_138259 |
LINCSCP_138259 |
MCF7 |
| 0.229625 |
3.927110e-13 |
975 |
CEFOTETAN |
LSM-45671 |
|
0.04uM |
24h |
LINCSCP_174880 |
LINCSCP_174880 |
YAPC |
| 0.229607 |
3.944441e-13 |
975 |
Alvocidib |
LSM-1011 |
CDK1|CDK2|CDK4|CDK5|CDK6|CDK7|CDK8|CDK9|EGFR|PYGM |
1.11uM |
24h |
LINCSCP_151107 |
LINCSCP_151107 |
PC3 |
| -0.2296 |
3.951128e-13 |
975 |
Amethopterin |
LSM-4285 |
DHFR |
10uM |
24h |
LINCSCP_243376 |
LINCSCP_243376 |
MCF7 |
| -0.229488 |
4.059077e-13 |
975 |
MLS002699336 |
LSM-2967 |
|
10uM |
24h |
LINCSCP_31608 |
LINCSCP_31608 |
MCF7 |
| -0.229432 |
4.113685e-13 |
975 |
GSK 1059615 |
LSM-42799 |
PIK3CA|PIK3CB|PIK3CD|PIK3CG |
0.04uM |
24h |
LINCSCP_81099 |
LINCSCP_81099 |
A549 |
| -0.229404 |
4.141509e-13 |
975 |
Acebutolol |
LSM-4384 |
ADRB1 |
10uM |
24h |
LINCSCP_271939 |
LINCSCP_271939 |
PC3 |
| -0.229401 |
4.144675e-13 |
975 |
Amperozide |
LSM-3159 |
DRD2|HTR2A |
10uM |
24h |
LINCSCP_32911 |
LINCSCP_32911 |
MCF7 |
| -0.22939 |
4.155021e-13 |
975 |
Famciclovir |
LSM-2990 |
|
0.04uM |
24h |
LINCSCP_172806 |
LINCSCP_172806 |
YAPC |
| -0.229383 |
4.162104e-13 |
975 |
BRD-K92300676 |
LSM-42292 |
|
5uM |
24h |
LINCSCP_48380 |
LINCSCP_48380 |
PC3 |
| -0.229372 |
4.173178e-13 |
975 |
CHEMBL1888222 |
LSM-3166 |
|
10uM |
24h |
LINCSCP_177858 |
LINCSCP_177858 |
A375 |
| 0.229368 |
4.176953e-13 |
975 |
BRD-K41513507 |
LSM-39567 |
|
1uM |
6h |
LINCSCP_38054 |
LINCSCP_38054 |
MCF7 |
| -0.22935 |
4.194905e-13 |
975 |
Plinabulin |
LSM-43250 |
TUBA1A|TUBA1B|TUBA1C|TUBA3E|TUBA4A|TUBB|TUBB1|TUBB2A|TUBB2B|TUBB3|TUBB4A|TUBB4B|TUBB6|TUBB8 |
10uM |
24h |
LINCSCP_46861 |
LINCSCP_46861 |
PC3 |
| -0.229327 |
4.218635e-13 |
975 |
Dasatinib |
LSM-1020 |
ABL1|BCR|BLK|EPHA2|FGR|FRK|FYN|HCK|KIT|LCK|LYN|PDGFRB|SRC|SRMS|YES1 |
0.04uM |
24h |
LINCSCP_99887 |
LINCSCP_99887 |
HCC515 |
| 0.229326 |
4.219695e-13 |
975 |
SPECTRUM_001418 |
LSM-1664 |
ADRB2 |
10uM |
6h |
LINCSCP_32976 |
LINCSCP_32976 |
MCF7 |
| 0.229281 |
4.265761e-13 |
975 |
Cediranib |
LSM-5926 |
FLT1|FLT4|KDR|KIT|PDGFRA|PDGFRB |
1.11uM |
24h |
LINCSCP_159658 |
LINCSCP_159658 |
PC3 |
| -0.229274 |
4.272722e-13 |
975 |
vincristine |
|
TUBB |
10uM |
24h |
LINCSCP_37613 |
LINCSCP_37613 |
MCF7 |
| -0.229271 |
4.275254e-13 |
975 |
Sildenafil |
LSM-3797 |
PDE5A |
100uM |
6h |
LINCSCP_218538 |
LINCSCP_218538 |
HCT116 |
| -0.22924 |
4.307892e-13 |
975 |
R-59022 |
LSM-3215 |
DGKA |
10uM |
24h |
LINCSCP_25289 |
LINCSCP_25289 |
HT29 |
| 0.229231 |
4.317033e-13 |
975 |
BRD-K29768655 |
LSM-38891 |
|
5uM |
24h |
LINCSCP_63022 |
LINCSCP_63022 |
VCAP |
| 0.229221 |
4.326587e-13 |
975 |
Calpeptin |
LSM-2570 |
|
10uM |
24h |
LINCSCP_33356 |
LINCSCP_33356 |
MCF7 |
| -0.229162 |
4.388963e-13 |
975 |
Podofilox |
LSM-3055 |
|
10uM |
24h |
LINCSCP_141623 |
LINCSCP_141623 |
MCF7 |
| 0.229131 |
4.421748e-13 |
975 |
ST092443 |
LSM-1481 |
ADORA1|ADORA2A|ADORA2B |
10uM |
6h |
LINCSCP_32963 |
LINCSCP_32963 |
MCF7 |
| 0.229128 |
4.424650e-13 |
975 |
MLS000680027 |
LSM-1646 |
|
10uM |
24h |
LINCSCP_4880 |
LINCSCP_4880 |
A549 |
| -0.229091 |
4.463948e-13 |
975 |
AC1LCS2I |
LSM-1738 |
|
10uM |
24h |
LINCSCP_45274 |
LINCSCP_45274 |
PC3 |
| -0.22908 |
4.475899e-13 |
975 |
BRD-K04986062 |
LSM-45341 |
|
10uM |
6h |
LINCSCP_24174 |
LINCSCP_24174 |
HL60 |
| -0.22906 |
4.497185e-13 |
975 |
2-(4-Nitro-phenylamino)-benzoic acid |
LSM-45307 |
|
3uM |
24h |
LINCSCP_12389 |
LINCSCP_12389 |
CD34 |
| -0.228991 |
4.571583e-13 |
975 |
Selumetinib |
LSM-1056 |
MAP2K1|MAP2K2 |
10uM |
24h |
LINCSCP_24337 |
LINCSCP_24337 |
HS578T |
| -0.228975 |
4.589767e-13 |
975 |
GSK 1059615 |
LSM-42799 |
PIK3CA|PIK3CB|PIK3CD|PIK3CG |
0.12uM |
24h |
LINCSCP_166178 |
LINCSCP_166178 |
SKL |
| 0.228969 |
4.596301e-13 |
975 |
Famciclovir |
LSM-2990 |
|
10uM |
6h |
LINCSCP_235865 |
LINCSCP_235865 |
MCF7 |
| 0.228937 |
4.631607e-13 |
975 |
SCHEMBL13991002 |
LSM-6278 |
|
40uM |
6h |
LINCSCP_10644 |
LINCSCP_10644 |
AGS |
| 0.228929 |
4.640509e-13 |
975 |
Vinpocetine |
LSM-3178 |
PDE1A |
10uM |
24h |
LINCSCP_44036 |
LINCSCP_44036 |
PC3 |
| 0.228883 |
4.691669e-13 |
975 |
Colforsin |
LSM-2193 |
ADCY2 |
10uM |
24h |
LINCSCP_33588 |
LINCSCP_33588 |
MCF7 |
| 0.228853 |
4.725403e-13 |
975 |
Lapatinib |
LSM-1051 |
EGFR|ERBB2 |
0.12uM |
3h |
LINCSCP_164118 |
LINCSCP_164118 |
SKBR3 |
| 0.228852 |
4.726113e-13 |
975 |
BRD-K00248931 |
LSM-8439 |
|
5uM |
24h |
LINCSCP_63327 |
LINCSCP_63327 |
VCAP |
| 0.228849 |
4.729753e-13 |
975 |
SC_I_004 |
LSM-45332 |
|
10uM |
6h |
LINCSCP_20101 |
LINCSCP_20101 |
HCC515 |
| 0.228815 |
4.768547e-13 |
975 |
BRD-K85724483 |
LSM-13676 |
|
5uM |
24h |
LINCSCP_63413 |
LINCSCP_63413 |
VCAP |
| -0.228795 |
4.791929e-13 |
975 |
Pimavanserin |
LSM-45960 |
HTR2A |
0.37uM |
24h |
LINCSCP_173144 |
LINCSCP_173144 |
YAPC |
| -0.228788 |
4.799895e-13 |
975 |
Mebendazole |
LSM-3749 |
|
40uM |
24h |
LINCSCP_67612 |
LINCSCP_67612 |
MCF7 |
| 0.22876 |
4.831948e-13 |
975 |
Cpccoet |
LSM-1360 |
GRM1 |
10uM |
24h |
LINCSCP_32808 |
LINCSCP_32808 |
MCF7 |
| 0.228737 |
4.858577e-13 |
975 |
BRD-K50131741 |
LSM-11477 |
|
5uM |
6h |
LINCSCP_63805 |
LINCSCP_63805 |
VCAP |
| -0.228682 |
4.923206e-13 |
975 |
Parbendazole |
LSM-4893 |
TUBB |
0.5uM |
24h |
LINCSCP_37423 |
LINCSCP_37423 |
MCF7 |
| -0.228667 |
4.940170e-13 |
975 |
BRD-K67829818 |
LSM-14902 |
|
5uM |
24h |
LINCSCP_309229 |
LINCSCP_309229 |
VCAP |
| -0.228652 |
4.958420e-13 |
975 |
AZD-5438 |
LSM-1159 |
CDK1|CDK10|CDK11B|CDK12|CDK13|CDK14|CDK15|CDK16|CDK17|CDK18|CDK19|CDK2|CDK20|CDK3|CDK4|CDK5|CDK6|CDK7|CDK8|CDK9 |
3.33uM |
24h |
LINCSCP_131331 |
LINCSCP_131331 |
MCF10A |
| -0.228626 |
4.989633e-13 |
975 |
NMS-1286937 |
LSM-45818 |
|
10uM |
24h |
LINCSCP_160070 |
LINCSCP_160070 |
PC3 |
| 0.228607 |
5.012283e-13 |
975 |
Cobalt (Ii) Chloride |
LSM-5958 |
HIF1A |
10uM |
6h |
LINCSCP_3123 |
LINCSCP_3123 |
A375 |
| 0.228604 |
5.015705e-13 |
975 |
Hydroxyprogesterone Caproate |
LSM-4900 |
AR|ESR1|ESR2|NR1H4|NR1I2|NR3C1|PGR |
0.04uM |
24h |
LINCSCP_101434 |
LINCSCP_101434 |
HELA |
| -0.228579 |
5.045768e-13 |
975 |
Mebendazole |
LSM-3749 |
|
10uM |
24h |
LINCSCP_139710 |
LINCSCP_139710 |
MCF7 |
| -0.22856 |
5.068051e-13 |
975 |
Danazol |
LSM-3073 |
AR|ESR1|GNRHR|PGR |
10uM |
6h |
LINCSCP_241838 |
LINCSCP_241838 |
MCF7 |
| 0.228557 |
5.071522e-13 |
975 |
Imatinib |
LSM-1023 |
ABL1|BCR|CSF1R|KIT|PDGFRA|PDGFRB |
0.12uM |
3h |
LINCSCP_116096 |
LINCSCP_116096 |
HS578T |
| -0.22851 |
5.128970e-13 |
975 |
BDBM43201 |
LSM-5018 |
|
10uM |
24h |
LINCSCP_45873 |
LINCSCP_45873 |
PC3 |
| -0.228503 |
5.137933e-13 |
975 |
BRD-K92096002 |
LSM-14087 |
|
5uM |
24h |
LINCSCP_61298 |
LINCSCP_61298 |
VCAP |
| 0.228423 |
5.236600e-13 |
975 |
ZINC03898662 |
LSM-4928 |
|
10uM |
6h |
LINCSCP_59366 |
LINCSCP_59366 |
VCAP |
| 0.228372 |
5.300447e-13 |
975 |
BRD-K94390774 |
LSM-14217 |
|
0.5uM |
24h |
LINCSCP_37498 |
LINCSCP_37498 |
MCF7 |
| 0.228359 |
5.317693e-13 |
975 |
ML100 |
LSM-6293 |
|
10uM |
6h |
LINCSCP_53629 |
LINCSCP_53629 |
SNGM |
| 0.228357 |
5.320464e-13 |
975 |
Etya |
LSM-5239 |
ALOX12|PPARA|PPARG|PTGS1 |
10uM |
24h |
LINCSCP_263813 |
LINCSCP_263813 |
NPC |
| -0.22834 |
5.341049e-13 |
975 |
BRD-A95504714 |
LSM-45336 |
|
10uM |
24h |
LINCSCP_55301 |
LINCSCP_55301 |
U937 |
| 0.228277 |
5.422913e-13 |
975 |
Gallocatechin Gallate |
LSM-6228 |
BACE1|FASN |
90uM |
6h |
LINCSCP_29321 |
LINCSCP_29321 |
LOVO |
| 0.228263 |
5.441022e-13 |
975 |
SPBIO_002561 |
LSM-2031 |
CHRNA2|HTR3A |
10uM |
24h |
LINCSCP_33318 |
LINCSCP_33318 |
MCF7 |
| -0.22824 |
5.471269e-13 |
975 |
LY2874455 |
LSM-45659 |
|
1.11uM |
24h |
LINCSCP_89886 |
LINCSCP_89886 |
HA1E |
| -0.228218 |
5.499450e-13 |
975 |
cortisone-acetate |
LSM-45387 |
TUBA1A|TUBA1B|TUBA1C|TUBA3E|TUBA4A|TUBB|TUBB1|TUBB2A|TUBB2B|TUBB3|TUBB4A|TUBB4B|TUBB6|TUBB8 |
0.12uM |
24h |
LINCSCP_126698 |
LINCSCP_126698 |
HT29 |
| -0.228216 |
5.501445e-13 |
975 |
TORIN1 |
LSM-1079 |
MTOR |
3.33uM |
24h |
LINCSCP_136999 |
LINCSCP_136999 |
MCF7 |
| -0.228215 |
5.502786e-13 |
975 |
ENMD-2076 |
LSM-45335 |
AURKA|AURKB|CSF1R|FGFR3|FLT3|KDR|KIT|PDGFRA|SRC |
10uM |
24h |
LINCSCP_97097 |
LINCSCP_97097 |
HA1E |
| 0.228198 |
5.526234e-13 |
975 |
MLS002264496 |
LSM-3730 |
|
10uM |
6h |
LINCSCP_292651 |
LINCSCP_292651 |
VCAP |
| 0.228144 |
5.596884e-13 |
975 |
Fccp |
LSM-2317 |
|
10uM |
24h |
LINCSCP_11417 |
LINCSCP_11417 |
ASC |
| -0.228142 |
5.599901e-13 |
975 |
Batimastat |
LSM-6276 |
|
3.33uM |
24h |
LINCSCP_101143 |
LINCSCP_101143 |
HELA |
| -0.228135 |
5.608828e-13 |
975 |
PD-98059 |
LSM-3394 |
MAP2K1 |
10uM |
6h |
LINCSCP_218769 |
LINCSCP_218769 |
HEC108 |
| -0.228119 |
5.630822e-13 |
975 |
Triazolothiadiazine, 36 |
LSM-1553 |
|
10uM |
24h |
LINCSCP_31315 |
LINCSCP_31315 |
MCF7 |
| 0.228062 |
5.708267e-13 |
975 |
JTE 013 |
LSM-2961 |
S1PR2 |
10uM |
24h |
LINCSCP_11438 |
LINCSCP_11438 |
ASC |
| -0.228059 |
5.712471e-13 |
975 |
Wortmannin |
LSM-3947 |
PIK3CA|PIK3CG|PLK1 |
3uM |
24h |
LINCSCP_55299 |
LINCSCP_55299 |
U937 |
| 0.228058 |
5.713866e-13 |
975 |
CHEMBL2203528 |
LSM-36795 |
|
0.01uM |
24h |
LINCSCP_288101 |
LINCSCP_288101 |
THP1 |
| -0.228035 |
5.744737e-13 |
975 |
CHEMBL1434137 |
LSM-6234 |
RARG |
40uM |
6h |
LINCSCP_4737 |
LINCSCP_4737 |
A549 |
| -0.227937 |
5.879663e-13 |
975 |
ZK-93426 |
LSM-3530 |
GABRA1 |
10uM |
6h |
LINCSCP_180119 |
LINCSCP_180119 |
A375 |
| 0.227923 |
5.900601e-13 |
975 |
GMX1778 |
LSM-6247 |
NAMPT |
0.1uM |
24h |
LINCSCP_4540 |
LINCSCP_4540 |
A549 |
| -0.227886 |
5.951820e-13 |
975 |
Selumetinib |
LSM-1056 |
MAP2K1|MAP2K2 |
0.1uM |
24h |
LINCSCP_24335 |
LINCSCP_24335 |
HS578T |
| -0.227879 |
5.962065e-13 |
975 |
PF-03758309 |
LSM-4254 |
PAK4 |
10uM |
24h |
LINCSCP_164954 |
LINCSCP_164954 |
SKL.C |
| 0.227868 |
5.977155e-13 |
975 |
AC1O9ATU |
LSM-1760 |
HMGCR |
10uM |
24h |
LINCSCP_32850 |
LINCSCP_32850 |
MCF7 |
| -0.227839 |
6.019720e-13 |
975 |
Velnacrine |
LSM-1959 |
|
10uM |
6h |
LINCSCP_467 |
LINCSCP_467 |
A375 |
| 0.227797 |
6.079937e-13 |
975 |
CHEMBL2359362 |
LSM-12720 |
|
5uM |
24h |
LINCSCP_61488 |
LINCSCP_61488 |
VCAP |
| -0.227793 |
6.085736e-13 |
975 |
BRD-K53407305 |
LSM-11686 |
|
5uM |
24h |
LINCSCP_27808 |
LINCSCP_27808 |
HT29 |
| -0.227778 |
6.106948e-13 |
975 |
Vitinoin |
LSM-2135 |
RARA|RARB|RARG|RORB |
3uM |
24h |
LINCSCP_37631 |
LINCSCP_37631 |
MCF7 |
| 0.22777 |
6.119412e-13 |
975 |
MLS002264419 |
LSM-3651 |
|
10uM |
6h |
LINCSCP_31511 |
LINCSCP_31511 |
MCF7 |
| 0.227762 |
6.131154e-13 |
975 |
Danusertib |
LSM-5253 |
AURKA|AURKB|AURKC|FGFR1|NTRK1|RET |
1.11uM |
24h |
LINCSCP_167746 |
LINCSCP_167746 |
YAPC |
| 0.227748 |
6.151105e-13 |
975 |
HY-11007 |
LSM-1022 |
ABL1|BCR |
10uM |
6h |
LINCSCP_32397 |
LINCSCP_32397 |
MCF7 |
| -0.227717 |
6.196550e-13 |
975 |
Hexamethoxyflavone |
LSM-4160 |
PIM1 |
10uM |
6h |
LINCSCP_290511 |
LINCSCP_290511 |
VCAP |
| 0.227716 |
6.197611e-13 |
975 |
Quinacrine |
LSM-1577 |
TP53 |
10uM |
6h |
LINCSCP_267363 |
LINCSCP_267363 |
PC3 |
| -0.227715 |
6.199827e-13 |
975 |
Broad-Sai-370 |
LSM-45321 |
|
3uM |
24h |
LINCSCP_250125 |
LINCSCP_250125 |
MCF7 |
| 0.227705 |
6.213840e-13 |
975 |
GSK-J2 |
LSM-44940 |
|
0.04uM |
24h |
LINCSCP_129007 |
LINCSCP_129007 |
HUVEC |
| 0.227693 |
6.232295e-13 |
975 |
Mocetinostat |
LSM-5344 |
HDAC1|HDAC11|HDAC2|HDAC3|HDAC8 |
0.04uM |
24h |
LINCSCP_82263 |
LINCSCP_82263 |
A549 |
| -0.227685 |
6.244440e-13 |
975 |
Veliparib |
LSM-1146 |
PARP1|PARP2 |
10uM |
6h |
LINCSCP_51234 |
LINCSCP_51234 |
RMUGS |
| -0.227666 |
6.272036e-13 |
975 |
Tacalcitol |
LSM-45518 |
|
10uM |
24h |
LINCSCP_108911 |
LINCSCP_108911 |
HELA |
| -0.227662 |
6.277825e-13 |
975 |
SA-427730 |
LSM-40726 |
|
10uM |
6h |
LINCSCP_37162 |
LINCSCP_37162 |
MCF7 |
| 0.227517 |
6.497991e-13 |
975 |
BRD-K94454791 |
LSM-14219 |
|
5uM |
24h |
LINCSCP_62192 |
LINCSCP_62192 |
VCAP |
| 0.227458 |
6.590120e-13 |
975 |
Resveratrol |
LSM-42917 |
PTGS1|PTGS2|SIRT1 |
0.12uM |
24h |
LINCSCP_168054 |
LINCSCP_168054 |
YAPC |
| 0.227449 |
6.603952e-13 |
975 |
amcinonide |
|
|
0.12uM |
24h |
LINCSCP_133999 |
LINCSCP_133999 |
MCF7 |
| 0.227433 |
6.630001e-13 |
975 |
BRD-K49276305 |
LSM-11423 |
|
5uM |
24h |
LINCSCP_62006 |
LINCSCP_62006 |
VCAP |
| -0.227367 |
6.734566e-13 |
975 |
BRD-A07407288 |
LSM-1460 |
|
10uM |
24h |
LINCSCP_242400 |
LINCSCP_242400 |
MCF7 |
| 0.227347 |
6.765569e-13 |
975 |
GSK-1070916 |
LSM-1062 |
AURKB|AURKC |
1uM |
6h |
LINCSCP_36630 |
LINCSCP_36630 |
MCF7 |
| 0.227334 |
6.787326e-13 |
975 |
MK-2206 |
LSM-1057 |
AKT1|AKT2|AKT3 |
0.12uM |
24h |
LINCSCP_113073 |
LINCSCP_113073 |
HME1 |
| 0.227321 |
6.807687e-13 |
975 |
THZ-2-98-01 |
LSM-44946 |
|
1.11uM |
24h |
LINCSCP_113220 |
LINCSCP_113220 |
HME1 |
| -0.227312 |
6.821952e-13 |
975 |
CHEMBL1271221 |
LSM-2596 |
|
10uM |
6h |
LINCSCP_5495 |
LINCSCP_5495 |
A549 |
| -0.227304 |
6.835155e-13 |
975 |
Ixabepilone |
LSM-43293 |
TUBA1A|TUBA1B|TUBA1C|TUBA3E|TUBA4A|TUBB|TUBB1|TUBB2A|TUBB2B|TUBB3|TUBB4A|TUBB4B|TUBB6|TUBB8 |
0.12uM |
24h |
LINCSCP_138118 |
LINCSCP_138118 |
MCF7 |
| -0.227274 |
6.885232e-13 |
975 |
CHEMBL2362317 |
LSM-12520 |
|
10uM |
24h |
LINCSCP_48560 |
LINCSCP_48560 |
PC3 |
| 0.227265 |
6.899619e-13 |
975 |
Quinine |
LSM-5109 |
SCN5A |
10uM |
6h |
LINCSCP_59547 |
LINCSCP_59547 |
VCAP |
| 0.227252 |
6.920625e-13 |
975 |
Naftifine |
LSM-43018 |
|
10uM |
6h |
LINCSCP_7519 |
LINCSCP_7519 |
A549 |
| 0.22725 |
6.923703e-13 |
975 |
SMR000651449 |
LSM-3511 |
|
10uM |
6h |
LINCSCP_29371 |
LINCSCP_29371 |
LOVO |
| 0.227241 |
6.937936e-13 |
975 |
BMS-345541 |
LSM-1028 |
IKBKB |
0.37uM |
3h |
LINCSCP_145696 |
LINCSCP_145696 |
MDAMB231 |
| -0.227219 |
6.974359e-13 |
975 |
Glimepiride |
LSM-2760 |
ABCC8|KCNJ11 |
10uM |
24h |
LINCSCP_52748 |
LINCSCP_52748 |
SKB |
| 0.227134 |
7.117344e-13 |
975 |
BRD-K13185593 |
LSM-9220 |
|
5uM |
6h |
LINCSCP_62505 |
LINCSCP_62505 |
VCAP |
| 0.227103 |
7.170421e-13 |
975 |
Diclofensine (hydrochloride) |
LSM-45632 |
|
1.11uM |
24h |
LINCSCP_139814 |
LINCSCP_139814 |
MCF7 |
| -0.227095 |
7.183681e-13 |
975 |
SR-02000000477 |
LSM-4204 |
|
10uM |
6h |
LINCSCP_45865 |
LINCSCP_45865 |
PC3 |
| -0.22708 |
7.209194e-13 |
975 |
Canertinib |
LSM-1120 |
EGFR|ERBB2|ERBB4 |
1.11uM |
24h |
LINCSCP_113118 |
LINCSCP_113118 |
HME1 |
| -0.227074 |
7.218987e-13 |
975 |
Dihydroorotate Dehydrogenase Inhibitor, Brequinar |
LSM-45952 |
|
10uM |
24h |
LINCSCP_144449 |
LINCSCP_144449 |
MCF7 |
| -0.227059 |
7.245189e-13 |
975 |
HMN-214 |
LSM-42802 |
CSF1R|FLT1|FLT3|FLT4|KDR|KIT|PDGFRB|RET |
3.33uM |
24h |
LINCSCP_150430 |
LINCSCP_150430 |
NPC.TAK |
| 0.227032 |
7.292119e-13 |
975 |
CHEMBL1495595 |
LSM-3294 |
|
10uM |
6h |
LINCSCP_5133 |
LINCSCP_5133 |
A549 |
| -0.227006 |
7.337279e-13 |
975 |
BRD-K86671899 |
LSM-13737 |
|
10uM |
24h |
LINCSCP_35257 |
LINCSCP_35257 |
MCF7 |
| -0.226961 |
7.414596e-13 |
975 |
MLS002473457 |
LSM-4212 |
|
10uM |
24h |
LINCSCP_31223 |
LINCSCP_31223 |
MCF7 |
| 0.226919 |
7.490083e-13 |
975 |
MLS000589843 |
LSM-43120 |
|
0.1uM |
24h |
LINCSCP_288171 |
LINCSCP_288171 |
THP1 |
| -0.226909 |
7.507930e-13 |
975 |
Vorinostat |
LSM-3828 |
HDAC1|HDAC2|HDAC3|HDAC6|HDAC8 |
10uM |
6h |
LINCSCP_66960 |
LINCSCP_66960 |
HCT116 |
| -0.226903 |
7.518083e-13 |
975 |
N9-Isopropylolomoucine |
LSM-3607 |
CDK1|CDK5 |
10uM |
24h |
LINCSCP_44249 |
LINCSCP_44249 |
PC3 |
| 0.226898 |
7.526509e-13 |
975 |
BRD-K10120618 |
LSM-9046 |
|
5uM |
6h |
LINCSCP_62499 |
LINCSCP_62499 |
VCAP |
| 0.226853 |
7.607395e-13 |
975 |
BRD-K96552587 |
LSM-42512 |
|
10uM |
24h |
LINCSCP_28320 |
LINCSCP_28320 |
HT29 |
| -0.226829 |
7.650250e-13 |
975 |
BRD-K76005220 |
LSM-15054 |
|
10uM |
24h |
LINCSCP_310052 |
LINCSCP_310052 |
VCAP |
| -0.22682 |
7.666303e-13 |
975 |
Wortmannin |
LSM-3947 |
PIK3CA|PIK3CG|PLK1 |
10uM |
24h |
LINCSCP_68951 |
LINCSCP_68951 |
VCAP |
| -0.226819 |
7.668772e-13 |
975 |
GW843682X |
LSM-1014 |
PLK1|PLK3 |
3uM |
24h |
LINCSCP_38252 |
LINCSCP_38252 |
MCF7 |
| -0.226817 |
7.672705e-13 |
975 |
FK888 |
LSM-3876 |
TACR1 |
0.37uM |
24h |
LINCSCP_173162 |
LINCSCP_173162 |
YAPC |
| -0.2268 |
7.703106e-13 |
975 |
Ponatinib |
LSM-1151 |
ABL1|BCR|FGFR1|FGFR2|FGFR3|FGFR4|FLT3|KIT|RET|TEK |
0.5uM |
24h |
LINCSCP_24748 |
LINCSCP_24748 |
HS578T |
| -0.2268 |
7.703175e-13 |
975 |
MG-132 |
LSM-1107 |
PSMB1 |
20uM |
24h |
LINCSCP_134815 |
LINCSCP_134815 |
MCF7 |
| -0.226791 |
7.720117e-13 |
975 |
R-59022 |
LSM-3215 |
DGKA |
10uM |
6h |
LINCSCP_223921 |
LINCSCP_223921 |
HT29 |
| 0.226785 |
7.730742e-13 |
975 |
CHEMBL565654 |
LSM-3666 |
|
10uM |
6h |
LINCSCP_5156 |
LINCSCP_5156 |
A549 |
| 0.226738 |
7.817477e-13 |
975 |
ipratropium |
LSM-45809 |
|
0.04uM |
24h |
LINCSCP_123152 |
LINCSCP_123152 |
HT29 |
| 0.226718 |
7.854355e-13 |
975 |
CHEBI:48565 |
LSM-1614 |
ADRA2A|ADRA2B|ADRA2C|HTR1A|HTR1B|HTR1D|HTR2B |
10uM |
6h |
LINCSCP_33175 |
LINCSCP_33175 |
MCF7 |
| 0.22671 |
7.869892e-13 |
975 |
BRD-K31462841 |
LSM-10335 |
|
5uM |
24h |
LINCSCP_62141 |
LINCSCP_62141 |
VCAP |
| -0.22667 |
7.943840e-13 |
975 |
Triazolothiadiazine, 29 |
LSM-3455 |
|
10uM |
24h |
LINCSCP_45727 |
LINCSCP_45727 |
PC3 |
| -0.226601 |
8.075292e-13 |
975 |
FR-180204 |
LSM-42790 |
MAPK1|MAPK3 |
10uM |
6h |
LINCSCP_5542 |
LINCSCP_5542 |
A549 |
| -0.226548 |
8.176941e-13 |
975 |
PRESTWICK3_000892 |
LSM-1968 |
|
10uM |
24h |
LINCSCP_262558 |
LINCSCP_262558 |
NPC |
| 0.226542 |
8.187945e-13 |
975 |
Torsemide |
LSM-2662 |
SLC12A1 |
0.04uM |
24h |
LINCSCP_134835 |
LINCSCP_134835 |
MCF7 |
| -0.226502 |
8.267066e-13 |
975 |
SA-85377 |
LSM-39088 |
|
0.5uM |
24h |
LINCSCP_252630 |
LINCSCP_252630 |
MCF7 |
| 0.226482 |
8.306032e-13 |
975 |
Mpep |
LSM-4678 |
GRM5 |
10uM |
24h |
LINCSCP_33645 |
LINCSCP_33645 |
MCF7 |
| -0.226471 |
8.327982e-13 |
975 |
SMR001317659 |
LSM-2094 |
|
0.5uM |
24h |
LINCSCP_30473 |
LINCSCP_30473 |
MCF7 |
| 0.226465 |
8.338912e-13 |
975 |
L-690330 |
LSM-4578 |
IMPA1 |
0.37uM |
24h |
LINCSCP_121130 |
LINCSCP_121130 |
HT29 |
| -0.226446 |
8.376160e-13 |
975 |
Alisertib |
LSM-37184 |
AURKA |
0.37uM |
24h |
LINCSCP_109512 |
LINCSCP_109512 |
HELA |
| 0.226404 |
8.459490e-13 |
975 |
CHEMBL2333346 |
LSM-36791 |
|
0.5uM |
6h |
LINCSCP_279898 |
LINCSCP_279898 |
PC3 |
| 0.226387 |
8.493597e-13 |
975 |
Felbamate |
LSM-4232 |
GRIN1|GRIN2A|GRIN2B|GRIN2C|GRIN2D|GRIN3A|GRIN3B |
10uM |
24h |
LINCSCP_11488 |
LINCSCP_11488 |
ASC |
| 0.226374 |
8.521421e-13 |
975 |
Indigo Red |
LSM-42899 |
CDK1|CDK5|GSK3A |
0.12uM |
24h |
LINCSCP_101762 |
LINCSCP_101762 |
HELA |
| -0.226365 |
8.539418e-13 |
975 |
Fraxidin Methyl Ether |
LSM-3489 |
CA12 |
10uM |
24h |
LINCSCP_284773 |
LINCSCP_284773 |
SKB |
| -0.226342 |
8.585062e-13 |
975 |
Alvocidib |
LSM-1011 |
CDK1|CDK2|CDK4|CDK5|CDK6|CDK7|CDK8|CDK9|EGFR|PYGM |
0.1uM |
24h |
LINCSCP_251095 |
LINCSCP_251095 |
MCF7 |
| 0.226339 |
8.591079e-13 |
975 |
BRD-K41931739 |
LSM-39588 |
|
10uM |
6h |
LINCSCP_22357 |
LINCSCP_22357 |
HEPG2 |
| -0.226326 |
8.618601e-13 |
975 |
AM 281 |
LSM-3318 |
CNR1 |
10uM |
6h |
LINCSCP_529 |
LINCSCP_529 |
A375 |
| -0.226324 |
8.622630e-13 |
975 |
Triazolothiadiazine, 23 |
LSM-3093 |
|
10uM |
24h |
LINCSCP_31169 |
LINCSCP_31169 |
MCF7 |
| 0.226316 |
8.638307e-13 |
975 |
BRD-K35247118 |
LSM-39203 |
|
10uM |
24h |
LINCSCP_48762 |
LINCSCP_48762 |
PC3 |
| 0.226286 |
8.699228e-13 |
975 |
PLX-4720 |
LSM-1049 |
BRAF |
0.37uM |
24h |
LINCSCP_130646 |
LINCSCP_130646 |
MCF10A |
| -0.226262 |
8.749492e-13 |
975 |
SCHEMBL16226068 |
LSM-43297 |
HSP90AA1 |
0.1uM |
6h |
LINCSCP_235629 |
LINCSCP_235629 |
MCF7 |
| 0.226255 |
8.764447e-13 |
975 |
AC1NWAUW |
LSM-1341 |
PRKACA |
10uM |
6h |
LINCSCP_14517 |
LINCSCP_14517 |
HA1E |
| 0.226243 |
8.789350e-13 |
975 |
Dexniguldipine |
LSM-15285 |
|
1.11uM |
24h |
LINCSCP_139148 |
LINCSCP_139148 |
MCF7 |
| -0.226213 |
8.850971e-13 |
975 |
Tiapride |
LSM-5676 |
DRD2|DRD3 |
1.11uM |
24h |
LINCSCP_171466 |
LINCSCP_171466 |
YAPC |
| -0.226207 |
8.863976e-13 |
975 |
BRD-K45392462 |
LSM-39787 |
|
5uM |
24h |
LINCSCP_185732 |
LINCSCP_185732 |
A375 |
| -0.226203 |
8.871332e-13 |
975 |
CGP 60474 |
LSM-1025 |
CDK1 |
10uM |
3h |
LINCSCP_113439 |
LINCSCP_113439 |
HME1 |
| 0.226192 |
8.895051e-13 |
975 |
citiolone |
LSM-45723 |
|
0.37uM |
24h |
LINCSCP_156633 |
LINCSCP_156633 |
PC3 |
| -0.226178 |
8.923612e-13 |
975 |
Repaglinide |
LSM-3863 |
ABCC8|KCNJ11 |
10uM |
6h |
LINCSCP_4411 |
LINCSCP_4411 |
A549 |
| -0.226167 |
8.947484e-13 |
975 |
Podofilox |
LSM-3055 |
|
1.11uM |
24h |
LINCSCP_141625 |
LINCSCP_141625 |
MCF7 |
| -0.226137 |
9.010449e-13 |
975 |
AC1OAATK |
LSM-4772 |
|
10uM |
6h |
LINCSCP_211494 |
LINCSCP_211494 |
HA1E |
| 0.226116 |
9.056033e-13 |
975 |
BRD-K22562809 |
LSM-9795 |
|
5uM |
24h |
LINCSCP_62131 |
LINCSCP_62131 |
VCAP |
| 0.226113 |
9.062353e-13 |
975 |
BRD-K31556224 |
LSM-10340 |
|
5uM |
24h |
LINCSCP_62271 |
LINCSCP_62271 |
VCAP |
| 0.226086 |
9.121679e-13 |
975 |
Dacarbazine |
LSM-5487 |
|
3.33uM |
24h |
LINCSCP_72012 |
LINCSCP_72012 |
A375 |
| 0.226036 |
9.227969e-13 |
975 |
CHEMBL2135770 |
LSM-38343 |
|
10uM |
6h |
LINCSCP_23154 |
LINCSCP_23154 |
HEPG2 |
| -0.226005 |
9.297747e-13 |
975 |
GP 2A |
LSM-2757 |
CNR2 |
10uM |
24h |
LINCSCP_7597 |
LINCSCP_7597 |
A549 |
| 0.225994 |
9.320093e-13 |
975 |
Sulfamerazine |
LSM-5979 |
|
10uM |
24h |
LINCSCP_34528 |
LINCSCP_34528 |
MCF7 |
| 0.225986 |
9.339542e-13 |
975 |
Erastin |
LSM-4914 |
VDAC2 |
5uM |
24h |
LINCSCP_25399 |
LINCSCP_25399 |
HT29 |
| -0.225969 |
9.376914e-13 |
975 |
E-3810 |
LSM-45728 |
FGFR1|FGFR2|FLT1|FLT4|KDR |
0.37uM |
24h |
LINCSCP_90066 |
LINCSCP_90066 |
HA1E |
| -0.225949 |
9.420163e-13 |
975 |
CI-1040 |
LSM-1048 |
MAP2K1|MAP2K2 |
3.33uM |
24h |
LINCSCP_121602 |
LINCSCP_121602 |
HT29 |
| 0.225908 |
9.511450e-13 |
975 |
Ingenol 3,20-dibenzoate |
LSM-4445 |
PRKCD|PRKCE |
10uM |
6h |
LINCSCP_21298 |
LINCSCP_21298 |
HEC108 |
| -0.225897 |
9.535958e-13 |
975 |
ML162 |
LSM-1493 |
|
3uM |
24h |
LINCSCP_37608 |
LINCSCP_37608 |
MCF7 |
| 0.225892 |
9.546805e-13 |
975 |
2-(4-Chlorophenyl)-4-propan-2-yloxyquinazoline |
LSM-3936 |
|
10uM |
6h |
LINCSCP_16376 |
LINCSCP_16376 |
HA1E |
| 0.225879 |
9.577401e-13 |
975 |
ST50998710 |
LSM-43133 |
|
10uM |
6h |
LINCSCP_16359 |
LINCSCP_16359 |
HA1E |
| -0.225856 |
9.629369e-13 |
975 |
BRD-K36959991 |
LSM-8215 |
|
1uM |
6h |
LINCSCP_37121 |
LINCSCP_37121 |
MCF7 |
| -0.225843 |
9.658221e-13 |
975 |
TORIN1 |
LSM-1079 |
MTOR |
10uM |
24h |
LINCSCP_29506 |
LINCSCP_29506 |
MCF10A |
| 0.225819 |
9.712624e-13 |
975 |
Fluspirilene |
LSM-3748 |
DRD2|HTR2A |
5uM |
6h |
LINCSCP_21257 |
LINCSCP_21257 |
HCT116 |
| -0.22581 |
9.734466e-13 |
975 |
Doxycycline |
LSM-5179 |
MMP8 |
10uM |
6h |
LINCSCP_16934 |
LINCSCP_16934 |
HA1E |
| -0.225786 |
9.788854e-13 |
975 |
13-Hydroxy-8,14,19-trimethoxy-4,10,12,16-tetramethyl-3,20,22-trioxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18-pentaen-9-yl carbamate |
LSM-42815 |
HSP90AA1 |
10uM |
6h |
LINCSCP_67863 |
LINCSCP_67863 |
PC3 |
| -0.225774 |
9.817117e-13 |
975 |
Tacedinaline |
LSM-19036 |
HDAC1|HDAC10|HDAC11|HDAC2|HDAC3|HDAC4|HDAC5|HDAC6|HDAC7|HDAC8|HDAC9 |
0.1uM |
6h |
LINCSCP_17160 |
LINCSCP_17160 |
HA1E |
| 0.225765 |
9.837376e-13 |
975 |
MLS003129913 |
LSM-10708 |
|
5uM |
24h |
LINCSCP_64187 |
LINCSCP_64187 |
VCAP |
| -0.225749 |
9.874908e-13 |
975 |
FPL64176 |
LSM-3777 |
CACNA1C |
10uM |
24h |
LINCSCP_42926 |
LINCSCP_42926 |
NPC |
| 0.225748 |
9.877125e-13 |
975 |
BRD-K03354784 |
LSM-8643 |
|
5uM |
6h |
LINCSCP_62960 |
LINCSCP_62960 |
VCAP |
| 0.225736 |
9.904686e-13 |
975 |
Quinapril |
LSM-3620 |
ACE |
10uM |
6h |
LINCSCP_226952 |
LINCSCP_226952 |
HT29 |
| -0.225731 |
9.918393e-13 |
975 |
PNU-99194A |
LSM-3568 |
DRD3 |
10uM |
6h |
LINCSCP_289881 |
LINCSCP_289881 |
VCAP |
| 0.225713 |
9.960324e-13 |
975 |
SMR000064811 |
LSM-22739 |
|
1uM |
24h |
LINCSCP_205430 |
LINCSCP_205430 |
CD34 |
| 0.225697 |
9.998095e-13 |
975 |
Bosutinib |
LSM-1190 |
ABL1|BCR|CAMK2G|HCK|LYN|SRC |
0.37uM |
24h |
LINCSCP_71674 |
LINCSCP_71674 |
A375 |
| 0.225673 |
1.005276e-12 |
975 |
Corticosterone |
LSM-5814 |
HSD11B1|NR3C2 |
10uM |
24h |
LINCSCP_31648 |
LINCSCP_31648 |
MCF7 |
| -0.225653 |
1.010172e-12 |
975 |
Fusaric acid |
LSM-3944 |
DBH |
10uM |
24h |
LINCSCP_262427 |
LINCSCP_262427 |
NPC |
| 0.225643 |
1.012453e-12 |
975 |
Foretinib |
LSM-1158 |
FLT1|FLT3|FLT4|KDR|KIT|MET|PDGFRA|PDGFRB|TEK |
0.1uM |
24h |
LINCSCP_39347 |
LINCSCP_39347 |
MDAMB231 |
| 0.22563 |
1.015674e-12 |
975 |
NU-7441 |
LSM-1061 |
PRKDC |
1uM |
24h |
LINCSCP_38914 |
LINCSCP_38914 |
MDAMB231 |
| -0.225585 |
1.026538e-12 |
975 |
Withaferin A |
LSM-6685 |
IKBKB|NAMPT |
0.5uM |
6h |
LINCSCP_201647 |
LINCSCP_201647 |
A549 |
| -0.225569 |
1.030427e-12 |
975 |
ST021200 |
LSM-4601 |
|
10uM |
24h |
LINCSCP_30539 |
LINCSCP_30539 |
MCF7 |
| -0.225561 |
1.032207e-12 |
975 |
AC1NWAML |
LSM-1325 |
NR3C1 |
10uM |
6h |
LINCSCP_44760 |
LINCSCP_44760 |
PC3 |
| 0.225557 |
1.033118e-12 |
975 |
AC1N9M1C |
LSM-4494 |
|
10uM |
6h |
LINCSCP_2113 |
LINCSCP_2113 |
A375 |
| 0.22555 |
1.034863e-12 |
975 |
BRD-K50929556 |
LSM-11535 |
|
5uM |
24h |
LINCSCP_62791 |
LINCSCP_62791 |
VCAP |
| 0.225542 |
1.036787e-12 |
975 |
Emedastine |
LSM-5331 |
HRH1 |
3.33uM |
24h |
LINCSCP_169819 |
LINCSCP_169819 |
YAPC |
| -0.225522 |
1.041805e-12 |
975 |
BRD-K62768020 |
LSM-45100 |
|
10uM |
6h |
LINCSCP_32355 |
LINCSCP_32355 |
MCF7 |
| -0.22552 |
1.042383e-12 |
975 |
MLS002276484 |
LSM-2585 |
|
10uM |
24h |
LINCSCP_30952 |
LINCSCP_30952 |
MCF7 |
| 0.225519 |
1.042404e-12 |
975 |
BRD-K57073585 |
LSM-14868 |
|
5uM |
24h |
LINCSCP_64200 |
LINCSCP_64200 |
VCAP |
| 0.225509 |
1.044879e-12 |
975 |
BRD-K50868745 |
LSM-11532 |
|
5uM |
24h |
LINCSCP_48245 |
LINCSCP_48245 |
PC3 |
| 0.225488 |
1.050151e-12 |
975 |
Rivaroxaban |
LSM-45951 |
|
0.12uM |
24h |
LINCSCP_141693 |
LINCSCP_141693 |
MCF7 |
| 0.225479 |
1.052460e-12 |
975 |
BRD-K82399474 |
LSM-13463 |
|
5uM |
24h |
LINCSCP_62177 |
LINCSCP_62177 |
VCAP |
| 0.225478 |
1.052551e-12 |
975 |
BRD-K29943481 |
LSM-38901 |
|
5uM |
24h |
LINCSCP_35108 |
LINCSCP_35108 |
MCF7 |
| -0.22545 |
1.059565e-12 |
975 |
BRD-A73558769 |
LSM-45352 |
|
10uM |
24h |
LINCSCP_288779 |
LINCSCP_288779 |
U937 |
| -0.225448 |
1.060165e-12 |
975 |
Racephedrine |
LSM-1633 |
ADRA1A|ADRA2A |
10uM |
6h |
LINCSCP_4300 |
LINCSCP_4300 |
A549 |
| -0.225437 |
1.062798e-12 |
975 |
TORIN-2 |
LSM-1080 |
MTOR |
0.5uM |
24h |
LINCSCP_29583 |
LINCSCP_29583 |
MCF10A |
| -0.225422 |
1.066690e-12 |
975 |
SMR000651464 |
LSM-2818 |
|
10uM |
6h |
LINCSCP_212171 |
LINCSCP_212171 |
HA1E |
| -0.225321 |
1.092203e-12 |
975 |
CHEMBL2057940 |
LSM-2409 |
|
10uM |
24h |
LINCSCP_31344 |
LINCSCP_31344 |
MCF7 |
| -0.225305 |
1.096292e-12 |
975 |
PF-03758309 |
LSM-4254 |
PAK4 |
10uM |
24h |
LINCSCP_114440 |
LINCSCP_114440 |
HME1 |
| -0.225265 |
1.106825e-12 |
975 |
BRD-K81156227 |
LSM-13391 |
|
10uM |
24h |
LINCSCP_312055 |
LINCSCP_312055 |
VCAP |
| 0.225247 |
1.111506e-12 |
975 |
BRD-K87167564 |
LSM-13774 |
|
5uM |
6h |
LINCSCP_62995 |
LINCSCP_62995 |
VCAP |
| -0.225245 |
1.112034e-12 |
975 |
SPECTRUM_000011 |
LSM-1767 |
|
0.04uM |
24h |
LINCSCP_109370 |
LINCSCP_109370 |
HELA |
| -0.225242 |
1.112761e-12 |
975 |
Telmisartan |
LSM-3657 |
AGTR1|PPARG |
10uM |
6h |
LINCSCP_270080 |
LINCSCP_270080 |
PC3 |
| -0.225203 |
1.123093e-12 |
975 |
Skiii |
LSM-2462 |
SPHK1 |
40uM |
6h |
LINCSCP_289035 |
LINCSCP_289035 |
U937 |
| 0.225201 |
1.123377e-12 |
975 |
(Z) Fluvoxamine |
LSM-3625 |
SLC6A4 |
10uM |
6h |
LINCSCP_31800 |
LINCSCP_31800 |
MCF7 |
| 0.225196 |
1.124951e-12 |
975 |
SCHEMBL17378613 |
LSM-5749 |
CSF1R |
3.33uM |
24h |
LINCSCP_100217 |
LINCSCP_100217 |
HCC515 |
| -0.225135 |
1.141038e-12 |
975 |
NSC 663284 |
LSM-2042 |
CDC25A|CDC25B |
10uM |
6h |
LINCSCP_220463 |
LINCSCP_220463 |
HEPG2 |
| 0.225134 |
1.141383e-12 |
975 |
BRD-K89697623 |
LSM-13963 |
|
5uM |
6h |
LINCSCP_62742 |
LINCSCP_62742 |
VCAP |
| -0.225114 |
1.146591e-12 |
975 |
ANISODAMINE HYDROBROMIDE |
LSM-45481 |
|
1.11uM |
24h |
LINCSCP_166594 |
LINCSCP_166594 |
YAPC |
| 0.225112 |
1.147359e-12 |
975 |
PF-04217903 |
LSM-1166 |
MET |
10uM |
24h |
LINCSCP_129482 |
LINCSCP_129482 |
JURKAT |
| -0.225111 |
1.147432e-12 |
975 |
Acarbose |
LSM-4631 |
AMY2A|GAA|MGAM |
10uM |
24h |
LINCSCP_47316 |
LINCSCP_47316 |
PC3 |
| 0.22509 |
1.153181e-12 |
975 |
TGX 221 |
LSM-1172 |
PIK3CB |
10uM |
24h |
LINCSCP_81178 |
LINCSCP_81178 |
A549 |
| -0.225063 |
1.160422e-12 |
975 |
PD-0325901 |
LSM-1101 |
MAP2K1|MAP2K2 |
10uM |
24h |
LINCSCP_81448 |
LINCSCP_81448 |
A549 |
| 0.225057 |
1.162092e-12 |
975 |
BRD-K53155533 |
LSM-11669 |
|
5uM |
24h |
LINCSCP_60894 |
LINCSCP_60894 |
VCAP |
| 0.224984 |
1.182215e-12 |
975 |
MLS002276498 |
LSM-3406 |
|
10uM |
6h |
LINCSCP_5141 |
LINCSCP_5141 |
A549 |
| 0.224982 |
1.182969e-12 |
975 |
AC1Q6JJ5 |
LSM-6192 |
TOP2A |
0.1uM |
6h |
LINCSCP_55422 |
LINCSCP_55422 |
U937 |
| -0.22498 |
1.183372e-12 |
975 |
ST-4062971 |
LSM-36806 |
|
1uM |
24h |
LINCSCP_37699 |
LINCSCP_37699 |
MCF7 |
| 0.224952 |
1.191105e-12 |
975 |
N-{3-[(4-methoxyphenyl)amino]-1,4-dioxo-1,4-dihydronaphthalen-2-yl}acetamide |
LSM-45353 |
|
0.5uM |
24h |
LINCSCP_222135 |
LINCSCP_222135 |
HL60 |
| 0.224949 |
1.191923e-12 |
975 |
MK-2866 (GTx-024) |
LSM-45447 |
AR |
10uM |
24h |
LINCSCP_71313 |
LINCSCP_71313 |
A375 |
| -0.224868 |
1.215004e-12 |
975 |
Palbociclib |
LSM-1071 |
CCND1|CDK4|CDK6 |
10uM |
6h |
LINCSCP_20464 |
LINCSCP_20464 |
HCC515 |
| 0.224865 |
1.215694e-12 |
975 |
Alpelisib |
LSM-4256 |
PIK3CA |
0.12uM |
3h |
LINCSCP_132484 |
LINCSCP_132484 |
MCF7 |
| -0.224845 |
1.221372e-12 |
975 |
Mepivacaine |
LSM-4306 |
SCN10A|SCN11A|SCN1A|SCN2A|SCN3A|SCN4A|SCN5A|SCN7A|SCN8A|SCN9A |
0.37uM |
24h |
LINCSCP_75258 |
LINCSCP_75258 |
A375 |
| 0.224807 |
1.232402e-12 |
975 |
MLS002276514 |
LSM-3561 |
|
10uM |
6h |
LINCSCP_1837 |
LINCSCP_1837 |
A375 |
| -0.224806 |
1.232746e-12 |
975 |
Tivantinib |
LSM-1131 |
MET |
3.33uM |
24h |
LINCSCP_135381 |
LINCSCP_135381 |
MCF7 |
| -0.224764 |
1.245041e-12 |
975 |
GW620972X |
LSM-1209 |
|
0.04uM |
24h |
LINCSCP_134270 |
LINCSCP_134270 |
MCF7 |
| -0.224762 |
1.245407e-12 |
975 |
NCGC00166323-01 |
LSM-6478 |
|
3.33uM |
24h |
LINCSCP_140430 |
LINCSCP_140430 |
MCF7 |
| -0.224749 |
1.249428e-12 |
975 |
bupivacaine |
LSM-45529 |
|
3.33uM |
24h |
LINCSCP_72256 |
LINCSCP_72256 |
A375 |
| 0.224738 |
1.252585e-12 |
975 |
BRD-K66814954 |
LSM-12499 |
|
5uM |
24h |
LINCSCP_63107 |
LINCSCP_63107 |
VCAP |
| 0.224737 |
1.252739e-12 |
975 |
CID755673 |
LSM-2050 |
|
10uM |
24h |
LINCSCP_1094 |
LINCSCP_1094 |
A375 |
| 0.22472 |
1.257942e-12 |
975 |
MLS002276500 |
LSM-3964 |
|
10uM |
24h |
LINCSCP_45962 |
LINCSCP_45962 |
PC3 |
| 0.224682 |
1.269050e-12 |
975 |
CO-1686 (AVL-301) |
LSM-45736 |
EGFR |
0.12uM |
24h |
LINCSCP_74158 |
LINCSCP_74158 |
A375 |
| 0.224672 |
1.272044e-12 |
975 |
Ziprasidone |
LSM-5433 |
DRD2|HRH1|HTR1A|HTR1B|HTR1D|HTR1E|HTR2A|HTR2C|HTR7 |
10uM |
6h |
LINCSCP_20433 |
LINCSCP_20433 |
HCC515 |
| -0.224662 |
1.275199e-12 |
975 |
Proglumide |
LSM-4439 |
CCKAR|CCKBR |
10uM |
24h |
LINCSCP_172789 |
LINCSCP_172789 |
YAPC |
| 0.224609 |
1.290972e-12 |
975 |
BRD-K14768034 |
LSM-38036 |
|
5uM |
24h |
LINCSCP_63010 |
LINCSCP_63010 |
VCAP |
| 0.224598 |
1.294248e-12 |
975 |
Gallocatechin Gallate |
LSM-6228 |
BACE1|FASN |
90uM |
6h |
LINCSCP_54911 |
LINCSCP_54911 |
THP1 |
| 0.224597 |
1.294545e-12 |
975 |
sorafenib |
|
BRAF|DDR2|FGFR1|FLT1|FLT3|FLT4|KDR|KIT|PDGFRB|RAF1|RET |
0.1uM |
24h |
LINCSCP_51382 |
LINCSCP_51382 |
SKBR3 |
| -0.224587 |
1.297701e-12 |
975 |
WH-4-025 |
LSM-44937 |
|
0.04uM |
24h |
LINCSCP_144890 |
LINCSCP_144890 |
MDAMB231 |
| -0.224559 |
1.306324e-12 |
975 |
BRD-K86838317 |
LSM-13751 |
|
5uM |
6h |
LINCSCP_306160 |
LINCSCP_306160 |
VCAP |
| -0.224547 |
1.310022e-12 |
975 |
Riluzole |
LSM-2471 |
SCN10A|SCN11A|SCN1A|SCN2A|SCN3A|SCN4A|SCN5A|SCN7A|SCN8A|SCN9A |
10uM |
6h |
LINCSCP_33201 |
LINCSCP_33201 |
MCF7 |
| -0.224526 |
1.316430e-12 |
975 |
Acetaminophen |
LSM-5533 |
FAAH|PTGS1|PTGS2|TRPV1 |
0.04uM |
24h |
LINCSCP_139031 |
LINCSCP_139031 |
MCF7 |
| -0.224488 |
1.328237e-12 |
975 |
CHEMBL2359949 |
LSM-39623 |
|
10uM |
24h |
LINCSCP_32177 |
LINCSCP_32177 |
MCF7 |
| -0.224486 |
1.328807e-12 |
975 |
CHEMBL566501 |
LSM-4112 |
|
10uM |
24h |
LINCSCP_5034 |
LINCSCP_5034 |
A549 |
| 0.224476 |
1.331965e-12 |
975 |
Imatinib |
LSM-1023 |
ABL1|BCR|CSF1R|KIT|PDGFRA|PDGFRB |
0.04uM |
3h |
LINCSCP_130379 |
LINCSCP_130379 |
LNCAP |
| 0.224437 |
1.343984e-12 |
975 |
Tretinoin |
LSM-42854 |
RARA|RARB|RARG|RORB |
1uM |
48h |
LINCSCP_64538 |
LINCSCP_64538 |
VCAP |
| -0.224435 |
1.344824e-12 |
975 |
BRD-K57200229-001-01-6 |
LSM-6809 |
|
10uM |
24h |
LINCSCP_33883 |
LINCSCP_33883 |
MCF7 |
| -0.224416 |
1.350841e-12 |
975 |
MW-STK33-97 |
LSM-44613 |
|
0.01uM |
24h |
LINCSCP_261240 |
LINCSCP_261240 |
NOMO1 |
| -0.224397 |
1.356784e-12 |
975 |
CHEMBL1619263 |
LSM-4840 |
|
10uM |
24h |
LINCSCP_239380 |
LINCSCP_239380 |
MCF7 |
| -0.224356 |
1.369831e-12 |
975 |
MLS000534605 |
LSM-4827 |
|
10uM |
24h |
LINCSCP_31958 |
LINCSCP_31958 |
MCF7 |
| 0.224325 |
1.379849e-12 |
975 |
Acetazolamide |
LSM-5543 |
CA1|CA12|CA14|CA2|CA4|CA7 |
0.12uM |
24h |
LINCSCP_105727 |
LINCSCP_105727 |
HELA |
| -0.224237 |
1.408589e-12 |
975 |
Manumycin-A |
LSM-43075 |
FNTA|IKBKB |
10uM |
24h |
LINCSCP_106788 |
LINCSCP_106788 |
HELA |
| -0.224218 |
1.414961e-12 |
975 |
altrenogest |
LSM-45498 |
|
0.37uM |
24h |
LINCSCP_139857 |
LINCSCP_139857 |
MCF7 |
| 0.224207 |
1.418425e-12 |
975 |
Amiloride |
LSM-4194 |
ASIC1|ASIC2|SCNN1A|SCNN1B|SCNN1G |
10uM |
6h |
LINCSCP_289945 |
LINCSCP_289945 |
VCAP |
| -0.22419 |
1.424260e-12 |
975 |
CHEMBL2355498 |
LSM-41978 |
|
5uM |
24h |
LINCSCP_231885 |
LINCSCP_231885 |
HT29 |
| -0.224188 |
1.424819e-12 |
975 |
Benzamil |
LSM-3945 |
PKD2L1|SCNN1A|SCNN1B|SCNN1D|SCNN1G|SLC8A1 |
10uM |
24h |
LINCSCP_11598 |
LINCSCP_11598 |
ASC |
| -0.22414 |
1.440888e-12 |
975 |
Infigratinib |
LSM-1184 |
FGFR1|FGFR2|FGFR3|FGFR4 |
0.1uM |
6h |
LINCSCP_36913 |
LINCSCP_36913 |
MCF7 |
| -0.224124 |
1.446216e-12 |
975 |
Forskolin, NKH477 |
LSM-45443 |
|
0.12uM |
24h |
LINCSCP_72147 |
LINCSCP_72147 |
A375 |
| -0.224062 |
1.467288e-12 |
975 |
BRD-K17666351 |
LSM-9492 |
|
5uM |
6h |
LINCSCP_306504 |
LINCSCP_306504 |
VCAP |
| -0.224043 |
1.473941e-12 |
975 |
BRD-K61202234 |
LSM-12134 |
|
5uM |
24h |
LINCSCP_62020 |
LINCSCP_62020 |
VCAP |
| -0.224016 |
1.483221e-12 |
975 |
ST023431 |
LSM-4327 |
|
10uM |
24h |
LINCSCP_46398 |
LINCSCP_46398 |
PC3 |
| -0.224014 |
1.484162e-12 |
975 |
BX-795 |
LSM-1189 |
PDK1|PDPK1 |
10uM |
6h |
LINCSCP_39760 |
LINCSCP_39760 |
MDST8 |
| 0.224 |
1.488923e-12 |
975 |
Curcumin |
LSM-43083 |
PTGS1|PTGS2 |
0.5uM |
24h |
LINCSCP_17226 |
LINCSCP_17226 |
HA1E |
| -0.223983 |
1.494702e-12 |
975 |
Tamatinib |
LSM-1040 |
SYK |
0.37uM |
24h |
LINCSCP_72163 |
LINCSCP_72163 |
A375 |
| -0.223971 |
1.499105e-12 |
975 |
FK888 |
LSM-3876 |
TACR1 |
0.04uM |
24h |
LINCSCP_173164 |
LINCSCP_173164 |
YAPC |
| 0.223956 |
1.504361e-12 |
975 |
Disopyramide |
LSM-1439 |
SCN10A|SCN11A|SCN1A|SCN2A|SCN3A|SCN4A|SCN5A|SCN7A|SCN8A|SCN9A |
10uM |
24h |
LINCSCP_71289 |
LINCSCP_71289 |
A375 |
| -0.223955 |
1.504531e-12 |
975 |
Dimethisoquin |
LSM-3647 |
|
10uM |
24h |
LINCSCP_11471 |
LINCSCP_11471 |
ASC |
| 0.223952 |
1.505508e-12 |
975 |
BRD-K49553303-001-01-8 |
LSM-40022 |
|
10uM |
6h |
LINCSCP_20625 |
LINCSCP_20625 |
HCC515 |
| -0.223934 |
1.511931e-12 |
975 |
Panobinostat |
LSM-43059 |
HDAC1|HDAC10|HDAC11|HDAC2|HDAC3|HDAC4|HDAC5|HDAC6|HDAC7|HDAC8|HDAC9 |
0.001uM |
24h |
LINCSCP_49296 |
LINCSCP_49296 |
PC3 |
| 0.223924 |
1.515412e-12 |
975 |
Oxybenzone |
LSM-3309 |
|
0.12uM |
24h |
LINCSCP_123169 |
LINCSCP_123169 |
HT29 |
| -0.223901 |
1.523806e-12 |
975 |
Tetrahydrouridine |
LSM-45757 |
|
1.11uM |
24h |
LINCSCP_160234 |
LINCSCP_160234 |
PC3 |
| 0.223823 |
1.551683e-12 |
975 |
AC1Q6JJ5 |
LSM-6192 |
TOP2A |
0.1uM |
6h |
LINCSCP_40163 |
LINCSCP_40163 |
NCIH508 |
| -0.223808 |
1.557095e-12 |
975 |
Albendazole |
LSM-3782 |
|
3uM |
24h |
LINCSCP_37948 |
LINCSCP_37948 |
MCF7 |
| 0.223797 |
1.561293e-12 |
975 |
CEFOTETAN |
LSM-45671 |
|
0.04uM |
24h |
LINCSCP_97869 |
LINCSCP_97869 |
HA1E |
| -0.22379 |
1.563579e-12 |
975 |
Epirubicin HCl |
LSM-45684 |
|
1.11uM |
24h |
LINCSCP_139628 |
LINCSCP_139628 |
MCF7 |
| 0.223779 |
1.567753e-12 |
975 |
GSK-3 Inhibitor IX |
LSM-42780 |
|
0.37uM |
24h |
LINCSCP_131179 |
LINCSCP_131179 |
MCF10A |
| -0.223706 |
1.594882e-12 |
975 |
MLS003128871 |
LSM-12917 |
|
5uM |
24h |
LINCSCP_64313 |
LINCSCP_64313 |
VCAP |
| 0.223698 |
1.597651e-12 |
975 |
BRD-A98888159 |
LSM-45917 |
|
0.04uM |
24h |
LINCSCP_124456 |
LINCSCP_124456 |
HT29 |
| 0.22369 |
1.600582e-12 |
975 |
Broad-Sai-424 |
LSM-45346 |
|
5uM |
24h |
LINCSCP_35522 |
LINCSCP_35522 |
MCF7 |
| 0.223654 |
1.614342e-12 |
975 |
Phenyl Biguanide |
LSM-4586 |
|
10uM |
6h |
LINCSCP_7694 |
LINCSCP_7694 |
A549 |
| 0.223608 |
1.631497e-12 |
975 |
BRD-K35669573 |
LSM-29348 |
|
0.5uM |
6h |
LINCSCP_42042 |
LINCSCP_42042 |
NOMO1 |
| -0.223566 |
1.647518e-12 |
975 |
Desmethylclomipramine |
LSM-36428 |
|
10uM |
24h |
LINCSCP_43462 |
LINCSCP_43462 |
NPC |
| 0.223557 |
1.651277e-12 |
975 |
MLS002725684 |
LSM-1500 |
|
10uM |
24h |
LINCSCP_238262 |
LINCSCP_238262 |
MCF7 |
| -0.223521 |
1.665241e-12 |
975 |
Mecamylamine |
LSM-4990 |
CHRNA2|CHRNA3|CHRNB4 |
0.04uM |
24h |
LINCSCP_72171 |
LINCSCP_72171 |
A375 |
| -0.223512 |
1.668453e-12 |
975 |
ENMD-2076 |
LSM-45335 |
AURKA|AURKB|CSF1R|FGFR3|FLT3|KDR|KIT|PDGFRA|SRC |
1.11uM |
24h |
LINCSCP_97099 |
LINCSCP_97099 |
HA1E |
| -0.223512 |
1.668659e-12 |
975 |
BRD-K76005220 |
LSM-15054 |
|
10uM |
6h |
LINCSCP_310177 |
LINCSCP_310177 |
VCAP |
| -0.223503 |
1.671980e-12 |
975 |
Rebastinib |
LSM-6708 |
ABL1 |
1.11uM |
24h |
LINCSCP_149724 |
LINCSCP_149724 |
NPC.TAK |
| -0.223485 |
1.678944e-12 |
975 |
BRD-A24396574-001-01-5 |
LSM-5006 |
|
0.37uM |
3h |
LINCSCP_130209 |
LINCSCP_130209 |
LNCAP |
| -0.223482 |
1.680160e-12 |
975 |
Galeterone |
LSM-45479 |
|
3.33uM |
24h |
LINCSCP_135945 |
LINCSCP_135945 |
MCF7 |
| 0.223453 |
1.691606e-12 |
975 |
Mosapride |
LSM-5042 |
HTR4 |
10uM |
24h |
LINCSCP_240235 |
LINCSCP_240235 |
MCF7 |
| 0.223425 |
1.702761e-12 |
975 |
BRD-K94241935 |
LSM-14207 |
|
5uM |
24h |
LINCSCP_62191 |
LINCSCP_62191 |
VCAP |
| -0.223424 |
1.702992e-12 |
975 |
Y-27632 |
LSM-44936 |
ROCK1|ROCK2 |
10uM |
6h |
LINCSCP_30371 |
LINCSCP_30371 |
MCF7 |
| -0.223423 |
1.703713e-12 |
975 |
Infigratinib |
LSM-1184 |
FGFR1|FGFR2|FGFR3|FGFR4 |
0.37uM |
24h |
LINCSCP_146338 |
LINCSCP_146338 |
MNEU.E |
| -0.223405 |
1.710567e-12 |
975 |
17-DMAG (Alvespimycin) HCl |
LSM-46133 |
|
0.12uM |
24h |
LINCSCP_101864 |
LINCSCP_101864 |
HELA |
| 0.2234 |
1.712705e-12 |
975 |
SPECTRUM5_002023 |
LSM-5041 |
|
10uM |
24h |
LINCSCP_10980 |
LINCSCP_10980 |
ASC |
| -0.223392 |
1.715963e-12 |
975 |
CHEMBL3188763 |
LSM-1698 |
|
10uM |
24h |
LINCSCP_1357 |
LINCSCP_1357 |
A375 |
| 0.223376 |
1.722299e-12 |
975 |
BRD-K94161851 |
LSM-14197 |
|
5uM |
24h |
LINCSCP_61668 |
LINCSCP_61668 |
VCAP |
| -0.22337 |
1.724511e-12 |
975 |
MLS002264387 |
LSM-2079 |
|
10uM |
6h |
LINCSCP_45777 |
LINCSCP_45777 |
PC3 |
| -0.223359 |
1.729322e-12 |
975 |
BRD-K02058097 |
LSM-8558 |
|
5uM |
6h |
LINCSCP_307861 |
LINCSCP_307861 |
VCAP |
| -0.22333 |
1.740733e-12 |
975 |
ZINC02121610 |
LSM-3277 |
|
10uM |
24h |
LINCSCP_1181 |
LINCSCP_1181 |
A375 |
| -0.223327 |
1.742174e-12 |
975 |
Falnidamol |
LSM-3584 |
EGFR |
0.04uM |
24h |
LINCSCP_160405 |
LINCSCP_160405 |
PC3 |
| -0.223327 |
1.742198e-12 |
975 |
MG-132 |
LSM-1107 |
PSMB1 |
1uM |
6h |
LINCSCP_251216 |
LINCSCP_251216 |
MCF7 |
| -0.223239 |
1.778342e-12 |
975 |
Tacedinaline |
LSM-19036 |
HDAC1|HDAC10|HDAC11|HDAC2|HDAC3|HDAC4|HDAC5|HDAC6|HDAC7|HDAC8|HDAC9 |
3uM |
24h |
LINCSCP_279727 |
LINCSCP_279727 |
PC3 |
| -0.223235 |
1.779654e-12 |
975 |
5-(6-Aminopurin-9-yl)-2-methyltetrahydrofuran-3-ol |
LSM-4354 |
|
0.04uM |
24h |
LINCSCP_73676 |
LINCSCP_73676 |
A375 |
| -0.223143 |
1.818511e-12 |
975 |
Selumetinib |
LSM-1056 |
MAP2K1|MAP2K2 |
0.04uM |
24h |
LINCSCP_99983 |
LINCSCP_99983 |
HCC515 |
| -0.223119 |
1.828422e-12 |
975 |
Foretinib |
LSM-1158 |
FLT1|FLT3|FLT4|KDR|KIT|MET|PDGFRA|PDGFRB|TEK |
10uM |
24h |
LINCSCP_105435 |
LINCSCP_105435 |
HELA |
| -0.223096 |
1.838337e-12 |
975 |
CHEMBL2220622 |
LSM-3841 |
|
10uM |
24h |
LINCSCP_31658 |
LINCSCP_31658 |
MCF7 |
| 0.223033 |
1.865511e-12 |
975 |
MLS002699429 |
LSM-44942 |
|
40uM |
6h |
LINCSCP_4760 |
LINCSCP_4760 |
A549 |
| 0.22303 |
1.866891e-12 |
975 |
Amonafide |
LSM-5667 |
TOP2A |
10uM |
6h |
LINCSCP_26507 |
LINCSCP_26507 |
HT29 |
| -0.223007 |
1.877023e-12 |
975 |
KW-2449 |
LSM-42803 |
ABL1|AURKA|AURKB|FLT3 |
10uM |
24h |
LINCSCP_165376 |
LINCSCP_165376 |
SKL |
| 0.222998 |
1.880598e-12 |
975 |
BRD-K74998149 |
LSM-41356 |
|
10uM |
6h |
LINCSCP_49175 |
LINCSCP_49175 |
PC3 |
| -0.222974 |
1.891207e-12 |
975 |
BRD-A28746609 |
LSM-1102 |
NR1I2|TUBB |
10uM |
24h |
LINCSCP_137544 |
LINCSCP_137544 |
MCF7 |
| -0.222961 |
1.896828e-12 |
975 |
SA-424170 |
LSM-39302 |
|
3uM |
24h |
LINCSCP_37239 |
LINCSCP_37239 |
MCF7 |
| -0.222952 |
1.901205e-12 |
975 |
INCA-6 |
LSM-2729 |
NFATC1 |
10uM |
24h |
LINCSCP_18889 |
LINCSCP_18889 |
HCC515 |
| -0.222945 |
1.904009e-12 |
975 |
BRD-K30802967 |
LSM-6102 |
|
10uM |
24h |
LINCSCP_295574 |
LINCSCP_295574 |
VCAP |
| 0.222937 |
1.907461e-12 |
975 |
Enzalutamide |
LSM-6254 |
AR |
0.1uM |
6h |
LINCSCP_51164 |
LINCSCP_51164 |
RMUGS |
| 0.222905 |
1.921698e-12 |
975 |
BI-2536 |
LSM-1041 |
PLK1 |
0.04uM |
3h |
LINCSCP_163909 |
LINCSCP_163909 |
SKBR3 |
| 0.222893 |
1.927331e-12 |
975 |
SCHEMBL16980224 |
LSM-1092 |
AURKA |
0.1uM |
24h |
LINCSCP_24826 |
LINCSCP_24826 |
HS578T |
| 0.222892 |
1.927667e-12 |
975 |
ST50426557 |
LSM-4770 |
|
10uM |
6h |
LINCSCP_16391 |
LINCSCP_16391 |
HA1E |
| 0.22284 |
1.951228e-12 |
975 |
Vorinostat |
LSM-3828 |
HDAC1|HDAC2|HDAC3|HDAC6|HDAC8 |
0.1uM |
24h |
LINCSCP_250247 |
LINCSCP_250247 |
MCF7 |
| -0.222839 |
1.951760e-12 |
975 |
CGP 60474 |
LSM-1025 |
CDK1 |
0.1uM |
24h |
LINCSCP_29605 |
LINCSCP_29605 |
MCF10A |
| -0.222829 |
1.955986e-12 |
975 |
SA-1459031 |
LSM-38951 |
|
3uM |
24h |
LINCSCP_41714 |
LINCSCP_41714 |
NKDBA |
| -0.222805 |
1.966882e-12 |
975 |
Colforsin |
LSM-2193 |
ADCY2 |
10uM |
24h |
LINCSCP_52845 |
LINCSCP_52845 |
SKB |
| -0.222805 |
1.966955e-12 |
975 |
Fenbendazole |
LSM-3134 |
TUBB |
3uM |
24h |
LINCSCP_38201 |
LINCSCP_38201 |
MCF7 |
| -0.222758 |
1.988928e-12 |
975 |
Carbazole, 9-(4-methylbenzoyl)- |
LSM-3597 |
|
10uM |
24h |
LINCSCP_25960 |
LINCSCP_25960 |
HT29 |
| -0.222702 |
2.014775e-12 |
975 |
HMN-214 |
LSM-42802 |
CSF1R|FLT1|FLT3|FLT4|KDR|KIT|PDGFRB|RET |
1.11uM |
24h |
LINCSCP_150431 |
LINCSCP_150431 |
NPC.TAK |
| -0.222695 |
2.018005e-12 |
975 |
Infigratinib |
LSM-1184 |
FGFR1|FGFR2|FGFR3|FGFR4 |
0.1uM |
24h |
LINCSCP_24737 |
LINCSCP_24737 |
HS578T |
| -0.222672 |
2.028761e-12 |
975 |
R-7128 |
LSM-45627 |
|
10uM |
24h |
LINCSCP_142547 |
LINCSCP_142547 |
MCF7 |
| 0.222666 |
2.031824e-12 |
975 |
Sulfadoxine |
LSM-5657 |
|
1.11uM |
24h |
LINCSCP_73405 |
LINCSCP_73405 |
A375 |
| -0.22264 |
2.043984e-12 |
975 |
Buparlisib |
LSM-1148 |
PIK3CA|PIK3CB|PIK3CD|PIK3CG|PIK3R1|PIK3R2|PIK3R3|PIK3R5 |
3.33uM |
24h |
LINCSCP_131989 |
LINCSCP_131989 |
MCF7 |
| 0.222638 |
2.045067e-12 |
975 |
Trifluoperazine |
LSM-4010 |
DRD2|DRD3|DRD4|HTR2A|HTR2C |
10uM |
6h |
LINCSCP_40252 |
LINCSCP_40252 |
NCIH508 |
| 0.222587 |
2.069382e-12 |
975 |
BRD-K78496556 |
LSM-41553 |
|
10uM |
24h |
LINCSCP_48829 |
LINCSCP_48829 |
PC3 |
| 0.222567 |
2.078697e-12 |
975 |
Indigo Red |
LSM-42899 |
CDK1|CDK5|GSK3A |
0.12uM |
24h |
LINCSCP_71639 |
LINCSCP_71639 |
A375 |
| -0.222566 |
2.079423e-12 |
975 |
Ursolic acid |
LSM-4889 |
HSD11B1|PTPN1 |
70uM |
6h |
LINCSCP_51191 |
LINCSCP_51191 |
RMUGS |
| 0.222518 |
2.102745e-12 |
975 |
AS601245 |
LSM-1034 |
MAPK10|MAPK8|MAPK9 |
0.12uM |
24h |
LINCSCP_81344 |
LINCSCP_81344 |
A549 |
| -0.222515 |
2.104103e-12 |
975 |
Pifithrin-beta |
LSM-2688 |
|
10uM |
6h |
LINCSCP_14237 |
LINCSCP_14237 |
HA1E |
| -0.222509 |
2.107315e-12 |
975 |
AZD4547 |
LSM-6308 |
|
10uM |
24h |
LINCSCP_128094 |
LINCSCP_128094 |
HUES3 |
| 0.22249 |
2.116300e-12 |
975 |
Labetalol |
LSM-1282 |
ADRA1A|ADRA1B|ADRA1D|ADRA2A|ADRA2B|ADRA2C|ADRB1|ADRB2|ADRB3 |
10uM |
24h |
LINCSCP_243336 |
LINCSCP_243336 |
MCF7 |
| -0.222489 |
2.116988e-12 |
975 |
Azathioprine |
LSM-42936 |
PPAT |
10uM |
6h |
LINCSCP_3085 |
LINCSCP_3085 |
A375 |
| -0.222488 |
2.117470e-12 |
975 |
Phylloquinone |
LSM-43150 |
|
10uM |
24h |
LINCSCP_271953 |
LINCSCP_271953 |
PC3 |
| -0.222487 |
2.117753e-12 |
975 |
omeprazole |
LSM-45749 |
|
10uM |
24h |
LINCSCP_121859 |
LINCSCP_121859 |
HT29 |
| 0.222471 |
2.125645e-12 |
975 |
(-)-Tramadol |
LSM-3125 |
OPRM1|SLC6A2|SLC6A4 |
10uM |
24h |
LINCSCP_73485 |
LINCSCP_73485 |
A375 |
| -0.222448 |
2.137009e-12 |
975 |
761437-28-9 |
LSM-1208 |
|
10uM |
24h |
LINCSCP_149805 |
LINCSCP_149805 |
NPC.TAK |
| -0.22243 |
2.145917e-12 |
975 |
Epigalocatechin Gallate |
LSM-5661 |
FASN |
0.04uM |
24h |
LINCSCP_87063 |
LINCSCP_87063 |
CD34 |
| 0.222428 |
2.146947e-12 |
975 |
Zileuton |
LSM-5084 |
ALOX5 |
0.04uM |
24h |
LINCSCP_120406 |
LINCSCP_120406 |
HT29 |
| 0.2224 |
2.161292e-12 |
975 |
CHEMBL1705549 |
LSM-2498 |
|
10uM |
24h |
LINCSCP_237832 |
LINCSCP_237832 |
MCF7 |
| 0.222397 |
2.162444e-12 |
975 |
Meclofenamic acid |
LSM-3108 |
ALOX5|PTGS1|PTGS2 |
10uM |
6h |
LINCSCP_193472 |
LINCSCP_193472 |
A549 |
| -0.222373 |
2.174482e-12 |
975 |
AC1M52QF |
LSM-43140 |
|
10uM |
6h |
LINCSCP_54019 |
LINCSCP_54019 |
SW480 |
| 0.222349 |
2.186955e-12 |
975 |
BRD-K66775134 |
LSM-12498 |
|
5uM |
6h |
LINCSCP_63823 |
LINCSCP_63823 |
VCAP |
| 0.222348 |
2.187186e-12 |
975 |
Retapamulin |
LSM-45949 |
|
0.04uM |
24h |
LINCSCP_71664 |
LINCSCP_71664 |
A375 |
| -0.222321 |
2.201143e-12 |
975 |
BRD-K30393343 |
LSM-14786 |
|
3uM |
6h |
LINCSCP_38026 |
LINCSCP_38026 |
MCF7 |
| -0.22232 |
2.201336e-12 |
975 |
BRD-K80368509 |
LSM-45306 |
|
3uM |
24h |
LINCSCP_222193 |
LINCSCP_222193 |
HL60 |
| 0.222304 |
2.209944e-12 |
975 |
BRD-K81415316 |
LSM-13399 |
|
5uM |
24h |
LINCSCP_61502 |
LINCSCP_61502 |
VCAP |
| -0.222292 |
2.215748e-12 |
975 |
BRD-A31180007 |
LSM-45646 |
|
10uM |
24h |
LINCSCP_154655 |
LINCSCP_154655 |
PC3 |
| -0.222288 |
2.218092e-12 |
975 |
naftidrofuryl |
LSM-45485 |
|
0.04uM |
24h |
LINCSCP_76390 |
LINCSCP_76390 |
A375 |
| -0.22228 |
2.221801e-12 |
975 |
BRD-K07820537 |
LSM-37695 |
|
10uM |
6h |
LINCSCP_64740 |
LINCSCP_64740 |
VCAP |
| -0.222269 |
2.227906e-12 |
975 |
1,3-Dipropyl-8-cyclopentylxanthine |
LSM-19971 |
|
3.33uM |
24h |
LINCSCP_170437 |
LINCSCP_170437 |
YAPC |
| -0.222256 |
2.234624e-12 |
975 |
Wortmannin |
LSM-3947 |
PIK3CA|PIK3CG|PLK1 |
0.5uM |
24h |
LINCSCP_310742 |
LINCSCP_310742 |
VCAP |
| 0.222235 |
2.245145e-12 |
975 |
SA-1939079 |
LSM-41390 |
|
3uM |
24h |
LINCSCP_252320 |
LINCSCP_252320 |
MCF7 |
| 0.222219 |
2.253933e-12 |
975 |
Nilotinib |
LSM-1099 |
ABL1|BCR|KIT |
0.04uM |
24h |
LINCSCP_144878 |
LINCSCP_144878 |
MDAMB231 |
| -0.222216 |
2.255179e-12 |
975 |
Erlotinib |
LSM-1097 |
EGFR |
1.11uM |
24h |
LINCSCP_96967 |
LINCSCP_96967 |
HA1E |
| 0.222183 |
2.272423e-12 |
975 |
Formoterol |
LSM-4251 |
ADRB2 |
3.33uM |
24h |
LINCSCP_171883 |
LINCSCP_171883 |
YAPC |
| 0.222171 |
2.278961e-12 |
975 |
Phenoxazine |
LSM-4657 |
|
10uM |
6h |
LINCSCP_53583 |
LINCSCP_53583 |
SNGM |
| 0.222166 |
2.281422e-12 |
975 |
BRD-K24754728 |
LSM-6092 |
|
10uM |
24h |
LINCSCP_7799 |
LINCSCP_7799 |
A549 |
| 0.222158 |
2.285774e-12 |
975 |
K-115 |
LSM-45986 |
|
1.11uM |
24h |
LINCSCP_76530 |
LINCSCP_76530 |
A375 |
| 0.222133 |
2.299215e-12 |
975 |
SMR000009277 |
LSM-3264 |
|
10uM |
6h |
LINCSCP_15882 |
LINCSCP_15882 |
HA1E |
| 0.222103 |
2.315314e-12 |
975 |
Tozasertib |
LSM-1021 |
ABL1|AURKA|AURKB|AURKC|BCR|FLT3|JAK2 |
0.1uM |
24h |
LINCSCP_11755 |
LINCSCP_11755 |
BT20 |
| -0.2221 |
2.316951e-12 |
975 |
PD-0325901 |
LSM-1101 |
MAP2K1|MAP2K2 |
0.37uM |
24h |
LINCSCP_165201 |
LINCSCP_165201 |
SKL.C |
| -0.222043 |
2.347329e-12 |
975 |
MLN-0128 |
LSM-1206 |
MTOR |
3.33uM |
24h |
LINCSCP_149777 |
LINCSCP_149777 |
NPC.TAK |
| 0.222043 |
2.347348e-12 |
975 |
BRD-K37434018 |
LSM-10689 |
|
5uM |
24h |
LINCSCP_303069 |
LINCSCP_303069 |
VCAP |
| -0.221974 |
2.385209e-12 |
975 |
PCI-34051 |
LSM-4812 |
HDAC1|HDAC10|HDAC6|HDAC8 |
3uM |
24h |
LINCSCP_49261 |
LINCSCP_49261 |
PC3 |
| -0.221965 |
2.390071e-12 |
975 |
Setiptiline |
LSM-45982 |
|
10uM |
24h |
LINCSCP_90393 |
LINCSCP_90393 |
HA1E |
| 0.221947 |
2.400371e-12 |
975 |
Sulconazole |
LSM-1751 |
|
10uM |
6h |
LINCSCP_32981 |
LINCSCP_32981 |
MCF7 |
| 0.221913 |
2.419078e-12 |
975 |
5807-14-7 |
LSM-5565 |
|
10uM |
6h |
LINCSCP_3090 |
LINCSCP_3090 |
A375 |
| 0.221911 |
2.420616e-12 |
975 |
BRD-K84797952 |
LSM-41900 |
|
5uM |
24h |
LINCSCP_28136 |
LINCSCP_28136 |
HT29 |
| -0.221903 |
2.424761e-12 |
975 |
Cortisone Acetate |
LSM-5917 |
NR3C1 |
10uM |
24h |
LINCSCP_47344 |
LINCSCP_47344 |
PC3 |
| 0.221893 |
2.430171e-12 |
975 |
Gefitinib |
LSM-1098 |
EGFR |
0.37uM |
3h |
LINCSCP_133196 |
LINCSCP_133196 |
MCF7 |
| 0.221881 |
2.436992e-12 |
975 |
ZK 756326 |
LSM-3253 |
CCR8 |
10uM |
6h |
LINCSCP_4395 |
LINCSCP_4395 |
A549 |
| -0.22188 |
2.437712e-12 |
975 |
SB-366791 |
LSM-3316 |
TRPV1 |
10uM |
24h |
LINCSCP_42646 |
LINCSCP_42646 |
NPC |
| -0.221848 |
2.455765e-12 |
975 |
MLS003129913 |
LSM-10708 |
|
5uM |
24h |
LINCSCP_309387 |
LINCSCP_309387 |
VCAP |
| -0.221843 |
2.458686e-12 |
975 |
ML175 |
LSM-3291 |
|
10uM |
24h |
LINCSCP_25945 |
LINCSCP_25945 |
HT29 |
| 0.221823 |
2.469864e-12 |
975 |
Roflumilast |
LSM-45821 |
PDE4A|PDE4B|PDE4C|PDE4D |
10uM |
24h |
LINCSCP_75203 |
LINCSCP_75203 |
A375 |
| -0.221795 |
2.486072e-12 |
975 |
AC1LWSL2 |
LSM-3096 |
|
10uM |
24h |
LINCSCP_34146 |
LINCSCP_34146 |
MCF7 |
| 0.22179 |
2.488779e-12 |
975 |
Crizotinib |
LSM-1027 |
ALK|MET |
0.5uM |
6h |
LINCSCP_51711 |
LINCSCP_51711 |
SKBR3 |
| -0.221786 |
2.491311e-12 |
975 |
4,11-Diethyl-4,9-dihydroxy-1H-pyrano[3',4':6,7]indolizino[1,2-b]quinoline-3,14(4H,12H)-dione |
LSM-6189 |
TOP1 |
1uM |
24h |
LINCSCP_35636 |
LINCSCP_35636 |
MCF7 |
| -0.221771 |
2.499877e-12 |
975 |
Iproniazid |
LSM-5940 |
|
10uM |
24h |
LINCSCP_47347 |
LINCSCP_47347 |
PC3 |
| -0.221758 |
2.507487e-12 |
975 |
SCHEMBL3954849 |
LSM-5982 |
|
3.33uM |
3h |
LINCSCP_163146 |
LINCSCP_163146 |
SKBR3 |
| 0.221747 |
2.514115e-12 |
975 |
AKT Inhibitor VIII |
LSM-1035 |
AKT1|AKT2 |
10uM |
6h |
LINCSCP_13456 |
LINCSCP_13456 |
H1299 |
| -0.22174 |
2.518204e-12 |
975 |
BRD-K63513868 |
LSM-45333 |
|
1uM |
24h |
LINCSCP_222175 |
LINCSCP_222175 |
HL60 |
| -0.221732 |
2.522688e-12 |
975 |
MLS006011051 |
LSM-42801 |
BRAF |
10uM |
24h |
LINCSCP_39456 |
LINCSCP_39456 |
MDAMB231 |
| -0.221727 |
2.525315e-12 |
975 |
Withaferin A |
LSM-6685 |
IKBKB|NAMPT |
0.5uM |
6h |
LINCSCP_201990 |
LINCSCP_201990 |
A549 |
| -0.221717 |
2.531485e-12 |
975 |
MLS002473428 |
LSM-2278 |
|
10uM |
24h |
LINCSCP_269117 |
LINCSCP_269117 |
PC3 |
| -0.221714 |
2.533080e-12 |
975 |
JSH-23 |
LSM-5897 |
RELA |
5uM |
6h |
LINCSCP_45238 |
LINCSCP_45238 |
PC3 |
| -0.221702 |
2.540015e-12 |
975 |
LY2228820 |
LSM-45439 |
MAPK14 |
0.37uM |
24h |
LINCSCP_171109 |
LINCSCP_171109 |
YAPC |
| -0.221702 |
2.540490e-12 |
975 |
AZD8931 (Sapitinib) |
LSM-45462 |
EGFR|ERBB2|ERBB3 |
10uM |
24h |
LINCSCP_144119 |
LINCSCP_144119 |
MCF7 |
| 0.221698 |
2.542717e-12 |
975 |
Diflunisal |
LSM-2490 |
PTGS1|PTGS2 |
10uM |
6h |
LINCSCP_243170 |
LINCSCP_243170 |
MCF7 |
| 0.221682 |
2.551884e-12 |
975 |
Methyl 1-hydroxy-7-(hydroxymethyl)-1,4a,5,7a-tetrahydrocyclopenta[c]pyran-4-carboxylate |
LSM-4955 |
|
10uM |
6h |
LINCSCP_34172 |
LINCSCP_34172 |
MCF7 |
| -0.221678 |
2.554282e-12 |
975 |
Ibrutinib (PCI-32765) |
LSM-45830 |
BTK |
0.04uM |
24h |
LINCSCP_142564 |
LINCSCP_142564 |
MCF7 |
| 0.221673 |
2.557202e-12 |
975 |
N-(3-Fluoro-4-((7-methoxyquinolin-4-yl)oxy)phenyl)-1-(2-hydroxy-2-methylpropyl)-5-methyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazole-4-carboxamide |
LSM-1113 |
|
0.1uM |
6h |
LINCSCP_39551 |
LINCSCP_39551 |
MDAMB231 |
| 0.221668 |
2.560301e-12 |
975 |
Bemegride |
LSM-2325 |
GABRA1 |
0.12uM |
24h |
LINCSCP_156239 |
LINCSCP_156239 |
PC3 |
| -0.221664 |
2.562938e-12 |
975 |
UNII-5J49Q6B70F |
LSM-5877 |
TUBB |
10uM |
24h |
LINCSCP_46120 |
LINCSCP_46120 |
PC3 |
| 0.221644 |
2.574382e-12 |
975 |
AC1Q6JJ5 |
LSM-6192 |
TOP2A |
0.1uM |
6h |
LINCSCP_41825 |
LINCSCP_41825 |
NOMO1 |
| -0.221639 |
2.577338e-12 |
975 |
Oxfendazole |
LSM-1466 |
|
10uM |
24h |
LINCSCP_32821 |
LINCSCP_32821 |
MCF7 |
| -0.221635 |
2.579861e-12 |
975 |
3,7-Bis(dimethylamino)phenothiazin-5-ium |
LSM-4555 |
ACHE |
10uM |
6h |
LINCSCP_19507 |
LINCSCP_19507 |
HCC515 |
| -0.22162 |
2.588559e-12 |
975 |
Rigosertib |
LSM-44531 |
CDK1|F2R|FLT1|FYN|PDGFRA|PLK1|PLK2|SRC |
0.04uM |
24h |
LINCSCP_148252 |
LINCSCP_148252 |
NPC.CAS9 |
| -0.221615 |
2.591577e-12 |
975 |
SR-142948 |
LSM-4038 |
|
10uM |
6h |
LINCSCP_289924 |
LINCSCP_289924 |
VCAP |
| -0.221588 |
2.608160e-12 |
975 |
BRD-K18183699 |
LSM-38235 |
|
10uM |
6h |
LINCSCP_49096 |
LINCSCP_49096 |
PC3 |
| -0.221583 |
2.610811e-12 |
975 |
EMF-sumo1-1 |
|
|
10uM |
24h |
LINCSCP_164919 |
LINCSCP_164919 |
SKL.C |
| 0.221578 |
2.614302e-12 |
975 |
Nilotinib |
LSM-1099 |
ABL1|BCR|KIT |
0.37uM |
3h |
LINCSCP_163430 |
LINCSCP_163430 |
SKBR3 |
| -0.221574 |
2.616743e-12 |
975 |
SA-1458163 |
LSM-36821 |
|
10uM |
24h |
LINCSCP_41804 |
LINCSCP_41804 |
NKDBA |
| 0.221559 |
2.625786e-12 |
975 |
BRD-K00954272 |
LSM-8495 |
|
5uM |
24h |
LINCSCP_61540 |
LINCSCP_61540 |
VCAP |
| -0.221548 |
2.632341e-12 |
975 |
ascorbic-acid |
LSM-45932 |
|
10uM |
24h |
LINCSCP_122074 |
LINCSCP_122074 |
HT29 |
| -0.221538 |
2.638611e-12 |
975 |
RO 16-6941 |
LSM-2985 |
|
10uM |
6h |
LINCSCP_7712 |
LINCSCP_7712 |
A549 |
| -0.221536 |
2.639351e-12 |
975 |
Chelidonine |
LSM-2715 |
|
10uM |
24h |
LINCSCP_25267 |
LINCSCP_25267 |
HT29 |
| -0.221513 |
2.653853e-12 |
975 |
Temozolomide |
LSM-4590 |
MGMT |
10uM |
24h |
LINCSCP_121013 |
LINCSCP_121013 |
HT29 |
| -0.221504 |
2.659247e-12 |
975 |
AZD-8330 |
LSM-1165 |
MAP2K1|MAP2K2 |
0.5uM |
24h |
LINCSCP_39386 |
LINCSCP_39386 |
MDAMB231 |
| -0.221493 |
2.665648e-12 |
975 |
RG 108 |
LSM-6283 |
DNMT1 |
80uM |
6h |
LINCSCP_223125 |
LINCSCP_223125 |
HT115 |
| -0.221444 |
2.696177e-12 |
975 |
LY-294002 |
LSM-2597 |
MTOR|PIK3CA|PIK3CB|PIK3CD|PIK3CG|PLK1|PRKDC |
10uM |
24h |
LINCSCP_67526 |
LINCSCP_67526 |
MCF7 |
| -0.221439 |
2.699361e-12 |
975 |
Deforolimus |
LSM-43190 |
MTOR |
10uM |
6h |
LINCSCP_32326 |
LINCSCP_32326 |
MCF7 |
| 0.221436 |
2.701360e-12 |
975 |
3-Chloro-l-alanine |
LSM-6205 |
RPS2 |
0.5uM |
6h |
LINCSCP_51078 |
LINCSCP_51078 |
RMUGS |
| -0.221434 |
2.702387e-12 |
975 |
CHEMBL3084797 |
LSM-1261 |
|
10uM |
6h |
LINCSCP_4257 |
LINCSCP_4257 |
A549 |
| 0.221333 |
2.766355e-12 |
975 |
Flurofamide |
LSM-3502 |
|
10uM |
6h |
LINCSCP_14585 |
LINCSCP_14585 |
HA1E |
| -0.221291 |
2.792995e-12 |
975 |
Perospirone |
LSM-5912 |
DRD2|HTR2A |
10uM |
24h |
LINCSCP_58201 |
LINCSCP_58201 |
VCAP |
| 0.22126 |
2.813460e-12 |
975 |
amlodipine |
|
CACNA1C|CACNA1D|CACNA1S|CACNA2D1 |
10uM |
6h |
LINCSCP_58231 |
LINCSCP_58231 |
VCAP |
| 0.221236 |
2.829058e-12 |
975 |
9-Cis retinol |
LSM-5317 |
RARA|RARB|RARG|RORB |
40uM |
6h |
LINCSCP_4793 |
LINCSCP_4793 |
A549 |
| 0.221218 |
2.840355e-12 |
975 |
ML179 |
LSM-3734 |
|
10uM |
6h |
LINCSCP_57703 |
LINCSCP_57703 |
VCAP |
| -0.221209 |
2.846437e-12 |
975 |
BRD-8899 |
LSM-29350 |
|
0.01uM |
24h |
LINCSCP_261224 |
LINCSCP_261224 |
NOMO1 |
| -0.221198 |
2.853471e-12 |
975 |
BML-278 |
LSM-37205 |
|
10uM |
24h |
LINCSCP_43502 |
LINCSCP_43502 |
NPC |
| -0.221184 |
2.862780e-12 |
975 |
SCHEMBL618594 |
LSM-1070 |
|
10uM |
24h |
LINCSCP_149880 |
LINCSCP_149880 |
NPC.TAK |
| -0.22117 |
2.872566e-12 |
975 |
Gabexate |
LSM-3314 |
PRSS1 |
10uM |
24h |
LINCSCP_293921 |
LINCSCP_293921 |
VCAP |
| -0.221155 |
2.882507e-12 |
975 |
Camptothecin |
LSM-4611 |
TOP1 |
1.11uM |
24h |
LINCSCP_138884 |
LINCSCP_138884 |
MCF7 |
| 0.221121 |
2.904689e-12 |
975 |
BRD-K09503339 |
LSM-9005 |
|
5uM |
24h |
LINCSCP_63338 |
LINCSCP_63338 |
VCAP |
| 0.221091 |
2.924985e-12 |
975 |
BRD-K05025838 |
LSM-8732 |
|
5uM |
24h |
LINCSCP_63331 |
LINCSCP_63331 |
VCAP |
| -0.221064 |
2.943437e-12 |
975 |
Ponatinib |
LSM-1151 |
ABL1|BCR|FGFR1|FGFR2|FGFR3|FGFR4|FLT3|KIT|RET|TEK |
3.33uM |
24h |
LINCSCP_150318 |
LINCSCP_150318 |
NPC.TAK |
| 0.221063 |
2.944297e-12 |
975 |
GAP-134 (Hydrochloride) |
LSM-45532 |
|
1.11uM |
24h |
LINCSCP_72019 |
LINCSCP_72019 |
A375 |
| 0.22106 |
2.946272e-12 |
975 |
ZINC03977910 |
LSM-5391 |
NR3C1 |
10uM |
24h |
LINCSCP_34275 |
LINCSCP_34275 |
MCF7 |
| -0.221059 |
2.946667e-12 |
975 |
Wortmannin |
LSM-3947 |
PIK3CA|PIK3CG|PLK1 |
0.1uM |
6h |
LINCSCP_264456 |
LINCSCP_264456 |
PC3 |
| -0.221032 |
2.965148e-12 |
975 |
Danusertib |
LSM-5253 |
AURKA|AURKB|AURKC|FGFR1|NTRK1|RET |
10uM |
24h |
LINCSCP_135938 |
LINCSCP_135938 |
MCF7 |
| 0.221029 |
2.966932e-12 |
975 |
MLS002276502 |
LSM-3802 |
|
10uM |
24h |
LINCSCP_5013 |
LINCSCP_5013 |
A549 |
| -0.221017 |
2.975265e-12 |
975 |
BRD-K79489641 |
LSM-41607 |
|
10uM |
6h |
LINCSCP_279528 |
LINCSCP_279528 |
PC3 |
| -0.221011 |
2.979665e-12 |
975 |
Radicicol |
LSM-43303 |
|
0.1uM |
24h |
LINCSCP_67971 |
LINCSCP_67971 |
PC3 |
| 0.221009 |
2.981098e-12 |
975 |
BRD-K99191181 |
LSM-14523 |
|
5uM |
24h |
LINCSCP_61521 |
LINCSCP_61521 |
VCAP |
| -0.221005 |
2.983289e-12 |
975 |
Dactolisib |
LSM-4255 |
MTOR|PIK3CA|PIK3CB|PIK3CD|PIK3CG|PIK3R1|PIK3R2|PIK3R3|PIK3R5 |
0.5uM |
24h |
LINCSCP_25477 |
LINCSCP_25477 |
HT29 |
| 0.221004 |
2.984462e-12 |
975 |
BRD-K12450081 |
LSM-37913 |
|
30uM |
6h |
LINCSCP_309859 |
LINCSCP_309859 |
VCAP |
| -0.220987 |
2.996345e-12 |
975 |
MLS000778276 |
LSM-43118 |
|
10uM |
6h |
LINCSCP_37319 |
LINCSCP_37319 |
MCF7 |
| -0.220981 |
3.000010e-12 |
975 |
Gangleoidin Acetate |
LSM-3750 |
|
10uM |
24h |
LINCSCP_44062 |
LINCSCP_44062 |
PC3 |
| 0.220957 |
3.017113e-12 |
975 |
MLS003128682 |
LSM-40989 |
|
5uM |
24h |
LINCSCP_64307 |
LINCSCP_64307 |
VCAP |
| 0.220953 |
3.019639e-12 |
975 |
KU-55933 |
LSM-1074 |
ATM |
0.12uM |
24h |
LINCSCP_133641 |
LINCSCP_133641 |
MCF7 |
| -0.220952 |
3.020006e-12 |
975 |
Dolastatin 10 |
LSM-45943 |
|
1.11uM |
24h |
LINCSCP_143053 |
LINCSCP_143053 |
MCF7 |
| 0.220951 |
3.021231e-12 |
975 |
EX-8678 |
LSM-1147 |
|
0.12uM |
3h |
LINCSCP_145925 |
LINCSCP_145925 |
MDAMB231 |
| -0.22094 |
3.028771e-12 |
975 |
AC1L24QB |
LSM-5372 |
ADRA1A|ADRA2A |
10uM |
6h |
LINCSCP_16950 |
LINCSCP_16950 |
HA1E |
| -0.220932 |
3.034103e-12 |
975 |
AC1M9EOE |
LSM-3145 |
|
10uM |
6h |
LINCSCP_267922 |
LINCSCP_267922 |
PC3 |
| -0.220929 |
3.036447e-12 |
975 |
Tenofovir |
LSM-5340 |
|
10uM |
24h |
LINCSCP_58845 |
LINCSCP_58845 |
VCAP |
| -0.220904 |
3.054171e-12 |
975 |
Albendazole |
LSM-3782 |
|
10uM |
24h |
LINCSCP_143471 |
LINCSCP_143471 |
MCF7 |
| 0.220903 |
3.054876e-12 |
975 |
MW-STK33-100 |
LSM-44614 |
|
0.5uM |
6h |
LINCSCP_42079 |
LINCSCP_42079 |
NOMO1 |
| -0.220885 |
3.067414e-12 |
975 |
BMS-794833 |
LSM-45864 |
|
0.12uM |
24h |
LINCSCP_154138 |
LINCSCP_154138 |
PC3 |
| 0.220883 |
3.068683e-12 |
975 |
Gefitinib |
LSM-1098 |
EGFR |
1.11uM |
24h |
LINCSCP_130016 |
LINCSCP_130016 |
LNCAP |
| -0.220881 |
3.069896e-12 |
975 |
PD-0325901 |
LSM-1101 |
MAP2K1|MAP2K2 |
10uM |
3h |
LINCSCP_130158 |
LINCSCP_130158 |
LNCAP |
| -0.220839 |
3.099610e-12 |
975 |
Nafadotride |
LSM-1755 |
DRD3 |
10uM |
24h |
LINCSCP_284615 |
LINCSCP_284615 |
SKB |
| -0.220832 |
3.104695e-12 |
975 |
GSK-1070916 |
LSM-1062 |
AURKB|AURKC |
3.33uM |
24h |
LINCSCP_149913 |
LINCSCP_149913 |
NPC.TAK |
| -0.220763 |
3.154458e-12 |
975 |
Neratinib |
LSM-42778 |
EGFR|ERBB2|ERBB4 |
1.11uM |
24h |
LINCSCP_114741 |
LINCSCP_114741 |
HS578T |
| -0.220757 |
3.158899e-12 |
975 |
522-11-2 |
LSM-3052 |
|
10uM |
24h |
LINCSCP_33377 |
LINCSCP_33377 |
MCF7 |
| -0.220753 |
3.161916e-12 |
975 |
SA-1938820 |
LSM-38649 |
|
10uM |
6h |
LINCSCP_37097 |
LINCSCP_37097 |
MCF7 |
| -0.220738 |
3.173087e-12 |
975 |
MLS000583957 |
LSM-1763 |
|
10uM |
24h |
LINCSCP_32431 |
LINCSCP_32431 |
MCF7 |
| 0.220694 |
3.205291e-12 |
975 |
Temefos |
LSM-3148 |
|
10uM |
6h |
LINCSCP_240938 |
LINCSCP_240938 |
MCF7 |
| 0.220657 |
3.232581e-12 |
975 |
CHEMBL568636 |
LSM-3576 |
|
10uM |
6h |
LINCSCP_1840 |
LINCSCP_1840 |
A375 |
| -0.220619 |
3.260687e-12 |
975 |
Linezolid |
LSM-5750 |
MAOA|MAOB |
10uM |
24h |
LINCSCP_203537 |
LINCSCP_203537 |
ASC |
| -0.220617 |
3.262380e-12 |
975 |
BRD-K63513868 |
LSM-45333 |
|
10uM |
24h |
LINCSCP_24138 |
LINCSCP_24138 |
HL60 |
| -0.220596 |
3.278405e-12 |
975 |
Amthamine |
LSM-2874 |
|
10uM |
24h |
LINCSCP_11562 |
LINCSCP_11562 |
ASC |
| -0.220583 |
3.288363e-12 |
975 |
Radicicol |
LSM-43303 |
|
0.1uM |
6h |
LINCSCP_273625 |
LINCSCP_273625 |
PC3 |
| 0.220582 |
3.288767e-12 |
975 |
Ziprasidone |
LSM-5433 |
DRD2|HRH1|HTR1A|HTR1B|HTR1D|HTR1E|HTR2A|HTR2C|HTR7 |
10uM |
6h |
LINCSCP_22529 |
LINCSCP_22529 |
HEPG2 |
| -0.220563 |
3.303329e-12 |
975 |
LY2801653 |
LSM-45706 |
MET |
10uM |
24h |
LINCSCP_91142 |
LINCSCP_91142 |
HA1E |
| 0.220561 |
3.304420e-12 |
975 |
Warfarin |
LSM-1405 |
VKORC1 |
10uM |
6h |
LINCSCP_243090 |
LINCSCP_243090 |
MCF7 |
| -0.220538 |
3.322407e-12 |
975 |
SCHEMBL570779 |
LSM-1149 |
|
10uM |
3h |
LINCSCP_163259 |
LINCSCP_163259 |
SKBR3 |
| 0.220523 |
3.333498e-12 |
975 |
BRD-K29181432 |
LSM-6771 |
|
5uM |
24h |
LINCSCP_63069 |
LINCSCP_63069 |
VCAP |
| 0.2205 |
3.351475e-12 |
975 |
VX-745 |
LSM-1169 |
MAPK14 |
0.12uM |
24h |
LINCSCP_134131 |
LINCSCP_134131 |
MCF7 |
| 0.220489 |
3.359760e-12 |
975 |
BRD-K31830150 |
LSM-10360 |
|
5uM |
24h |
LINCSCP_63487 |
LINCSCP_63487 |
VCAP |
| -0.220488 |
3.360258e-12 |
975 |
Mebendazole |
LSM-3749 |
|
20uM |
24h |
LINCSCP_67611 |
LINCSCP_67611 |
MCF7 |
| 0.220463 |
3.380060e-12 |
975 |
YM 201636 |
LSM-1109 |
|
0.37uM |
24h |
LINCSCP_132135 |
LINCSCP_132135 |
MCF7 |
| -0.220452 |
3.388586e-12 |
975 |
Irinotecan |
LSM-2167 |
TOP1 |
10uM |
24h |
LINCSCP_52570 |
LINCSCP_52570 |
SKB |
| 0.220445 |
3.394367e-12 |
975 |
CHEMBL2002102 |
LSM-39063 |
|
10uM |
24h |
LINCSCP_59470 |
LINCSCP_59470 |
VCAP |
| -0.22043 |
3.405400e-12 |
975 |
SCHEMBL722708 |
LSM-4983 |
OPRD1|OPRK1|OPRM1 |
10uM |
24h |
LINCSCP_58060 |
LINCSCP_58060 |
VCAP |
| 0.220424 |
3.410196e-12 |
975 |
Retapamulin |
LSM-45949 |
|
0.12uM |
24h |
LINCSCP_71663 |
LINCSCP_71663 |
A375 |
| -0.22042 |
3.413443e-12 |
975 |
UK 356618 |
LSM-4940 |
MMP3 |
10uM |
6h |
LINCSCP_40092 |
LINCSCP_40092 |
NCIH2073 |
| -0.220417 |
3.416140e-12 |
975 |
ABT737 |
LSM-1180 |
BCL2|BCL2L1|BCL2L2 |
3.33uM |
24h |
LINCSCP_114114 |
LINCSCP_114114 |
HME1 |
| -0.22041 |
3.421479e-12 |
975 |
MLS001065903 |
LSM-2501 |
|
10uM |
6h |
LINCSCP_5098 |
LINCSCP_5098 |
A549 |
| 0.220397 |
3.431805e-12 |
975 |
CHEMBL2136735 |
LSM-1152 |
FGFR1|FGFR3|FLT1|FLT4|KDR|PDGFRA|PDGFRB |
0.12uM |
24h |
LINCSCP_69468 |
LINCSCP_69468 |
A375 |
| -0.220363 |
3.458374e-12 |
975 |
Gliclazide |
LSM-5096 |
ABCC8 |
3.33uM |
24h |
LINCSCP_171675 |
LINCSCP_171675 |
YAPC |
| -0.220361 |
3.459923e-12 |
975 |
CTK8H3236 |
LSM-1838 |
TACR1 |
10uM |
24h |
LINCSCP_43983 |
LINCSCP_43983 |
PC3 |
| 0.220344 |
3.473457e-12 |
975 |
Gallocatechin Gallate |
LSM-6228 |
BACE1|FASN |
90uM |
6h |
LINCSCP_13486 |
LINCSCP_13486 |
H1299 |
| -0.220321 |
3.492079e-12 |
975 |
Flurandrenolide |
LSM-1993 |
NR3C1 |
10uM |
24h |
LINCSCP_42823 |
LINCSCP_42823 |
NPC |
| 0.220289 |
3.517626e-12 |
975 |
BRD-K86948282 |
LSM-42014 |
|
10uM |
24h |
LINCSCP_48840 |
LINCSCP_48840 |
PC3 |
| 0.220255 |
3.545419e-12 |
975 |
BRD-K88334823 |
LSM-13858 |
|
5uM |
24h |
LINCSCP_63119 |
LINCSCP_63119 |
VCAP |
| -0.220242 |
3.555776e-12 |
975 |
Ivacaftor (VX-770) |
LSM-45975 |
CFTR |
0.04uM |
24h |
LINCSCP_158222 |
LINCSCP_158222 |
PC3 |
| -0.220218 |
3.575570e-12 |
975 |
Perhexiline |
LSM-4353 |
CPT1A|CPT2 |
1.11uM |
24h |
LINCSCP_72156 |
LINCSCP_72156 |
A375 |
| -0.220208 |
3.583716e-12 |
975 |
MLS001065872 |
LSM-3213 |
|
10uM |
24h |
LINCSCP_4972 |
LINCSCP_4972 |
A549 |
| -0.220202 |
3.589009e-12 |
975 |
AS-605240 |
LSM-42784 |
PIK3CG |
1uM |
24h |
LINCSCP_24299 |
LINCSCP_24299 |
HS578T |
| 0.220194 |
3.595503e-12 |
975 |
ALD1-H_001117 |
LSM-45107 |
|
10uM |
6h |
LINCSCP_32715 |
LINCSCP_32715 |
MCF7 |
| 0.220181 |
3.605971e-12 |
975 |
SCHEMBL16226502 |
LSM-43056 |
HSP90AA1 |
0.001uM |
24h |
LINCSCP_250719 |
LINCSCP_250719 |
MCF7 |
| 0.220179 |
3.607894e-12 |
975 |
Metaraminol |
LSM-6000 |
ADRA1A|ADRA1B|ADRA1D |
10uM |
24h |
LINCSCP_243581 |
LINCSCP_243581 |
MCF7 |
| -0.220169 |
3.615691e-12 |
975 |
Sepantronium |
LSM-5399 |
BIRC5 |
0.37uM |
24h |
LINCSCP_155388 |
LINCSCP_155388 |
PC3 |
| -0.220137 |
3.642415e-12 |
975 |
Perindopril |
LSM-4080 |
ACE |
0.12uM |
24h |
LINCSCP_103857 |
LINCSCP_103857 |
HELA |
| 0.220125 |
3.652435e-12 |
975 |
Cytarabine |
LSM-5470 |
POLA1|POLB|POLD1|POLE |
0.37uM |
24h |
LINCSCP_74127 |
LINCSCP_74127 |
A375 |
| 0.220058 |
3.709185e-12 |
975 |
GSK-J2 |
LSM-44940 |
|
0.37uM |
24h |
LINCSCP_87193 |
LINCSCP_87193 |
CD34 |
| -0.220056 |
3.710707e-12 |
975 |
Masitinib |
LSM-1130 |
FGFR3|KIT|LYN|PDGFRA|PDGFRB |
10uM |
24h |
LINCSCP_271194 |
LINCSCP_271194 |
PC3 |
| -0.220052 |
3.714755e-12 |
975 |
Olanzapine |
LSM-5359 |
DRD1|DRD2|DRD3|DRD4|HRH1|HTR1A|HTR1B|HTR1D|HTR1E|HTR2A|HTR2C|HTR6|HTR7 |
3.33uM |
24h |
LINCSCP_154507 |
LINCSCP_154507 |
PC3 |
| -0.22002 |
3.741750e-12 |
975 |
CHEMBL1478888 |
LSM-6413 |
|
10uM |
6h |
LINCSCP_33961 |
LINCSCP_33961 |
MCF7 |
| -0.219987 |
3.770211e-12 |
975 |
TAS-103 (dihydrochloride) |
LSM-45292 |
|
10uM |
24h |
LINCSCP_136082 |
LINCSCP_136082 |
MCF7 |
| -0.219981 |
3.775098e-12 |
975 |
MLS000778276 |
LSM-43118 |
|
3uM |
24h |
LINCSCP_37235 |
LINCSCP_37235 |
MCF7 |
| 0.219944 |
3.807922e-12 |
975 |
CHEMBL3182395 |
LSM-1164 |
MAP2K5|MAPK7 |
0.12uM |
24h |
LINCSCP_113747 |
LINCSCP_113747 |
HME1 |
| -0.219848 |
3.892605e-12 |
975 |
Broad-Sai-560 |
LSM-45991 |
|
10uM |
24h |
LINCSCP_43508 |
LINCSCP_43508 |
NPC |
| -0.219836 |
3.903263e-12 |
975 |
BRD-K05174693 |
LSM-37543 |
|
10uM |
24h |
LINCSCP_309974 |
LINCSCP_309974 |
VCAP |
| 0.219813 |
3.923483e-12 |
975 |
MLS002474283 |
LSM-6132 |
|
10uM |
6h |
LINCSCP_32345 |
LINCSCP_32345 |
MCF7 |
| 0.219813 |
3.924058e-12 |
975 |
MLS000589843 |
LSM-43120 |
|
1uM |
24h |
LINCSCP_55117 |
LINCSCP_55117 |
THP1 |
| 0.219773 |
3.959955e-12 |
975 |
BRD-K40506152 |
LSM-10901 |
|
5uM |
24h |
LINCSCP_61778 |
LINCSCP_61778 |
VCAP |
| 0.219762 |
3.969690e-12 |
975 |
Masitinib |
LSM-1130 |
FGFR3|KIT|LYN|PDGFRA|PDGFRB |
10uM |
6h |
LINCSCP_32735 |
LINCSCP_32735 |
MCF7 |
| -0.219758 |
3.973299e-12 |
975 |
BRD-K71387353 |
LSM-12794 |
|
10uM |
24h |
LINCSCP_28286 |
LINCSCP_28286 |
HT29 |
| -0.219756 |
3.975056e-12 |
975 |
PLX-4720 |
LSM-1049 |
BRAF |
10uM |
24h |
LINCSCP_116361 |
LINCSCP_116361 |
HT29 |
| 0.219756 |
3.975325e-12 |
975 |
BRD-K55612480 |
LSM-40319 |
|
10uM |
6h |
LINCSCP_32343 |
LINCSCP_32343 |
MCF7 |
| 0.219741 |
3.988464e-12 |
975 |
2-Cyano-3-(3,4-dihydroxyphenyl)-n-phenylprop-2-enamide |
LSM-2755 |
EGFR |
10uM |
24h |
LINCSCP_52650 |
LINCSCP_52650 |
SKB |
| 0.219707 |
4.020186e-12 |
975 |
BRD-K66186977 |
LSM-8320 |
|
5uM |
24h |
LINCSCP_60794 |
LINCSCP_60794 |
VCAP |
| 0.219702 |
4.024758e-12 |
975 |
ICI 162846 |
LSM-3484 |
|
0.37uM |
24h |
LINCSCP_72719 |
LINCSCP_72719 |
A375 |
| -0.219696 |
4.030234e-12 |
975 |
MK-5108 |
LSM-36812 |
AURKA|AURKB |
1.11uM |
24h |
LINCSCP_136874 |
LINCSCP_136874 |
MCF7 |
| -0.219631 |
4.090539e-12 |
975 |
CHEMBL2143415 |
LSM-6085 |
|
3uM |
6h |
LINCSCP_37082 |
LINCSCP_37082 |
MCF7 |
| -0.219619 |
4.102183e-12 |
975 |
AM 281 |
LSM-3318 |
CNR1 |
10uM |
6h |
LINCSCP_25372 |
LINCSCP_25372 |
HT29 |
| 0.219616 |
4.104947e-12 |
975 |
BRD-K93779718 |
LSM-15076 |
|
3uM |
6h |
LINCSCP_38112 |
LINCSCP_38112 |
MCF7 |
| -0.219612 |
4.108544e-12 |
975 |
Buparlisib |
LSM-1148 |
PIK3CA|PIK3CB|PIK3CD|PIK3CG|PIK3R1|PIK3R2|PIK3R3|PIK3R5 |
10uM |
24h |
LINCSCP_116295 |
LINCSCP_116295 |
HT29 |
| -0.219585 |
4.133932e-12 |
975 |
BRD-K24026396 |
LSM-14766 |
|
5uM |
24h |
LINCSCP_64177 |
LINCSCP_64177 |
VCAP |
| 0.219575 |
4.143600e-12 |
975 |
BRD-8899 |
LSM-29350 |
|
10uM |
24h |
LINCSCP_239426 |
LINCSCP_239426 |
MCF7 |
| -0.219555 |
4.162436e-12 |
975 |
PF-03758309 |
LSM-4254 |
PAK4 |
3.33uM |
24h |
LINCSCP_114441 |
LINCSCP_114441 |
HME1 |
| -0.219552 |
4.165732e-12 |
975 |
NSC95397 |
LSM-3521 |
|
10uM |
24h |
LINCSCP_267320 |
LINCSCP_267320 |
PC3 |
| -0.219545 |
4.171653e-12 |
975 |
Dapivirine (TMC120) |
LSM-45463 |
|
3.33uM |
24h |
LINCSCP_104448 |
LINCSCP_104448 |
HELA |
| -0.219544 |
4.172813e-12 |
975 |
SA-97110 |
LSM-37431 |
|
3uM |
6h |
LINCSCP_37070 |
LINCSCP_37070 |
MCF7 |
| 0.219501 |
4.213909e-12 |
975 |
ZINC21986197 |
LSM-5392 |
|
10uM |
24h |
LINCSCP_34276 |
LINCSCP_34276 |
MCF7 |
| -0.219499 |
4.215880e-12 |
975 |
IOX2 |
LSM-6339 |
|
0.04uM |
24h |
LINCSCP_114106 |
LINCSCP_114106 |
HME1 |
| 0.219493 |
4.222121e-12 |
975 |
ethyl 6-(2,3-dihydro-1H-indol-1-ylmethyl)-4-(3-nitrophenyl)-2-oxo-1,2,3,4-tetrahydro-5-pyrimidinecarboxylate |
LSM-45350 |
|
0.5uM |
24h |
LINCSCP_222102 |
LINCSCP_222102 |
HL60 |
| -0.219468 |
4.245890e-12 |
975 |
SA-1919710 |
LSM-39226 |
|
3uM |
24h |
LINCSCP_41723 |
LINCSCP_41723 |
NKDBA |
| -0.219447 |
4.266923e-12 |
975 |
CHEMBL1965031 |
LSM-6684 |
|
10uM |
6h |
LINCSCP_16900 |
LINCSCP_16900 |
HA1E |
| -0.219442 |
4.271738e-12 |
975 |
Methyllycaconitine |
LSM-1457 |
CHRNA7 |
10uM |
6h |
LINCSCP_241722 |
LINCSCP_241722 |
MCF7 |
| -0.219437 |
4.276489e-12 |
975 |
Calcitriol |
LSM-45950 |
|
0.37uM |
24h |
LINCSCP_89509 |
LINCSCP_89509 |
HA1E |
| -0.219401 |
4.311377e-12 |
975 |
CHEMBL1593913 |
LSM-3929 |
|
10uM |
6h |
LINCSCP_225502 |
LINCSCP_225502 |
HT29 |
| -0.2194 |
4.312525e-12 |
975 |
Pinacidil |
LSM-1557 |
ABCC8|ABCC9 |
0.12uM |
24h |
LINCSCP_122576 |
LINCSCP_122576 |
HT29 |
| 0.2194 |
4.312882e-12 |
975 |
Mifobate |
LSM-1761 |
PPARG |
3.33uM |
24h |
LINCSCP_97500 |
LINCSCP_97500 |
HA1E |
| -0.219388 |
4.324085e-12 |
975 |
BRD-K74671783 |
LSM-13005 |
|
1uM |
6h |
LINCSCP_37824 |
LINCSCP_37824 |
MCF7 |
| 0.219388 |
4.324985e-12 |
975 |
Pranoprofen |
LSM-5110 |
|
10uM |
24h |
LINCSCP_34454 |
LINCSCP_34454 |
MCF7 |
| -0.219387 |
4.325762e-12 |
975 |
BRD-K81732150 |
LSM-43610 |
|
10uM |
24h |
LINCSCP_65708 |
LINCSCP_65708 |
VCAP |
| -0.219375 |
4.337258e-12 |
975 |
MLS002264379 |
LSM-2753 |
|
10uM |
6h |
LINCSCP_45807 |
LINCSCP_45807 |
PC3 |
| 0.219371 |
4.341131e-12 |
975 |
4-[(6-Amino-4-pyrimidinyl)amino]benzenesulfonamide |
LSM-3612 |
|
10uM |
24h |
LINCSCP_284788 |
LINCSCP_284788 |
SKB |
| -0.219369 |
4.343810e-12 |
975 |
Ponatinib |
LSM-1151 |
ABL1|BCR|FGFR1|FGFR2|FGFR3|FGFR4|FLT3|KIT|RET|TEK |
0.1uM |
24h |
LINCSCP_39413 |
LINCSCP_39413 |
MDAMB231 |
| -0.219364 |
4.348610e-12 |
975 |
Genz-644282 |
LSM-45838 |
|
0.04uM |
24h |
LINCSCP_143224 |
LINCSCP_143224 |
MCF7 |
| 0.219349 |
4.363338e-12 |
975 |
Lamivudine |
LSM-5215 |
|
10uM |
6h |
LINCSCP_292994 |
LINCSCP_292994 |
VCAP |
| 0.219348 |
4.363989e-12 |
975 |
Indigo Red |
LSM-42899 |
CDK1|CDK5|GSK3A |
10uM |
24h |
LINCSCP_71635 |
LINCSCP_71635 |
A375 |
| -0.21934 |
4.372607e-12 |
975 |
MLS001065900 |
LSM-3925 |
|
10uM |
24h |
LINCSCP_31662 |
LINCSCP_31662 |
MCF7 |
| 0.219322 |
4.389983e-12 |
975 |
Imatinib |
LSM-1023 |
ABL1|BCR|CSF1R|KIT|PDGFRA|PDGFRB |
10uM |
24h |
LINCSCP_131432 |
LINCSCP_131432 |
MCF10A |
| 0.219321 |
4.391285e-12 |
975 |
Indomethacin |
LSM-3275 |
PPARG|PTGDR2|PTGS1|PTGS2 |
0.12uM |
24h |
LINCSCP_157449 |
LINCSCP_157449 |
PC3 |
| -0.21925 |
4.463072e-12 |
975 |
GSK-1070916 |
LSM-1062 |
AURKB|AURKC |
3.33uM |
24h |
LINCSCP_147757 |
LINCSCP_147757 |
NPC.CAS9 |
| -0.219217 |
4.496970e-12 |
975 |
BRD-K37299375 |
LSM-10679 |
|
10uM |
24h |
LINCSCP_312309 |
LINCSCP_312309 |
VCAP |
| -0.219213 |
4.501320e-12 |
975 |
Regorafenib |
LSM-1226 |
ABL1|BRAF|DDR2|FGFR1|FGFR2|FLT1|FLT4|FRK|KDR|KIT|MAPK11|PDGFRA|PDGFRB|RAF1|RET|TEK |
0.12uM |
24h |
LINCSCP_153191 |
LINCSCP_153191 |
PC3 |
| 0.219196 |
4.518382e-12 |
975 |
BRD-K52111234 |
LSM-40150 |
|
10uM |
24h |
LINCSCP_272057 |
LINCSCP_272057 |
PC3 |
| 0.219179 |
4.536133e-12 |
975 |
AT 7867 |
LSM-1155 |
|
0.12uM |
24h |
LINCSCP_86848 |
LINCSCP_86848 |
CD34 |
| -0.219157 |
4.558817e-12 |
975 |
Benzonatate |
LSM-4052 |
SCN5A |
10uM |
24h |
LINCSCP_21433 |
LINCSCP_21433 |
HEK293T |
| 0.219154 |
4.562161e-12 |
975 |
UCL 2077 |
LSM-3106 |
|
10uM |
6h |
LINCSCP_14273 |
LINCSCP_14273 |
HA1E |
| -0.219147 |
4.569054e-12 |
975 |
Dacomitinib |
LSM-42808 |
EGFR|ERBB2|ERBB3|ERBB4 |
10uM |
24h |
LINCSCP_123075 |
LINCSCP_123075 |
HT29 |
| -0.219147 |
4.569370e-12 |
975 |
AC1Q6JJ5 |
LSM-6192 |
TOP2A |
1uM |
24h |
LINCSCP_9673 |
LINCSCP_9673 |
A549 |
| 0.21914 |
4.576468e-12 |
975 |
Antazoline |
LSM-6023 |
HRH1 |
10uM |
24h |
LINCSCP_243591 |
LINCSCP_243591 |
MCF7 |
| -0.219134 |
4.583264e-12 |
975 |
AC1MJ3VH |
LSM-1731 |
TOP2A |
1.11uM |
24h |
LINCSCP_137018 |
LINCSCP_137018 |
MCF7 |
| 0.21909 |
4.628882e-12 |
975 |
179324-69-7 |
LSM-6281 |
ADRM1|PSMA1|PSMA2|PSMA3|PSMA4|PSMA5|PSMA6|PSMA7|PSMA8|PSMB1|PSMB10|PSMB11|PSMB2|PSMB3|PSMB4|PSMB5|PSMB6|PSMB7|PSMB8|PSMB9|PSMC1|PSMC2|PSMC3|PSMC4|PSMC5|PSMC6|PSMD1|PSMD11|PSMD12|PSMD13|PSMD14|PSMD2|PSMD3|PSMD4|PSMD6|PSMD7|PSMD8|SEM1 |
0.01uM |
6h |
LINCSCP_53512 |
LINCSCP_53512 |
SKMEL28 |
| -0.219074 |
4.646408e-12 |
975 |
MLS003448162 |
LSM-3552 |
|
10uM |
24h |
LINCSCP_237408 |
LINCSCP_237408 |
MCF7 |
| 0.219068 |
4.651974e-12 |
975 |
BRD-K19724753 |
LSM-43375 |
|
5uM |
24h |
LINCSCP_60010 |
LINCSCP_60010 |
VCAP |
| 0.219061 |
4.660321e-12 |
975 |
AT 7867 |
LSM-1155 |
|
0.04uM |
24h |
LINCSCP_84369 |
LINCSCP_84369 |
ASC |
| -0.219058 |
4.663335e-12 |
975 |
Dinoprostone |
LSM-42919 |
PTGER1|PTGER2|PTGER3|PTGER4 |
10uM |
24h |
LINCSCP_262611 |
LINCSCP_262611 |
NPC |
| -0.219022 |
4.701942e-12 |
975 |
Thioguanosine |
LSM-5832 |
|
0.37uM |
24h |
LINCSCP_175141 |
LINCSCP_175141 |
YAPC |
| 0.219021 |
4.702760e-12 |
975 |
MLS001065877 |
LSM-3888 |
|
10uM |
6h |
LINCSCP_5171 |
LINCSCP_5171 |
A549 |
| 0.219006 |
4.718481e-12 |
975 |
Linsitinib |
LSM-1135 |
IGF1R|INSR |
0.1uM |
24h |
LINCSCP_39360 |
LINCSCP_39360 |
MDAMB231 |
| -0.218994 |
4.731313e-12 |
975 |
Selumetinib |
LSM-1056 |
MAP2K1|MAP2K2 |
80uM |
24h |
LINCSCP_4559 |
LINCSCP_4559 |
A549 |
| 0.218983 |
4.743736e-12 |
975 |
BRD-K64877338 |
LSM-45344 |
|
10uM |
24h |
LINCSCP_205487 |
LINCSCP_205487 |
CD34 |
| -0.218959 |
4.770158e-12 |
975 |
PLX-4720 |
LSM-1049 |
BRAF |
10uM |
3h |
LINCSCP_132408 |
LINCSCP_132408 |
MCF7 |
| 0.218929 |
4.802660e-12 |
975 |
BRD-K11787592 |
LSM-9142 |
|
5uM |
24h |
LINCSCP_61555 |
LINCSCP_61555 |
VCAP |
| -0.218898 |
4.836759e-12 |
975 |
COT-10B |
LSM-6226 |
|
1uM |
6h |
LINCSCP_9570 |
LINCSCP_9570 |
A549 |
| 0.218879 |
4.857205e-12 |
975 |
(1S,2R)-Phenylpropanolamine |
LSM-5416 |
|
10uM |
24h |
LINCSCP_34279 |
LINCSCP_34279 |
MCF7 |
| -0.218876 |
4.861114e-12 |
975 |
BRD-K81860076 |
LSM-41740 |
|
5uM |
24h |
LINCSCP_231877 |
LINCSCP_231877 |
HT29 |
| -0.218835 |
4.906949e-12 |
975 |
Erlotinib |
LSM-1097 |
EGFR |
1.11uM |
24h |
LINCSCP_99638 |
LINCSCP_99638 |
HCC515 |
| -0.218797 |
4.948843e-12 |
975 |
BAS 09531330 |
LSM-32192 |
|
0.5uM |
24h |
LINCSCP_12380 |
LINCSCP_12380 |
CD34 |
| 0.218784 |
4.964005e-12 |
975 |
AZD-1775 |
LSM-1153 |
WEE1 |
10uM |
6h |
LINCSCP_53587 |
LINCSCP_53587 |
SNGM |
| 0.218774 |
4.974927e-12 |
975 |
BRD-K70711508 |
LSM-41121 |
|
10uM |
24h |
LINCSCP_35237 |
LINCSCP_35237 |
MCF7 |
| 0.218767 |
4.983550e-12 |
975 |
Propranolol |
LSM-4329 |
ADRB1|ADRB2|ADRB3 |
0.04uM |
24h |
LINCSCP_154391 |
LINCSCP_154391 |
PC3 |
| 0.218758 |
4.993078e-12 |
975 |
17-DMAG (Alvespimycin) HCl |
LSM-46133 |
|
0.04uM |
24h |
LINCSCP_167041 |
LINCSCP_167041 |
YAPC |
| -0.218725 |
5.031377e-12 |
975 |
SA-1939064 |
LSM-40654 |
|
10uM |
6h |
LINCSCP_37157 |
LINCSCP_37157 |
MCF7 |
| -0.21872 |
5.036985e-12 |
975 |
Alvocidib |
LSM-1011 |
CDK1|CDK2|CDK4|CDK5|CDK6|CDK7|CDK8|CDK9|EGFR|PYGM |
0.01uM |
24h |
LINCSCP_9749 |
LINCSCP_9749 |
A549 |
| 0.218717 |
5.040624e-12 |
975 |
BRD-K38311495 |
LSM-10749 |
|
5uM |
24h |
LINCSCP_61226 |
LINCSCP_61226 |
VCAP |
| -0.218716 |
5.040889e-12 |
975 |
1,4-Diamino-2,3-dicyano-1,4-bis(methylthio)butadiene |
LSM-42967 |
|
10uM |
6h |
LINCSCP_223900 |
LINCSCP_223900 |
HT29 |
| 0.21871 |
5.047903e-12 |
975 |
BRD-K22080587 |
LSM-9765 |
|
5uM |
24h |
LINCSCP_48235 |
LINCSCP_48235 |
PC3 |
| 0.218698 |
5.061598e-12 |
975 |
FPA1_000301 |
LSM-36736 |
|
10uM |
24h |
LINCSCP_239969 |
LINCSCP_239969 |
MCF7 |
| -0.218682 |
5.081194e-12 |
975 |
Carfilzomib (PR-171) |
LSM-45547 |
ADRM1|PSMA1|PSMA2|PSMA3|PSMA4|PSMA5|PSMA6|PSMA7|PSMA8|PSMB1|PSMB10|PSMB11|PSMB2|PSMB3|PSMB4|PSMB5|PSMB6|PSMB7|PSMB8|PSMB9|PSMC1|PSMC2|PSMC3|PSMC4|PSMC5|PSMC6|PSMD1|PSMD11|PSMD12|PSMD13|PSMD14|PSMD2|PSMD3|PSMD4|PSMD6|PSMD7|PSMD8|SEM1 |
3.33uM |
24h |
LINCSCP_169879 |
LINCSCP_169879 |
YAPC |
| 0.218675 |
5.089171e-12 |
975 |
STK327831 |
LSM-2865 |
|
10uM |
6h |
LINCSCP_31066 |
LINCSCP_31066 |
MCF7 |
| -0.218673 |
5.091486e-12 |
975 |
ABT-751 |
LSM-6285 |
|
10uM |
24h |
LINCSCP_45052 |
LINCSCP_45052 |
PC3 |
| 0.218664 |
5.101319e-12 |
975 |
Yohimbine |
LSM-2779 |
ADRA2A|ADRA2B|ADRA2C|HTR1A|HTR1B|HTR1D|HTR2B |
1.11uM |
24h |
LINCSCP_71995 |
LINCSCP_71995 |
A375 |
| -0.218662 |
5.103467e-12 |
975 |
CHEMBL1982812 |
LSM-6576 |
|
10uM |
6h |
LINCSCP_295791 |
LINCSCP_295791 |
VCAP |
| -0.218643 |
5.126005e-12 |
975 |
SMR000250171 |
LSM-4145 |
|
10uM |
24h |
LINCSCP_268263 |
LINCSCP_268263 |
PC3 |
| -0.218641 |
5.128435e-12 |
975 |
SCHEMBL3958507 |
LSM-5245 |
COQ8B|EGFR |
0.04uM |
3h |
LINCSCP_131501 |
LINCSCP_131501 |
MCF10A |
| -0.218627 |
5.144768e-12 |
975 |
BRD-K68319707 |
LSM-40988 |
|
10uM |
24h |
LINCSCP_43036 |
LINCSCP_43036 |
NPC |
| -0.218623 |
5.149380e-12 |
975 |
Epirubicin HCl |
LSM-45684 |
|
0.37uM |
24h |
LINCSCP_139629 |
LINCSCP_139629 |
MCF7 |
| 0.218619 |
5.154170e-12 |
975 |
Risperidone |
LSM-3193 |
ADRA1A|ADRA1B|DRD2|DRD3|DRD4|HRH1|HTR1A|HTR1D|HTR2A|HTR2C |
1.11uM |
24h |
LINCSCP_76554 |
LINCSCP_76554 |
A375 |
| -0.218611 |
5.163341e-12 |
975 |
BRD-K43226598 |
LSM-39644 |
|
10uM |
6h |
LINCSCP_47213 |
LINCSCP_47213 |
PC3 |
| 0.21858 |
5.200439e-12 |
975 |
SCHEMBL17052537 |
LSM-5803 |
BTK|JAK3|MKNK2|MTOR|PRKDC |
0.12uM |
3h |
LINCSCP_113437 |
LINCSCP_113437 |
HME1 |
| -0.218577 |
5.203944e-12 |
975 |
VX-702 |
LSM-5252 |
MAPK14 |
10uM |
6h |
LINCSCP_46937 |
LINCSCP_46937 |
PC3 |
| -0.218557 |
5.227553e-12 |
975 |
GW843682X |
LSM-1014 |
PLK1|PLK3 |
1uM |
24h |
LINCSCP_254365 |
LINCSCP_254365 |
MCF7 |
| 0.218538 |
5.249842e-12 |
975 |
L-161,982 |
LSM-2875 |
PTGER4 |
10uM |
6h |
LINCSCP_220525 |
LINCSCP_220525 |
HEPG2 |
| -0.218533 |
5.256150e-12 |
975 |
BAY 61-3606 |
LSM-1167 |
SYK |
10uM |
24h |
LINCSCP_112758 |
LINCSCP_112758 |
HEPG2 |
| -0.218522 |
5.269274e-12 |
975 |
1,3-Dipropyl-8-cyclopentylxanthine |
LSM-19971 |
|
0.12uM |
24h |
LINCSCP_170440 |
LINCSCP_170440 |
YAPC |
| -0.218521 |
5.270129e-12 |
975 |
Trichlorfon |
LSM-4995 |
ACHE |
10uM |
24h |
LINCSCP_243345 |
LINCSCP_243345 |
MCF7 |
| -0.2185 |
5.296167e-12 |
975 |
nifedipine |
LSM-4176 |
CACNA1C|CACNA1D|CACNA1F|CACNA1S|CACNA2D1 |
10uM |
6h |
LINCSCP_46133 |
LINCSCP_46133 |
PC3 |
| 0.21849 |
5.307911e-12 |
975 |
CHEMBL2203528 |
LSM-36795 |
|
3uM |
6h |
LINCSCP_261281 |
LINCSCP_261281 |
NOMO1 |
| -0.218476 |
5.325095e-12 |
975 |
Tamatinib |
LSM-1040 |
SYK |
10uM |
6h |
LINCSCP_4730 |
LINCSCP_4730 |
A549 |
| -0.218456 |
5.349180e-12 |
975 |
DOCETAXEL |
LSM-45649 |
|
0.04uM |
24h |
LINCSCP_138263 |
LINCSCP_138263 |
MCF7 |
| -0.218441 |
5.367762e-12 |
975 |
BRD-K97235918 |
LSM-14404 |
|
5uM |
6h |
LINCSCP_62600 |
LINCSCP_62600 |
VCAP |
| -0.218432 |
5.377784e-12 |
975 |
Thioridazine |
LSM-1863 |
DRD1|DRD2|DRD3|DRD4|HTR2A|HTR2C |
10uM |
6h |
LINCSCP_257288 |
LINCSCP_257288 |
NCIH508 |
| -0.21843 |
5.381237e-12 |
975 |
MLS001065891 |
LSM-3963 |
|
10uM |
24h |
LINCSCP_31020 |
LINCSCP_31020 |
MCF7 |
| 0.218427 |
5.384222e-12 |
975 |
ZINC01045466 |
LSM-4913 |
|
10uM |
6h |
LINCSCP_217368 |
LINCSCP_217368 |
HCC515 |
| -0.218411 |
5.404450e-12 |
975 |
CHEMBL2134588 |
LSM-42520 |
|
5uM |
24h |
LINCSCP_3468 |
LINCSCP_3468 |
A375 |
| -0.2184 |
5.417499e-12 |
975 |
CDK4 Inhibitor III |
LSM-2121 |
CDK4 |
10uM |
24h |
LINCSCP_284651 |
LINCSCP_284651 |
SKB |
| 0.21838 |
5.441992e-12 |
975 |
Dexniguldipine |
LSM-15285 |
|
0.37uM |
24h |
LINCSCP_122569 |
LINCSCP_122569 |
HT29 |
| 0.218374 |
5.449608e-12 |
975 |
BRD-K76688030 |
LSM-13122 |
|
5uM |
24h |
LINCSCP_302168 |
LINCSCP_302168 |
VCAP |
| -0.218351 |
5.478202e-12 |
975 |
AZD-1152-HQPA |
LSM-1067 |
AURKA|AURKB |
1uM |
24h |
LINCSCP_11764 |
LINCSCP_11764 |
BT20 |
| 0.218348 |
5.482317e-12 |
975 |
GW843682X |
LSM-1014 |
PLK1|PLK3 |
10uM |
6h |
LINCSCP_55550 |
LINCSCP_55550 |
U937 |
| 0.218346 |
5.484064e-12 |
975 |
MK-8245 |
LSM-45756 |
|
0.12uM |
24h |
LINCSCP_71305 |
LINCSCP_71305 |
A375 |
| -0.218334 |
5.499229e-12 |
975 |
BRD-K80213755 |
LSM-13329 |
|
5uM |
24h |
LINCSCP_62044 |
LINCSCP_62044 |
VCAP |
| -0.218234 |
5.625478e-12 |
975 |
Setiptiline |
LSM-45982 |
|
0.04uM |
24h |
LINCSCP_72082 |
LINCSCP_72082 |
A375 |
| 0.218234 |
5.626376e-12 |
975 |
Pracinostat |
LSM-43290 |
|
0.12uM |
24h |
LINCSCP_108639 |
LINCSCP_108639 |
HELA |
| 0.218224 |
5.639013e-12 |
975 |
AT-9283 |
LSM-37023 |
ABL1|AURKA|AURKB|FLT3|JAK2|JAK3 |
0.04uM |
24h |
LINCSCP_168462 |
LINCSCP_168462 |
YAPC |
| 0.218218 |
5.646752e-12 |
975 |
Ranitidine |
LSM-42886 |
HRH2 |
10uM |
6h |
LINCSCP_2638 |
LINCSCP_2638 |
A375 |
| 0.218217 |
5.648019e-12 |
975 |
BRD-K41087962 |
LSM-42690 |
|
0.5uM |
6h |
LINCSCP_29340 |
LINCSCP_29340 |
LOVO |
| 0.218215 |
5.650332e-12 |
975 |
BRD-K71714567 |
LSM-41172 |
|
10uM |
6h |
LINCSCP_38086 |
LINCSCP_38086 |
MCF7 |
| 0.218202 |
5.667594e-12 |
975 |
Erlotinib |
LSM-1097 |
EGFR |
10uM |
3h |
LINCSCP_145209 |
LINCSCP_145209 |
MDAMB231 |
| 0.218182 |
5.692837e-12 |
975 |
BRD-K84145110 |
LSM-41871 |
|
5uM |
24h |
LINCSCP_3418 |
LINCSCP_3418 |
A375 |
| 0.218134 |
5.755354e-12 |
975 |
Fadrozole |
LSM-5015 |
CYP19A1 |
1.11uM |
24h |
LINCSCP_72383 |
LINCSCP_72383 |
A375 |
| 0.218131 |
5.759286e-12 |
975 |
Proparacaine |
LSM-3780 |
SCN10A|SCN11A|SCN1A|SCN2A|SCN3A|SCN4A|SCN5A|SCN7A|SCN8A|SCN9A |
10uM |
6h |
LINCSCP_228014 |
LINCSCP_228014 |
HT29 |
| 0.218124 |
5.768647e-12 |
975 |
Phenothiazine |
LSM-3324 |
|
10uM |
6h |
LINCSCP_216500 |
LINCSCP_216500 |
HCC515 |
| -0.218119 |
5.774632e-12 |
975 |
CHEMBL2359886 |
LSM-6824 |
|
10uM |
24h |
LINCSCP_49488 |
LINCSCP_49488 |
PC3 |
| 0.218106 |
5.792636e-12 |
975 |
MK-8245 |
LSM-45756 |
|
0.37uM |
24h |
LINCSCP_71304 |
LINCSCP_71304 |
A375 |
| 0.218087 |
5.817033e-12 |
975 |
Quizartinib |
LSM-1037 |
CSF1R|FLT3|KIT|PDGFRA|PDGFRB|RET |
0.5uM |
6h |
LINCSCP_39307 |
LINCSCP_39307 |
MDAMB231 |
| 0.218077 |
5.830901e-12 |
975 |
SA-84512 |
LSM-39138 |
|
10uM |
6h |
LINCSCP_20610 |
LINCSCP_20610 |
HCC515 |
| -0.218035 |
5.886252e-12 |
975 |
CHEMBL3186447 |
LSM-42507 |
|
10uM |
6h |
LINCSCP_65895 |
LINCSCP_65895 |
VCAP |
| -0.218017 |
5.910111e-12 |
975 |
altrenogest |
LSM-45498 |
|
3.33uM |
24h |
LINCSCP_123272 |
LINCSCP_123272 |
HT29 |
| 0.218004 |
5.927270e-12 |
975 |
TGX 221 |
LSM-1172 |
PIK3CB |
0.12uM |
24h |
LINCSCP_130599 |
LINCSCP_130599 |
MCF10A |
| -0.217993 |
5.942153e-12 |
975 |
PCL2_000154 |
LSM-36683 |
|
10uM |
24h |
LINCSCP_32178 |
LINCSCP_32178 |
MCF7 |
| 0.217989 |
5.948637e-12 |
975 |
MLS003649983 |
LSM-12616 |
|
5uM |
24h |
LINCSCP_61812 |
LINCSCP_61812 |
VCAP |
| 0.217984 |
5.955248e-12 |
975 |
MLS-0091943.0001 |
LSM-42868 |
|
10uM |
6h |
LINCSCP_20406 |
LINCSCP_20406 |
HCC515 |
| -0.217959 |
5.988167e-12 |
975 |
SA-1939064 |
LSM-40654 |
|
3uM |
6h |
LINCSCP_37159 |
LINCSCP_37159 |
MCF7 |
| 0.217956 |
5.992248e-12 |
975 |
Indigo Red |
LSM-42899 |
CDK1|CDK5|GSK3A |
0.04uM |
24h |
LINCSCP_71640 |
LINCSCP_71640 |
A375 |
| -0.217951 |
5.999510e-12 |
975 |
Practolol |
LSM-1531 |
ADRB1 |
10uM |
24h |
LINCSCP_272427 |
LINCSCP_272427 |
PC3 |
| 0.217939 |
6.016662e-12 |
975 |
ICI 162846 |
LSM-3484 |
|
10uM |
24h |
LINCSCP_72716 |
LINCSCP_72716 |
A375 |
| -0.217921 |
6.040906e-12 |
975 |
Colchicine |
LSM-5199 |
TUBA1A|TUBA1B|TUBA1C|TUBA3E|TUBA4A|TUBB|TUBB1|TUBB2A|TUBB2B|TUBB3|TUBB4A|TUBB4B|TUBB6|TUBB8 |
0.37uM |
24h |
LINCSCP_156675 |
LINCSCP_156675 |
PC3 |
| 0.217919 |
6.043515e-12 |
975 |
CP466722 |
LSM-1009 |
ATM |
0.5uM |
24h |
LINCSCP_51321 |
LINCSCP_51321 |
SKBR3 |
| -0.217891 |
6.082379e-12 |
975 |
altrenogest |
LSM-45498 |
|
1.11uM |
24h |
LINCSCP_139856 |
LINCSCP_139856 |
MCF7 |
| -0.217878 |
6.099482e-12 |
975 |
MG-132 |
LSM-1107 |
PSMB1 |
3uM |
24h |
LINCSCP_36274 |
LINCSCP_36274 |
MCF7 |
| 0.217848 |
6.141797e-12 |
975 |
GSK-1904529A |
LSM-1134 |
IGF1R|INSR |
0.37uM |
24h |
LINCSCP_69485 |
LINCSCP_69485 |
A375 |
| 0.217828 |
6.169607e-12 |
975 |
Glipizide |
LSM-2251 |
ABCC8|KCNJ11 |
0.37uM |
24h |
LINCSCP_92580 |
LINCSCP_92580 |
HA1E |
| -0.217827 |
6.170713e-12 |
975 |
Lurasidone |
LSM-45843 |
DRD2|HTR2A |
10uM |
24h |
LINCSCP_123319 |
LINCSCP_123319 |
HT29 |
| 0.217827 |
6.171640e-12 |
975 |
BMS-345541 |
LSM-1028 |
IKBKB |
0.37uM |
24h |
LINCSCP_131197 |
LINCSCP_131197 |
MCF10A |
| -0.217826 |
6.172381e-12 |
975 |
SA-1939126 |
LSM-39500 |
|
10uM |
6h |
LINCSCP_37128 |
LINCSCP_37128 |
MCF7 |
| 0.217808 |
6.198023e-12 |
975 |
SMR000068650 |
LSM-2859 |
|
100uM |
24h |
LINCSCP_710 |
LINCSCP_710 |
A375 |
| -0.21778 |
6.236537e-12 |
975 |
CHEMBL1083527 |
LSM-1122 |
|
1.11uM |
24h |
LINCSCP_114831 |
LINCSCP_114831 |
HS578T |
| 0.217768 |
6.254773e-12 |
975 |
Nimodipine |
LSM-1659 |
CACNA1C|CACNA1D|CACNA1F|CACNA1S|NR3C2 |
0.12uM |
24h |
LINCSCP_123103 |
LINCSCP_123103 |
HT29 |
| -0.217752 |
6.276788e-12 |
975 |
GW843682X |
LSM-1014 |
PLK1|PLK3 |
0.5uM |
24h |
LINCSCP_38250 |
LINCSCP_38250 |
MCF7 |
| -0.217741 |
6.292667e-12 |
975 |
Quinoclamine |
LSM-6261 |
|
3uM |
24h |
LINCSCP_37250 |
LINCSCP_37250 |
MCF7 |
| -0.217714 |
6.330598e-12 |
975 |
BRD-K19919069 |
LSM-38339 |
|
10uM |
6h |
LINCSCP_49100 |
LINCSCP_49100 |
PC3 |
| -0.217687 |
6.369770e-12 |
975 |
Dienestrol |
LSM-43043 |
ESR1 |
10uM |
24h |
LINCSCP_284818 |
LINCSCP_284818 |
SKB |
| -0.217687 |
6.369850e-12 |
975 |
Lapatinib |
LSM-1051 |
EGFR|ERBB2 |
0.12uM |
24h |
LINCSCP_72153 |
LINCSCP_72153 |
A375 |
| -0.217678 |
6.383706e-12 |
975 |
Dihydroorotate Dehydrogenase Inhibitor, Brequinar |
LSM-45952 |
|
0.12uM |
24h |
LINCSCP_111065 |
LINCSCP_111065 |
HELA |
| -0.217669 |
6.396608e-12 |
975 |
MLS003271309 |
LSM-3432 |
|
10uM |
6h |
LINCSCP_16339 |
LINCSCP_16339 |
HA1E |
| -0.217656 |
6.415436e-12 |
975 |
Irinotecan |
LSM-2167 |
TOP1 |
10uM |
24h |
LINCSCP_135986 |
LINCSCP_135986 |
MCF7 |
| -0.217647 |
6.427882e-12 |
975 |
BRD-K27113545 |
LSM-10069 |
|
5uM |
24h |
LINCSCP_63988 |
LINCSCP_63988 |
VCAP |
| -0.217646 |
6.428966e-12 |
975 |
BRD-K25990552 |
LSM-38695 |
|
10uM |
24h |
LINCSCP_28343 |
LINCSCP_28343 |
HT29 |
| -0.217639 |
6.439273e-12 |
975 |
CHIR-99021 |
LSM-1181 |
|
0.04uM |
3h |
LINCSCP_130421 |
LINCSCP_130421 |
LNCAP |
| -0.217617 |
6.472566e-12 |
975 |
GSK-1070916 |
LSM-1062 |
AURKB|AURKC |
0.1uM |
24h |
LINCSCP_38798 |
LINCSCP_38798 |
MCF7 |
| 0.217591 |
6.510610e-12 |
975 |
SA-440832 |
LSM-40344 |
|
1uM |
6h |
LINCSCP_253743 |
LINCSCP_253743 |
MCF7 |
| -0.21759 |
6.512429e-12 |
975 |
CHEMBL2361187 |
LSM-12338 |
|
10uM |
24h |
LINCSCP_312497 |
LINCSCP_312497 |
VCAP |
| 0.217562 |
6.552731e-12 |
975 |
Alectinib |
LSM-1202 |
ALK|RET |
3.33uM |
24h |
LINCSCP_91101 |
LINCSCP_91101 |
HA1E |
| -0.217562 |
6.553118e-12 |
975 |
Oxaprozin |
LSM-2553 |
PTGS1|PTGS2 |
3uM |
24h |
LINCSCP_23373 |
LINCSCP_23373 |
HEPG2 |
| -0.21755 |
6.570928e-12 |
975 |
AC1LUIBL |
LSM-6693 |
|
10uM |
6h |
LINCSCP_22622 |
LINCSCP_22622 |
HEPG2 |
| -0.217542 |
6.583284e-12 |
975 |
Simvastatin |
LSM-2492 |
HMGCR |
10uM |
24h |
LINCSCP_52497 |
LINCSCP_52497 |
SKB |
| -0.217532 |
6.597530e-12 |
975 |
N6-Methyladenosine |
LSM-3835 |
|
10uM |
24h |
LINCSCP_47565 |
LINCSCP_47565 |
PC3 |
| -0.217531 |
6.599775e-12 |
975 |
BRD-K82041810-001-01-8 |
LSM-13438 |
|
5uM |
24h |
LINCSCP_62050 |
LINCSCP_62050 |
VCAP |
| -0.217522 |
6.612123e-12 |
975 |
CHEMBL1495595 |
LSM-3294 |
|
10uM |
24h |
LINCSCP_188324 |
LINCSCP_188324 |
A549 |
| -0.217514 |
6.625501e-12 |
975 |
Sorafenib |
LSM-1008 |
BRAF|DDR2|FGFR1|FLT1|FLT3|FLT4|KDR|KIT|PDGFRB|RAF1|RET |
10uM |
24h |
LINCSCP_103260 |
LINCSCP_103260 |
HELA |
| 0.217458 |
6.709125e-12 |
975 |
GSK-2334470 |
LSM-1222 |
PDK1|PDPK1 |
0.1uM |
6h |
LINCSCP_53600 |
LINCSCP_53600 |
SNGM |
| 0.217457 |
6.711431e-12 |
975 |
Pfmrk inhibitor, wr 216174 |
LSM-42921 |
|
10uM |
24h |
LINCSCP_52741 |
LINCSCP_52741 |
SKB |
| 0.217449 |
6.722767e-12 |
975 |
TWS 119 |
LSM-1111 |
GSK3B |
0.12uM |
24h |
LINCSCP_115001 |
LINCSCP_115001 |
HS578T |
| 0.217405 |
6.790435e-12 |
975 |
Piperacillin |
LSM-5924 |
|
10uM |
6h |
LINCSCP_272363 |
LINCSCP_272363 |
PC3 |
| -0.217373 |
6.839961e-12 |
975 |
AZD-1775 |
LSM-1153 |
WEE1 |
3.33uM |
24h |
LINCSCP_112268 |
LINCSCP_112268 |
HEPG2 |
| 0.217355 |
6.867767e-12 |
975 |
BRD-K84994827 |
LSM-13620 |
|
5uM |
24h |
LINCSCP_62478 |
LINCSCP_62478 |
VCAP |
| -0.217354 |
6.869139e-12 |
975 |
Deoxycholic acid |
LSM-5529 |
GPBAR1 |
1.11uM |
24h |
LINCSCP_75974 |
LINCSCP_75974 |
A375 |
| -0.217327 |
6.911023e-12 |
975 |
TUL_XX087 |
LSM-36794 |
|
0.01uM |
6h |
LINCSCP_42021 |
LINCSCP_42021 |
NOMO1 |
| -0.217323 |
6.917298e-12 |
975 |
Lenvatinib (E7080) |
LSM-45581 |
FLT1|FLT4|KDR |
3.33uM |
24h |
LINCSCP_93739 |
LINCSCP_93739 |
HA1E |
| 0.217317 |
6.927526e-12 |
975 |
BRD-K99307487 |
LSM-14529 |
|
5uM |
24h |
LINCSCP_62958 |
LINCSCP_62958 |
VCAP |
| -0.217298 |
6.956645e-12 |
975 |
Tipifarnib |
LSM-6258 |
CHURC1-FNTB|FNTA|FNTB |
1.11uM |
24h |
LINCSCP_158579 |
LINCSCP_158579 |
PC3 |
| -0.217292 |
6.967122e-12 |
975 |
GSK 1059615 |
LSM-42799 |
PIK3CA|PIK3CB|PIK3CD|PIK3CG |
10uM |
24h |
LINCSCP_81400 |
LINCSCP_81400 |
A549 |
| -0.217286 |
6.976224e-12 |
975 |
Cabazitaxel |
LSM-46002 |
|
3.33uM |
24h |
LINCSCP_138307 |
LINCSCP_138307 |
MCF7 |
| -0.21727 |
7.001227e-12 |
975 |
Hydralazine |
LSM-15370 |
|
10uM |
24h |
LINCSCP_47456 |
LINCSCP_47456 |
PC3 |
| 0.217252 |
7.030281e-12 |
975 |
BRD-K94454791 |
LSM-14219 |
|
5uM |
6h |
LINCSCP_62240 |
LINCSCP_62240 |
VCAP |
| 0.217208 |
7.100616e-12 |
975 |
BRD-K94685656 |
LSM-14229 |
|
5uM |
24h |
LINCSCP_304626 |
LINCSCP_304626 |
VCAP |
| -0.217185 |
7.136916e-12 |
975 |
cortisone-acetate |
LSM-45387 |
TUBA1A|TUBA1B|TUBA1C|TUBA3E|TUBA4A|TUBB|TUBB1|TUBB2A|TUBB2B|TUBB3|TUBB4A|TUBB4B|TUBB6|TUBB8 |
0.37uM |
24h |
LINCSCP_109896 |
LINCSCP_109896 |
HELA |
| 0.217183 |
7.140974e-12 |
975 |
BRD-K71714567 |
LSM-41172 |
|
1uM |
6h |
LINCSCP_254157 |
LINCSCP_254157 |
MCF7 |
| -0.217168 |
7.164447e-12 |
975 |
BRD-K59730983 |
LSM-7638 |
|
5uM |
24h |
LINCSCP_60215 |
LINCSCP_60215 |
VCAP |
| -0.217117 |
7.248431e-12 |
975 |
BRD-A41986761 |
LSM-45957 |
|
3.33uM |
24h |
LINCSCP_90016 |
LINCSCP_90016 |
HA1E |
| 0.217055 |
7.349218e-12 |
975 |
Rilmenidine |
LSM-4253 |
ADRA2A|NISCH |
0.37uM |
24h |
LINCSCP_138045 |
LINCSCP_138045 |
MCF7 |
| -0.217031 |
7.390043e-12 |
975 |
Auraptene |
LSM-43035 |
MAOB |
10uM |
24h |
LINCSCP_42931 |
LINCSCP_42931 |
NPC |
| -0.217008 |
7.427795e-12 |
975 |
Wortmannin |
LSM-3947 |
PIK3CA|PIK3CG|PLK1 |
10uM |
24h |
LINCSCP_67768 |
LINCSCP_67768 |
NPC |
| -0.217006 |
7.432200e-12 |
975 |
CHEMBL1555138 |
LSM-3692 |
|
10uM |
24h |
LINCSCP_31197 |
LINCSCP_31197 |
MCF7 |
| -0.216964 |
7.502024e-12 |
975 |
MLS003179192 |
LSM-3532 |
|
10uM |
6h |
LINCSCP_22406 |
LINCSCP_22406 |
HEPG2 |
| 0.216926 |
7.567806e-12 |
975 |
Roflumilast |
LSM-45821 |
PDE4A|PDE4B|PDE4C|PDE4D |
3.33uM |
24h |
LINCSCP_75204 |
LINCSCP_75204 |
A375 |
| -0.216863 |
7.675073e-12 |
975 |
Genistein |
LSM-5549 |
CFTR|ESR2 |
10uM |
24h |
LINCSCP_309398 |
LINCSCP_309398 |
VCAP |
| 0.216859 |
7.682815e-12 |
975 |
BRD-K25866499 |
LSM-9996 |
|
5uM |
24h |
LINCSCP_63064 |
LINCSCP_63064 |
VCAP |
| -0.216858 |
7.684118e-12 |
975 |
Mitoxantrone |
LSM-2481 |
TOP2A |
0.01uM |
24h |
LINCSCP_9456 |
LINCSCP_9456 |
A549 |
| -0.216856 |
7.687305e-12 |
975 |
KU-C104137 |
LSM-2101 |
|
10uM |
6h |
LINCSCP_1492 |
LINCSCP_1492 |
A375 |
| 0.216852 |
7.695234e-12 |
975 |
AMD-070 (hydrochloride) |
LSM-45591 |
|
3.33uM |
24h |
LINCSCP_75543 |
LINCSCP_75543 |
A375 |
| -0.216773 |
7.833391e-12 |
975 |
FK888 |
LSM-3876 |
TACR1 |
3.33uM |
24h |
LINCSCP_124782 |
LINCSCP_124782 |
HT29 |
| -0.216764 |
7.849951e-12 |
975 |
Rhizocarpic-acid |
LSM-42811 |
|
10uM |
6h |
LINCSCP_14519 |
LINCSCP_14519 |
HA1E |
| -0.216737 |
7.896691e-12 |
975 |
SCHEMBL17497626 |
LSM-44605 |
|
0.5uM |
24h |
LINCSCP_17243 |
LINCSCP_17243 |
HA1E |
| -0.216733 |
7.903772e-12 |
975 |
Albendazole |
LSM-3782 |
|
0.37uM |
24h |
LINCSCP_110087 |
LINCSCP_110087 |
HELA |
| -0.2167 |
7.963452e-12 |
975 |
Aliskiren |
LSM-2653 |
REN |
10uM |
24h |
LINCSCP_262120 |
LINCSCP_262120 |
NPC |
| -0.216684 |
7.991802e-12 |
975 |
CHEMBL2359798 |
LSM-6796 |
|
10uM |
24h |
LINCSCP_37861 |
LINCSCP_37861 |
MCF7 |
| -0.216665 |
8.026937e-12 |
975 |
OTSSP167 |
LSM-6340 |
|
3.33uM |
24h |
LINCSCP_140214 |
LINCSCP_140214 |
MCF7 |
| -0.216653 |
8.048746e-12 |
975 |
Phorbol 12-myristate-13-acetate |
LSM-4341 |
PRKCA |
10uM |
24h |
LINCSCP_25393 |
LINCSCP_25393 |
HT29 |
| -0.216627 |
8.095124e-12 |
975 |
792173-99-0 |
LSM-2924 |
HCRTR1 |
10uM |
24h |
LINCSCP_42893 |
LINCSCP_42893 |
NPC |
| -0.216603 |
8.140485e-12 |
975 |
GSK 1059615 |
LSM-42799 |
PIK3CA|PIK3CB|PIK3CD|PIK3CG |
3.33uM |
24h |
LINCSCP_81401 |
LINCSCP_81401 |
A549 |
| 0.216567 |
8.206152e-12 |
975 |
TRAP-101 |
LSM-3563 |
OPRL1 |
10uM |
24h |
LINCSCP_11314 |
LINCSCP_11314 |
ASC |
| -0.216567 |
8.207108e-12 |
975 |
TL_HRAS26 |
LSM-2013 |
|
10uM |
6h |
LINCSCP_45109 |
LINCSCP_45109 |
PC3 |
| -0.216557 |
8.224796e-12 |
975 |
LY2228820 |
LSM-45439 |
MAPK14 |
0.37uM |
24h |
LINCSCP_157508 |
LINCSCP_157508 |
PC3 |
| -0.216549 |
8.239222e-12 |
975 |
SA-1456170 |
LSM-40904 |
|
1uM |
24h |
LINCSCP_37720 |
LINCSCP_37720 |
MCF7 |
| 0.216523 |
8.288778e-12 |
975 |
AC1NXRFO |
LSM-43270 |
|
0.1uM |
24h |
LINCSCP_9171 |
LINCSCP_9171 |
A549 |
| -0.216482 |
8.365338e-12 |
975 |
Tamoxifen |
LSM-42959 |
ESR1|ESR2 |
10uM |
24h |
LINCSCP_55329 |
LINCSCP_55329 |
U937 |
| -0.216453 |
8.419440e-12 |
975 |
SCHEMBL3363896 |
LSM-3789 |
ENTPD1|ENTPD2|ENTPD3 |
10uM |
24h |
LINCSCP_14784 |
LINCSCP_14784 |
HA1E |
| 0.216441 |
8.442882e-12 |
975 |
Thiabendazole |
LSM-3741 |
|
10uM |
24h |
LINCSCP_47661 |
LINCSCP_47661 |
PC3 |
| 0.216409 |
8.502947e-12 |
975 |
JSH-23 |
LSM-5897 |
RELA |
5uM |
6h |
LINCSCP_40246 |
LINCSCP_40246 |
NCIH508 |
| -0.216404 |
8.513416e-12 |
975 |
BRD-K48918933 |
LSM-7478 |
|
5uM |
24h |
LINCSCP_60042 |
LINCSCP_60042 |
VCAP |
| -0.216387 |
8.545995e-12 |
975 |
ST074627 |
LSM-4732 |
|
10uM |
6h |
LINCSCP_2074 |
LINCSCP_2074 |
A375 |
| 0.216387 |
8.546812e-12 |
975 |
ARTESUNATE |
LSM-45731 |
|
0.04uM |
24h |
LINCSCP_71646 |
LINCSCP_71646 |
A375 |
| 0.216383 |
8.553728e-12 |
975 |
AT-9283 |
LSM-37023 |
ABL1|AURKA|AURKB|FLT3|JAK2|JAK3 |
0.04uM |
24h |
LINCSCP_91473 |
LINCSCP_91473 |
HA1E |
| 0.216376 |
8.567557e-12 |
975 |
Mesoridazine |
LSM-1329 |
DRD2|HTR2A |
10uM |
24h |
LINCSCP_52794 |
LINCSCP_52794 |
SKB |
| 0.21637 |
8.579292e-12 |
975 |
SCHEMBL3958507 |
LSM-5245 |
COQ8B|EGFR |
1.11uM |
24h |
LINCSCP_99722 |
LINCSCP_99722 |
HCC515 |
| -0.216346 |
8.626237e-12 |
975 |
MG-132 |
LSM-1107 |
PSMB1 |
20uM |
24h |
LINCSCP_71231 |
LINCSCP_71231 |
A375 |
| -0.216338 |
8.640787e-12 |
975 |
Afuresertib |
LSM-42768 |
AKT1|AKT2|AKT3 |
10uM |
24h |
LINCSCP_104003 |
LINCSCP_104003 |
HELA |
| 0.216338 |
8.640791e-12 |
975 |
Amuvatinib |
LSM-1118 |
FLT3|KIT|MET|PDGFRA |
0.37uM |
24h |
LINCSCP_133263 |
LINCSCP_133263 |
MCF7 |
| -0.216311 |
8.694171e-12 |
975 |
Withaferin A |
LSM-6685 |
IKBKB|NAMPT |
10uM |
24h |
LINCSCP_111325 |
LINCSCP_111325 |
HEPG2 |
| -0.216301 |
8.713034e-12 |
975 |
BRD-K36620425 |
LSM-39274 |
|
10uM |
24h |
LINCSCP_310012 |
LINCSCP_310012 |
VCAP |
| 0.216299 |
8.716699e-12 |
975 |
GW-5074 |
LSM-42779 |
RAF1 |
10uM |
24h |
LINCSCP_6824 |
LINCSCP_6824 |
A549 |
| 0.216294 |
8.725988e-12 |
975 |
Pinacidil |
LSM-1557 |
ABCC8|ABCC9 |
10uM |
24h |
LINCSCP_31538 |
LINCSCP_31538 |
MCF7 |
| -0.216284 |
8.747276e-12 |
975 |
Clofibric acid |
LSM-2427 |
PPARA |
0.12uM |
24h |
LINCSCP_125126 |
LINCSCP_125126 |
HT29 |
| -0.216279 |
8.755806e-12 |
975 |
SPECTRUM_000897 |
LSM-1378 |
NR3C1 |
10uM |
24h |
LINCSCP_90507 |
LINCSCP_90507 |
HA1E |
| 0.21627 |
8.774678e-12 |
975 |
Doramapimod |
LSM-1170 |
MAPK11|MAPK12|MAPK14 |
3.33uM |
24h |
LINCSCP_126227 |
LINCSCP_126227 |
HT29 |
| 0.21623 |
8.853759e-12 |
975 |
SMR000068650 |
LSM-2859 |
|
10uM |
24h |
LINCSCP_31602 |
LINCSCP_31602 |
MCF7 |
| -0.216186 |
8.942621e-12 |
975 |
AMG-517 |
LSM-45865 |
TRPV1 |
3.33uM |
24h |
LINCSCP_121134 |
LINCSCP_121134 |
HT29 |
| -0.216178 |
8.956989e-12 |
975 |
Menadione |
LSM-3755 |
|
10uM |
24h |
LINCSCP_260634 |
LINCSCP_260634 |
NKDBA |
| -0.216178 |
8.957677e-12 |
975 |
BRD-K38044934 |
LSM-39361 |
|
0.5uM |
6h |
LINCSCP_48656 |
LINCSCP_48656 |
PC3 |
| -0.216175 |
8.964164e-12 |
975 |
Selumetinib |
LSM-1056 |
MAP2K1|MAP2K2 |
1uM |
24h |
LINCSCP_24338 |
LINCSCP_24338 |
HS578T |
| -0.216168 |
8.977332e-12 |
975 |
2,3-Diamino-1-phenylpropan-1-one |
LSM-1452 |
|
10uM |
24h |
LINCSCP_33045 |
LINCSCP_33045 |
MCF7 |
| -0.216165 |
8.985094e-12 |
975 |
NVP-AUY922 |
LSM-1162 |
|
1.11uM |
24h |
LINCSCP_116309 |
LINCSCP_116309 |
HT29 |
| 0.216159 |
8.995736e-12 |
975 |
Palbociclib |
LSM-1071 |
CCND1|CDK4|CDK6 |
0.12uM |
24h |
LINCSCP_88008 |
LINCSCP_88008 |
HA1E |
| -0.216141 |
9.032213e-12 |
975 |
Dienestrol |
LSM-43043 |
ESR1 |
10uM |
24h |
LINCSCP_33424 |
LINCSCP_33424 |
MCF7 |
| -0.216085 |
9.146528e-12 |
975 |
Mebendazole |
LSM-3749 |
|
20uM |
24h |
LINCSCP_252327 |
LINCSCP_252327 |
MCF7 |
| 0.21607 |
9.178138e-12 |
975 |
ZINC00969081 |
LSM-3555 |
|
10uM |
6h |
LINCSCP_20022 |
LINCSCP_20022 |
HCC515 |
| 0.216069 |
9.180438e-12 |
975 |
Triamcinolone Acetonide |
LSM-5641 |
NR3C1 |
10uM |
6h |
LINCSCP_16979 |
LINCSCP_16979 |
HA1E |
| -0.216049 |
9.221627e-12 |
975 |
Guanadrel |
LSM-43257 |
SLC6A2 |
0.12uM |
24h |
LINCSCP_104577 |
LINCSCP_104577 |
HELA |
| -0.216036 |
9.247940e-12 |
975 |
PD-0325901 |
LSM-1101 |
MAP2K1|MAP2K2 |
0.37uM |
24h |
LINCSCP_144614 |
LINCSCP_144614 |
MDAMB231 |
| -0.216024 |
9.273171e-12 |
975 |
Glyburide |
LSM-2811 |
ABCC8|CFTR|KCNJ11|KCNJ5|KCNJ8 |
10uM |
24h |
LINCSCP_272031 |
LINCSCP_272031 |
PC3 |
| -0.215993 |
9.338755e-12 |
975 |
1-[2-(4-Methylphenyl)indolizin-3-yl]-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethanone |
LSM-4511 |
|
10uM |
24h |
LINCSCP_49831 |
LINCSCP_49831 |
PHH |
| -0.21595 |
9.430261e-12 |
975 |
KW-2449 |
LSM-42803 |
ABL1|AURKA|AURKB|FLT3 |
10uM |
24h |
LINCSCP_81847 |
LINCSCP_81847 |
A549 |
| -0.215936 |
9.458008e-12 |
975 |
TUL_XX087 |
LSM-36794 |
|
0.01uM |
6h |
LINCSCP_288188 |
LINCSCP_288188 |
THP1 |
| -0.215928 |
9.475069e-12 |
975 |
BRD-K10211010 |
LSM-9049 |
|
10uM |
24h |
LINCSCP_8998 |
LINCSCP_8998 |
A549 |
| 0.215896 |
9.544843e-12 |
975 |
BRD-K08663380 |
LSM-8951 |
|
0.01uM |
24h |
LINCSCP_65084 |
LINCSCP_65084 |
VCAP |
| -0.215895 |
9.547244e-12 |
975 |
CHEMBL2360382 |
LSM-41340 |
|
10uM |
24h |
LINCSCP_47333 |
LINCSCP_47333 |
PC3 |
| 0.215888 |
9.561727e-12 |
975 |
BRD-K22828860 |
LSM-6090 |
|
10uM |
6h |
LINCSCP_16277 |
LINCSCP_16277 |
HA1E |
| -0.215883 |
9.571997e-12 |
975 |
PD-0325901 |
LSM-1101 |
MAP2K1|MAP2K2 |
10uM |
24h |
LINCSCP_131874 |
LINCSCP_131874 |
MCF7 |
| 0.215875 |
9.588705e-12 |
975 |
IWR-1-ENDO |
LSM-5707 |
TNKS|TNKS2 |
10uM |
24h |
LINCSCP_188042 |
LINCSCP_188042 |
A549 |
| 0.215866 |
9.609102e-12 |
975 |
apicidin |
LSM-45760 |
|
3.33uM |
24h |
LINCSCP_139561 |
LINCSCP_139561 |
MCF7 |
| 0.215866 |
9.609362e-12 |
975 |
MK-2866 (GTx-024) |
LSM-45447 |
AR |
1.11uM |
24h |
LINCSCP_71315 |
LINCSCP_71315 |
A375 |
| -0.215858 |
9.625353e-12 |
975 |
AC1O7M2R |
LSM-3745 |
ADCY2 |
10uM |
24h |
LINCSCP_263900 |
LINCSCP_263900 |
NPC |
| 0.215851 |
9.641371e-12 |
975 |
Cytarabine |
LSM-5470 |
POLA1|POLB|POLD1|POLE |
10uM |
24h |
LINCSCP_74124 |
LINCSCP_74124 |
A375 |
| -0.215839 |
9.668074e-12 |
975 |
DOCETAXEL |
LSM-45649 |
|
10uM |
24h |
LINCSCP_170064 |
LINCSCP_170064 |
YAPC |
| -0.215811 |
9.728449e-12 |
975 |
Mepivacaine |
LSM-4306 |
SCN10A|SCN11A|SCN1A|SCN2A|SCN3A|SCN4A|SCN5A|SCN7A|SCN8A|SCN9A |
3.33uM |
24h |
LINCSCP_75256 |
LINCSCP_75256 |
A375 |
| -0.21579 |
9.774096e-12 |
975 |
MG-132 |
LSM-1107 |
PSMB1 |
20uM |
24h |
LINCSCP_136251 |
LINCSCP_136251 |
MCF7 |
| -0.215759 |
9.843819e-12 |
975 |
179324-69-7 |
LSM-6281 |
ADRM1|PSMA1|PSMA2|PSMA3|PSMA4|PSMA5|PSMA6|PSMA7|PSMA8|PSMB1|PSMB10|PSMB11|PSMB2|PSMB3|PSMB4|PSMB5|PSMB6|PSMB7|PSMB8|PSMB9|PSMC1|PSMC2|PSMC3|PSMC4|PSMC5|PSMC6|PSMD1|PSMD11|PSMD12|PSMD13|PSMD14|PSMD2|PSMD3|PSMD4|PSMD6|PSMD7|PSMD8|SEM1 |
20uM |
24h |
LINCSCP_71505 |
LINCSCP_71505 |
A375 |
| 0.215722 |
9.925528e-12 |
975 |
BRD-K42694358 |
LSM-14827 |
|
5uM |
24h |
LINCSCP_64193 |
LINCSCP_64193 |
VCAP |
| -0.215672 |
1.003737e-11 |
975 |
PJ34 |
LSM-4937 |
|
10uM |
24h |
LINCSCP_251023 |
LINCSCP_251023 |
MCF7 |
| -0.215671 |
1.003872e-11 |
975 |
Tozasertib |
LSM-1021 |
ABL1|AURKA|AURKB|AURKC|BCR|FLT3|JAK2 |
10uM |
3h |
LINCSCP_130805 |
LINCSCP_130805 |
MCF10A |
| 0.215633 |
1.012444e-11 |
975 |
GAP-134 (Hydrochloride) |
LSM-45532 |
|
0.12uM |
24h |
LINCSCP_72021 |
LINCSCP_72021 |
A375 |
| 0.215628 |
1.013602e-11 |
975 |
Axitinib |
LSM-43191 |
FLT1|FLT4|KDR |
10uM |
6h |
LINCSCP_32327 |
LINCSCP_32327 |
MCF7 |
| 0.215624 |
1.014641e-11 |
975 |
CHEMBL567331 |
LSM-3577 |
CLK1|CLK4|DYRK1A |
10uM |
24h |
LINCSCP_4995 |
LINCSCP_4995 |
A549 |
| -0.215602 |
1.019713e-11 |
975 |
PF477736 |
LSM-1112 |
CHEK1 |
3.33uM |
24h |
LINCSCP_132049 |
LINCSCP_132049 |
MCF7 |
| -0.215594 |
1.021510e-11 |
975 |
MLS003179196 |
LSM-1356 |
|
10uM |
6h |
LINCSCP_31436 |
LINCSCP_31436 |
MCF7 |
| -0.215591 |
1.022043e-11 |
975 |
STK054715 |
LSM-1925 |
|
10uM |
6h |
LINCSCP_5464 |
LINCSCP_5464 |
A549 |
| -0.215572 |
1.026576e-11 |
975 |
MLS002264406 |
LSM-1675 |
|
10uM |
6h |
LINCSCP_45764 |
LINCSCP_45764 |
PC3 |
| -0.215571 |
1.026733e-11 |
975 |
PF-03758309 |
LSM-4254 |
PAK4 |
1.11uM |
24h |
LINCSCP_150277 |
LINCSCP_150277 |
NPC.TAK |
| -0.215565 |
1.028179e-11 |
975 |
nimodipine |
LSM-45413 |
|
0.37uM |
24h |
LINCSCP_138489 |
LINCSCP_138489 |
MCF7 |
| -0.215563 |
1.028649e-11 |
975 |
Olanzapine |
LSM-5359 |
DRD1|DRD2|DRD3|DRD4|HRH1|HTR1A|HTR1B|HTR1D|HTR1E|HTR2A|HTR2C|HTR6|HTR7 |
10uM |
24h |
LINCSCP_168104 |
LINCSCP_168104 |
YAPC |
| -0.215558 |
1.029769e-11 |
975 |
FK888 |
LSM-3876 |
TACR1 |
0.12uM |
24h |
LINCSCP_173163 |
LINCSCP_173163 |
YAPC |
| -0.215533 |
1.035461e-11 |
975 |
HG-5-88-01 |
LSM-42725 |
COQ8B|EGFR |
10uM |
24h |
LINCSCP_10964 |
LINCSCP_10964 |
ASC |
| -0.215501 |
1.042986e-11 |
975 |
Sunitinib |
LSM-42800 |
CSF1R|FLT1|FLT3|FLT4|KDR|KIT|PDGFRA|PDGFRB|RET |
10uM |
24h |
LINCSCP_113845 |
LINCSCP_113845 |
HME1 |
| 0.215469 |
1.050466e-11 |
975 |
AC1MSUFC |
LSM-6191 |
HMGCR |
40uM |
6h |
LINCSCP_21143 |
LINCSCP_21143 |
HCT116 |
| 0.215445 |
1.056126e-11 |
975 |
BRD-K71151012 |
LSM-12772 |
|
5uM |
24h |
LINCSCP_62917 |
LINCSCP_62917 |
VCAP |
| 0.215423 |
1.061326e-11 |
975 |
Trametinib |
LSM-1143 |
MAP2K1|MAP2K2 |
0.12uM |
3h |
LINCSCP_115438 |
LINCSCP_115438 |
HS578T |
| -0.215413 |
1.063664e-11 |
975 |
MLS000862515 |
LSM-3487 |
|
10uM |
6h |
LINCSCP_16042 |
LINCSCP_16042 |
HA1E |
| -0.215406 |
1.065429e-11 |
975 |
Seliciclib |
LSM-1001 |
CDK1|CDK2|CDK5|CDK7|CDK9 |
10uM |
24h |
LINCSCP_38936 |
LINCSCP_38936 |
MDAMB231 |
| 0.215384 |
1.070812e-11 |
975 |
Imatinib |
LSM-1023 |
ABL1|BCR|CSF1R|KIT|PDGFRA|PDGFRB |
0.37uM |
3h |
LINCSCP_145936 |
LINCSCP_145936 |
MDAMB231 |
| -0.215367 |
1.074846e-11 |
975 |
Wortmannin |
LSM-3947 |
PIK3CA|PIK3CG|PLK1 |
0.5uM |
6h |
LINCSCP_43941 |
LINCSCP_43941 |
PC3 |
| -0.215366 |
1.075037e-11 |
975 |
Neratinib |
LSM-42778 |
EGFR|ERBB2|ERBB4 |
10uM |
24h |
LINCSCP_51475 |
LINCSCP_51475 |
SKBR3 |
| 0.215347 |
1.079664e-11 |
975 |
GSK2636771 |
LSM-45667 |
PIK3CB |
0.12uM |
24h |
LINCSCP_124623 |
LINCSCP_124623 |
HT29 |
| -0.215337 |
1.081994e-11 |
975 |
KX2-391 |
LSM-45890 |
SRC |
0.12uM |
24h |
LINCSCP_155706 |
LINCSCP_155706 |
PC3 |
| -0.215334 |
1.082898e-11 |
975 |
Solifenacin succinate |
LSM-45423 |
CHRM2|CHRM3 |
10uM |
24h |
LINCSCP_102447 |
LINCSCP_102447 |
HELA |
| -0.215327 |
1.084538e-11 |
975 |
SCHEMBL6465902 |
LSM-3544 |
PDE5A |
10uM |
6h |
LINCSCP_2637 |
LINCSCP_2637 |
A375 |
| -0.215242 |
1.105430e-11 |
975 |
Vinblastine |
LSM-1647 |
TUBB |
0.5uM |
24h |
LINCSCP_38130 |
LINCSCP_38130 |
MCF7 |
| -0.215239 |
1.106190e-11 |
975 |
N,N-Dimethyl-n'-{5-[(2-methyl-4-quinolyl)thio]-1,3,4-thiadiazol-2-yl}iminoformamide |
LSM-4930 |
|
10uM |
24h |
LINCSCP_32253 |
LINCSCP_32253 |
MCF7 |
| -0.215226 |
1.109356e-11 |
975 |
BRD-K89390280 |
LSM-15064 |
|
10uM |
6h |
LINCSCP_64815 |
LINCSCP_64815 |
VCAP |
| -0.215221 |
1.110549e-11 |
975 |
C30H33N3O5S |
LSM-1156 |
ATM |
3.33uM |
24h |
LINCSCP_148779 |
LINCSCP_148779 |
NPC |
| 0.215204 |
1.114684e-11 |
975 |
Swainsonine |
LSM-45602 |
|
3.85uM |
24h |
LINCSCP_74495 |
LINCSCP_74495 |
A375 |
| -0.215187 |
1.119026e-11 |
975 |
PF-03758309 |
LSM-4254 |
PAK4 |
3.33uM |
24h |
LINCSCP_89029 |
LINCSCP_89029 |
HA1E |
| -0.215161 |
1.125678e-11 |
975 |
CHEMBL2131454 |
LSM-38019 |
|
10uM |
6h |
LINCSCP_55568 |
LINCSCP_55568 |
U937 |
| -0.215159 |
1.126163e-11 |
975 |
4-[(5-Bromoquinolin-8-yl)amino]-4-oxobutanoic acid |
LSM-4561 |
|
10uM |
24h |
LINCSCP_31892 |
LINCSCP_31892 |
MCF7 |
| 0.215138 |
1.131294e-11 |
975 |
Resveratrol |
LSM-42917 |
PTGS1|PTGS2|SIRT1 |
0.12uM |
24h |
LINCSCP_72750 |
LINCSCP_72750 |
A375 |
| -0.215107 |
1.139349e-11 |
975 |
SCHEMBL17497626 |
LSM-44605 |
|
1uM |
24h |
LINCSCP_17245 |
LINCSCP_17245 |
HA1E |
| -0.215077 |
1.146970e-11 |
975 |
A-443654 |
LSM-1045 |
|
0.12uM |
24h |
LINCSCP_81559 |
LINCSCP_81559 |
A549 |
| -0.215077 |
1.146994e-11 |
975 |
SB225002 |
LSM-3367 |
CXCR2 |
10uM |
24h |
LINCSCP_44980 |
LINCSCP_44980 |
PC3 |
| -0.215064 |
1.150243e-11 |
975 |
AT-7519 |
LSM-1004 |
CDK1|CDK10|CDK11B|CDK12|CDK13|CDK14|CDK15|CDK16|CDK17|CDK18|CDK19|CDK2|CDK20|CDK3|CDK4|CDK5|CDK6|CDK7|CDK8|CDK9 |
0.04uM |
24h |
LINCSCP_121330 |
LINCSCP_121330 |
HT29 |
| 0.21505 |
1.153800e-11 |
975 |
Gelsemine |
LSM-1353 |
GLRA3 |
10uM |
24h |
LINCSCP_25216 |
LINCSCP_25216 |
HT29 |
| 0.215033 |
1.158307e-11 |
975 |
rifampicin |
|
|
0.12uM |
24h |
LINCSCP_145632 |
LINCSCP_145632 |
MDAMB231 |
| -0.215031 |
1.158952e-11 |
975 |
CGS-15943 |
LSM-3076 |
ADORA1|ADORA2A|ADORA2B |
40uM |
24h |
LINCSCP_67593 |
LINCSCP_67593 |
MCF7 |
| 0.215014 |
1.163174e-11 |
975 |
Carmoxirole |
LSM-3850 |
DRD2 |
10uM |
6h |
LINCSCP_18444 |
LINCSCP_18444 |
HCC515 |
| -0.214992 |
1.168996e-11 |
975 |
altrenogest |
LSM-45498 |
|
3.33uM |
24h |
LINCSCP_139855 |
LINCSCP_139855 |
MCF7 |
| 0.214983 |
1.171277e-11 |
975 |
SPECTRUM2_001084 |
LSM-1740 |
ATP1A1 |
10uM |
24h |
LINCSCP_11140 |
LINCSCP_11140 |
ASC |
| -0.214943 |
1.181948e-11 |
975 |
INOSITOL |
LSM-45237 |
|
1.11uM |
24h |
LINCSCP_158435 |
LINCSCP_158435 |
PC3 |
| 0.214929 |
1.185554e-11 |
975 |
Erlotinib |
LSM-1097 |
EGFR |
0.1uM |
6h |
LINCSCP_39625 |
LINCSCP_39625 |
MDAMB231 |
| -0.214909 |
1.190832e-11 |
975 |
Ropinirole |
LSM-2351 |
DRD2|DRD3|DRD4 |
10uM |
24h |
LINCSCP_101525 |
LINCSCP_101525 |
HELA |
| -0.214864 |
1.202896e-11 |
975 |
L 168049 |
LSM-2394 |
GCGR |
10uM |
6h |
LINCSCP_480 |
LINCSCP_480 |
A375 |
| 0.214847 |
1.207554e-11 |
975 |
Oxedrine |
LSM-4956 |
ADRA1A |
10uM |
24h |
LINCSCP_31534 |
LINCSCP_31534 |
MCF7 |
| -0.214842 |
1.208830e-11 |
975 |
Dactolisib |
LSM-4255 |
MTOR|PIK3CA|PIK3CB|PIK3CD|PIK3CG|PIK3R1|PIK3R2|PIK3R3|PIK3R5 |
0.04uM |
24h |
LINCSCP_90008 |
LINCSCP_90008 |
HA1E |
| 0.214821 |
1.214694e-11 |
975 |
cucurbitacin-i |
LSM-45610 |
|
1.11uM |
24h |
LINCSCP_72742 |
LINCSCP_72742 |
A375 |
| 0.214753 |
1.233288e-11 |
975 |
Vorinostat |
LSM-3828 |
HDAC1|HDAC2|HDAC3|HDAC6|HDAC8 |
0.37uM |
24h |
LINCSCP_164679 |
LINCSCP_164679 |
SKL.C |
| 0.214751 |
1.233797e-11 |
975 |
BRD-K96269157 |
LSM-14336 |
|
5uM |
24h |
LINCSCP_61854 |
LINCSCP_61854 |
VCAP |
| -0.214742 |
1.236247e-11 |
975 |
T5832551 |
LSM-2617 |
|
10uM |
24h |
LINCSCP_31140 |
LINCSCP_31140 |
MCF7 |
| -0.21473 |
1.239423e-11 |
975 |
lapatinib |
|
EGFR|ERBB2 |
10uM |
6h |
LINCSCP_6129 |
LINCSCP_6129 |
A549 |
| -0.214721 |
1.242114e-11 |
975 |
Risperidone |
LSM-3193 |
ADRA1A|ADRA1B|DRD2|DRD3|DRD4|HRH1|HTR1A|HTR1D|HTR2A|HTR2C |
0.37uM |
24h |
LINCSCP_158298 |
LINCSCP_158298 |
PC3 |
| 0.214717 |
1.243110e-11 |
975 |
BRD-K49441594 |
LSM-11434 |
|
10uM |
6h |
LINCSCP_279488 |
LINCSCP_279488 |
PC3 |
| -0.214716 |
1.243285e-11 |
975 |
TUL_XX087 |
LSM-36794 |
|
1uM |
24h |
LINCSCP_41939 |
LINCSCP_41939 |
NOMO1 |
| -0.214697 |
1.248814e-11 |
975 |
Phenelzine |
LSM-5928 |
AOC3|MAOA|MAOB |
10uM |
24h |
LINCSCP_47571 |
LINCSCP_47571 |
PC3 |
| -0.214688 |
1.251188e-11 |
975 |
SMR000075623 |
LSM-4644 |
|
10uM |
6h |
LINCSCP_211428 |
LINCSCP_211428 |
HA1E |
| 0.214658 |
1.259539e-11 |
975 |
3-(4-Pyridyl)indole |
LSM-4569 |
ROCK1 |
10uM |
24h |
LINCSCP_123642 |
LINCSCP_123642 |
HT29 |
| -0.214654 |
1.260692e-11 |
975 |
Glycocholic acid |
LSM-3222 |
|
10uM |
24h |
LINCSCP_43465 |
LINCSCP_43465 |
NPC |
| -0.214647 |
1.262851e-11 |
975 |
Leflunomide |
LSM-3771 |
DHODH |
10uM |
24h |
LINCSCP_44063 |
LINCSCP_44063 |
PC3 |
| 0.214638 |
1.265281e-11 |
975 |
BRD-K45265806 |
LSM-11183 |
|
5uM |
24h |
LINCSCP_61605 |
LINCSCP_61605 |
VCAP |
| 0.21459 |
1.278864e-11 |
975 |
NU1025 |
LSM-4643 |
PARP1 |
0.01uM |
6h |
LINCSCP_36391 |
LINCSCP_36391 |
MCF7 |
| 0.214589 |
1.279104e-11 |
975 |
BRD-K08920503 |
LSM-8964 |
|
5uM |
24h |
LINCSCP_61938 |
LINCSCP_61938 |
VCAP |
| -0.214579 |
1.281974e-11 |
975 |
Methimazole |
LSM-5646 |
TPO |
10uM |
24h |
LINCSCP_34504 |
LINCSCP_34504 |
MCF7 |
| -0.214576 |
1.282881e-11 |
975 |
Mebendazole |
LSM-3749 |
|
10uM |
24h |
LINCSCP_67610 |
LINCSCP_67610 |
MCF7 |
| -0.214568 |
1.285286e-11 |
975 |
BRD-K78976513 |
LSM-7884 |
|
5uM |
24h |
LINCSCP_60236 |
LINCSCP_60236 |
VCAP |
| -0.214557 |
1.288317e-11 |
975 |
XMD 8-92 |
LSM-1094 |
MAPK7 |
10uM |
6h |
LINCSCP_20463 |
LINCSCP_20463 |
HCC515 |
| -0.214503 |
1.304145e-11 |
975 |
Escitalopram |
LSM-3569 |
SLC6A4 |
10uM |
6h |
LINCSCP_239290 |
LINCSCP_239290 |
MCF7 |
| -0.214499 |
1.305133e-11 |
975 |
PCI-32765 |
LSM-1129 |
BTK |
1uM |
6h |
LINCSCP_39503 |
LINCSCP_39503 |
MDAMB231 |
| -0.214485 |
1.309354e-11 |
975 |
BI-2536 |
LSM-1041 |
PLK1 |
0.12uM |
24h |
LINCSCP_124227 |
LINCSCP_124227 |
HT29 |
| -0.214463 |
1.315552e-11 |
975 |
TL_HRAS26 |
LSM-2013 |
|
10uM |
24h |
LINCSCP_202327 |
LINCSCP_202327 |
A549 |
| -0.214451 |
1.319334e-11 |
975 |
Panobinostat |
LSM-43059 |
HDAC1|HDAC10|HDAC11|HDAC2|HDAC3|HDAC4|HDAC5|HDAC6|HDAC7|HDAC8|HDAC9 |
0.01uM |
24h |
LINCSCP_35485 |
LINCSCP_35485 |
MCF7 |
| -0.214449 |
1.319719e-11 |
975 |
AC1OFCDP |
LSM-5348 |
HMGCR |
10uM |
24h |
LINCSCP_34475 |
LINCSCP_34475 |
MCF7 |
| -0.214445 |
1.321047e-11 |
975 |
GSK 1059615 |
LSM-42799 |
PIK3CA|PIK3CB|PIK3CD|PIK3CG |
3.33uM |
24h |
LINCSCP_147936 |
LINCSCP_147936 |
NPC.CAS9 |
| 0.214415 |
1.329835e-11 |
975 |
AZD-1152-HQPA |
LSM-1067 |
AURKA|AURKB |
0.01uM |
24h |
LINCSCP_201159 |
LINCSCP_201159 |
A549 |
| -0.214379 |
1.340470e-11 |
975 |
MLS002276504 |
LSM-2291 |
|
10uM |
24h |
LINCSCP_267571 |
LINCSCP_267571 |
PC3 |
| 0.214332 |
1.354639e-11 |
975 |
Imatinib |
LSM-1023 |
ABL1|BCR|CSF1R|KIT|PDGFRA|PDGFRB |
0.04uM |
3h |
LINCSCP_113618 |
LINCSCP_113618 |
HME1 |
| -0.214325 |
1.356812e-11 |
975 |
SMR000651449 |
LSM-3511 |
|
10uM |
6h |
LINCSCP_51187 |
LINCSCP_51187 |
RMUGS |
| 0.214323 |
1.357424e-11 |
975 |
SR 33805 oxalate |
LSM-45933 |
|
0.37uM |
24h |
LINCSCP_105714 |
LINCSCP_105714 |
HELA |
| -0.214317 |
1.359217e-11 |
975 |
SB705498 |
LSM-45502 |
TRPV1 |
10uM |
24h |
LINCSCP_172270 |
LINCSCP_172270 |
YAPC |
| 0.214276 |
1.371613e-11 |
975 |
Fenretinide |
LSM-42925 |
RARA |
10uM |
6h |
LINCSCP_13397 |
LINCSCP_13397 |
FIBRNPC |
| 0.214264 |
1.375505e-11 |
975 |
VX-745 |
LSM-1169 |
MAPK14 |
0.37uM |
24h |
LINCSCP_134130 |
LINCSCP_134130 |
MCF7 |
| -0.214262 |
1.376157e-11 |
975 |
BRD-K41431262 |
LSM-39564 |
|
10uM |
24h |
LINCSCP_47314 |
LINCSCP_47314 |
PC3 |
| -0.214235 |
1.384448e-11 |
975 |
CHEMBL2135537 |
LSM-6149 |
|
10uM |
24h |
LINCSCP_59263 |
LINCSCP_59263 |
VCAP |
| -0.214227 |
1.386700e-11 |
975 |
7-Bromo-1,2,3,9-tetrahydropyrrolo[2,1-b]quinazoline |
LSM-3873 |
|
10uM |
6h |
LINCSCP_5168 |
LINCSCP_5168 |
A549 |
| 0.214213 |
1.391062e-11 |
975 |
Levomethorphan |
LSM-2525 |
SIGMAR1|SLC6A4 |
10uM |
24h |
LINCSCP_44544 |
LINCSCP_44544 |
PC3 |
| -0.214211 |
1.391626e-11 |
975 |
BG-51 |
LSM-45301 |
HDAC3 |
0.1uM |
24h |
LINCSCP_35505 |
LINCSCP_35505 |
MCF7 |
| -0.21421 |
1.392105e-11 |
975 |
Wortmannin |
LSM-3947 |
PIK3CA|PIK3CG|PLK1 |
0.1uM |
24h |
LINCSCP_264404 |
LINCSCP_264404 |
PC3 |
| 0.214201 |
1.394851e-11 |
975 |
EX-8678 |
LSM-1147 |
|
0.04uM |
3h |
LINCSCP_145926 |
LINCSCP_145926 |
MDAMB231 |
| -0.2142 |
1.395110e-11 |
975 |
IC 261 |
LSM-42870 |
|
10uM |
24h |
LINCSCP_37639 |
LINCSCP_37639 |
MCF7 |
| -0.214134 |
1.415905e-11 |
975 |
AS-605240 |
LSM-42784 |
PIK3CG |
3.33uM |
24h |
LINCSCP_76661 |
LINCSCP_76661 |
A375 |
| 0.214132 |
1.416556e-11 |
975 |
STK222600 |
LSM-3535 |
|
10uM |
6h |
LINCSCP_211453 |
LINCSCP_211453 |
HA1E |
| -0.214124 |
1.419117e-11 |
975 |
BRD-K08777248 |
LSM-37743 |
|
10uM |
24h |
LINCSCP_59173 |
LINCSCP_59173 |
VCAP |
| -0.214121 |
1.419905e-11 |
975 |
GSK-1070916 |
LSM-1062 |
AURKB|AURKC |
1uM |
6h |
LINCSCP_4102 |
LINCSCP_4102 |
A375 |
| 0.214078 |
1.433690e-11 |
975 |
Luteolin |
LSM-5229 |
|
1uM |
24h |
LINCSCP_254206 |
LINCSCP_254206 |
MCF7 |
| 0.214056 |
1.440636e-11 |
975 |
Nebivolol |
LSM-45235 |
|
3.33uM |
24h |
LINCSCP_169975 |
LINCSCP_169975 |
YAPC |
| -0.214051 |
1.442329e-11 |
975 |
Temoporfin |
LSM-45995 |
|
1.11uM |
24h |
LINCSCP_155237 |
LINCSCP_155237 |
PC3 |
| -0.214043 |
1.444851e-11 |
975 |
I-BET151 |
LSM-6335 |
|
10uM |
24h |
LINCSCP_164760 |
LINCSCP_164760 |
SKL.C |
| -0.214028 |
1.449852e-11 |
975 |
Idebenone |
LSM-5505 |
|
10uM |
6h |
LINCSCP_269994 |
LINCSCP_269994 |
PC3 |
| 0.214003 |
1.457703e-11 |
975 |
Imiloxan |
LSM-1308 |
ADRA2A|ADRA2B |
10uM |
24h |
LINCSCP_168008 |
LINCSCP_168008 |
YAPC |
| 0.213995 |
1.460293e-11 |
975 |
noscapine |
|
|
0.12uM |
3h |
LINCSCP_145901 |
LINCSCP_145901 |
MDAMB231 |
| -0.213985 |
1.463807e-11 |
975 |
PD-173074 |
LSM-1026 |
FGFR1|FGFR3 |
3.33uM |
24h |
LINCSCP_115621 |
LINCSCP_115621 |
HS578T |
| -0.213973 |
1.467408e-11 |
975 |
PNU-74654 |
LSM-44945 |
CTNNB1|TCF4 |
80uM |
24h |
LINCSCP_44929 |
LINCSCP_44929 |
PC3 |
| -0.213972 |
1.467869e-11 |
975 |
NMS-1286937 |
LSM-45818 |
|
3.33uM |
24h |
LINCSCP_125285 |
LINCSCP_125285 |
HT29 |
| 0.213968 |
1.469074e-11 |
975 |
Acetazolamide |
LSM-5543 |
CA1|CA12|CA14|CA2|CA4|CA7 |
3.33uM |
24h |
LINCSCP_122519 |
LINCSCP_122519 |
HT29 |
| -0.213962 |
1.471162e-11 |
975 |
Y-39983 |
LSM-1150 |
ROCK1|ROCK2 |
1.11uM |
3h |
LINCSCP_133230 |
LINCSCP_133230 |
MCF7 |
| 0.21395 |
1.475096e-11 |
975 |
Seliciclib |
LSM-1001 |
CDK1|CDK2|CDK5|CDK7|CDK9 |
3.33uM |
24h |
LINCSCP_130626 |
LINCSCP_130626 |
MCF10A |
| -0.213928 |
1.482502e-11 |
975 |
CX-5461 |
LSM-6342 |
|
1.11uM |
24h |
LINCSCP_147955 |
LINCSCP_147955 |
NPC.CAS9 |
| 0.213888 |
1.495640e-11 |
975 |
Pimobendan |
LSM-45256 |
|
0.12uM |
24h |
LINCSCP_159606 |
LINCSCP_159606 |
PC3 |
| 0.213847 |
1.509406e-11 |
975 |
376348-65-1, Uk-427857, uk427857 |
LSM-6182 |
CCR5 |
10uM |
6h |
LINCSCP_19448 |
LINCSCP_19448 |
HCC515 |
| 0.213845 |
1.509902e-11 |
975 |
AC1Q5RFA |
LSM-43063 |
|
1.11uM |
24h |
LINCSCP_104976 |
LINCSCP_104976 |
HELA |
| -0.213826 |
1.516240e-11 |
975 |
MLS000778276 |
LSM-43118 |
|
10uM |
24h |
LINCSCP_37234 |
LINCSCP_37234 |
MCF7 |
| -0.213818 |
1.519242e-11 |
975 |
Batimastat |
LSM-6276 |
|
0.12uM |
24h |
LINCSCP_152723 |
LINCSCP_152723 |
PC3 |
| -0.213804 |
1.523676e-11 |
975 |
K784-3187 |
LSM-45465 |
ESR2 |
3.33uM |
24h |
LINCSCP_96511 |
LINCSCP_96511 |
HA1E |
| 0.213797 |
1.526122e-11 |
975 |
BRD-A00474148 |
LSM-45242 |
|
1.11uM |
24h |
LINCSCP_90778 |
LINCSCP_90778 |
HA1E |
| -0.213792 |
1.527960e-11 |
975 |
AC1NS4S0 |
LSM-43073 |
ATP2A1 |
10uM |
6h |
LINCSCP_12685 |
LINCSCP_12685 |
COV644 |
| 0.213788 |
1.529154e-11 |
975 |
BRD-K04086909 |
LSM-8681 |
|
5uM |
24h |
LINCSCP_61402 |
LINCSCP_61402 |
VCAP |
| -0.213761 |
1.538627e-11 |
975 |
GSK-461364 |
LSM-1013 |
PLK1 |
0.04uM |
24h |
LINCSCP_144238 |
LINCSCP_144238 |
MCF7 |
| -0.213756 |
1.540160e-11 |
975 |
Ergothioneine |
LSM-45829 |
|
10uM |
24h |
LINCSCP_102543 |
LINCSCP_102543 |
HELA |
| -0.213727 |
1.550082e-11 |
975 |
LY 2183240 |
LSM-2839 |
FAAH |
10uM |
24h |
LINCSCP_44940 |
LINCSCP_44940 |
PC3 |
| -0.213702 |
1.558628e-11 |
975 |
4449-51-8 |
LSM-4304 |
SMO |
10uM |
24h |
LINCSCP_261560 |
LINCSCP_261560 |
NPC |
| -0.213658 |
1.573972e-11 |
975 |
MG-132 |
LSM-1107 |
PSMB1 |
20uM |
24h |
LINCSCP_134726 |
LINCSCP_134726 |
MCF7 |
| -0.213621 |
1.586995e-11 |
975 |
BRD-K65093687 |
LSM-40822 |
|
10uM |
24h |
LINCSCP_193633 |
LINCSCP_193633 |
A549 |
| 0.213599 |
1.595002e-11 |
975 |
Vorinostat |
LSM-3828 |
HDAC1|HDAC2|HDAC3|HDAC6|HDAC8 |
0.1uM |
24h |
LINCSCP_176431 |
LINCSCP_176431 |
A375 |
| 0.213586 |
1.599581e-11 |
975 |
AZD-1152-HQPA |
LSM-1067 |
AURKA|AURKB |
0.5uM |
24h |
LINCSCP_51423 |
LINCSCP_51423 |
SKBR3 |
| -0.213562 |
1.607943e-11 |
975 |
Aloisine A |
LSM-4110 |
CDK2 |
10uM |
24h |
LINCSCP_44269 |
LINCSCP_44269 |
PC3 |
| -0.213559 |
1.609302e-11 |
975 |
Camptothecin |
LSM-4611 |
TOP1 |
0.12uM |
24h |
LINCSCP_138886 |
LINCSCP_138886 |
MCF7 |
| -0.213526 |
1.621079e-11 |
975 |
HG-9-91-01 |
LSM-6343 |
|
1.11uM |
24h |
LINCSCP_129603 |
LINCSCP_129603 |
JURKAT |
| -0.213514 |
1.625134e-11 |
975 |
SB-216763 |
LSM-1161 |
GSK3B |
10uM |
6h |
LINCSCP_54968 |
LINCSCP_54968 |
THP1 |
| -0.213509 |
1.627004e-11 |
975 |
Palbociclib |
LSM-1071 |
CCND1|CDK4|CDK6 |
1.11uM |
3h |
LINCSCP_130172 |
LINCSCP_130172 |
LNCAP |
| -0.213481 |
1.637377e-11 |
975 |
LY2874455 |
LSM-45659 |
|
10uM |
24h |
LINCSCP_71570 |
LINCSCP_71570 |
A375 |
| -0.213459 |
1.645241e-11 |
975 |
WH-4-025 |
LSM-44937 |
|
3.33uM |
3h |
LINCSCP_163440 |
LINCSCP_163440 |
SKBR3 |
| -0.213455 |
1.646900e-11 |
975 |
CHEMBL489621 |
LSM-4059 |
|
10uM |
6h |
LINCSCP_22260 |
LINCSCP_22260 |
HEPG2 |
| -0.213437 |
1.653308e-11 |
975 |
Clozapine |
LSM-2823 |
ADRA1A|ADRA1B|CHRM1|CHRM2|CHRM3|CHRM4|DRD1|DRD2|DRD3|DRD4|HRH1|HRH4|HTR1A|HTR1B|HTR1D|HTR1E|HTR2A|HTR2C|HTR6|HTR7 |
0.12uM |
24h |
LINCSCP_122240 |
LINCSCP_122240 |
HT29 |
| 0.213402 |
1.666380e-11 |
975 |
BRD-K41431262 |
LSM-39564 |
|
10uM |
6h |
LINCSCP_16965 |
LINCSCP_16965 |
HA1E |
| -0.213395 |
1.668888e-11 |
975 |
Primidone |
LSM-2700 |
GABRA1|GABRA2|GABRA3|GABRA4|GABRA5|GABRA6|GABRB1|GABRB2|GABRB3|GABRD|GABRE|GABRG1|GABRG2|GABRG3|GABRP|GABRQ|SCN10A|SCN11A|SCN1A|SCN2A|SCN3A|SCN4A|SCN5A|SCN7A|SCN8A|SCN9A |
10uM |
6h |
LINCSCP_212166 |
LINCSCP_212166 |
HA1E |
| -0.213393 |
1.669576e-11 |
975 |
PD-0325901 |
LSM-1101 |
MAP2K1|MAP2K2 |
10uM |
24h |
LINCSCP_166258 |
LINCSCP_166258 |
SKL |
| -0.213383 |
1.673397e-11 |
975 |
galantamine |
|
|
10uM |
24h |
LINCSCP_152275 |
LINCSCP_152275 |
PC3 |
| -0.213382 |
1.673589e-11 |
975 |
LY-294002 |
LSM-2597 |
MTOR|PIK3CA|PIK3CB|PIK3CD|PIK3CG|PLK1|PRKDC |
0.5uM |
24h |
LINCSCP_311989 |
LINCSCP_311989 |
VCAP |
| -0.21338 |
1.674485e-11 |
975 |
MLS002699810 |
LSM-4058 |
|
10uM |
24h |
LINCSCP_57587 |
LINCSCP_57587 |
VCAP |
| 0.21335 |
1.685744e-11 |
975 |
Lenalidomide |
LSM-6187 |
CRBN|CUL4A|DDB1|RBX1|TNF |
0.37uM |
24h |
LINCSCP_71656 |
LINCSCP_71656 |
A375 |
| -0.213349 |
1.685919e-11 |
975 |
KUC104493 |
LSM-2344 |
|
10uM |
24h |
LINCSCP_5376 |
LINCSCP_5376 |
A549 |
| 0.213337 |
1.690492e-11 |
975 |
Neostigmine |
LSM-5360 |
ACHE |
10uM |
24h |
LINCSCP_243951 |
LINCSCP_243951 |
MCF7 |
| 0.213333 |
1.691882e-11 |
975 |
Perphenazine |
LSM-2224 |
DRD2 |
10uM |
6h |
LINCSCP_8024 |
LINCSCP_8024 |
A549 |
| 0.213327 |
1.694083e-11 |
975 |
Linopirdine |
LSM-3317 |
KCNQ2|KCNQ3 |
10uM |
6h |
LINCSCP_528 |
LINCSCP_528 |
A375 |
| 0.213316 |
1.698435e-11 |
975 |
BRD-K22912836 |
LSM-38513 |
|
5uM |
24h |
LINCSCP_64257 |
LINCSCP_64257 |
VCAP |
| -0.213313 |
1.699659e-11 |
975 |
K784-3187 |
LSM-45465 |
ESR2 |
1.11uM |
24h |
LINCSCP_141727 |
LINCSCP_141727 |
MCF7 |
| -0.213258 |
1.720309e-11 |
975 |
CHEMBL1270504 |
LSM-2324 |
|
10uM |
6h |
LINCSCP_5480 |
LINCSCP_5480 |
A549 |
| 0.213245 |
1.725450e-11 |
975 |
SB525334 |
LSM-1121 |
TGFBR1 |
0.1uM |
24h |
LINCSCP_39389 |
LINCSCP_39389 |
MDAMB231 |
| -0.213243 |
1.726003e-11 |
975 |
Withaferin A |
LSM-6685 |
IKBKB|NAMPT |
5uM |
24h |
LINCSCP_67407 |
LINCSCP_67407 |
MCF7 |
| -0.213242 |
1.726667e-11 |
975 |
BRD-A35207501 |
LSM-45361 |
|
10uM |
6h |
LINCSCP_24161 |
LINCSCP_24161 |
HL60 |
| -0.213239 |
1.727790e-11 |
975 |
BRD-K71604153 |
LSM-12811 |
|
5uM |
6h |
LINCSCP_61369 |
LINCSCP_61369 |
VCAP |
| -0.213228 |
1.731749e-11 |
975 |
Syrosingopine |
LSM-2297 |
|
10uM |
6h |
LINCSCP_33478 |
LINCSCP_33478 |
MCF7 |
| -0.213221 |
1.734723e-11 |
975 |
13-Hydroxy-8,14,19-trimethoxy-4,10,12,16-tetramethyl-3,20,22-trioxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18-pentaen-9-yl carbamate |
LSM-42815 |
HSP90AA1 |
10uM |
24h |
LINCSCP_262745 |
LINCSCP_262745 |
NPC |
| -0.213195 |
1.744582e-11 |
975 |
Crizotinib |
LSM-1027 |
ALK|MET |
10uM |
6h |
LINCSCP_20508 |
LINCSCP_20508 |
HCC515 |
| 0.213125 |
1.772061e-11 |
975 |
YM 201636 |
LSM-1109 |
|
0.04uM |
24h |
LINCSCP_144872 |
LINCSCP_144872 |
MDAMB231 |
| 0.213104 |
1.780108e-11 |
975 |
MK-2206 |
LSM-1057 |
AKT1|AKT2|AKT3 |
1.11uM |
3h |
LINCSCP_131594 |
LINCSCP_131594 |
MCF10A |
| -0.213098 |
1.782511e-11 |
975 |
Toremifene |
LSM-42973 |
ESR1|ESR2 |
10uM |
6h |
LINCSCP_179556 |
LINCSCP_179556 |
A375 |
| 0.213081 |
1.789160e-11 |
975 |
BSPBIO_001542 |
LSM-42823 |
PPP1CA|PPP2CA |
10uM |
24h |
LINCSCP_44681 |
LINCSCP_44681 |
PC3 |
| -0.213062 |
1.796720e-11 |
975 |
NS-3694 |
LSM-2591 |
CASP9 |
10uM |
6h |
LINCSCP_4351 |
LINCSCP_4351 |
A549 |
| 0.213051 |
1.801067e-11 |
975 |
Eugenol |
LSM-2720 |
|
10uM |
24h |
LINCSCP_30272 |
LINCSCP_30272 |
MCF7 |
| -0.213043 |
1.804390e-11 |
975 |
Fcodpguefhccia-Uhfffaoysa-N |
LSM-42689 |
CASP3 |
10uM |
24h |
LINCSCP_44927 |
LINCSCP_44927 |
PC3 |
| 0.213027 |
1.810761e-11 |
975 |
SJ 172550 |
LSM-43286 |
MDM4 |
10uM |
6h |
LINCSCP_13603 |
LINCSCP_13603 |
H1299 |
| -0.212997 |
1.822767e-11 |
975 |
BAY 61-3606 |
LSM-1167 |
SYK |
3.33uM |
24h |
LINCSCP_82579 |
LINCSCP_82579 |
A549 |
| 0.21296 |
1.837876e-11 |
975 |
BRD-K36910796 |
LSM-15073 |
|
10uM |
24h |
LINCSCP_253922 |
LINCSCP_253922 |
MCF7 |
| 0.212955 |
1.839954e-11 |
975 |
Linsitinib |
LSM-1135 |
IGF1R|INSR |
0.1uM |
6h |
LINCSCP_36879 |
LINCSCP_36879 |
MCF7 |
| -0.212949 |
1.842216e-11 |
975 |
GSK-461364 |
LSM-1013 |
PLK1 |
3.33uM |
24h |
LINCSCP_86884 |
LINCSCP_86884 |
CD34 |
| -0.212947 |
1.843069e-11 |
975 |
BRD-K38986089 |
LSM-14809 |
|
5uM |
24h |
LINCSCP_309156 |
LINCSCP_309156 |
VCAP |
| -0.212939 |
1.846564e-11 |
975 |
Mebendazole |
LSM-3749 |
|
1.11uM |
24h |
LINCSCP_139712 |
LINCSCP_139712 |
MCF7 |
| -0.212929 |
1.850472e-11 |
975 |
SB-216763 |
LSM-1161 |
GSK3B |
10uM |
6h |
LINCSCP_10593 |
LINCSCP_10593 |
AGS |
| 0.21292 |
1.854237e-11 |
975 |
CHEMBL1270506 |
LSM-4218 |
|
10uM |
6h |
LINCSCP_5574 |
LINCSCP_5574 |
A549 |
| 0.212877 |
1.872137e-11 |
975 |
SCHEMBL13991002 |
LSM-6278 |
|
40uM |
6h |
LINCSCP_13588 |
LINCSCP_13588 |
H1299 |
| -0.212858 |
1.879839e-11 |
975 |
Fluphenazine |
LSM-3226 |
DRD1|DRD2 |
0.12uM |
24h |
LINCSCP_76592 |
LINCSCP_76592 |
A375 |
| 0.212811 |
1.899511e-11 |
975 |
BRD-K87159745 |
LSM-13773 |
|
5uM |
24h |
LINCSCP_63414 |
LINCSCP_63414 |
VCAP |
| 0.21281 |
1.900032e-11 |
975 |
Tamatinib |
LSM-1040 |
SYK |
0.1uM |
24h |
LINCSCP_36471 |
LINCSCP_36471 |
MCF7 |
| -0.212797 |
1.905235e-11 |
975 |
13-Methyl-7-[9-(4,4,5,5,5-pentafluoropentylsulfinyl)nonyl]-6,7,8,9,11,12,14,15,16,17-decahydrocyclopenta[a]phenanthrene-3,17-diol |
LSM-1895 |
ESR1 |
10uM |
24h |
LINCSCP_67197 |
LINCSCP_67197 |
HT29 |
| 0.212785 |
1.910619e-11 |
975 |
BRD-K20718732 |
LSM-38389 |
|
10uM |
6h |
LINCSCP_8031 |
LINCSCP_8031 |
A549 |
| -0.212779 |
1.912954e-11 |
975 |
SCHEMBL15422156 |
LSM-43123 |
|
10uM |
24h |
LINCSCP_31975 |
LINCSCP_31975 |
MCF7 |
| -0.212771 |
1.916467e-11 |
975 |
COT-10B |
LSM-6226 |
|
40uM |
24h |
LINCSCP_30507 |
LINCSCP_30507 |
MCF7 |
| 0.212766 |
1.918611e-11 |
975 |
BRD-A02747686 |
LSM-45850 |
|
1.11uM |
24h |
LINCSCP_174103 |
LINCSCP_174103 |
YAPC |
| -0.212731 |
1.933590e-11 |
975 |
AZ628 |
LSM-1050 |
BRAF|RAF1 |
10uM |
24h |
LINCSCP_170058 |
LINCSCP_170058 |
YAPC |
| -0.21272 |
1.938291e-11 |
975 |
Vinblastine |
LSM-1647 |
TUBB |
3uM |
24h |
LINCSCP_38133 |
LINCSCP_38133 |
MCF7 |
| -0.212682 |
1.954724e-11 |
975 |
Pentobarbital |
LSM-1566 |
GABRA1|GABRA2|GABRA3|GABRA4|GABRA5|GABRA6|GABRB1|GABRB2|GABRB3|GABRD|GABRE|GABRG1|GABRG2|GABRG3|GABRP|GABRQ |
0.04uM |
24h |
LINCSCP_136740 |
LINCSCP_136740 |
MCF7 |
| -0.212674 |
1.957933e-11 |
975 |
AS601245 |
LSM-1034 |
MAPK10|MAPK8|MAPK9 |
0.1uM |
24h |
LINCSCP_51270 |
LINCSCP_51270 |
SKBR3 |
| -0.212626 |
1.979064e-11 |
975 |
BRD-A24396574-001-01-5 |
LSM-5006 |
|
10uM |
3h |
LINCSCP_131616 |
LINCSCP_131616 |
MCF10A |
| 0.212623 |
1.980409e-11 |
975 |
Ticrynafen |
LSM-5478 |
CYP2C9|SLC12A1 |
10uM |
6h |
LINCSCP_3086 |
LINCSCP_3086 |
A375 |
| -0.212619 |
1.982135e-11 |
975 |
Y-39983 |
LSM-1150 |
ROCK1|ROCK2 |
10uM |
24h |
LINCSCP_36816 |
LINCSCP_36816 |
MCF7 |
| -0.212599 |
1.990754e-11 |
975 |
BRD-K98803880 |
LSM-6858 |
|
10uM |
6h |
LINCSCP_23752 |
LINCSCP_23752 |
HEPG2 |
| -0.212596 |
1.992136e-11 |
975 |
MLS002264449 |
LSM-3136 |
|
10uM |
6h |
LINCSCP_268936 |
LINCSCP_268936 |
PC3 |
| 0.212587 |
1.996045e-11 |
975 |
Y-39983 |
LSM-1150 |
ROCK1|ROCK2 |
0.12uM |
24h |
LINCSCP_115772 |
LINCSCP_115772 |
HS578T |
| -0.212579 |
1.999555e-11 |
975 |
ZINC01063165 |
LSM-4679 |
|
10uM |
24h |
LINCSCP_52261 |
LINCSCP_52261 |
SKB |
| 0.212571 |
2.003232e-11 |
975 |
Selumetinib |
LSM-1056 |
MAP2K1|MAP2K2 |
0.12uM |
3h |
LINCSCP_164106 |
LINCSCP_164106 |
SKBR3 |
| 0.212567 |
2.005009e-11 |
975 |
Imatinib |
LSM-1023 |
ABL1|BCR|CSF1R|KIT|PDGFRA|PDGFRB |
0.04uM |
24h |
LINCSCP_131437 |
LINCSCP_131437 |
MCF10A |
| 0.212562 |
2.007182e-11 |
975 |
Kenpaullone |
LSM-2824 |
CDK1|CDK5|GSK3B |
10uM |
6h |
LINCSCP_2704 |
LINCSCP_2704 |
A375 |
| 0.212561 |
2.007734e-11 |
975 |
Disopyramide |
LSM-1439 |
SCN10A|SCN11A|SCN1A|SCN2A|SCN3A|SCN4A|SCN5A|SCN7A|SCN8A|SCN9A |
0.12uM |
24h |
LINCSCP_71293 |
LINCSCP_71293 |
A375 |
| 0.212559 |
2.008372e-11 |
975 |
TWS 119 |
LSM-1111 |
GSK3B |
1.11uM |
24h |
LINCSCP_132104 |
LINCSCP_132104 |
MCF7 |
| -0.212557 |
2.009189e-11 |
975 |
Famciclovir |
LSM-2990 |
|
0.37uM |
24h |
LINCSCP_141008 |
LINCSCP_141008 |
MCF7 |
| -0.212508 |
2.031315e-11 |
975 |
SA-102042 |
LSM-40575 |
|
0.5uM |
24h |
LINCSCP_38211 |
LINCSCP_38211 |
MCF7 |
| -0.212501 |
2.034436e-11 |
975 |
MLS000038113 |
LSM-4839 |
|
10uM |
24h |
LINCSCP_32435 |
LINCSCP_32435 |
MCF7 |
| 0.212483 |
2.042435e-11 |
975 |
Strophanthidin |
LSM-3891 |
ATP1A1 |
10uM |
6h |
LINCSCP_7737 |
LINCSCP_7737 |
A549 |
| 0.212483 |
2.042522e-11 |
975 |
Mocetinostat |
LSM-5344 |
HDAC1|HDAC11|HDAC2|HDAC3|HDAC8 |
1.11uM |
24h |
LINCSCP_146863 |
LINCSCP_146863 |
NEU |
| 0.212479 |
2.044423e-11 |
975 |
BRD-K32381042 |
LSM-10395 |
|
5uM |
24h |
LINCSCP_62643 |
LINCSCP_62643 |
VCAP |
| -0.212468 |
2.049125e-11 |
975 |
MLS002264447 |
LSM-2942 |
|
10uM |
6h |
LINCSCP_45816 |
LINCSCP_45816 |
PC3 |
| 0.21246 |
2.053082e-11 |
975 |
MLS000626949 |
LSM-43326 |
|
10uM |
6h |
LINCSCP_16847 |
LINCSCP_16847 |
HA1E |
| -0.212459 |
2.053386e-11 |
975 |
HMN-214 |
LSM-42802 |
CSF1R|FLT1|FLT3|FLT4|KDR|KIT|PDGFRB|RET |
1.11uM |
24h |
LINCSCP_142603 |
LINCSCP_142603 |
MCF7 |
| -0.212452 |
2.056682e-11 |
975 |
MLS002264489 |
LSM-2871 |
|
10uM |
6h |
LINCSCP_19731 |
LINCSCP_19731 |
HCC515 |
| 0.212385 |
2.087003e-11 |
975 |
Dorzolamide HCL |
LSM-45672 |
|
0.12uM |
24h |
LINCSCP_142647 |
LINCSCP_142647 |
MCF7 |
| 0.212365 |
2.096206e-11 |
975 |
MLS003370610 |
LSM-1383 |
|
10uM |
6h |
LINCSCP_219414 |
LINCSCP_219414 |
HEPG2 |
| 0.212343 |
2.106604e-11 |
975 |
MK-8245 |
LSM-45756 |
|
10uM |
24h |
LINCSCP_71301 |
LINCSCP_71301 |
A375 |
| -0.212333 |
2.111153e-11 |
975 |
BRD-K35995762 |
LSM-10594 |
|
5uM |
24h |
LINCSCP_62448 |
LINCSCP_62448 |
VCAP |
| 0.212307 |
2.123332e-11 |
975 |
Erismodegib |
LSM-4938 |
SMO |
10uM |
6h |
LINCSCP_4727 |
LINCSCP_4727 |
A549 |
| 0.212248 |
2.151427e-11 |
975 |
Chloroxine |
LSM-2371 |
|
3.33uM |
24h |
LINCSCP_89861 |
LINCSCP_89861 |
HA1E |
| -0.212244 |
2.153258e-11 |
975 |
AC1NR4QJ |
LSM-43144 |
CYSLTR1 |
10uM |
24h |
LINCSCP_271943 |
LINCSCP_271943 |
PC3 |
| -0.21224 |
2.154996e-11 |
975 |
Tomelukast |
LSM-3675 |
CYSLTR1 |
10uM |
6h |
LINCSCP_537 |
LINCSCP_537 |
A375 |
| 0.212239 |
2.155379e-11 |
975 |
BRD-K60595380 |
LSM-12089 |
|
5uM |
24h |
LINCSCP_63716 |
LINCSCP_63716 |
VCAP |
| -0.212233 |
2.158458e-11 |
975 |
UNII-884KT10YB7 |
LSM-2298 |
HRH2 |
10uM |
24h |
LINCSCP_262847 |
LINCSCP_262847 |
NPC |
| -0.212216 |
2.166767e-11 |
975 |
TORIN-2 |
LSM-1080 |
MTOR |
1uM |
24h |
LINCSCP_29585 |
LINCSCP_29585 |
MCF10A |
| -0.212211 |
2.168913e-11 |
975 |
Ruxolitinib |
LSM-1139 |
JAK1|JAK2|TYK2 |
10uM |
6h |
LINCSCP_20468 |
LINCSCP_20468 |
HCC515 |
| -0.212202 |
2.173448e-11 |
975 |
BRD-K82927587 |
LSM-41804 |
|
5uM |
24h |
LINCSCP_48313 |
LINCSCP_48313 |
PC3 |
| -0.212196 |
2.176145e-11 |
975 |
MK-0812 |
LSM-45856 |
|
0.37uM |
24h |
LINCSCP_169737 |
LINCSCP_169737 |
YAPC |
| -0.212186 |
2.180928e-11 |
975 |
MLN-0128 |
LSM-1206 |
MTOR |
0.12uM |
24h |
LINCSCP_106404 |
LINCSCP_106404 |
HELA |
| -0.212171 |
2.188391e-11 |
975 |
Dactolisib |
LSM-4255 |
MTOR|PIK3CA|PIK3CB|PIK3CD|PIK3CG|PIK3R1|PIK3R2|PIK3R3|PIK3R5 |
0.5uM |
6h |
LINCSCP_40183 |
LINCSCP_40183 |
NCIH508 |
| 0.212152 |
2.197484e-11 |
975 |
SA-243276 |
LSM-41502 |
|
0.5uM |
24h |
LINCSCP_37732 |
LINCSCP_37732 |
MCF7 |
| -0.212152 |
2.197573e-11 |
975 |
Withaferin A |
LSM-6685 |
IKBKB|NAMPT |
10uM |
6h |
LINCSCP_68446 |
LINCSCP_68446 |
VCAP |
| -0.212142 |
2.202045e-11 |
975 |
3-(Diphenylmethoxy)-8-methyl-8-azabicyclo[3.2.1]octane |
LSM-5012 |
CHRM1 |
10uM |
24h |
LINCSCP_47270 |
LINCSCP_47270 |
PC3 |
| 0.212141 |
2.202640e-11 |
975 |
Iguratimod |
LSM-45469 |
|
1.11uM |
24h |
LINCSCP_138068 |
LINCSCP_138068 |
MCF7 |
| -0.212141 |
2.202901e-11 |
975 |
GSK 1059615 |
LSM-42799 |
PIK3CA|PIK3CB|PIK3CD|PIK3CG |
3.33uM |
24h |
LINCSCP_69046 |
LINCSCP_69046 |
A375 |
| -0.212128 |
2.209017e-11 |
975 |
C28H30CIN5O4S |
LSM-42791 |
MET |
0.1uM |
24h |
LINCSCP_12187 |
LINCSCP_12187 |
BT20 |
| -0.21211 |
2.217794e-11 |
975 |
CX-5461 |
LSM-6342 |
|
10uM |
24h |
LINCSCP_137808 |
LINCSCP_137808 |
MCF7 |
| 0.212093 |
2.226267e-11 |
975 |
BRD-K96922741 |
LSM-14379 |
|
5uM |
24h |
LINCSCP_62482 |
LINCSCP_62482 |
VCAP |
| -0.212082 |
2.231390e-11 |
975 |
BRD-K56842656 |
LSM-40388 |
|
10uM |
24h |
LINCSCP_65665 |
LINCSCP_65665 |
VCAP |
| 0.212077 |
2.234185e-11 |
975 |
BRD-K54822214 |
LSM-40272 |
|
10uM |
6h |
LINCSCP_16322 |
LINCSCP_16322 |
HA1E |
| 0.212047 |
2.248661e-11 |
975 |
BRD-K22345692 |
LSM-9782 |
|
5uM |
24h |
LINCSCP_62634 |
LINCSCP_62634 |
VCAP |
| -0.212046 |
2.249442e-11 |
975 |
MLS002264447 |
LSM-2942 |
|
10uM |
6h |
LINCSCP_31485 |
LINCSCP_31485 |
MCF7 |
| 0.212034 |
2.255272e-11 |
975 |
sorafenib |
|
BRAF|DDR2|FGFR1|FLT1|FLT3|FLT4|KDR|KIT|PDGFRB|RAF1|RET |
0.1uM |
24h |
LINCSCP_11721 |
LINCSCP_11721 |
BT20 |
| 0.212033 |
2.255963e-11 |
975 |
Clenbuterol |
LSM-5144 |
ADRB2 |
10uM |
6h |
LINCSCP_34344 |
LINCSCP_34344 |
MCF7 |
| -0.212005 |
2.269714e-11 |
975 |
KW-2478 |
LSM-45404 |
|
1.11uM |
24h |
LINCSCP_105641 |
LINCSCP_105641 |
HELA |
| 0.212003 |
2.270914e-11 |
975 |
MLS002703290 |
LSM-1784 |
|
10uM |
24h |
LINCSCP_31555 |
LINCSCP_31555 |
MCF7 |
| -0.211999 |
2.272717e-11 |
975 |
172985-18-1 |
LSM-4563 |
|
10uM |
24h |
LINCSCP_32149 |
LINCSCP_32149 |
MCF7 |
| -0.211991 |
2.276955e-11 |
975 |
Withaferin A |
LSM-6685 |
IKBKB|NAMPT |
0.01uM |
6h |
LINCSCP_9362 |
LINCSCP_9362 |
A549 |
| -0.211986 |
2.279094e-11 |
975 |
Volasertib (BI 6727) |
LSM-45277 |
PLK1 |
0.37uM |
24h |
LINCSCP_142574 |
LINCSCP_142574 |
MCF7 |
| -0.211974 |
2.285280e-11 |
975 |
I-BET151 |
LSM-6335 |
|
3.33uM |
24h |
LINCSCP_164761 |
LINCSCP_164761 |
SKL.C |
| -0.21197 |
2.287459e-11 |
975 |
13-Hydroxy-8,14,19-trimethoxy-4,10,12,16-tetramethyl-3,20,22-trioxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18-pentaen-9-yl carbamate |
LSM-42815 |
HSP90AA1 |
1uM |
6h |
LINCSCP_43933 |
LINCSCP_43933 |
PC3 |
| 0.211968 |
2.288534e-11 |
975 |
Irsogladine |
LSM-3663 |
PDE4A |
0.12uM |
24h |
LINCSCP_142845 |
LINCSCP_142845 |
MCF7 |
| -0.211915 |
2.315502e-11 |
975 |
Clofilium |
LSM-5214 |
|
10uM |
6h |
LINCSCP_34352 |
LINCSCP_34352 |
MCF7 |
| -0.211914 |
2.315716e-11 |
975 |
R-N-Propylnorapomorphine |
LSM-2281 |
DRD1|DRD2 |
10uM |
24h |
LINCSCP_14691 |
LINCSCP_14691 |
HA1E |
| -0.211913 |
2.316529e-11 |
975 |
ITK Inhibitor |
LSM-1043 |
ITK |
10uM |
24h |
LINCSCP_52321 |
LINCSCP_52321 |
SKB |
| 0.211905 |
2.320156e-11 |
975 |
ZIDOVUDINE [AZT] |
LSM-45628 |
|
10uM |
24h |
LINCSCP_74136 |
LINCSCP_74136 |
A375 |
| -0.211877 |
2.334839e-11 |
975 |
Diperodon |
LSM-4393 |
|
10uM |
6h |
LINCSCP_34336 |
LINCSCP_34336 |
MCF7 |
| -0.211871 |
2.337962e-11 |
975 |
Arachidonyl Trifluoromethylketone |
LSM-43275 |
PLA2G4A |
0.1uM |
24h |
LINCSCP_36244 |
LINCSCP_36244 |
MCF7 |
| -0.21187 |
2.338618e-11 |
975 |
BRD-K98064019 |
LSM-6170 |
|
10uM |
6h |
LINCSCP_16396 |
LINCSCP_16396 |
HA1E |
| -0.211857 |
2.345038e-11 |
975 |
MLS003587249 |
LSM-44616 |
|
10uM |
24h |
LINCSCP_242531 |
LINCSCP_242531 |
MCF7 |
| -0.211852 |
2.347722e-11 |
975 |
PF-03758309 |
LSM-4254 |
PAK4 |
3.33uM |
24h |
LINCSCP_139405 |
LINCSCP_139405 |
MCF7 |
| 0.211852 |
2.347780e-11 |
975 |
Entinostat |
LSM-4811 |
HDAC1|HDAC10|HDAC11|HDAC2|HDAC3|HDAC4|HDAC5|HDAC6|HDAC7|HDAC8|HDAC9 |
0.1uM |
24h |
LINCSCP_35524 |
LINCSCP_35524 |
MCF7 |
| -0.211843 |
2.352084e-11 |
975 |
Arctigenin |
LSM-3183 |
CHUK|MAP2K1 |
10uM |
24h |
LINCSCP_233968 |
LINCSCP_233968 |
HUH7 |
| 0.211811 |
2.369033e-11 |
975 |
Gliclazide |
LSM-5096 |
ABCC8 |
0.04uM |
24h |
LINCSCP_139877 |
LINCSCP_139877 |
MCF7 |
| -0.211802 |
2.373890e-11 |
975 |
BRD-K06589444 |
LSM-37625 |
|
10uM |
24h |
LINCSCP_42947 |
LINCSCP_42947 |
NPC |
| 0.211801 |
2.374001e-11 |
975 |
Brinzolamide |
LSM-3677 |
CA1|CA2|CA7 |
10uM |
6h |
LINCSCP_34403 |
LINCSCP_34403 |
MCF7 |
| -0.211801 |
2.374344e-11 |
975 |
Butoconazole |
LSM-1344 |
|
0.12uM |
24h |
LINCSCP_153173 |
LINCSCP_153173 |
PC3 |
| -0.211784 |
2.383181e-11 |
975 |
BRD-K35095050 |
LSM-43607 |
|
10uM |
6h |
LINCSCP_49122 |
LINCSCP_49122 |
PC3 |
| -0.211769 |
2.390972e-11 |
975 |
AZ628 |
LSM-1050 |
BRAF|RAF1 |
3.33uM |
24h |
LINCSCP_93069 |
LINCSCP_93069 |
HA1E |
| -0.211705 |
2.424763e-11 |
975 |
Rigosertib |
LSM-44531 |
CDK1|F2R|FLT1|FYN|PDGFRA|PLK1|PLK2|SRC |
0.12uM |
24h |
LINCSCP_148251 |
LINCSCP_148251 |
NPC.CAS9 |
| -0.211698 |
2.428683e-11 |
975 |
Iniparib |
LSM-6317 |
PARP1 |
0.04uM |
24h |
LINCSCP_154487 |
LINCSCP_154487 |
PC3 |
| 0.211697 |
2.429454e-11 |
975 |
Lithocholic acid |
LSM-5371 |
NR1I2|VDR |
10uM |
24h |
LINCSCP_263823 |
LINCSCP_263823 |
NPC |
| -0.211693 |
2.431331e-11 |
975 |
BRN 1088760 |
LSM-43335 |
|
10uM |
6h |
LINCSCP_32384 |
LINCSCP_32384 |
MCF7 |
| 0.211655 |
2.451546e-11 |
975 |
Alizapride |
LSM-4953 |
DRD2 |
10uM |
24h |
LINCSCP_75197 |
LINCSCP_75197 |
A375 |
| 0.211649 |
2.454934e-11 |
975 |
Calpeptin |
LSM-2570 |
|
10uM |
6h |
LINCSCP_13896 |
LINCSCP_13896 |
HA1E |
| -0.211637 |
2.461448e-11 |
975 |
Epirubicin HCl |
LSM-45684 |
|
3.33uM |
24h |
LINCSCP_139627 |
LINCSCP_139627 |
MCF7 |
| -0.21163 |
2.465521e-11 |
975 |
Doxorubicin |
LSM-4062 |
TOP2A |
10uM |
24h |
LINCSCP_191833 |
LINCSCP_191833 |
A549 |
| 0.211624 |
2.468317e-11 |
975 |
CHEMBL2135770 |
LSM-38343 |
|
10uM |
6h |
LINCSCP_211897 |
LINCSCP_211897 |
HA1E |
| 0.211606 |
2.478484e-11 |
975 |
Methyl 1-hydroxy-7-(hydroxymethyl)-1,4a,5,7a-tetrahydrocyclopenta[c]pyran-4-carboxylate |
LSM-4955 |
|
10uM |
6h |
LINCSCP_3052 |
LINCSCP_3052 |
A375 |
| -0.211599 |
2.482216e-11 |
975 |
CHEMBL3186688 |
LSM-3014 |
|
10uM |
24h |
LINCSCP_177847 |
LINCSCP_177847 |
A375 |
| 0.211577 |
2.494478e-11 |
975 |
GSK 1059615 |
LSM-42799 |
PIK3CA|PIK3CB|PIK3CD|PIK3CG |
0.04uM |
3h |
LINCSCP_130115 |
LINCSCP_130115 |
LNCAP |
| -0.211555 |
2.506419e-11 |
975 |
Canertinib |
LSM-1120 |
EGFR|ERBB2|ERBB4 |
10uM |
24h |
LINCSCP_240315 |
LINCSCP_240315 |
MCF7 |
| 0.211554 |
2.506606e-11 |
975 |
Sirolimus |
LSM-42783 |
FKBP1A|MTOR |
0.5uM |
24h |
LINCSCP_251282 |
LINCSCP_251282 |
MCF7 |
| -0.211533 |
2.518341e-11 |
975 |
Gliquidone |
LSM-3809 |
ABCC8 |
0.04uM |
24h |
LINCSCP_78177 |
LINCSCP_78177 |
A375 |
| -0.211519 |
2.525975e-11 |
975 |
4,11-Diethyl-4,9-dihydroxy-1H-pyrano[3',4':6,7]indolizino[1,2-b]quinoline-3,14(4H,12H)-dione |
LSM-6189 |
TOP1 |
0.1uM |
24h |
LINCSCP_35633 |
LINCSCP_35633 |
MCF7 |
| -0.211492 |
2.541412e-11 |
975 |
HSCI1_000313 |
LSM-2211 |
|
10uM |
6h |
LINCSCP_55785 |
LINCSCP_55785 |
VCAP |
| -0.211487 |
2.544289e-11 |
975 |
Camptothecin |
LSM-4611 |
TOP1 |
10uM |
24h |
LINCSCP_138882 |
LINCSCP_138882 |
MCF7 |
| -0.211472 |
2.552592e-11 |
975 |
Sepantronium |
LSM-5399 |
BIRC5 |
3.33uM |
24h |
LINCSCP_155386 |
LINCSCP_155386 |
PC3 |
| -0.211463 |
2.557713e-11 |
975 |
Withaferin A |
LSM-6685 |
IKBKB|NAMPT |
20uM |
6h |
LINCSCP_64598 |
LINCSCP_64598 |
VCAP |
| 0.211433 |
2.574647e-11 |
975 |
MLS001065836 |
LSM-2813 |
|
10uM |
6h |
LINCSCP_1811 |
LINCSCP_1811 |
A375 |
| 0.211428 |
2.577354e-11 |
975 |
Chaetocin |
LSM-6198 |
SUV39H1 |
0.1uM |
6h |
LINCSCP_51071 |
LINCSCP_51071 |
RMUGS |
| -0.21141 |
2.587658e-11 |
975 |
HMN-214 |
LSM-42802 |
CSF1R|FLT1|FLT3|FLT4|KDR|KIT|PDGFRB|RET |
1.11uM |
24h |
LINCSCP_148279 |
LINCSCP_148279 |
NPC.CAS9 |
| -0.211399 |
2.593971e-11 |
975 |
Cisapride |
LSM-6397 |
HTR4 |
3.33uM |
24h |
LINCSCP_74322 |
LINCSCP_74322 |
A375 |
| 0.211358 |
2.617133e-11 |
975 |
Linsitinib |
LSM-1135 |
IGF1R|INSR |
0.5uM |
24h |
LINCSCP_36771 |
LINCSCP_36771 |
MCF7 |
| -0.21134 |
2.627362e-11 |
975 |
PD-0325901 |
LSM-1101 |
MAP2K1|MAP2K2 |
10uM |
3h |
LINCSCP_145717 |
LINCSCP_145717 |
MDAMB231 |
| 0.211308 |
2.646132e-11 |
975 |
MLN 2480 |
LSM-45644 |
ARAF|BRAF|RAF1 |
0.37uM |
24h |
LINCSCP_75581 |
LINCSCP_75581 |
A375 |
| -0.2113 |
2.650671e-11 |
975 |
ZINC02121610 |
LSM-3277 |
|
10uM |
6h |
LINCSCP_26019 |
LINCSCP_26019 |
HT29 |
| 0.211292 |
2.655500e-11 |
975 |
4-Hydroxytamoxifen |
LSM-42848 |
ESR1|ESR2 |
10uM |
6h |
LINCSCP_30355 |
LINCSCP_30355 |
MCF7 |
| 0.211283 |
2.660614e-11 |
975 |
Cevimeline hydrochloride |
LSM-45454 |
|
1.11uM |
24h |
LINCSCP_73751 |
LINCSCP_73751 |
A375 |
| -0.211278 |
2.663540e-11 |
975 |
Ofloxacin |
LSM-4370 |
|
1.11uM |
24h |
LINCSCP_154076 |
LINCSCP_154076 |
PC3 |
| -0.211261 |
2.673412e-11 |
975 |
Afatinib |
LSM-43226 |
EGFR|ERBB2|ERBB4 |
10uM |
24h |
LINCSCP_32221 |
LINCSCP_32221 |
MCF7 |
| -0.211254 |
2.677690e-11 |
975 |
BRD-K69040870-001-01-4 |
LSM-41026 |
|
10uM |
24h |
LINCSCP_28382 |
LINCSCP_28382 |
HT29 |
| -0.211248 |
2.681143e-11 |
975 |
BRD-K56664261 |
LSM-40382 |
|
10uM |
24h |
LINCSCP_312028 |
LINCSCP_312028 |
VCAP |
| 0.211244 |
2.683818e-11 |
975 |
BRD-K13448237 |
LSM-9234 |
|
5uM |
24h |
LINCSCP_63666 |
LINCSCP_63666 |
VCAP |
| 0.211236 |
2.688581e-11 |
975 |
BRD-K28431278 |
LSM-38818 |
|
5uM |
24h |
LINCSCP_64267 |
LINCSCP_64267 |
VCAP |
| 0.211227 |
2.693774e-11 |
975 |
2,3-Diamino-1-phenylpropan-1-one |
LSM-1452 |
|
10uM |
24h |
LINCSCP_11228 |
LINCSCP_11228 |
ASC |
| -0.211179 |
2.722347e-11 |
975 |
Calcitriol |
LSM-45950 |
|
0.37uM |
24h |
LINCSCP_71196 |
LINCSCP_71196 |
A375 |
| 0.211176 |
2.724285e-11 |
975 |
Imatinib |
LSM-1023 |
ABL1|BCR|CSF1R|KIT|PDGFRA|PDGFRB |
0.12uM |
24h |
LINCSCP_113263 |
LINCSCP_113263 |
HME1 |
| -0.211169 |
2.728300e-11 |
975 |
1-{1-[4-(Morpholine-4-sulfonyl)-phenyl]-piperidin-4-ylmethyl}-3-o-tolyl-urea |
LSM-4851 |
|
10uM |
24h |
LINCSCP_33832 |
LINCSCP_33832 |
MCF7 |
| 0.211161 |
2.733175e-11 |
975 |
GSK-3 Inhibitor II |
LSM-1030 |
GSK3B |
10uM |
24h |
LINCSCP_129661 |
LINCSCP_129661 |
JURKAT |
| -0.211158 |
2.734964e-11 |
975 |
BRD-K20139170 |
LSM-14748 |
|
5uM |
24h |
LINCSCP_64171 |
LINCSCP_64171 |
VCAP |
| 0.211145 |
2.742486e-11 |
975 |
rifampicin |
|
|
1.11uM |
24h |
LINCSCP_115788 |
LINCSCP_115788 |
HS578T |
| 0.211127 |
2.753420e-11 |
975 |
Fipronil |
LSM-1608 |
|
0.37uM |
24h |
LINCSCP_141308 |
LINCSCP_141308 |
MCF7 |
| -0.211123 |
2.755660e-11 |
975 |
SA-1458571 |
LSM-38001 |
|
3uM |
24h |
LINCSCP_252592 |
LINCSCP_252592 |
MCF7 |
| 0.211121 |
2.756965e-11 |
975 |
ipratropium |
LSM-45809 |
|
0.37uM |
24h |
LINCSCP_123150 |
LINCSCP_123150 |
HT29 |
| 0.211121 |
2.757105e-11 |
975 |
Acetyl-Farnesyl-Cysteine |
LSM-43236 |
PPARG |
10uM |
6h |
LINCSCP_32750 |
LINCSCP_32750 |
MCF7 |
| -0.211096 |
2.772532e-11 |
975 |
DOCETAXEL |
LSM-45649 |
|
0.37uM |
24h |
LINCSCP_138261 |
LINCSCP_138261 |
MCF7 |
| -0.21109 |
2.775716e-11 |
975 |
Hydroxyprogesterone Caproate |
LSM-4900 |
AR|ESR1|ESR2|NR1H4|NR1I2|NR3C1|PGR |
10uM |
6h |
LINCSCP_217147 |
LINCSCP_217147 |
HCC515 |
| 0.211071 |
2.787549e-11 |
975 |
Etravirine (TMC125) |
LSM-45824 |
|
0.04uM |
24h |
LINCSCP_109934 |
LINCSCP_109934 |
HELA |
| -0.21105 |
2.800452e-11 |
975 |
Aurora A Inhibitor I |
LSM-1065 |
AURKA |
10uM |
24h |
LINCSCP_134079 |
LINCSCP_134079 |
MCF7 |
| -0.211009 |
2.825556e-11 |
975 |
BRD-K73276569 |
LSM-41250 |
|
10uM |
24h |
LINCSCP_233164 |
LINCSCP_233164 |
HT29 |
| -0.211008 |
2.826366e-11 |
975 |
Epothilone B (EPO906, Patupilone) |
LSM-46001 |
|
0.04uM |
24h |
LINCSCP_142102 |
LINCSCP_142102 |
MCF7 |
| -0.210962 |
2.855273e-11 |
975 |
BRD-K37852224 |
LSM-6792 |
|
10uM |
24h |
LINCSCP_31913 |
LINCSCP_31913 |
MCF7 |
| -0.210942 |
2.867458e-11 |
975 |
N-[(1-Ethylpyrrolidin-3-yl)methyl]-2-methoxy-5-sulfamoylbenzamide |
LSM-1307 |
CA7|DRD2|DRD3 |
10uM |
24h |
LINCSCP_44336 |
LINCSCP_44336 |
PC3 |
| 0.210917 |
2.883631e-11 |
975 |
SCHEMBL2554399 |
LSM-3303 |
|
10uM |
6h |
LINCSCP_219715 |
LINCSCP_219715 |
HEPG2 |
| -0.210916 |
2.884204e-11 |
975 |
Camptothecin |
LSM-4611 |
TOP1 |
3.33uM |
24h |
LINCSCP_138883 |
LINCSCP_138883 |
MCF7 |
| -0.210891 |
2.899706e-11 |
975 |
LDN 193189 |
LSM-1115 |
ACVR1|BMPR1A |
0.37uM |
24h |
LINCSCP_150874 |
LINCSCP_150874 |
PC3 |
| 0.210864 |
2.917189e-11 |
975 |
Indoprofen |
LSM-1564 |
PTGS1|PTGS2 |
0.37uM |
24h |
LINCSCP_75605 |
LINCSCP_75605 |
A375 |
| -0.210826 |
2.941421e-11 |
975 |
Zafirlukast |
LSM-5792 |
CYSLTR1 |
10uM |
24h |
LINCSCP_108869 |
LINCSCP_108869 |
HELA |
| 0.210821 |
2.944541e-11 |
975 |
Pictilisib |
LSM-1047 |
PIK3CA|PIK3CB|PIK3CD|PIK3CG|PIK3R1|PIK3R2|PIK3R3|PIK3R5 |
3.33uM |
3h |
LINCSCP_113392 |
LINCSCP_113392 |
HME1 |
| -0.210821 |
2.944644e-11 |
975 |
NG,NG-Dimethyl-L-arginine, Dihydrochloride |
LSM-45294 |
|
3.33uM |
24h |
LINCSCP_103674 |
LINCSCP_103674 |
HELA |
| -0.210821 |
2.944934e-11 |
975 |
SCHEMBL10583556 |
LSM-1657 |
PTGS1|PTGS2 |
10uM |
6h |
LINCSCP_252812 |
LINCSCP_252812 |
MCF7 |
| -0.210808 |
2.952917e-11 |
975 |
BRD-K45322187 |
LSM-39781 |
|
10uM |
6h |
LINCSCP_65153 |
LINCSCP_65153 |
VCAP |
| -0.210774 |
2.975301e-11 |
975 |
TORIN1 |
LSM-1079 |
MTOR |
10uM |
24h |
LINCSCP_111859 |
LINCSCP_111859 |
HEPG2 |
| 0.210767 |
2.979712e-11 |
975 |
Hypericin |
LSM-2650 |
|
1.11uM |
24h |
LINCSCP_71285 |
LINCSCP_71285 |
A375 |
| -0.210753 |
2.988674e-11 |
975 |
Withaferin A |
LSM-6685 |
IKBKB|NAMPT |
10uM |
24h |
LINCSCP_131976 |
LINCSCP_131976 |
MCF7 |
| -0.210735 |
3.000886e-11 |
975 |
NMS-1286937 |
LSM-45818 |
|
0.04uM |
24h |
LINCSCP_141874 |
LINCSCP_141874 |
MCF7 |
| 0.210723 |
3.008559e-11 |
975 |
BRD-K29660619 |
LSM-38887 |
|
5uM |
24h |
LINCSCP_63021 |
LINCSCP_63021 |
VCAP |
| -0.210702 |
3.022825e-11 |
975 |
MG-132 |
LSM-1107 |
PSMB1 |
20uM |
24h |
LINCSCP_134724 |
LINCSCP_134724 |
MCF7 |
| -0.2107 |
3.023682e-11 |
975 |
Wortmannin |
LSM-3947 |
PIK3CA|PIK3CG|PLK1 |
10uM |
6h |
LINCSCP_30142 |
LINCSCP_30142 |
MCF7 |
| 0.210698 |
3.025188e-11 |
975 |
Simvastatin |
LSM-2492 |
HMGCR |
10uM |
24h |
LINCSCP_28748 |
LINCSCP_28748 |
HUH7 |
| -0.210668 |
3.045050e-11 |
975 |
BRD-K07907451 |
LSM-37697 |
|
10uM |
24h |
LINCSCP_3518 |
LINCSCP_3518 |
A375 |
| 0.21065 |
3.056887e-11 |
975 |
Fluspirilene |
LSM-3748 |
DRD2|HTR2A |
5uM |
6h |
LINCSCP_12860 |
LINCSCP_12860 |
DV90 |
| -0.210628 |
3.071772e-11 |
975 |
BRD-K84245233 |
LSM-6856 |
|
5uM |
24h |
LINCSCP_34965 |
LINCSCP_34965 |
MCF7 |
| -0.210619 |
3.078139e-11 |
975 |
PD-0325901 |
LSM-1101 |
MAP2K1|MAP2K2 |
10uM |
24h |
LINCSCP_164850 |
LINCSCP_164850 |
SKL.C |
| -0.210603 |
3.088543e-11 |
975 |
COT Inhibitor-2 |
LSM-1154 |
|
0.1uM |
6h |
LINCSCP_39579 |
LINCSCP_39579 |
MDAMB231 |
| -0.210598 |
3.092159e-11 |
975 |
MLS002474240 |
LSM-39599 |
|
10uM |
24h |
LINCSCP_28251 |
LINCSCP_28251 |
HT29 |
| -0.210578 |
3.105425e-11 |
975 |
GSK-3 Inhibitor IX |
LSM-42780 |
|
0.12uM |
3h |
LINCSCP_131530 |
LINCSCP_131530 |
MCF10A |
| 0.210563 |
3.116237e-11 |
975 |
Rimonabant |
LSM-36994 |
CNR1 |
0.04uM |
24h |
LINCSCP_92720 |
LINCSCP_92720 |
HA1E |
| 0.210549 |
3.125632e-11 |
975 |
ICI 192,605 |
LSM-1887 |
|
10uM |
6h |
LINCSCP_26890 |
LINCSCP_26890 |
HT29 |
| 0.210532 |
3.137259e-11 |
975 |
BRD-K63947990 |
LSM-40766 |
|
0.5uM |
24h |
LINCSCP_37932 |
LINCSCP_37932 |
MCF7 |
| -0.210523 |
3.143432e-11 |
975 |
CO-1686 (AVL-301) |
LSM-45736 |
EGFR |
10uM |
24h |
LINCSCP_104303 |
LINCSCP_104303 |
HELA |
| 0.210505 |
3.155417e-11 |
975 |
VE-821 |
LSM-36358 |
|
0.04uM |
24h |
LINCSCP_87201 |
LINCSCP_87201 |
CD34 |
| -0.210474 |
3.177538e-11 |
975 |
BRD-K57962577 |
LSM-11931 |
|
10uM |
24h |
LINCSCP_200973 |
LINCSCP_200973 |
A549 |
| -0.210421 |
3.214276e-11 |
975 |
MLS002474203 |
LSM-6069 |
|
10uM |
6h |
LINCSCP_59312 |
LINCSCP_59312 |
VCAP |
| -0.210382 |
3.242014e-11 |
975 |
Y-39983 |
LSM-1150 |
ROCK1|ROCK2 |
10uM |
24h |
LINCSCP_139218 |
LINCSCP_139218 |
MCF7 |
| -0.210376 |
3.246192e-11 |
975 |
Selamectin |
LSM-44969 |
|
0.37uM |
24h |
LINCSCP_139737 |
LINCSCP_139737 |
MCF7 |
| -0.210366 |
3.253241e-11 |
975 |
UNC0638 |
LSM-6325 |
|
10uM |
24h |
LINCSCP_149015 |
LINCSCP_149015 |
NPC |
| 0.210361 |
3.256793e-11 |
975 |
BRD-K91745259 |
LSM-14065 |
|
10uM |
24h |
LINCSCP_9095 |
LINCSCP_9095 |
A549 |
| 0.21035 |
3.264722e-11 |
975 |
SR-02000000448 |
LSM-2483 |
|
10uM |
6h |
LINCSCP_26208 |
LINCSCP_26208 |
HT29 |
| 0.210301 |
3.299716e-11 |
975 |
BRD-K75368232 |
LSM-13037 |
|
0.5uM |
6h |
LINCSCP_37829 |
LINCSCP_37829 |
MCF7 |
| -0.210301 |
3.299893e-11 |
975 |
NCGC00012588 |
LSM-2552 |
|
10uM |
6h |
LINCSCP_5102 |
LINCSCP_5102 |
A549 |
| -0.21028 |
3.314685e-11 |
975 |
Dactolisib |
LSM-4255 |
MTOR|PIK3CA|PIK3CB|PIK3CD|PIK3CG|PIK3R1|PIK3R2|PIK3R3|PIK3R5 |
10uM |
24h |
LINCSCP_43409 |
LINCSCP_43409 |
NPC |
| -0.210262 |
3.328100e-11 |
975 |
Infigratinib |
LSM-1184 |
FGFR1|FGFR2|FGFR3|FGFR4 |
0.1uM |
24h |
LINCSCP_39401 |
LINCSCP_39401 |
MDAMB231 |
| -0.210255 |
3.333039e-11 |
975 |
Nicotine |
LSM-2093 |
CHRNA10|CHRNA4|CHRNA9|CHRNB2 |
1.11uM |
24h |
LINCSCP_74683 |
LINCSCP_74683 |
A375 |
| 0.210207 |
3.368643e-11 |
975 |
Atipamezole (hydrochloride) |
LSM-45983 |
|
0.37uM |
24h |
LINCSCP_93729 |
LINCSCP_93729 |
HA1E |
| 0.210195 |
3.376928e-11 |
975 |
PF477736 |
LSM-1112 |
CHEK1 |
0.1uM |
6h |
LINCSCP_29951 |
LINCSCP_29951 |
MCF10A |
| 0.210171 |
3.394902e-11 |
975 |
EX-8678 |
LSM-1147 |
|
3.33uM |
3h |
LINCSCP_164121 |
LINCSCP_164121 |
SKBR3 |
| -0.210143 |
3.415791e-11 |
975 |
SB743921 |
LSM-45775 |
|
1.11uM |
24h |
LINCSCP_142105 |
LINCSCP_142105 |
MCF7 |
| -0.210142 |
3.416460e-11 |
975 |
BRD-K98437249 |
LSM-15009 |
|
10uM |
24h |
LINCSCP_9101 |
LINCSCP_9101 |
A549 |
| 0.210128 |
3.426586e-11 |
975 |
GSK-3 Inhibitor IX |
LSM-42780 |
|
0.04uM |
24h |
LINCSCP_131181 |
LINCSCP_131181 |
MCF10A |
| -0.210097 |
3.449909e-11 |
975 |
CHEMBL2355586 |
LSM-6779 |
|
10uM |
6h |
LINCSCP_16897 |
LINCSCP_16897 |
HA1E |
| -0.210094 |
3.452573e-11 |
975 |
Dactolisib |
LSM-4255 |
MTOR|PIK3CA|PIK3CB|PIK3CD|PIK3CG|PIK3R1|PIK3R2|PIK3R3|PIK3R5 |
0.12uM |
24h |
LINCSCP_144853 |
LINCSCP_144853 |
MDAMB231 |
| -0.210089 |
3.455939e-11 |
975 |
PD153035 (Hydrochloride) |
LSM-45421 |
|
1.11uM |
24h |
LINCSCP_89407 |
LINCSCP_89407 |
HA1E |
| -0.210058 |
3.479903e-11 |
975 |
Trichostatin A, Streptomyces Sp. |
LSM-42814 |
HDAC1|HDAC10|HDAC3|HDAC4|HDAC6|HDAC7|HDAC8 |
0.5uM |
24h |
LINCSCP_30098 |
LINCSCP_30098 |
MCF7 |
| -0.210055 |
3.481785e-11 |
975 |
CHEMBL73824 |
LSM-2649 |
SIGMAR1 |
10uM |
24h |
LINCSCP_52745 |
LINCSCP_52745 |
SKB |
| -0.210051 |
3.485422e-11 |
975 |
SMR001317659 |
LSM-2094 |
|
10uM |
24h |
LINCSCP_30929 |
LINCSCP_30929 |
MCF7 |
| -0.210048 |
3.487683e-11 |
975 |
AZD-8055 |
LSM-1007 |
MTOR |
10uM |
24h |
LINCSCP_4587 |
LINCSCP_4587 |
A549 |
| -0.210044 |
3.490012e-11 |
975 |
Dolastatin 10 |
LSM-45943 |
|
0.04uM |
24h |
LINCSCP_143056 |
LINCSCP_143056 |
MCF7 |
| -0.21004 |
3.493572e-11 |
975 |
Panobinostat |
LSM-43059 |
HDAC1|HDAC10|HDAC11|HDAC2|HDAC3|HDAC4|HDAC5|HDAC6|HDAC7|HDAC8|HDAC9 |
0.001uM |
6h |
LINCSCP_35555 |
LINCSCP_35555 |
MCF7 |
| -0.210032 |
3.499387e-11 |
975 |
BRD-K68765796-001-01-8 |
LSM-41011 |
|
1uM |
24h |
LINCSCP_37479 |
LINCSCP_37479 |
MCF7 |
| 0.210032 |
3.499906e-11 |
975 |
Phensuximide |
LSM-1359 |
CACNA1G|CACNA1H|CACNA1I |
3.33uM |
24h |
LINCSCP_71648 |
LINCSCP_71648 |
A375 |
| -0.210026 |
3.503783e-11 |
975 |
ZM-241385 |
LSM-2444 |
ADORA1|ADORA2A|ADORA2B |
10uM |
24h |
LINCSCP_204616 |
LINCSCP_204616 |
ASC |
| -0.210025 |
3.504888e-11 |
975 |
BRD-K53325797 |
LSM-45342 |
|
3uM |
6h |
LINCSCP_205554 |
LINCSCP_205554 |
CD34 |
| -0.209996 |
3.526932e-11 |
975 |
CP-724714 |
LSM-42777 |
ERBB2 |
0.37uM |
3h |
LINCSCP_163130 |
LINCSCP_163130 |
SKBR3 |
| -0.209985 |
3.535519e-11 |
975 |
Wortmannin |
LSM-3947 |
PIK3CA|PIK3CG|PLK1 |
10uM |
24h |
LINCSCP_66549 |
LINCSCP_66549 |
A549 |
| -0.20997 |
3.546992e-11 |
975 |
BRD-K72299443 |
LSM-12860 |
|
5uM |
6h |
LINCSCP_61908 |
LINCSCP_61908 |
VCAP |
| -0.209965 |
3.551370e-11 |
975 |
BRD-A41986761 |
LSM-45957 |
|
0.37uM |
24h |
LINCSCP_101827 |
LINCSCP_101827 |
HELA |
| 0.209905 |
3.597571e-11 |
975 |
Cimetidine |
LSM-2404 |
HRH2 |
10uM |
24h |
LINCSCP_243459 |
LINCSCP_243459 |
MCF7 |
| 0.2099 |
3.601780e-11 |
975 |
ZSTK 474 |
LSM-1053 |
PIK3CG |
0.12uM |
3h |
LINCSCP_145913 |
LINCSCP_145913 |
MDAMB231 |
| -0.209893 |
3.607377e-11 |
975 |
AZD1208 |
LSM-45651 |
|
10uM |
24h |
LINCSCP_102334 |
LINCSCP_102334 |
HELA |
| -0.209873 |
3.623099e-11 |
975 |
SCHEMBL618594 |
LSM-1070 |
|
0.5uM |
24h |
LINCSCP_11614 |
LINCSCP_11614 |
BT20 |
| -0.20987 |
3.625139e-11 |
975 |
galantamine |
|
|
10uM |
24h |
LINCSCP_134073 |
LINCSCP_134073 |
MCF7 |
| 0.209864 |
3.630191e-11 |
975 |
C24H25CLFN5O3 |
LSM-42794 |
EGFR|ERBB2|ERBB4 |
0.04uM |
24h |
LINCSCP_88056 |
LINCSCP_88056 |
HA1E |
| 0.209855 |
3.637484e-11 |
975 |
CHEMBL1405981 |
LSM-2930 |
|
10uM |
24h |
LINCSCP_45307 |
LINCSCP_45307 |
PC3 |
| -0.209851 |
3.640833e-11 |
975 |
Thioproperazine |
LSM-2170 |
|
10uM |
24h |
LINCSCP_42838 |
LINCSCP_42838 |
NPC |
| -0.209829 |
3.657730e-11 |
975 |
CGS-12066A |
LSM-2420 |
HTR1B |
10uM |
24h |
LINCSCP_52579 |
LINCSCP_52579 |
SKB |
| 0.209822 |
3.663816e-11 |
975 |
N6-Methyladenosine |
LSM-3835 |
|
10uM |
24h |
LINCSCP_34317 |
LINCSCP_34317 |
MCF7 |
| -0.209777 |
3.699698e-11 |
975 |
BRD-A24396574-001-01-5 |
LSM-5006 |
|
10uM |
3h |
LINCSCP_86286 |
LINCSCP_86286 |
BT20 |
| 0.209759 |
3.714210e-11 |
975 |
L-Sulforaphane |
LSM-4919 |
NFE2L2 |
10uM |
6h |
LINCSCP_4667 |
LINCSCP_4667 |
A549 |
| 0.209748 |
3.723249e-11 |
975 |
BRD-K80553643 |
LSM-14944 |
|
5uM |
24h |
LINCSCP_64224 |
LINCSCP_64224 |
VCAP |
| -0.209746 |
3.724755e-11 |
975 |
GSK 1059615 |
LSM-42799 |
PIK3CA|PIK3CB|PIK3CD|PIK3CG |
3.33uM |
24h |
LINCSCP_114602 |
LINCSCP_114602 |
HME1 |
| -0.209735 |
3.733935e-11 |
975 |
BRD-A69951442-001-01-3 |
LSM-4466 |
NR3C1 |
10uM |
6h |
LINCSCP_54851 |
LINCSCP_54851 |
THP1 |
| -0.209732 |
3.736602e-11 |
975 |
Parthenolide |
LSM-43090 |
|
10uM |
24h |
LINCSCP_242165 |
LINCSCP_242165 |
MCF7 |
| -0.209703 |
3.759790e-11 |
975 |
Ipratropium |
LSM-1497 |
CHRM1|CHRM2|CHRM3|CHRM4 |
10uM |
6h |
LINCSCP_19163 |
LINCSCP_19163 |
HCC515 |
| -0.209701 |
3.761926e-11 |
975 |
Blebbistatin |
LSM-6195 |
MYH2 |
40uM |
6h |
LINCSCP_30719 |
LINCSCP_30719 |
MCF7 |
| -0.209694 |
3.767499e-11 |
975 |
VX-765 |
LSM-45578 |
|
0.04uM |
24h |
LINCSCP_101255 |
LINCSCP_101255 |
HELA |
| 0.209692 |
3.769151e-11 |
975 |
BRD-K90141430 |
LSM-13990 |
|
5uM |
24h |
LINCSCP_63757 |
LINCSCP_63757 |
VCAP |
| 0.209685 |
3.775021e-11 |
975 |
THIOCTIC ACID |
LSM-45889 |
|
0.04uM |
24h |
LINCSCP_153180 |
LINCSCP_153180 |
PC3 |
| 0.209679 |
3.780078e-11 |
975 |
BRD-K79522563 |
LSM-13287 |
|
5uM |
24h |
LINCSCP_62690 |
LINCSCP_62690 |
VCAP |
| -0.209675 |
3.782725e-11 |
975 |
BRD-K84245233 |
LSM-6856 |
|
3uM |
6h |
LINCSCP_23740 |
LINCSCP_23740 |
HEPG2 |
| -0.209669 |
3.788122e-11 |
975 |
ZINC01792951 |
LSM-2717 |
|
10uM |
24h |
LINCSCP_30958 |
LINCSCP_30958 |
MCF7 |
| 0.209659 |
3.796416e-11 |
975 |
MILNACIPRAN HYDROCHLORIDE |
LSM-45870 |
SLC6A2|SLC6A4 |
0.04uM |
24h |
LINCSCP_74533 |
LINCSCP_74533 |
A375 |
| 0.20964 |
3.811700e-11 |
975 |
CHEMBL472694 |
LSM-42830 |
GABBR1|GABBR2|SLC52A2 |
10uM |
6h |
LINCSCP_7646 |
LINCSCP_7646 |
A549 |
| 0.209639 |
3.812996e-11 |
975 |
SA-1939079 |
LSM-41390 |
|
0.5uM |
24h |
LINCSCP_37043 |
LINCSCP_37043 |
MCF7 |
| -0.209634 |
3.817020e-11 |
975 |
CEP-32496 |
LSM-45568 |
BRAF|EGFR|RET |
10uM |
24h |
LINCSCP_72923 |
LINCSCP_72923 |
A375 |
| 0.209621 |
3.827471e-11 |
975 |
Indoprofen |
LSM-1564 |
PTGS1|PTGS2 |
10uM |
24h |
LINCSCP_75602 |
LINCSCP_75602 |
A375 |
| -0.209603 |
3.842808e-11 |
975 |
Ergothioneine |
LSM-45829 |
|
0.12uM |
24h |
LINCSCP_72421 |
LINCSCP_72421 |
A375 |
| -0.209596 |
3.848461e-11 |
975 |
BRD-K47419679 |
LSM-39895 |
|
10uM |
6h |
LINCSCP_65829 |
LINCSCP_65829 |
VCAP |
| -0.209596 |
3.848936e-11 |
975 |
BRD-K31000214 |
LSM-10298 |
|
5uM |
6h |
LINCSCP_63146 |
LINCSCP_63146 |
VCAP |
| -0.209583 |
3.859862e-11 |
975 |
Benzylpenicillin |
LSM-3229 |
|
0.04uM |
24h |
LINCSCP_76617 |
LINCSCP_76617 |
A375 |
| -0.209569 |
3.871174e-11 |
975 |
Saracatinib |
LSM-1032 |
ABL1|SRC |
0.04uM |
3h |
LINCSCP_131555 |
LINCSCP_131555 |
MCF10A |
| -0.209564 |
3.875547e-11 |
975 |
Chelidonine |
LSM-2715 |
|
10uM |
6h |
LINCSCP_30367 |
LINCSCP_30367 |
MCF7 |
| 0.209545 |
3.891845e-11 |
975 |
BRD-K31815095 |
LSM-10358 |
|
5uM |
24h |
LINCSCP_63217 |
LINCSCP_63217 |
VCAP |
| -0.209544 |
3.892477e-11 |
975 |
PLX-4720 |
LSM-1049 |
BRAF |
3uM |
6h |
LINCSCP_39 |
LINCSCP_39 |
A375 |
| 0.209541 |
3.894779e-11 |
975 |
GMX1778 |
LSM-6247 |
NAMPT |
0.1uM |
24h |
LINCSCP_15327 |
LINCSCP_15327 |
HA1E |
| 0.209538 |
3.897893e-11 |
975 |
BRD-K62595167 |
LSM-12228 |
|
5uM |
24h |
LINCSCP_61630 |
LINCSCP_61630 |
VCAP |
| -0.209508 |
3.923563e-11 |
975 |
Vinblastine |
LSM-1647 |
TUBB |
1uM |
24h |
LINCSCP_38132 |
LINCSCP_38132 |
MCF7 |
| 0.209503 |
3.927776e-11 |
975 |
Alectinib |
LSM-1202 |
ALK|RET |
3.33uM |
24h |
LINCSCP_102910 |
LINCSCP_102910 |
HELA |
| -0.209502 |
3.928544e-11 |
975 |
Physostigmine |
LSM-2558 |
ACHE |
10uM |
24h |
LINCSCP_203943 |
LINCSCP_203943 |
ASC |
| -0.209499 |
3.930939e-11 |
975 |
Neratinib |
LSM-42778 |
EGFR|ERBB2|ERBB4 |
3.33uM |
24h |
LINCSCP_114740 |
LINCSCP_114740 |
HS578T |
| 0.209448 |
3.974462e-11 |
975 |
Hypericin |
LSM-2650 |
|
0.04uM |
24h |
LINCSCP_71288 |
LINCSCP_71288 |
A375 |
| 0.209444 |
3.977981e-11 |
975 |
Lapatinib |
LSM-1051 |
EGFR|ERBB2 |
0.5uM |
6h |
LINCSCP_11918 |
LINCSCP_11918 |
BT20 |
| -0.209443 |
3.978772e-11 |
975 |
Phorbol 12-myristate-13-acetate |
LSM-4341 |
PRKCA |
10uM |
24h |
LINCSCP_44821 |
LINCSCP_44821 |
PC3 |
| -0.20943 |
3.990437e-11 |
975 |
Sepantronium |
LSM-5399 |
BIRC5 |
0.12uM |
24h |
LINCSCP_137182 |
LINCSCP_137182 |
MCF7 |
| 0.209398 |
4.018628e-11 |
975 |
BRD-K79260832 |
LSM-14938 |
|
5uM |
24h |
LINCSCP_64220 |
LINCSCP_64220 |
VCAP |
| 0.209396 |
4.019700e-11 |
975 |
Pyrazolanthrone |
LSM-1163 |
MAPK10|MAPK8|MAPK9|TTK |
10uM |
6h |
LINCSCP_56118 |
LINCSCP_56118 |
VCAP |
| 0.209387 |
4.027772e-11 |
975 |
SA-427069 |
LSM-39453 |
|
3uM |
6h |
LINCSCP_37123 |
LINCSCP_37123 |
MCF7 |
| -0.209383 |
4.031316e-11 |
975 |
Rabusertib |
LSM-36359 |
CHEK1 |
3.33uM |
24h |
LINCSCP_148056 |
LINCSCP_148056 |
NPC.CAS9 |
| -0.209367 |
4.045128e-11 |
975 |
Thiorphan |
LSM-1652 |
MME |
10uM |
6h |
LINCSCP_33692 |
LINCSCP_33692 |
MCF7 |
| -0.209358 |
4.053340e-11 |
975 |
cortisone-acetate |
LSM-45387 |
TUBA1A|TUBA1B|TUBA1C|TUBA3E|TUBA4A|TUBB|TUBB1|TUBB2A|TUBB2B|TUBB3|TUBB4A|TUBB4B|TUBB6|TUBB8 |
0.04uM |
24h |
LINCSCP_143284 |
LINCSCP_143284 |
MCF7 |
| -0.209357 |
4.054453e-11 |
975 |
Trichostatin A, Streptomyces Sp. |
LSM-42814 |
HDAC1|HDAC10|HDAC3|HDAC4|HDAC6|HDAC7|HDAC8 |
10uM |
6h |
LINCSCP_68236 |
LINCSCP_68236 |
SNGM |
| 0.209349 |
4.060930e-11 |
975 |
noscapine |
|
|
0.12uM |
24h |
LINCSCP_129988 |
LINCSCP_129988 |
LNCAP |
| -0.209339 |
4.070207e-11 |
975 |
MLN-8054 |
LSM-1066 |
AURKA |
1.11uM |
24h |
LINCSCP_148143 |
LINCSCP_148143 |
NPC.CAS9 |
| 0.209337 |
4.071558e-11 |
975 |
KUC111774N |
LSM-36810 |
|
3uM |
6h |
LINCSCP_280134 |
LINCSCP_280134 |
PC3 |
| -0.209335 |
4.073874e-11 |
975 |
ML162 |
LSM-1493 |
|
10uM |
24h |
LINCSCP_44828 |
LINCSCP_44828 |
PC3 |
| -0.209333 |
4.075810e-11 |
975 |
Tipifarnib |
LSM-6258 |
CHURC1-FNTB|FNTA|FNTB |
10uM |
6h |
LINCSCP_12724 |
LINCSCP_12724 |
COV644 |
| 0.209326 |
4.081805e-11 |
975 |
Tamatinib |
LSM-1040 |
SYK |
0.04uM |
3h |
LINCSCP_145686 |
LINCSCP_145686 |
MDAMB231 |
| 0.209318 |
4.088762e-11 |
975 |
Pomalidomide |
LSM-45637 |
CRBN|CUL4A|DDB1|RBX1 |
0.04uM |
24h |
LINCSCP_74314 |
LINCSCP_74314 |
A375 |
| 0.209316 |
4.090935e-11 |
975 |
BRD-M88044810 |
LSM-45075 |
|
5uM |
24h |
LINCSCP_64053 |
LINCSCP_64053 |
VCAP |
| -0.209316 |
4.091002e-11 |
975 |
GSK 1059615 |
LSM-42799 |
PIK3CA|PIK3CB|PIK3CD|PIK3CG |
10uM |
24h |
LINCSCP_149313 |
LINCSCP_149313 |
NPC |
| 0.209308 |
4.097551e-11 |
975 |
Tivozanib |
LSM-1005 |
FLT1|FLT4|KDR|KIT|PDGFRA|PDGFRB |
1uM |
24h |
LINCSCP_39029 |
LINCSCP_39029 |
MDAMB231 |
| 0.209301 |
4.103763e-11 |
975 |
Benfluorex |
LSM-4365 |
HMGCR |
3uM |
24h |
LINCSCP_252547 |
LINCSCP_252547 |
MCF7 |
| -0.209278 |
4.124467e-11 |
975 |
Albendazole |
LSM-3782 |
|
3.33uM |
24h |
LINCSCP_143472 |
LINCSCP_143472 |
MCF7 |
| -0.209259 |
4.141651e-11 |
975 |
Dihydrocapsaicin |
LSM-37095 |
|
10uM |
24h |
LINCSCP_43451 |
LINCSCP_43451 |
NPC |
| -0.209258 |
4.142547e-11 |
975 |
Vidofludimus |
LSM-45600 |
|
10uM |
24h |
LINCSCP_106119 |
LINCSCP_106119 |
HELA |
| -0.209216 |
4.180365e-11 |
975 |
CHEMBL2137429 |
LSM-7427 |
|
5uM |
24h |
LINCSCP_60037 |
LINCSCP_60037 |
VCAP |
| -0.209213 |
4.183356e-11 |
975 |
Cilnidipine |
LSM-1284 |
CACNA1B |
10uM |
6h |
LINCSCP_227070 |
LINCSCP_227070 |
HT29 |
| 0.209212 |
4.184342e-11 |
975 |
SA-84905 |
LSM-38061 |
|
3uM |
24h |
LINCSCP_38154 |
LINCSCP_38154 |
MCF7 |
| -0.209195 |
4.199377e-11 |
975 |
Delcorine |
LSM-1882 |
|
10uM |
24h |
LINCSCP_204318 |
LINCSCP_204318 |
ASC |
| -0.209186 |
4.207554e-11 |
975 |
GSK 1059615 |
LSM-42799 |
PIK3CA|PIK3CB|PIK3CD|PIK3CG |
0.37uM |
24h |
LINCSCP_164769 |
LINCSCP_164769 |
SKL.C |
| 0.209186 |
4.207832e-11 |
975 |
Fenipentol |
LSM-5117 |
|
10uM |
24h |
LINCSCP_34455 |
LINCSCP_34455 |
MCF7 |
| -0.209181 |
4.212707e-11 |
975 |
Rabeprazole |
LSM-5045 |
ATP4A|ATP4B |
10uM |
24h |
LINCSCP_46058 |
LINCSCP_46058 |
PC3 |
| 0.209173 |
4.220240e-11 |
975 |
Carvedilol |
LSM-1310 |
ADRA1A|ADRA1B|ADRA1D|ADRB1|ADRB2|ADRB3 |
0.37uM |
24h |
LINCSCP_72737 |
LINCSCP_72737 |
A375 |
| 0.209146 |
4.244310e-11 |
975 |
Raloxifene |
LSM-3425 |
ESR1|ESR2 |
0.04uM |
24h |
LINCSCP_202639 |
LINCSCP_202639 |
A549 |
| -0.209145 |
4.245147e-11 |
975 |
Clorgiline |
LSM-5808 |
MAOA |
10uM |
24h |
LINCSCP_47555 |
LINCSCP_47555 |
PC3 |
| 0.209142 |
4.247913e-11 |
975 |
GSK-1904529A |
LSM-1134 |
IGF1R|INSR |
10uM |
24h |
LINCSCP_39352 |
LINCSCP_39352 |
MDAMB231 |
| -0.209139 |
4.250817e-11 |
975 |
Dihydroorotate Dehydrogenase Inhibitor, Brequinar |
LSM-45952 |
|
3.33uM |
24h |
LINCSCP_144450 |
LINCSCP_144450 |
MCF7 |
| -0.209135 |
4.255204e-11 |
975 |
JX401 |
LSM-2097 |
MAPK14 |
10uM |
6h |
LINCSCP_7413 |
LINCSCP_7413 |
A549 |
| -0.209133 |
4.256468e-11 |
975 |
Pimasertib |
LSM-5946 |
MAP2K1|MAP2K2 |
3.33uM |
24h |
LINCSCP_120774 |
LINCSCP_120774 |
HT29 |
| -0.209116 |
4.272780e-11 |
975 |
PI-103 |
LSM-1126 |
MTOR|PIK3CA|PIK3CB|PIK3CD|PIK3CG |
0.37uM |
24h |
LINCSCP_81553 |
LINCSCP_81553 |
A549 |
| -0.209113 |
4.275425e-11 |
975 |
BRD-K17139610 |
LSM-9464 |
|
10uM |
24h |
LINCSCP_48427 |
LINCSCP_48427 |
PC3 |
| -0.209082 |
4.304036e-11 |
975 |
BRD-A84327315-001-01-1 |
LSM-43157 |
VDR |
10uM |
24h |
LINCSCP_52339 |
LINCSCP_52339 |
SKB |
| -0.209081 |
4.304953e-11 |
975 |
TORIN1 |
LSM-1079 |
MTOR |
10uM |
24h |
LINCSCP_136998 |
LINCSCP_136998 |
MCF7 |
| -0.209065 |
4.320043e-11 |
975 |
17-DMAG (Alvespimycin) HCl |
LSM-46133 |
|
10uM |
24h |
LINCSCP_101860 |
LINCSCP_101860 |
HELA |
| 0.209063 |
4.322228e-11 |
975 |
Buparlisib |
LSM-1148 |
PIK3CA|PIK3CB|PIK3CD|PIK3CG|PIK3R1|PIK3R2|PIK3R3|PIK3R5 |
1uM |
6h |
LINCSCP_12289 |
LINCSCP_12289 |
BT20 |
| -0.209049 |
4.334652e-11 |
975 |
Indinavir |
LSM-5471 |
CYP3A4|CYP3A5|CYP3A7 |
10uM |
6h |
LINCSCP_46154 |
LINCSCP_46154 |
PC3 |
| -0.209039 |
4.344424e-11 |
975 |
Doxylamine |
LSM-1563 |
HRH1 |
10uM |
24h |
LINCSCP_284601 |
LINCSCP_284601 |
SKB |
| -0.209034 |
4.349343e-11 |
975 |
Foretinib |
LSM-1158 |
FLT1|FLT3|FLT4|KDR|KIT|MET|PDGFRA|PDGFRB|TEK |
3.33uM |
24h |
LINCSCP_99511 |
LINCSCP_99511 |
HCC515 |
| -0.209024 |
4.358839e-11 |
975 |
BRD-K46047563 |
LSM-39824 |
|
10uM |
6h |
LINCSCP_279076 |
LINCSCP_279076 |
PC3 |
| -0.209012 |
4.370414e-11 |
975 |
methiazole |
LSM-46021 |
|
10uM |
6h |
LINCSCP_55564 |
LINCSCP_55564 |
U937 |
| -0.209003 |
4.378238e-11 |
975 |
GSK-461364 |
LSM-1013 |
PLK1 |
0.37uM |
24h |
LINCSCP_82099 |
LINCSCP_82099 |
A549 |
| -0.20899 |
4.391006e-11 |
975 |
Griseofulvin |
LSM-5259 |
|
1.11uM |
24h |
LINCSCP_74251 |
LINCSCP_74251 |
A375 |
| 0.20895 |
4.429720e-11 |
975 |
BRD-K65997856 |
LSM-43352 |
|
10uM |
6h |
LINCSCP_23696 |
LINCSCP_23696 |
HEPG2 |
| 0.208936 |
4.443035e-11 |
975 |
2-(4-chlorophenyl)-3-(2-methoxyphenyl)hexahydro-1H-pyrrolo[1,2-c]imidazol-1-one |
LSM-45309 |
|
1uM |
24h |
LINCSCP_288758 |
LINCSCP_288758 |
U937 |
| -0.208932 |
4.446798e-11 |
975 |
CHEMBL490083 |
LSM-2547 |
|
10uM |
6h |
LINCSCP_45381 |
LINCSCP_45381 |
PC3 |
| -0.20893 |
4.448859e-11 |
975 |
Targinine |
LSM-36418 |
|
1.11uM |
24h |
LINCSCP_157531 |
LINCSCP_157531 |
PC3 |
| -0.208928 |
4.450859e-11 |
975 |
Calcipotriene |
LSM-42986 |
VDR |
10uM |
6h |
LINCSCP_270041 |
LINCSCP_270041 |
PC3 |
| -0.208881 |
4.495944e-11 |
975 |
179324-69-7 |
LSM-6281 |
ADRM1|PSMA1|PSMA2|PSMA3|PSMA4|PSMA5|PSMA6|PSMA7|PSMA8|PSMB1|PSMB10|PSMB11|PSMB2|PSMB3|PSMB4|PSMB5|PSMB6|PSMB7|PSMB8|PSMB9|PSMC1|PSMC2|PSMC3|PSMC4|PSMC5|PSMC6|PSMD1|PSMD11|PSMD12|PSMD13|PSMD14|PSMD2|PSMD3|PSMD4|PSMD6|PSMD7|PSMD8|SEM1 |
20uM |
24h |
LINCSCP_71507 |
LINCSCP_71507 |
A375 |
| -0.208874 |
4.503439e-11 |
975 |
AC1M43RN |
LSM-3363 |
|
10uM |
6h |
LINCSCP_15886 |
LINCSCP_15886 |
HA1E |
| -0.208837 |
4.538902e-11 |
975 |
KX2-391 |
LSM-45890 |
SRC |
0.37uM |
24h |
LINCSCP_155705 |
LINCSCP_155705 |
PC3 |
| 0.20883 |
4.546224e-11 |
975 |
9-Fluoro-11,17,21-trihydroxy-16-methylpregna-1,4-diene-3,20-dione |
LSM-4412 |
NR3C1 |
10uM |
6h |
LINCSCP_210578 |
LINCSCP_210578 |
HA1E |
| -0.2088 |
4.575511e-11 |
975 |
CHEMBL3182395 |
LSM-1164 |
MAP2K5|MAPK7 |
1uM |
24h |
LINCSCP_12217 |
LINCSCP_12217 |
BT20 |
| 0.208763 |
4.612631e-11 |
975 |
BRD-K20718732 |
LSM-38389 |
|
10uM |
6h |
LINCSCP_59576 |
LINCSCP_59576 |
VCAP |
| 0.208755 |
4.621154e-11 |
975 |
LRRK2-IN-1 |
LSM-1086 |
LRRK2 |
0.12uM |
24h |
LINCSCP_151439 |
LINCSCP_151439 |
PC3 |
| -0.208719 |
4.657083e-11 |
975 |
MLS002264463 |
LSM-3956 |
|
10uM |
6h |
LINCSCP_45625 |
LINCSCP_45625 |
PC3 |
| -0.208711 |
4.665610e-11 |
975 |
Infigratinib |
LSM-1184 |
FGFR1|FGFR2|FGFR3|FGFR4 |
0.5uM |
24h |
LINCSCP_24738 |
LINCSCP_24738 |
HS578T |
| -0.208709 |
4.667239e-11 |
975 |
SA-424380 |
LSM-37422 |
|
10uM |
24h |
LINCSCP_38135 |
LINCSCP_38135 |
MCF7 |
| 0.208705 |
4.670915e-11 |
975 |
HG6-64-1 |
LSM-43248 |
|
0.5uM |
24h |
LINCSCP_39124 |
LINCSCP_39124 |
MDAMB231 |
| -0.208702 |
4.674638e-11 |
975 |
CGS-15943 |
LSM-3076 |
ADORA1|ADORA2A|ADORA2B |
40uM |
6h |
LINCSCP_67582 |
LINCSCP_67582 |
MCF7 |
| 0.208676 |
4.701208e-11 |
975 |
Withaferin A |
LSM-6685 |
IKBKB|NAMPT |
0.5uM |
24h |
LINCSCP_43925 |
LINCSCP_43925 |
PC3 |
| 0.208668 |
4.708433e-11 |
975 |
Saracatinib |
LSM-1032 |
ABL1|SRC |
10uM |
3h |
LINCSCP_145699 |
LINCSCP_145699 |
MDAMB231 |
| -0.208668 |
4.708912e-11 |
975 |
761437-28-9 |
LSM-1208 |
|
1.11uM |
24h |
LINCSCP_149807 |
LINCSCP_149807 |
NPC.TAK |
| 0.208667 |
4.710020e-11 |
975 |
BRD-K32755775 |
LSM-10414 |
|
5uM |
24h |
LINCSCP_63362 |
LINCSCP_63362 |
VCAP |
| -0.208652 |
4.725460e-11 |
975 |
Isoreserpine |
LSM-2816 |
SLC18A1|SLC18A2 |
10uM |
24h |
LINCSCP_55979 |
LINCSCP_55979 |
VCAP |
| -0.208608 |
4.770915e-11 |
975 |
Masitinib |
LSM-1130 |
FGFR3|KIT|LYN|PDGFRA|PDGFRB |
0.37uM |
24h |
LINCSCP_86699 |
LINCSCP_86699 |
CD34 |
| -0.208601 |
4.777547e-11 |
975 |
Bosutinib |
LSM-1190 |
ABL1|BCR|CAMK2G|HCK|LYN|SRC |
10uM |
24h |
LINCSCP_148491 |
LINCSCP_148491 |
NPC |
| 0.208596 |
4.782883e-11 |
975 |
BRD-K47284302 |
LSM-11317 |
|
5uM |
24h |
LINCSCP_63699 |
LINCSCP_63699 |
VCAP |
| -0.208586 |
4.793400e-11 |
975 |
1,4-Diamino-2,3-dicyano-1,4-bis(methylthio)butadiene |
LSM-42967 |
|
10uM |
24h |
LINCSCP_324 |
LINCSCP_324 |
A375 |
| -0.208563 |
4.817360e-11 |
975 |
BRD-K86948282 |
LSM-42014 |
|
10uM |
24h |
LINCSCP_311770 |
LINCSCP_311770 |
VCAP |
| -0.208536 |
4.845093e-11 |
975 |
BRD-K59201357 |
LSM-40508 |
|
10uM |
24h |
LINCSCP_65318 |
LINCSCP_65318 |
VCAP |
| -0.208532 |
4.849902e-11 |
975 |
Leu-Enkephalin |
LSM-1461 |
OPRD1|OPRM1 |
10uM |
6h |
LINCSCP_25319 |
LINCSCP_25319 |
HT29 |
| -0.208504 |
4.879545e-11 |
975 |
AC1NX97Q |
LSM-45125 |
|
0.1uM |
24h |
LINCSCP_48083 |
LINCSCP_48083 |
PC3 |
| 0.208493 |
4.890538e-11 |
975 |
Petcm |
LSM-1917 |
|
10uM |
6h |
LINCSCP_4329 |
LINCSCP_4329 |
A549 |
| -0.208486 |
4.898590e-11 |
975 |
172516-41-5 |
LSM-3332 |
|
10uM |
24h |
LINCSCP_4980 |
LINCSCP_4980 |
A549 |
| -0.208453 |
4.933865e-11 |
975 |
CGS-12066A |
LSM-2420 |
HTR1B |
10uM |
6h |
LINCSCP_269954 |
LINCSCP_269954 |
PC3 |
| -0.208452 |
4.934087e-11 |
975 |
Vemurafenib |
LSM-1068 |
BRAF |
10uM |
6h |
LINCSCP_188167 |
LINCSCP_188167 |
A549 |
| 0.208447 |
4.939841e-11 |
975 |
BRD-K73602693 |
LSM-41271 |
|
1uM |
6h |
LINCSCP_254162 |
LINCSCP_254162 |
MCF7 |
| 0.208443 |
4.944088e-11 |
975 |
TWS 119 |
LSM-1111 |
GSK3B |
0.12uM |
24h |
LINCSCP_130695 |
LINCSCP_130695 |
MCF10A |
| -0.208421 |
4.968217e-11 |
975 |
BRD-K23001296 |
LSM-8169 |
|
5uM |
24h |
LINCSCP_60742 |
LINCSCP_60742 |
VCAP |
| -0.208416 |
4.972847e-11 |
975 |
SCHEMBL15422032 |
LSM-43336 |
|
10uM |
6h |
LINCSCP_16375 |
LINCSCP_16375 |
HA1E |
| -0.208415 |
4.974492e-11 |
975 |
PFI-1 |
LSM-6331 |
|
10uM |
24h |
LINCSCP_164670 |
LINCSCP_164670 |
SKL.C |
| 0.208384 |
5.007910e-11 |
975 |
BRD-K19890875 |
LSM-9633 |
|
5uM |
24h |
LINCSCP_62127 |
LINCSCP_62127 |
VCAP |
| -0.208358 |
5.036109e-11 |
975 |
Deoxycholic acid |
LSM-5529 |
GPBAR1 |
1.11uM |
24h |
LINCSCP_106139 |
LINCSCP_106139 |
HELA |
| 0.20833 |
5.066877e-11 |
975 |
HY-11007 |
LSM-1022 |
ABL1|BCR |
1.11uM |
24h |
LINCSCP_152211 |
LINCSCP_152211 |
PC3 |
| -0.208315 |
5.083343e-11 |
975 |
CHEMBL2139002 |
LSM-39211 |
|
10uM |
6h |
LINCSCP_23183 |
LINCSCP_23183 |
HEPG2 |
| -0.208308 |
5.091188e-11 |
975 |
Wortmannin |
LSM-3947 |
PIK3CA|PIK3CG|PLK1 |
10uM |
24h |
LINCSCP_67771 |
LINCSCP_67771 |
NPC |
| 0.208307 |
5.092005e-11 |
975 |
Endecaphyllin X |
LSM-3220 |
|
10uM |
6h |
LINCSCP_22946 |
LINCSCP_22946 |
HEPG2 |
| -0.208303 |
5.096709e-11 |
975 |
Ponatinib |
LSM-1151 |
ABL1|BCR|FGFR1|FGFR2|FGFR3|FGFR4|FLT3|KIT|RET|TEK |
10uM |
24h |
LINCSCP_166055 |
LINCSCP_166055 |
SKL |
| -0.2083 |
5.100074e-11 |
975 |
Mebendazole |
LSM-3749 |
|
10uM |
24h |
LINCSCP_67631 |
LINCSCP_67631 |
MCF7 |
| 0.208287 |
5.114310e-11 |
975 |
Lapatinib |
LSM-1051 |
EGFR|ERBB2 |
10uM |
3h |
LINCSCP_86436 |
LINCSCP_86436 |
BT20 |
| 0.208285 |
5.116300e-11 |
975 |
AMD-070 (hydrochloride) |
LSM-45591 |
|
0.12uM |
24h |
LINCSCP_75546 |
LINCSCP_75546 |
A375 |
| 0.208277 |
5.125532e-11 |
975 |
PF477736 |
LSM-1112 |
CHEK1 |
0.5uM |
6h |
LINCSCP_39522 |
LINCSCP_39522 |
MDAMB231 |
| 0.208274 |
5.128961e-11 |
975 |
Cilomilast |
LSM-5719 |
PDE4A|PDE4B|PDE4D |
10uM |
6h |
LINCSCP_32357 |
LINCSCP_32357 |
MCF7 |
| 0.208256 |
5.148994e-11 |
975 |
MLS003129153 |
LSM-7923 |
|
5uM |
24h |
LINCSCP_60628 |
LINCSCP_60628 |
VCAP |
| 0.208255 |
5.149477e-11 |
975 |
Trametinib |
LSM-1143 |
MAP2K1|MAP2K2 |
0.04uM |
3h |
LINCSCP_163480 |
LINCSCP_163480 |
SKBR3 |
| 0.208246 |
5.159785e-11 |
975 |
BRD-K57732441 |
LSM-40434 |
|
10uM |
6h |
LINCSCP_217283 |
LINCSCP_217283 |
HCC515 |
| -0.208224 |
5.184662e-11 |
975 |
Broad-Sai-560 |
LSM-45991 |
|
5uM |
24h |
LINCSCP_35539 |
LINCSCP_35539 |
MCF7 |
| -0.208205 |
5.206065e-11 |
975 |
MLS003128681 |
LSM-12649 |
|
5uM |
24h |
LINCSCP_309451 |
LINCSCP_309451 |
VCAP |
| -0.20817 |
5.245728e-11 |
975 |
AT-7519 |
LSM-1004 |
CDK1|CDK10|CDK11B|CDK12|CDK13|CDK14|CDK15|CDK16|CDK17|CDK18|CDK19|CDK2|CDK20|CDK3|CDK4|CDK5|CDK6|CDK7|CDK8|CDK9 |
0.04uM |
24h |
LINCSCP_169715 |
LINCSCP_169715 |
YAPC |
| 0.208155 |
5.262111e-11 |
975 |
MLS003448141 |
LSM-2187 |
|
10uM |
6h |
LINCSCP_19691 |
LINCSCP_19691 |
HCC515 |
| -0.20815 |
5.268078e-11 |
975 |
Broad-Sai-424 |
LSM-45346 |
|
3uM |
6h |
LINCSCP_35457 |
LINCSCP_35457 |
MCF7 |
| 0.208136 |
5.283424e-11 |
975 |
BRD-K01497355 |
LSM-37354 |
|
10uM |
24h |
LINCSCP_8985 |
LINCSCP_8985 |
A549 |
| 0.208134 |
5.285728e-11 |
975 |
BRD-K01289045 |
LSM-8512 |
|
5uM |
24h |
LINCSCP_61398 |
LINCSCP_61398 |
VCAP |
| 0.208127 |
5.294722e-11 |
975 |
Antipyrine |
LSM-3038 |
|
3uM |
24h |
LINCSCP_23424 |
LINCSCP_23424 |
HEPG2 |
| 0.208119 |
5.303031e-11 |
975 |
NCGC00025312-01 |
LSM-2901 |
PPARD |
10uM |
24h |
LINCSCP_52893 |
LINCSCP_52893 |
SKB |
| -0.208111 |
5.312191e-11 |
975 |
GSK-1070916 |
LSM-1062 |
AURKB|AURKC |
10uM |
24h |
LINCSCP_120473 |
LINCSCP_120473 |
HT29 |
| 0.208069 |
5.361310e-11 |
975 |
Dorzolamide HCL |
LSM-45672 |
|
0.37uM |
24h |
LINCSCP_142646 |
LINCSCP_142646 |
MCF7 |
| -0.208055 |
5.377653e-11 |
975 |
Deoxycholic acid |
LSM-5529 |
GPBAR1 |
3.33uM |
24h |
LINCSCP_75973 |
LINCSCP_75973 |
A375 |
| -0.208041 |
5.393933e-11 |
975 |
MLS002473641 |
LSM-3855 |
|
10uM |
24h |
LINCSCP_31408 |
LINCSCP_31408 |
MCF7 |
| 0.20803 |
5.406385e-11 |
975 |
YM-298198 |
LSM-3328 |
GRM1 |
10uM |
24h |
LINCSCP_55667 |
LINCSCP_55667 |
VCAP |
| 0.20799 |
5.453033e-11 |
975 |
BRD-K20093888 |
LSM-7114 |
|
5uM |
24h |
LINCSCP_60145 |
LINCSCP_60145 |
VCAP |
| -0.207989 |
5.454191e-11 |
975 |
L 741,742 |
LSM-2276 |
DRD4 |
10uM |
6h |
LINCSCP_477 |
LINCSCP_477 |
A375 |
| -0.207971 |
5.476286e-11 |
975 |
Broad-Sai-560 |
LSM-45991 |
|
0.5uM |
24h |
LINCSCP_35537 |
LINCSCP_35537 |
MCF7 |
| 0.207968 |
5.479923e-11 |
975 |
Inolitazone (dihydrochloride) |
LSM-45726 |
PPARG |
1.11uM |
24h |
LINCSCP_168435 |
LINCSCP_168435 |
YAPC |
| 0.207963 |
5.485861e-11 |
975 |
BMS-345541 |
LSM-1028 |
IKBKB |
0.12uM |
24h |
LINCSCP_131198 |
LINCSCP_131198 |
MCF10A |
| -0.207962 |
5.486674e-11 |
975 |
CHEMBL607856 |
LSM-3321 |
|
10uM |
6h |
LINCSCP_50975 |
LINCSCP_50975 |
RMGI |
| -0.20796 |
5.489322e-11 |
975 |
IDOXURIDINE |
LSM-45784 |
|
1.11uM |
24h |
LINCSCP_78426 |
LINCSCP_78426 |
A375 |
| -0.207956 |
5.494017e-11 |
975 |
179324-69-7 |
LSM-6281 |
ADRM1|PSMA1|PSMA2|PSMA3|PSMA4|PSMA5|PSMA6|PSMA7|PSMA8|PSMB1|PSMB10|PSMB11|PSMB2|PSMB3|PSMB4|PSMB5|PSMB6|PSMB7|PSMB8|PSMB9|PSMC1|PSMC2|PSMC3|PSMC4|PSMC5|PSMC6|PSMD1|PSMD11|PSMD12|PSMD13|PSMD14|PSMD2|PSMD3|PSMD4|PSMD6|PSMD7|PSMD8|SEM1 |
20uM |
24h |
LINCSCP_134556 |
LINCSCP_134556 |
MCF7 |
| 0.207941 |
5.511043e-11 |
975 |
Tranilast |
LSM-42898 |
|
0.04uM |
24h |
LINCSCP_71634 |
LINCSCP_71634 |
A375 |
| 0.207923 |
5.532506e-11 |
975 |
Latanoprost |
LSM-43170 |
PTGFR |
0.12uM |
24h |
LINCSCP_102859 |
LINCSCP_102859 |
HELA |
| -0.207923 |
5.533319e-11 |
975 |
Avrainvillamide Analog 5 |
LSM-45314 |
|
0.37uM |
24h |
LINCSCP_38447 |
LINCSCP_38447 |
MCF7 |
| -0.207918 |
5.538303e-11 |
975 |
IDOXURIDINE |
LSM-45784 |
|
3.33uM |
24h |
LINCSCP_78425 |
LINCSCP_78425 |
A375 |
| -0.207893 |
5.568797e-11 |
975 |
SN-38 |
LSM-45563 |
|
3.33uM |
24h |
LINCSCP_137341 |
LINCSCP_137341 |
MCF7 |
| 0.207892 |
5.570084e-11 |
975 |
BRD-K66142238 |
LSM-12461 |
|
5uM |
24h |
LINCSCP_63396 |
LINCSCP_63396 |
VCAP |
| 0.207889 |
5.573152e-11 |
975 |
Alpelisib |
LSM-4256 |
PIK3CA |
0.12uM |
3h |
LINCSCP_115378 |
LINCSCP_115378 |
HS578T |
| 0.207886 |
5.577226e-11 |
975 |
Lofexidine |
LSM-4951 |
ADRA2A |
3.33uM |
24h |
LINCSCP_75192 |
LINCSCP_75192 |
A375 |
| -0.207881 |
5.582980e-11 |
975 |
CHEMBL1394132 |
LSM-3090 |
|
10uM |
6h |
LINCSCP_57429 |
LINCSCP_57429 |
VCAP |
| -0.207872 |
5.593885e-11 |
975 |
AS-605240 |
LSM-42784 |
PIK3CG |
3.33uM |
24h |
LINCSCP_88218 |
LINCSCP_88218 |
HA1E |
| 0.20787 |
5.597206e-11 |
975 |
WHI-P97 |
LSM-1033 |
JAK3 |
10uM |
24h |
LINCSCP_11785 |
LINCSCP_11785 |
BT20 |
| 0.207848 |
5.623667e-11 |
975 |
Cholic acid |
LSM-5541 |
CES1|FECH|PLA2G1B |
3.33uM |
24h |
LINCSCP_75555 |
LINCSCP_75555 |
A375 |
| 0.207834 |
5.640543e-11 |
975 |
Alectinib |
LSM-1202 |
ALK|RET |
3.33uM |
24h |
LINCSCP_82621 |
LINCSCP_82621 |
A549 |
| 0.207826 |
5.650136e-11 |
975 |
Gefitinib |
LSM-1098 |
EGFR |
0.37uM |
24h |
LINCSCP_69611 |
LINCSCP_69611 |
A375 |
| -0.207819 |
5.658533e-11 |
975 |
VX-661 |
LSM-45570 |
CFTR |
10uM |
24h |
LINCSCP_80460 |
LINCSCP_80460 |
A375 |
| -0.207813 |
5.665858e-11 |
975 |
SCHEMBL16226502 |
LSM-43056 |
HSP90AA1 |
0.1uM |
6h |
LINCSCP_9303 |
LINCSCP_9303 |
A549 |
| 0.207798 |
5.684442e-11 |
975 |
T5715534 |
LSM-2466 |
|
10uM |
6h |
LINCSCP_20088 |
LINCSCP_20088 |
HCC515 |
| -0.207767 |
5.722233e-11 |
975 |
BD-1047 |
LSM-2810 |
SIGMAR1 |
10uM |
24h |
LINCSCP_11557 |
LINCSCP_11557 |
ASC |
| 0.207765 |
5.725037e-11 |
975 |
C24H25CLFN5O3 |
LSM-42794 |
EGFR|ERBB2|ERBB4 |
0.04uM |
24h |
LINCSCP_151248 |
LINCSCP_151248 |
PC3 |
| -0.20776 |
5.731341e-11 |
975 |
SB271046 |
LSM-45888 |
|
0.37uM |
24h |
LINCSCP_78271 |
LINCSCP_78271 |
A375 |
| -0.207747 |
5.747278e-11 |
975 |
BRD-K90446118 |
LSM-42207 |
|
10uM |
6h |
LINCSCP_16387 |
LINCSCP_16387 |
HA1E |
| -0.207739 |
5.756642e-11 |
975 |
Withaferin A |
LSM-6685 |
IKBKB|NAMPT |
10uM |
24h |
LINCSCP_150883 |
LINCSCP_150883 |
PC3 |
| 0.207736 |
5.761325e-11 |
975 |
STK219801 |
LSM-43281 |
|
20uM |
6h |
LINCSCP_29377 |
LINCSCP_29377 |
LOVO |
| -0.207733 |
5.764882e-11 |
975 |
BRD-K72269288 |
LSM-14911 |
|
5uM |
24h |
LINCSCP_64212 |
LINCSCP_64212 |
VCAP |
| -0.207711 |
5.792159e-11 |
975 |
AZD-5438 |
LSM-1159 |
CDK1|CDK10|CDK11B|CDK12|CDK13|CDK14|CDK15|CDK16|CDK17|CDK18|CDK19|CDK2|CDK20|CDK3|CDK4|CDK5|CDK6|CDK7|CDK8|CDK9 |
3.33uM |
24h |
LINCSCP_69513 |
LINCSCP_69513 |
A375 |
| -0.20771 |
5.793331e-11 |
975 |
MLS003079540 |
LSM-3507 |
|
10uM |
24h |
LINCSCP_177886 |
LINCSCP_177886 |
A375 |
| -0.207703 |
5.802143e-11 |
975 |
Alisertib |
LSM-37184 |
AURKA |
10uM |
24h |
LINCSCP_109509 |
LINCSCP_109509 |
HELA |
| -0.207701 |
5.804045e-11 |
975 |
Palbociclib |
LSM-1071 |
CCND1|CDK4|CDK6 |
0.12uM |
24h |
LINCSCP_76371 |
LINCSCP_76371 |
A375 |
| -0.207686 |
5.823665e-11 |
975 |
Meisoindigo |
LSM-45840 |
|
10uM |
24h |
LINCSCP_156157 |
LINCSCP_156157 |
PC3 |
| -0.207684 |
5.825623e-11 |
975 |
Ibrutinib (PCI-32765) |
LSM-45830 |
BTK |
0.04uM |
24h |
LINCSCP_125979 |
LINCSCP_125979 |
HT29 |
| -0.207676 |
5.836577e-11 |
975 |
Tivozanib |
LSM-1005 |
FLT1|FLT4|KDR|KIT|PDGFRA|PDGFRB |
10uM |
24h |
LINCSCP_149577 |
LINCSCP_149577 |
NPC.TAK |
| 0.207671 |
5.842765e-11 |
975 |
Methylprednisolone |
LSM-5485 |
NR3C1 |
10uM |
6h |
LINCSCP_22033 |
LINCSCP_22033 |
HEPG2 |
| -0.207668 |
5.846024e-11 |
975 |
2-(4-Chlorophenyl)-6-(methylthio)-4-oxo-3,4-dihydro-2H-1,3-thiazine-5-carbonitrile |
LSM-4328 |
|
10uM |
24h |
LINCSCP_42219 |
LINCSCP_42219 |
NPC |
| -0.207658 |
5.859145e-11 |
975 |
BRD-K37184875 |
LSM-39311 |
|
5uM |
24h |
LINCSCP_28077 |
LINCSCP_28077 |
HT29 |
| -0.20764 |
5.882082e-11 |
975 |
23979-41-1 |
LSM-5472 |
PTGS1|PTGS2 |
10uM |
24h |
LINCSCP_47633 |
LINCSCP_47633 |
PC3 |
| 0.207624 |
5.901245e-11 |
975 |
Gefitinib |
LSM-1098 |
EGFR |
0.37uM |
3h |
LINCSCP_164129 |
LINCSCP_164129 |
SKBR3 |
| 0.207593 |
5.941818e-11 |
975 |
WYE 125132 |
LSM-1064 |
MTOR |
3.33uM |
3h |
LINCSCP_145880 |
LINCSCP_145880 |
MDAMB231 |
| 0.207585 |
5.951503e-11 |
975 |
BRD-K89895693 |
LSM-13971 |
|
5uM |
6h |
LINCSCP_63194 |
LINCSCP_63194 |
VCAP |
| 0.207585 |
5.952167e-11 |
975 |
BRD-K47977047-001-01-2 |
LSM-6836 |
|
5uM |
6h |
LINCSCP_63165 |
LINCSCP_63165 |
VCAP |
| -0.207574 |
5.966468e-11 |
975 |
PF-03814735 |
LSM-45437 |
|
3.33uM |
24h |
LINCSCP_96924 |
LINCSCP_96924 |
HA1E |
| -0.207565 |
5.977123e-11 |
975 |
13-Hydroxy-8,14,19-trimethoxy-4,10,12,16-tetramethyl-3,20,22-trioxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18-pentaen-9-yl carbamate |
LSM-42815 |
HSP90AA1 |
10uM |
6h |
LINCSCP_68290 |
LINCSCP_68290 |
VCAP |
| -0.207558 |
5.985889e-11 |
975 |
Cucurbitacin-I |
LSM-43115 |
JAK2|STAT3 |
0.5uM |
24h |
LINCSCP_35628 |
LINCSCP_35628 |
MCF7 |
| -0.207548 |
5.999284e-11 |
975 |
Hycanthone |
LSM-5614 |
|
10uM |
24h |
LINCSCP_34293 |
LINCSCP_34293 |
MCF7 |
| -0.207535 |
6.015906e-11 |
975 |
856437-59-7 |
LSM-4751 |
|
10uM |
24h |
LINCSCP_42471 |
LINCSCP_42471 |
NPC |
| -0.207534 |
6.016890e-11 |
975 |
LY-294002 |
LSM-2597 |
MTOR|PIK3CA|PIK3CB|PIK3CD|PIK3CG|PLK1|PRKDC |
1uM |
24h |
LINCSCP_200926 |
LINCSCP_200926 |
A549 |
| -0.207528 |
6.025520e-11 |
975 |
Benactyzine |
LSM-5908 |
|
10uM |
6h |
LINCSCP_46175 |
LINCSCP_46175 |
PC3 |
| -0.207526 |
6.027806e-11 |
975 |
OTSSP167 |
LSM-6340 |
|
0.12uM |
24h |
LINCSCP_146309 |
LINCSCP_146309 |
MNEU.E |
| -0.207511 |
6.046885e-11 |
975 |
Brazilin |
LSM-1844 |
|
10uM |
24h |
LINCSCP_32857 |
LINCSCP_32857 |
MCF7 |
| 0.207505 |
6.055213e-11 |
975 |
Marimastat |
LSM-45636 |
|
0.04uM |
24h |
LINCSCP_72201 |
LINCSCP_72201 |
A375 |
| -0.207504 |
6.055984e-11 |
975 |
altrenogest |
LSM-45498 |
|
1.11uM |
24h |
LINCSCP_123273 |
LINCSCP_123273 |
HT29 |
| -0.207497 |
6.065395e-11 |
975 |
BRD-K74316684 |
LSM-41315 |
|
10uM |
24h |
LINCSCP_43163 |
LINCSCP_43163 |
NPC |
| -0.207492 |
6.071988e-11 |
975 |
MG-132 |
LSM-1107 |
PSMB1 |
20uM |
24h |
LINCSCP_134722 |
LINCSCP_134722 |
MCF7 |
| -0.207471 |
6.100414e-11 |
975 |
Mepivacaine |
LSM-4306 |
SCN10A|SCN11A|SCN1A|SCN2A|SCN3A|SCN4A|SCN5A|SCN7A|SCN8A|SCN9A |
1.11uM |
24h |
LINCSCP_156998 |
LINCSCP_156998 |
PC3 |
| 0.20747 |
6.100929e-11 |
975 |
MLS003672589 |
LSM-36804 |
|
10uM |
6h |
LINCSCP_282819 |
LINCSCP_282819 |
PL21 |
| -0.207465 |
6.107689e-11 |
975 |
Batimastat |
LSM-6276 |
|
0.04uM |
24h |
LINCSCP_71024 |
LINCSCP_71024 |
A375 |
| -0.207464 |
6.108533e-11 |
975 |
Lestaurtinib |
LSM-1231 |
FLT3|JAK2|NTRK1|NTRK2|NTRK3|RET |
1uM |
6h |
LINCSCP_37542 |
LINCSCP_37542 |
MCF7 |
| -0.207447 |
6.130814e-11 |
975 |
Erlotinib |
LSM-1097 |
EGFR |
3.33uM |
24h |
LINCSCP_96966 |
LINCSCP_96966 |
HA1E |
| -0.207431 |
6.152459e-11 |
975 |
GSK-J1 |
LSM-44939 |
|
0.12uM |
24h |
LINCSCP_86956 |
LINCSCP_86956 |
CD34 |
| 0.207412 |
6.177853e-11 |
975 |
Tranilast |
LSM-42898 |
|
1.11uM |
24h |
LINCSCP_71631 |
LINCSCP_71631 |
A375 |
| 0.207407 |
6.183896e-11 |
975 |
6Alpha-fluorotestosterone |
LSM-5881 |
|
10uM |
6h |
LINCSCP_211830 |
LINCSCP_211830 |
HA1E |
| 0.207407 |
6.184873e-11 |
975 |
DG-041 |
LSM-43279 |
PTGER3 |
40uM |
6h |
LINCSCP_51135 |
LINCSCP_51135 |
RMUGS |
| 0.207384 |
6.215482e-11 |
975 |
Brefeldin A |
LSM-42812 |
|
0.1uM |
24h |
LINCSCP_19217 |
LINCSCP_19217 |
HCC515 |
| 0.207381 |
6.219615e-11 |
975 |
LY-344864 |
LSM-4161 |
HTR1F |
10uM |
6h |
LINCSCP_4421 |
LINCSCP_4421 |
A549 |
| -0.207341 |
6.273252e-11 |
975 |
Wortmannin |
LSM-3947 |
PIK3CA|PIK3CG|PLK1 |
10uM |
24h |
LINCSCP_67285 |
LINCSCP_67285 |
MCF7 |
| -0.207329 |
6.288912e-11 |
975 |
BRD-A97035593 |
LSM-1947 |
XIAP |
10uM |
24h |
LINCSCP_30918 |
LINCSCP_30918 |
MCF7 |
| 0.207329 |
6.289736e-11 |
975 |
Tedizolid |
LSM-45778 |
|
0.37uM |
24h |
LINCSCP_123215 |
LINCSCP_123215 |
HT29 |
| -0.207326 |
6.293803e-11 |
975 |
Fedratinib |
LSM-1142 |
FLT3|JAK2 |
0.5uM |
24h |
LINCSCP_39369 |
LINCSCP_39369 |
MDAMB231 |
| -0.207319 |
6.302878e-11 |
975 |
GSK 1059615 |
LSM-42799 |
PIK3CA|PIK3CB|PIK3CD|PIK3CG |
3.33uM |
24h |
LINCSCP_149314 |
LINCSCP_149314 |
NPC |
| -0.207318 |
6.304759e-11 |
975 |
CHEMBL3185081 |
LSM-38200 |
|
5uM |
24h |
LINCSCP_8780 |
LINCSCP_8780 |
A549 |
| -0.20731 |
6.314805e-11 |
975 |
Celecoxib |
LSM-2032 |
PTGS2 |
10uM |
6h |
LINCSCP_32989 |
LINCSCP_32989 |
MCF7 |
| 0.207308 |
6.317281e-11 |
975 |
Indigo Red |
LSM-42899 |
CDK1|CDK5|GSK3A |
0.37uM |
24h |
LINCSCP_71638 |
LINCSCP_71638 |
A375 |
| 0.207289 |
6.344045e-11 |
975 |
SCHEMBL3958507 |
LSM-5245 |
COQ8B|EGFR |
0.1uM |
24h |
LINCSCP_51303 |
LINCSCP_51303 |
SKBR3 |
| -0.207275 |
6.362865e-11 |
975 |
BRD-K85592362 |
LSM-41939 |
|
10uM |
24h |
LINCSCP_47342 |
LINCSCP_47342 |
PC3 |
| -0.207272 |
6.366709e-11 |
975 |
Piplartine |
LSM-42914 |
|
10uM |
24h |
LINCSCP_25502 |
LINCSCP_25502 |
HT29 |
| -0.207239 |
6.411983e-11 |
975 |
SA-441487 |
LSM-37962 |
|
10uM |
6h |
LINCSCP_38280 |
LINCSCP_38280 |
MCF7 |
| -0.207232 |
6.421654e-11 |
975 |
Radicicol |
LSM-43303 |
|
1uM |
48h |
LINCSCP_64515 |
LINCSCP_64515 |
VCAP |
| -0.20722 |
6.438216e-11 |
975 |
BRD-K65148580 |
LSM-40829 |
|
10uM |
24h |
LINCSCP_3605 |
LINCSCP_3605 |
A375 |
| -0.207218 |
6.441920e-11 |
975 |
179324-69-7 |
LSM-6281 |
ADRM1|PSMA1|PSMA2|PSMA3|PSMA4|PSMA5|PSMA6|PSMA7|PSMA8|PSMB1|PSMB10|PSMB11|PSMB2|PSMB3|PSMB4|PSMB5|PSMB6|PSMB7|PSMB8|PSMB9|PSMC1|PSMC2|PSMC3|PSMC4|PSMC5|PSMC6|PSMD1|PSMD11|PSMD12|PSMD13|PSMD14|PSMD2|PSMD3|PSMD4|PSMD6|PSMD7|PSMD8|SEM1 |
20uM |
24h |
LINCSCP_71148 |
LINCSCP_71148 |
A375 |
| -0.207215 |
6.445248e-11 |
975 |
Tiapride |
LSM-5676 |
DRD2|DRD3 |
3.33uM |
24h |
LINCSCP_139663 |
LINCSCP_139663 |
MCF7 |
| -0.207199 |
6.467413e-11 |
975 |
Aminosalicylic acid |
LSM-5862 |
PTGS1|PTGS2 |
1.11uM |
24h |
LINCSCP_108331 |
LINCSCP_108331 |
HELA |
| -0.207193 |
6.475726e-11 |
975 |
92394-00-8 |
LSM-2622 |
|
10uM |
6h |
LINCSCP_19713 |
LINCSCP_19713 |
HCC515 |
| -0.207162 |
6.518978e-11 |
975 |
PCI-34051 |
LSM-4812 |
HDAC1|HDAC10|HDAC6|HDAC8 |
10uM |
24h |
LINCSCP_43515 |
LINCSCP_43515 |
NPC |
| 0.207162 |
6.519837e-11 |
975 |
GW843682X |
LSM-1014 |
PLK1|PLK3 |
10uM |
6h |
LINCSCP_41913 |
LINCSCP_41913 |
NOMO1 |
| -0.207156 |
6.528569e-11 |
975 |
Sepantronium |
LSM-5399 |
BIRC5 |
0.5uM |
24h |
LINCSCP_45017 |
LINCSCP_45017 |
PC3 |
| -0.207118 |
6.581144e-11 |
975 |
BRD-K74042299 |
LSM-44849 |
|
10uM |
6h |
LINCSCP_311902 |
LINCSCP_311902 |
VCAP |
| -0.207107 |
6.597711e-11 |
975 |
PDK1 Inhibitor |
LSM-1081 |
PDPK1 |
10uM |
24h |
LINCSCP_11649 |
LINCSCP_11649 |
BT20 |
| -0.207106 |
6.599347e-11 |
975 |
CP466722 |
LSM-1009 |
ATM |
3.33uM |
24h |
LINCSCP_111368 |
LINCSCP_111368 |
HEPG2 |
| -0.207101 |
6.605429e-11 |
975 |
AMBCB17415880 |
LSM-6488 |
|
10uM |
24h |
LINCSCP_193534 |
LINCSCP_193534 |
A549 |
| 0.207101 |
6.606356e-11 |
975 |
BRD-K41571462 |
LSM-10953 |
|
5uM |
24h |
LINCSCP_61993 |
LINCSCP_61993 |
VCAP |
| -0.207092 |
6.618035e-11 |
975 |
BX-795 |
LSM-1189 |
PDK1|PDPK1 |
10uM |
24h |
LINCSCP_84918 |
LINCSCP_84918 |
ASC |
| 0.207087 |
6.626321e-11 |
975 |
Actarit |
LSM-5475 |
|
3.33uM |
24h |
LINCSCP_121074 |
LINCSCP_121074 |
HT29 |
| 0.207083 |
6.631322e-11 |
975 |
BRD-K30802967 |
LSM-6102 |
|
10uM |
6h |
LINCSCP_59335 |
LINCSCP_59335 |
VCAP |
| -0.207056 |
6.669599e-11 |
975 |
Flubendazole |
LSM-5916 |
TUBB |
10uM |
24h |
LINCSCP_269803 |
LINCSCP_269803 |
PC3 |
| -0.207025 |
6.715022e-11 |
975 |
BRD-K44802037 |
LSM-39748 |
|
5uM |
24h |
LINCSCP_3477 |
LINCSCP_3477 |
A375 |
| -0.207014 |
6.731163e-11 |
975 |
BMS-536924 |
LSM-1210 |
IGF1R |
10uM |
24h |
LINCSCP_9474 |
LINCSCP_9474 |
A549 |
| 0.207008 |
6.739145e-11 |
975 |
PD-173074 |
LSM-1026 |
FGFR1|FGFR3 |
0.37uM |
3h |
LINCSCP_131667 |
LINCSCP_131667 |
MCF10A |
| 0.206991 |
6.764435e-11 |
975 |
AZD-6482 |
LSM-1059 |
PIK3CA|PIK3CB|PIK3CD|PIK3CG|PIK3R1|PIK3R2|PIK3R3|PIK3R5 |
0.04uM |
24h |
LINCSCP_130606 |
LINCSCP_130606 |
MCF10A |
| -0.206984 |
6.774073e-11 |
975 |
GW-5074 |
LSM-42779 |
RAF1 |
10uM |
24h |
LINCSCP_11153 |
LINCSCP_11153 |
ASC |
| -0.206981 |
6.778923e-11 |
975 |
SA-1920756 |
LSM-38561 |
|
1uM |
6h |
LINCSCP_37783 |
LINCSCP_37783 |
MCF7 |
| -0.206975 |
6.787306e-11 |
975 |
Proglumide |
LSM-4439 |
CCKAR|CCKBR |
3.33uM |
24h |
LINCSCP_172790 |
LINCSCP_172790 |
YAPC |
| -0.206972 |
6.791592e-11 |
975 |
TCB2 |
LSM-45588 |
|
10uM |
24h |
LINCSCP_160022 |
LINCSCP_160022 |
PC3 |
| 0.206942 |
6.835678e-11 |
975 |
SCHEMBL2559243 |
LSM-3225 |
|
10uM |
6h |
LINCSCP_5530 |
LINCSCP_5530 |
A549 |
| -0.206934 |
6.846697e-11 |
975 |
13-Hydroxy-8,14,19-trimethoxy-4,10,12,16-tetramethyl-3,20,22-trioxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18-pentaen-9-yl carbamate |
LSM-42815 |
HSP90AA1 |
10uM |
6h |
LINCSCP_68512 |
LINCSCP_68512 |
VCAP |
| -0.206932 |
6.850425e-11 |
975 |
Parthenolide |
LSM-43090 |
|
10uM |
24h |
LINCSCP_34463 |
LINCSCP_34463 |
MCF7 |
| -0.206913 |
6.878773e-11 |
975 |
Griseofulvin |
LSM-5259 |
|
0.37uM |
24h |
LINCSCP_74252 |
LINCSCP_74252 |
A375 |
| -0.206897 |
6.901738e-11 |
975 |
GSK429286A |
LSM-1012 |
ROCK1 |
10uM |
24h |
LINCSCP_51265 |
LINCSCP_51265 |
SKBR3 |
| -0.206891 |
6.911398e-11 |
975 |
BRD-K11359987 |
LSM-9119 |
|
5uM |
24h |
LINCSCP_27792 |
LINCSCP_27792 |
HT29 |
| -0.206865 |
6.949710e-11 |
975 |
amisulpride |
LSM-45926 |
|
0.04uM |
24h |
LINCSCP_74248 |
LINCSCP_74248 |
A375 |
| -0.206837 |
6.990986e-11 |
975 |
BRD-K07922534 |
LSM-15106 |
|
10uM |
6h |
LINCSCP_278960 |
LINCSCP_278960 |
PC3 |
| -0.206833 |
6.997104e-11 |
975 |
MLS003129123 |
LSM-7618 |
|
5uM |
24h |
LINCSCP_60584 |
LINCSCP_60584 |
VCAP |
| -0.206828 |
7.005763e-11 |
975 |
MLS002264397 |
LSM-1315 |
|
10uM |
6h |
LINCSCP_1457 |
LINCSCP_1457 |
A375 |
| 0.206819 |
7.018622e-11 |
975 |
Lofexidine |
LSM-4951 |
ADRA2A |
1.11uM |
24h |
LINCSCP_75193 |
LINCSCP_75193 |
A375 |
| 0.206814 |
7.026222e-11 |
975 |
EX-8678 |
LSM-1147 |
|
0.5uM |
6h |
LINCSCP_39565 |
LINCSCP_39565 |
MDAMB231 |
| -0.206791 |
7.061175e-11 |
975 |
SB225002 |
LSM-3367 |
CXCR2 |
1uM |
24h |
LINCSCP_37927 |
LINCSCP_37927 |
MCF7 |
| -0.206789 |
7.063393e-11 |
975 |
Lenvatinib (E7080) |
LSM-45581 |
FLT1|FLT4|KDR |
10uM |
24h |
LINCSCP_105567 |
LINCSCP_105567 |
HELA |
| -0.206771 |
7.090740e-11 |
975 |
CHEMBL2359949 |
LSM-39623 |
|
10uM |
6h |
LINCSCP_26495 |
LINCSCP_26495 |
HT29 |
| 0.206757 |
7.112987e-11 |
975 |
TUL_XIX002 |
LSM-36793 |
|
0.1uM |
24h |
LINCSCP_55067 |
LINCSCP_55067 |
THP1 |
| -0.206753 |
7.118600e-11 |
975 |
Tofacitinib (CP-690550) Citrate |
LSM-45505 |
|
10uM |
24h |
LINCSCP_153762 |
LINCSCP_153762 |
PC3 |
| -0.206751 |
7.122629e-11 |
975 |
SA-247582 |
LSM-40758 |
|
1uM |
24h |
LINCSCP_37247 |
LINCSCP_37247 |
MCF7 |
| 0.20675 |
7.124117e-11 |
975 |
TWS 119 |
LSM-1111 |
GSK3B |
0.12uM |
3h |
LINCSCP_132460 |
LINCSCP_132460 |
MCF7 |
| -0.206745 |
7.130706e-11 |
975 |
CHEMBL3182405 |
LSM-4793 |
|
10uM |
24h |
LINCSCP_10090 |
LINCSCP_10090 |
A549 |
| -0.206711 |
7.183102e-11 |
975 |
ST-4062971 |
LSM-36806 |
|
10uM |
24h |
LINCSCP_32490 |
LINCSCP_32490 |
MCF7 |
| -0.206703 |
7.196299e-11 |
975 |
MG-132 |
LSM-1107 |
PSMB1 |
20uM |
24h |
LINCSCP_72396 |
LINCSCP_72396 |
A375 |
| 0.206671 |
7.245671e-11 |
975 |
2-Methoxy-3-methyl-9H-carbazole |
LSM-36673 |
|
10uM |
24h |
LINCSCP_50307 |
LINCSCP_50307 |
PHH |
| -0.206666 |
7.253418e-11 |
975 |
Canertinib |
LSM-1120 |
EGFR|ERBB2|ERBB4 |
10uM |
3h |
LINCSCP_113469 |
LINCSCP_113469 |
HME1 |
| -0.206659 |
7.263948e-11 |
975 |
PD-0325901 |
LSM-1101 |
MAP2K1|MAP2K2 |
3.33uM |
24h |
LINCSCP_165199 |
LINCSCP_165199 |
SKL.C |
| 0.206656 |
7.269449e-11 |
975 |
BRD-K90970920 |
LSM-6165 |
|
10uM |
6h |
LINCSCP_59410 |
LINCSCP_59410 |
VCAP |
| 0.206652 |
7.274548e-11 |
975 |
BRD-K89895693 |
LSM-13971 |
|
5uM |
24h |
LINCSCP_63121 |
LINCSCP_63121 |
VCAP |
| 0.206649 |
7.279047e-11 |
975 |
Meclofenoxate |
LSM-5273 |
|
10uM |
24h |
LINCSCP_34466 |
LINCSCP_34466 |
MCF7 |
| 0.206641 |
7.292225e-11 |
975 |
Sulfadoxine |
LSM-5657 |
|
10uM |
24h |
LINCSCP_73403 |
LINCSCP_73403 |
A375 |
| -0.206639 |
7.295729e-11 |
975 |
Panobinostat |
LSM-43059 |
HDAC1|HDAC10|HDAC11|HDAC2|HDAC3|HDAC4|HDAC5|HDAC6|HDAC7|HDAC8|HDAC9 |
0.01uM |
24h |
LINCSCP_279676 |
LINCSCP_279676 |
PC3 |
| 0.206608 |
7.344312e-11 |
975 |
BRD-A69951442-001-01-3 |
LSM-4466 |
NR3C1 |
10uM |
6h |
LINCSCP_45091 |
LINCSCP_45091 |
PC3 |
| 0.206574 |
7.398478e-11 |
975 |
Hydrastinine |
LSM-4079 |
|
10uM |
24h |
LINCSCP_11348 |
LINCSCP_11348 |
ASC |
| 0.206546 |
7.442823e-11 |
975 |
CAY-10415 |
LSM-5100 |
INS |
10uM |
6h |
LINCSCP_239566 |
LINCSCP_239566 |
MCF7 |
| 0.206545 |
7.444172e-11 |
975 |
C19H19FN4O3 |
LSM-1178 |
FGFR1|FLT1|KDR |
3.33uM |
24h |
LINCSCP_81353 |
LINCSCP_81353 |
A549 |
| 0.206531 |
7.466935e-11 |
975 |
BRD-K49512493 |
LSM-11438 |
|
5uM |
24h |
LINCSCP_63702 |
LINCSCP_63702 |
VCAP |
| -0.206515 |
7.491237e-11 |
975 |
BRD-K91016007 |
LSM-42231 |
|
5uM |
24h |
LINCSCP_64335 |
LINCSCP_64335 |
VCAP |
| -0.206484 |
7.541652e-11 |
975 |
BRD-K46746428 |
LSM-39868 |
|
5uM |
24h |
LINCSCP_185735 |
LINCSCP_185735 |
A375 |
| -0.206472 |
7.562010e-11 |
975 |
MG-132 |
LSM-1107 |
PSMB1 |
20uM |
24h |
LINCSCP_71230 |
LINCSCP_71230 |
A375 |
| -0.206471 |
7.563489e-11 |
975 |
SA-103006 |
LSM-42617 |
|
10uM |
6h |
LINCSCP_32399 |
LINCSCP_32399 |
MCF7 |
| -0.206457 |
7.585435e-11 |
975 |
Denbufylline |
LSM-2837 |
|
10uM |
24h |
LINCSCP_241114 |
LINCSCP_241114 |
MCF7 |
| -0.206451 |
7.596192e-11 |
975 |
RO-3306 |
LSM-42788 |
CDK1 |
10uM |
24h |
LINCSCP_47337 |
LINCSCP_47337 |
PC3 |
| 0.206444 |
7.606945e-11 |
975 |
Imiloxan |
LSM-1308 |
ADRA2A|ADRA2B |
0.37uM |
24h |
LINCSCP_102834 |
LINCSCP_102834 |
HELA |
| -0.20643 |
7.629160e-11 |
975 |
Volasertib (BI 6727) |
LSM-45277 |
PLK1 |
0.12uM |
24h |
LINCSCP_142575 |
LINCSCP_142575 |
MCF7 |
| 0.206412 |
7.659883e-11 |
975 |
BRD-K99950451 |
LSM-14573 |
|
5uM |
24h |
LINCSCP_61309 |
LINCSCP_61309 |
VCAP |
| 0.206404 |
7.673290e-11 |
975 |
Gefitinib |
LSM-1098 |
EGFR |
0.37uM |
24h |
LINCSCP_130017 |
LINCSCP_130017 |
LNCAP |
| 0.206398 |
7.681917e-11 |
975 |
JNK-IN-2 |
LSM-43288 |
IRAK1 |
0.1uM |
6h |
LINCSCP_256251 |
LINCSCP_256251 |
MDAMB231 |
| -0.206384 |
7.706268e-11 |
975 |
Ifosfamide |
LSM-5118 |
CYP2A6|CYP2B6|CYP2C18|CYP2C19|CYP2C8|CYP2C9|CYP3A4|CYP3A5|CYP3A7|PTGS1 |
1.11uM |
24h |
LINCSCP_159154 |
LINCSCP_159154 |
PC3 |
| -0.206381 |
7.710503e-11 |
975 |
SPECTRUM_001418 |
LSM-1664 |
ADRB2 |
10uM |
24h |
LINCSCP_265619 |
LINCSCP_265619 |
PC3 |
| 0.206379 |
7.713419e-11 |
975 |
BRD-K78438907 |
LSM-41549 |
|
10uM |
24h |
LINCSCP_49020 |
LINCSCP_49020 |
PC3 |
| -0.206337 |
7.783871e-11 |
975 |
BRD-K45319854 |
LSM-11186 |
|
5uM |
6h |
LINCSCP_63159 |
LINCSCP_63159 |
VCAP |
| -0.206332 |
7.791581e-11 |
975 |
BRD-K83929831 |
LSM-6160 |
|
10uM |
24h |
LINCSCP_242571 |
LINCSCP_242571 |
MCF7 |
| -0.206332 |
7.792171e-11 |
975 |
Aminosalicylic acid |
LSM-5862 |
PTGS1|PTGS2 |
0.12uM |
24h |
LINCSCP_108333 |
LINCSCP_108333 |
HELA |
| 0.20633 |
7.795765e-11 |
975 |
CHEMBL2360924 |
LSM-10623 |
|
5uM |
24h |
LINCSCP_61592 |
LINCSCP_61592 |
VCAP |
| -0.206327 |
7.800456e-11 |
975 |
GSK-1070916 |
LSM-1062 |
AURKB|AURKC |
10uM |
24h |
LINCSCP_148784 |
LINCSCP_148784 |
NPC |
| -0.206317 |
7.816777e-11 |
975 |
CGS-15943 |
LSM-3076 |
ADORA1|ADORA2A|ADORA2B |
10uM |
24h |
LINCSCP_67628 |
LINCSCP_67628 |
MCF7 |
| -0.206311 |
7.827388e-11 |
975 |
CEP-701 |
LSM-45844 |
|
1.11uM |
24h |
LINCSCP_89448 |
LINCSCP_89448 |
HA1E |
| 0.206303 |
7.840604e-11 |
975 |
Vorinostat |
LSM-3828 |
HDAC1|HDAC2|HDAC3|HDAC6|HDAC8 |
1uM |
24h |
LINCSCP_66694 |
LINCSCP_66694 |
A549 |
| -0.206273 |
7.890480e-11 |
975 |
NMS-1286937 |
LSM-45818 |
|
3.33uM |
24h |
LINCSCP_160071 |
LINCSCP_160071 |
PC3 |
| -0.206268 |
7.899411e-11 |
975 |
HMN-214 |
LSM-42802 |
CSF1R|FLT1|FLT3|FLT4|KDR|KIT|PDGFRB|RET |
3.33uM |
24h |
LINCSCP_148278 |
LINCSCP_148278 |
NPC.CAS9 |
| -0.206262 |
7.910384e-11 |
975 |
BRD-K68319707 |
LSM-40988 |
|
10uM |
24h |
LINCSCP_249832 |
LINCSCP_249832 |
MCF7 |
| 0.206259 |
7.914822e-11 |
975 |
PD-173074 |
LSM-1026 |
FGFR1|FGFR3 |
0.04uM |
3h |
LINCSCP_145818 |
LINCSCP_145818 |
MDAMB231 |
| -0.206249 |
7.932236e-11 |
975 |
CHEMBL2357852 |
LSM-40442 |
|
10uM |
24h |
LINCSCP_37031 |
LINCSCP_37031 |
MCF7 |
| 0.206243 |
7.942677e-11 |
975 |
BRD-K84218095 |
LSM-13577 |
|
5uM |
24h |
LINCSCP_63533 |
LINCSCP_63533 |
VCAP |
| -0.206231 |
7.961739e-11 |
975 |
Rotenone |
LSM-5260 |
MT-ND1 |
0.5uM |
24h |
LINCSCP_25468 |
LINCSCP_25468 |
HT29 |
| -0.20622 |
7.980648e-11 |
975 |
BRD-K23985857 |
LSM-14765 |
|
10uM |
24h |
LINCSCP_42969 |
LINCSCP_42969 |
NPC |
| -0.206219 |
7.983299e-11 |
975 |
BRD-K00819343 |
LSM-37327 |
|
10uM |
6h |
LINCSCP_311793 |
LINCSCP_311793 |
VCAP |
| -0.206202 |
8.012197e-11 |
975 |
MLS003126519 |
LSM-3676 |
|
10uM |
6h |
LINCSCP_224916 |
LINCSCP_224916 |
HT29 |
| 0.206166 |
8.073578e-11 |
975 |
CHEMBL1617726 |
LSM-6255 |
|
80uM |
24h |
LINCSCP_30590 |
LINCSCP_30590 |
MCF7 |
| 0.20616 |
8.085024e-11 |
975 |
Rilmenidine |
LSM-4253 |
ADRA2A|NISCH |
10uM |
6h |
LINCSCP_40033 |
LINCSCP_40033 |
NCIH2073 |
| -0.20615 |
8.102239e-11 |
975 |
BRD-K43786699 |
LSM-11101 |
|
5uM |
24h |
LINCSCP_62286 |
LINCSCP_62286 |
VCAP |
| -0.20614 |
8.119725e-11 |
975 |
SA-84869 |
LSM-41398 |
|
3uM |
6h |
LINCSCP_37181 |
LINCSCP_37181 |
MCF7 |
| -0.206133 |
8.130445e-11 |
975 |
DICUMAROL |
LSM-45761 |
NQO1|VKORC1 |
0.04uM |
24h |
LINCSCP_141484 |
LINCSCP_141484 |
MCF7 |
| -0.206125 |
8.145373e-11 |
975 |
BRD-K09054764 |
LSM-37757 |
|
10uM |
6h |
LINCSCP_65764 |
LINCSCP_65764 |
VCAP |
| 0.206105 |
8.180268e-11 |
975 |
Milrinone |
LSM-3493 |
PDE3A |
10uM |
6h |
LINCSCP_33523 |
LINCSCP_33523 |
MCF7 |
| -0.20609 |
8.206067e-11 |
975 |
WZ 4002 |
LSM-1085 |
EGFR|ERBB2 |
10uM |
24h |
LINCSCP_149787 |
LINCSCP_149787 |
NPC.TAK |
| 0.206085 |
8.214538e-11 |
975 |
BRD-K99380810-001-01-1 |
LSM-6787 |
|
10uM |
6h |
LINCSCP_295952 |
LINCSCP_295952 |
VCAP |
| -0.206067 |
8.246375e-11 |
975 |
BRD-K86671899 |
LSM-13737 |
|
10uM |
24h |
LINCSCP_43064 |
LINCSCP_43064 |
NPC |
| -0.206067 |
8.247385e-11 |
975 |
BRD-K16752617 |
LSM-9440 |
|
5uM |
6h |
LINCSCP_61863 |
LINCSCP_61863 |
VCAP |
| -0.206043 |
8.289612e-11 |
975 |
Apilimod |
LSM-45286 |
|
3.33uM |
24h |
LINCSCP_122453 |
LINCSCP_122453 |
HT29 |
| -0.20604 |
8.294391e-11 |
975 |
AZ20 |
LSM-36357 |
|
10uM |
24h |
LINCSCP_149057 |
LINCSCP_149057 |
NPC |
| 0.206022 |
8.326163e-11 |
975 |
BRD-K51981081 |
LSM-14853 |
|
5uM |
24h |
LINCSCP_309194 |
LINCSCP_309194 |
VCAP |
| -0.206013 |
8.341871e-11 |
975 |
AZD1981 |
LSM-45513 |
PTGDR2 |
0.12uM |
24h |
LINCSCP_173157 |
LINCSCP_173157 |
YAPC |
| -0.205988 |
8.386988e-11 |
975 |
17-DMAG (Alvespimycin) HCl |
LSM-46133 |
|
3.33uM |
24h |
LINCSCP_71736 |
LINCSCP_71736 |
A375 |
| -0.205961 |
8.436528e-11 |
975 |
BRD-A84327315-001-01-1 |
LSM-43157 |
VDR |
10uM |
24h |
LINCSCP_46703 |
LINCSCP_46703 |
PC3 |
| -0.205932 |
8.487939e-11 |
975 |
K784-3187 |
LSM-45465 |
ESR2 |
0.12uM |
24h |
LINCSCP_125144 |
LINCSCP_125144 |
HT29 |
| -0.20593 |
8.492378e-11 |
975 |
Panobinostat |
LSM-43059 |
HDAC1|HDAC10|HDAC11|HDAC2|HDAC3|HDAC4|HDAC5|HDAC6|HDAC7|HDAC8|HDAC9 |
0.01uM |
24h |
LINCSCP_250182 |
LINCSCP_250182 |
MCF7 |
| -0.205909 |
8.531275e-11 |
975 |
PD-0325901 |
LSM-1101 |
MAP2K1|MAP2K2 |
0.12uM |
24h |
LINCSCP_165202 |
LINCSCP_165202 |
SKL.C |
| -0.2059 |
8.547049e-11 |
975 |
Idebenone |
LSM-5505 |
|
10uM |
6h |
LINCSCP_239215 |
LINCSCP_239215 |
MCF7 |
| -0.205895 |
8.556096e-11 |
975 |
galantamine |
|
|
10uM |
24h |
LINCSCP_114488 |
LINCSCP_114488 |
HME1 |
| -0.205883 |
8.578279e-11 |
975 |
Reserpine |
LSM-4162 |
SLC18A1|SLC18A2 |
10uM |
6h |
LINCSCP_33034 |
LINCSCP_33034 |
MCF7 |
| 0.205871 |
8.600566e-11 |
975 |
BRD-K54343811 |
LSM-44966 |
|
0.1uM |
24h |
LINCSCP_250225 |
LINCSCP_250225 |
MCF7 |
| -0.205845 |
8.647178e-11 |
975 |
GSK 525762A |
LSM-6334 |
|
3.33uM |
24h |
LINCSCP_164719 |
LINCSCP_164719 |
SKL.C |
| -0.20584 |
8.658085e-11 |
975 |
MG-132 |
LSM-1107 |
PSMB1 |
20uM |
24h |
LINCSCP_134727 |
LINCSCP_134727 |
MCF7 |
| 0.205823 |
8.688243e-11 |
975 |
XL-147 |
LSM-45674 |
PIK3CA|PIK3CB|PIK3CD|PIK3CG|PIK3R1|PIK3R2|PIK3R3|PIK3R5 |
0.37uM |
24h |
LINCSCP_141662 |
LINCSCP_141662 |
MCF7 |
| 0.205822 |
8.691023e-11 |
975 |
COT Inhibitor-2 |
LSM-1154 |
|
0.04uM |
24h |
LINCSCP_84201 |
LINCSCP_84201 |
ASC |
| -0.20579 |
8.749350e-11 |
975 |
PROTIRELIN |
LSM-45252 |
|
1.11uM |
24h |
LINCSCP_153237 |
LINCSCP_153237 |
PC3 |
| -0.20579 |
8.749577e-11 |
975 |
Sorafenib |
LSM-1008 |
BRAF|DDR2|FGFR1|FLT1|FLT3|FLT4|KDR|KIT|PDGFRB|RAF1|RET |
1.11uM |
24h |
LINCSCP_73129 |
LINCSCP_73129 |
A375 |
| -0.205776 |
8.776021e-11 |
975 |
BRD-K55077180 |
LSM-40286 |
|
5uM |
24h |
LINCSCP_8168 |
LINCSCP_8168 |
A549 |
| -0.205773 |
8.782054e-11 |
975 |
HMS2093P09 |
LSM-44968 |
PGR |
10uM |
6h |
LINCSCP_18997 |
LINCSCP_18997 |
HCC515 |
| -0.205773 |
8.782543e-11 |
975 |
Cyclosporine |
LSM-42883 |
PPIA|PPP3CA |
10uM |
24h |
LINCSCP_44010 |
LINCSCP_44010 |
PC3 |
| 0.205772 |
8.783367e-11 |
975 |
BRD-K21918725 |
LSM-45229 |
|
3uM |
24h |
LINCSCP_55306 |
LINCSCP_55306 |
U937 |
| 0.205768 |
8.791762e-11 |
975 |
CHEMBL2355186 |
LSM-8441 |
|
5uM |
6h |
LINCSCP_62488 |
LINCSCP_62488 |
VCAP |
| -0.20575 |
8.825264e-11 |
975 |
Dacomitinib |
LSM-42808 |
EGFR|ERBB2|ERBB3|ERBB4 |
10uM |
24h |
LINCSCP_139656 |
LINCSCP_139656 |
MCF7 |
| -0.205743 |
8.839021e-11 |
975 |
KUC103423N |
LSM-1819 |
|
10uM |
24h |
LINCSCP_31556 |
LINCSCP_31556 |
MCF7 |
| 0.205714 |
8.892687e-11 |
975 |
Dexamethasone Acetate |
LSM-1915 |
NR3C1 |
10uM |
24h |
LINCSCP_284627 |
LINCSCP_284627 |
SKB |
| -0.205712 |
8.897890e-11 |
975 |
ACON1_002471 |
LSM-36614 |
|
30uM |
24h |
LINCSCP_309965 |
LINCSCP_309965 |
VCAP |
| 0.205698 |
8.924332e-11 |
975 |
SB590885 |
LSM-42746 |
BRAF |
10uM |
6h |
LINCSCP_240402 |
LINCSCP_240402 |
MCF7 |
| 0.20569 |
8.939954e-11 |
975 |
SGI-1776 |
LSM-6307 |
PIM1|PIM2|PIM3 |
1.11uM |
24h |
LINCSCP_128385 |
LINCSCP_128385 |
HUVEC |
| -0.205678 |
8.962485e-11 |
975 |
Allantoin |
LSM-5190 |
|
10uM |
24h |
LINCSCP_34259 |
LINCSCP_34259 |
MCF7 |
| -0.205674 |
8.969282e-11 |
975 |
MLS002264395 |
LSM-3615 |
|
10uM |
6h |
LINCSCP_1612 |
LINCSCP_1612 |
A375 |
| -0.205674 |
8.970622e-11 |
975 |
TAE-684 |
LSM-1024 |
ALK |
10uM |
24h |
LINCSCP_32186 |
LINCSCP_32186 |
MCF7 |
| -0.205673 |
8.971487e-11 |
975 |
noscapine |
|
|
3.33uM |
24h |
LINCSCP_69579 |
LINCSCP_69579 |
A375 |
| -0.205663 |
8.990180e-11 |
975 |
PFI-1 |
LSM-6331 |
|
3.33uM |
24h |
LINCSCP_164671 |
LINCSCP_164671 |
SKL.C |
| -0.205642 |
9.031806e-11 |
975 |
CHEMBL41721 |
LSM-4978 |
CNR1|CNR2|GRIN1 |
10uM |
24h |
LINCSCP_31836 |
LINCSCP_31836 |
MCF7 |
| 0.205583 |
9.145115e-11 |
975 |
TAK-242 |
LSM-45934 |
|
0.04uM |
24h |
LINCSCP_139894 |
LINCSCP_139894 |
MCF7 |
| -0.205577 |
9.156704e-11 |
975 |
BRD-K34952911 |
LSM-45367 |
|
30uM |
24h |
LINCSCP_310011 |
LINCSCP_310011 |
VCAP |
| -0.205574 |
9.164122e-11 |
975 |
SCHEMBL16980224 |
LSM-1092 |
AURKA |
3.33uM |
24h |
LINCSCP_117604 |
LINCSCP_117604 |
HT29 |
| -0.205571 |
9.170109e-11 |
975 |
GSK-2334470 |
LSM-1222 |
PDK1|PDPK1 |
3.33uM |
24h |
LINCSCP_149332 |
LINCSCP_149332 |
NPC |
| 0.205565 |
9.180145e-11 |
975 |
Sasapyrine |
LSM-45517 |
|
1.11uM |
24h |
LINCSCP_141655 |
LINCSCP_141655 |
MCF7 |
| -0.205564 |
9.182210e-11 |
975 |
SMR001317659 |
LSM-2094 |
|
0.5uM |
6h |
LINCSCP_19490 |
LINCSCP_19490 |
HCC515 |
| -0.205545 |
9.221127e-11 |
975 |
Epothilone A |
LSM-43229 |
|
10uM |
24h |
LINCSCP_270819 |
LINCSCP_270819 |
PC3 |
| 0.205537 |
9.235856e-11 |
975 |
BRD-K76352008 |
LSM-41440 |
|
5uM |
6h |
LINCSCP_64443 |
LINCSCP_64443 |
VCAP |
| -0.205534 |
9.241643e-11 |
975 |
Wortmannin |
LSM-3947 |
PIK3CA|PIK3CG|PLK1 |
0.5uM |
24h |
LINCSCP_24122 |
LINCSCP_24122 |
HL60 |
| 0.205531 |
9.247650e-11 |
975 |
MLS002607722 |
LSM-3924 |
|
10uM |
24h |
LINCSCP_189031 |
LINCSCP_189031 |
A549 |
| -0.205524 |
9.261578e-11 |
975 |
PD-0325901 |
LSM-1101 |
MAP2K1|MAP2K2 |
1uM |
6h |
LINCSCP_36934 |
LINCSCP_36934 |
MCF7 |
| -0.205519 |
9.272222e-11 |
975 |
Seliciclib |
LSM-1001 |
CDK1|CDK2|CDK5|CDK7|CDK9 |
10uM |
24h |
LINCSCP_87753 |
LINCSCP_87753 |
HA1E |
| 0.205513 |
9.283541e-11 |
975 |
GSK429286A |
LSM-1012 |
ROCK1 |
10uM |
6h |
LINCSCP_219995 |
LINCSCP_219995 |
HEPG2 |
| -0.205505 |
9.299631e-11 |
975 |
Wortmannin |
LSM-3947 |
PIK3CA|PIK3CG|PLK1 |
10uM |
24h |
LINCSCP_222116 |
LINCSCP_222116 |
HL60 |
| -0.205505 |
9.299842e-11 |
975 |
Triacetylresveratrol |
LSM-44077 |
|
10uM |
24h |
LINCSCP_43498 |
LINCSCP_43498 |
NPC |
| -0.205496 |
9.317728e-11 |
975 |
PD-0325901 |
LSM-1101 |
MAP2K1|MAP2K2 |
1.11uM |
24h |
LINCSCP_165200 |
LINCSCP_165200 |
SKL.C |
| -0.205495 |
9.318940e-11 |
975 |
Albendazole |
LSM-3782 |
|
10uM |
24h |
LINCSCP_37946 |
LINCSCP_37946 |
MCF7 |
| -0.205482 |
9.344395e-11 |
975 |
BRD-K40397365 |
LSM-39496 |
|
10uM |
24h |
LINCSCP_66107 |
LINCSCP_66107 |
VCAP |
| -0.205478 |
9.352940e-11 |
975 |
Tizanidine |
LSM-5242 |
ADRA2A|ADRA2B|ADRA2C |
10uM |
24h |
LINCSCP_59456 |
LINCSCP_59456 |
VCAP |
| -0.205455 |
9.398715e-11 |
975 |
Guanadrel |
LSM-43257 |
SLC6A2 |
0.12uM |
24h |
LINCSCP_169756 |
LINCSCP_169756 |
YAPC |
| -0.205455 |
9.399007e-11 |
975 |
TAK-700 (Orteronel) |
LSM-45634 |
|
3.33uM |
24h |
LINCSCP_170347 |
LINCSCP_170347 |
YAPC |
| 0.205447 |
9.414643e-11 |
975 |
848193-68-0 |
LSM-6271 |
SIRT1 |
0.37uM |
24h |
LINCSCP_83403 |
LINCSCP_83403 |
ASC.C |
| -0.205443 |
9.422502e-11 |
975 |
Broad-Sai-560 |
LSM-45991 |
|
1uM |
24h |
LINCSCP_250253 |
LINCSCP_250253 |
MCF7 |
| -0.205422 |
9.465247e-11 |
975 |
galantamine |
|
|
10uM |
24h |
LINCSCP_148170 |
LINCSCP_148170 |
NPC.CAS9 |
| 0.205372 |
9.568016e-11 |
975 |
LDN 193189 |
LSM-1115 |
ACVR1|BMPR1A |
1uM |
24h |
LINCSCP_251715 |
LINCSCP_251715 |
MCF7 |
| -0.205354 |
9.604235e-11 |
975 |
Palbociclib |
LSM-1071 |
CCND1|CDK4|CDK6 |
0.04uM |
3h |
LINCSCP_86255 |
LINCSCP_86255 |
BT20 |
| -0.205346 |
9.620470e-11 |
975 |
AN-329/41044431 |
LSM-4512 |
|
10uM |
6h |
LINCSCP_46548 |
LINCSCP_46548 |
PC3 |
| -0.205337 |
9.638478e-11 |
975 |
AZD-1152-HQPA |
LSM-1067 |
AURKA|AURKB |
0.12uM |
24h |
LINCSCP_81080 |
LINCSCP_81080 |
A549 |
| 0.205329 |
9.655624e-11 |
975 |
BRD-K21033948 |
LSM-9708 |
|
5uM |
24h |
LINCSCP_61955 |
LINCSCP_61955 |
VCAP |
| -0.205319 |
9.675307e-11 |
975 |
OTSSP167 |
LSM-6340 |
|
0.12uM |
24h |
LINCSCP_140217 |
LINCSCP_140217 |
MCF7 |
| 0.205291 |
9.733901e-11 |
975 |
2-(4,5-Dihydro-1H-imidazol-2-yl)quinoxaline |
LSM-2238 |
|
10uM |
6h |
LINCSCP_26979 |
LINCSCP_26979 |
HT29 |
| 0.20528 |
9.755849e-11 |
975 |
STK009254 |
LSM-1910 |
INS |
10uM |
6h |
LINCSCP_14855 |
LINCSCP_14855 |
HA1E |
| -0.205271 |
9.775500e-11 |
975 |
Purvalanola |
LSM-3118 |
CDK1|CDK2|CDK4|CDK5 |
10uM |
24h |
LINCSCP_25284 |
LINCSCP_25284 |
HT29 |
| -0.205262 |
9.793984e-11 |
975 |
Vinblastine |
LSM-1647 |
TUBB |
10uM |
24h |
LINCSCP_32842 |
LINCSCP_32842 |
MCF7 |
| 0.205257 |
9.805230e-11 |
975 |
AKT Inhibitor VIII |
LSM-1035 |
AKT1|AKT2 |
3.33uM |
24h |
LINCSCP_68992 |
LINCSCP_68992 |
A375 |
| -0.205247 |
9.826047e-11 |
975 |
Dasatinib |
LSM-1020 |
ABL1|BCR|BLK|EPHA2|FGR|FRK|FYN|HCK|KIT|LCK|LYN|PDGFRB|SRC|SRMS|YES1 |
1.11uM |
24h |
LINCSCP_129514 |
LINCSCP_129514 |
JURKAT |
| 0.205244 |
9.832646e-11 |
975 |
THZ-2-98-01 |
LSM-44946 |
|
0.04uM |
24h |
LINCSCP_145543 |
LINCSCP_145543 |
MDAMB231 |
| 0.205174 |
9.979390e-11 |
975 |
GSK-319347A |
LSM-1216 |
IKBKG |
5uM |
6h |
LINCSCP_51151 |
LINCSCP_51151 |
RMUGS |
| -0.205161 |
1.000696e-10 |
975 |
BRD-K39839146 |
LSM-10855 |
|
5uM |
24h |
LINCSCP_27999 |
LINCSCP_27999 |
HT29 |
| -0.20515 |
1.002971e-10 |
975 |
Temsirolimus (CCI-779, NSC 683864) |
LSM-45994 |
MTOR |
1.11uM |
24h |
LINCSCP_120092 |
LINCSCP_120092 |
HT29 |
| -0.205129 |
1.007534e-10 |
975 |
PF-03758309 |
LSM-4254 |
PAK4 |
0.37uM |
24h |
LINCSCP_114443 |
LINCSCP_114443 |
HME1 |
| -0.205062 |
1.022043e-10 |
975 |
BRD-K90827020 |
LSM-8000 |
|
5uM |
24h |
LINCSCP_60094 |
LINCSCP_60094 |
VCAP |
| -0.20505 |
1.024698e-10 |
975 |
BRD-K04534322 |
LSM-36643 |
|
10uM |
24h |
LINCSCP_46211 |
LINCSCP_46211 |
PC3 |
| -0.205045 |
1.025717e-10 |
975 |
PF431396 |
LSM-1116 |
|
0.5uM |
24h |
LINCSCP_39486 |
LINCSCP_39486 |
MDAMB231 |
| 0.205037 |
1.027442e-10 |
975 |
MLS003271344 |
LSM-2697 |
|
10uM |
6h |
LINCSCP_212164 |
LINCSCP_212164 |
HA1E |
| -0.205028 |
1.029470e-10 |
975 |
SCH-23390 |
LSM-3005 |
DRD1|DRD5|HTR2C |
10uM |
24h |
LINCSCP_31377 |
LINCSCP_31377 |
MCF7 |
| 0.205025 |
1.030155e-10 |
975 |
XMD 8-92 |
LSM-1094 |
MAPK7 |
10uM |
24h |
LINCSCP_87216 |
LINCSCP_87216 |
CD34 |
| -0.205022 |
1.030830e-10 |
975 |
Tofacitinib (CP-690550) Citrate |
LSM-45505 |
|
1.11uM |
24h |
LINCSCP_102186 |
LINCSCP_102186 |
HELA |
| 0.205011 |
1.033140e-10 |
975 |
Carbacyclin |
LSM-42923 |
PPARD|PTGIR |
1uM |
24h |
LINCSCP_205462 |
LINCSCP_205462 |
CD34 |
| -0.204978 |
1.040494e-10 |
975 |
BRD-K01425431 |
|
|
1.11uM |
24h |
LINCSCP_151311 |
LINCSCP_151311 |
PC3 |
| -0.204973 |
1.041564e-10 |
975 |
BRD-K01621458 |
LSM-45313 |
|
0.1uM |
6h |
LINCSCP_279796 |
LINCSCP_279796 |
PC3 |
| 0.204918 |
1.053842e-10 |
975 |
Chlordiazepoxide |
LSM-5922 |
GABRA1|GABRA2|GABRA3|GABRA4|GABRA5|GABRA6|GABRB1|GABRB2|GABRB3|GABRD|GABRE|GABRG1|GABRG2|GABRG3|GABRP|GABRQ |
10uM |
6h |
LINCSCP_26314 |
LINCSCP_26314 |
HT29 |
| -0.204907 |
1.056260e-10 |
975 |
Clozapine |
LSM-2823 |
ADRA1A|ADRA1B|CHRM1|CHRM2|CHRM3|CHRM4|DRD1|DRD2|DRD3|DRD4|HRH1|HRH4|HTR1A|HTR1B|HTR1D|HTR1E|HTR2A|HTR2C|HTR6|HTR7 |
10uM |
24h |
LINCSCP_122236 |
LINCSCP_122236 |
HT29 |
| -0.204882 |
1.061881e-10 |
975 |
Mepivacaine |
LSM-4306 |
SCN10A|SCN11A|SCN1A|SCN2A|SCN3A|SCN4A|SCN5A|SCN7A|SCN8A|SCN9A |
1.11uM |
24h |
LINCSCP_75257 |
LINCSCP_75257 |
A375 |
| 0.204858 |
1.067483e-10 |
975 |
Tamatinib |
LSM-1040 |
SYK |
0.04uM |
3h |
LINCSCP_163885 |
LINCSCP_163885 |
SKBR3 |
| 0.204854 |
1.068332e-10 |
975 |
331771-20-1 |
LSM-1096 |
AURKA|AURKB |
0.5uM |
6h |
LINCSCP_39636 |
LINCSCP_39636 |
MDAMB231 |
| -0.204854 |
1.068419e-10 |
975 |
N-Pentanoyl-n-{[2'-(2H-tetrazol-5-yl)biphenyl-4-yl]methyl}valine |
LSM-4977 |
AGTR1 |
10uM |
6h |
LINCSCP_20694 |
LINCSCP_20694 |
HCC515 |
| -0.204845 |
1.070284e-10 |
975 |
MDL 72832 |
LSM-1352 |
HTR1A |
10uM |
24h |
LINCSCP_262499 |
LINCSCP_262499 |
NPC |
| 0.204844 |
1.070524e-10 |
975 |
rifampicin |
|
|
0.12uM |
24h |
LINCSCP_131483 |
LINCSCP_131483 |
MCF10A |
| -0.204843 |
1.070751e-10 |
975 |
AS-605240 |
LSM-42784 |
PIK3CG |
3.33uM |
24h |
LINCSCP_86113 |
LINCSCP_86113 |
BT20 |
| 0.204815 |
1.077097e-10 |
975 |
SCHEMBL13991002 |
LSM-6278 |
|
40uM |
6h |
LINCSCP_30871 |
LINCSCP_30871 |
MCF7 |
| -0.204814 |
1.077514e-10 |
975 |
SA-1925996 |
LSM-42061 |
|
1uM |
24h |
LINCSCP_254358 |
LINCSCP_254358 |
MCF7 |
| -0.204804 |
1.079681e-10 |
975 |
BRD-K53293903 |
LSM-40198 |
|
10uM |
6h |
LINCSCP_65485 |
LINCSCP_65485 |
VCAP |
| -0.204798 |
1.081178e-10 |
975 |
MLS002607743 |
LSM-4089 |
|
10uM |
6h |
LINCSCP_22117 |
LINCSCP_22117 |
HEPG2 |
| -0.204756 |
1.090695e-10 |
975 |
Tigecycline |
LSM-36875 |
|
0.1uM |
6h |
LINCSCP_3768 |
LINCSCP_3768 |
A375 |
| 0.204735 |
1.095802e-10 |
975 |
4LY1 |
LSM-6529 |
HDAC1|HDAC2 |
10uM |
24h |
LINCSCP_7771 |
LINCSCP_7771 |
A549 |
| -0.204733 |
1.096206e-10 |
975 |
Amylocaine |
LSM-1292 |
|
10uM |
6h |
LINCSCP_401 |
LINCSCP_401 |
A375 |
| -0.204728 |
1.097382e-10 |
975 |
Phorbol Myristate Acetate |
LSM-25630 |
|
10uM |
24h |
LINCSCP_28847 |
LINCSCP_28847 |
HUH7 |
| 0.20472 |
1.099183e-10 |
975 |
MLS003129601 |
LSM-7829 |
|
5uM |
24h |
LINCSCP_60616 |
LINCSCP_60616 |
VCAP |
| -0.204711 |
1.101340e-10 |
975 |
SCHEMBL8922766 |
LSM-1595 |
ADORA3 |
10uM |
6h |
LINCSCP_25324 |
LINCSCP_25324 |
HT29 |
| -0.204679 |
1.108733e-10 |
975 |
SCHEMBL618594 |
LSM-1070 |
|
10uM |
24h |
LINCSCP_147725 |
LINCSCP_147725 |
NPC.CAS9 |
| 0.204668 |
1.111489e-10 |
975 |
ST51005413 |
LSM-4948 |
|
30uM |
6h |
LINCSCP_310202 |
LINCSCP_310202 |
VCAP |
| -0.204661 |
1.113150e-10 |
975 |
MLS003429132 |
LSM-42893 |
|
10uM |
24h |
LINCSCP_57525 |
LINCSCP_57525 |
VCAP |
| 0.204615 |
1.123929e-10 |
975 |
Benzohydroxamate |
LSM-36789 |
|
0.1uM |
24h |
LINCSCP_250118 |
LINCSCP_250118 |
MCF7 |
| -0.204552 |
1.139130e-10 |
975 |
BRD-K08777248 |
LSM-37743 |
|
10uM |
24h |
LINCSCP_242425 |
LINCSCP_242425 |
MCF7 |
| -0.204522 |
1.146315e-10 |
975 |
Riluzole |
LSM-2471 |
SCN10A|SCN11A|SCN1A|SCN2A|SCN3A|SCN4A|SCN5A|SCN7A|SCN8A|SCN9A |
10uM |
24h |
LINCSCP_136465 |
LINCSCP_136465 |
MCF7 |
| -0.204515 |
1.148156e-10 |
975 |
Epothilone B (EPO906, Patupilone) |
LSM-46001 |
|
3.33uM |
24h |
LINCSCP_142098 |
LINCSCP_142098 |
MCF7 |
| 0.204509 |
1.149488e-10 |
975 |
Tyrphostin AG 1288 |
LSM-5257 |
TNF |
10uM |
6h |
LINCSCP_46938 |
LINCSCP_46938 |
PC3 |
| -0.204502 |
1.151197e-10 |
975 |
Wortmannin |
LSM-3947 |
PIK3CA|PIK3CG|PLK1 |
3uM |
24h |
LINCSCP_9398 |
LINCSCP_9398 |
A549 |
| -0.204473 |
1.158505e-10 |
975 |
KUC104123 |
LSM-2866 |
|
10uM |
6h |
LINCSCP_5511 |
LINCSCP_5511 |
A549 |
| 0.204466 |
1.160087e-10 |
975 |
PD-160170 |
LSM-2247 |
NPY1R |
10uM |
6h |
LINCSCP_26897 |
LINCSCP_26897 |
HT29 |
| 0.204455 |
1.162783e-10 |
975 |
BRD-K12559526 |
LSM-14723 |
|
5uM |
24h |
LINCSCP_64160 |
LINCSCP_64160 |
VCAP |
| -0.204451 |
1.163774e-10 |
975 |
KF 38789 |
LSM-1641 |
SELP |
10uM |
6h |
LINCSCP_44096 |
LINCSCP_44096 |
PC3 |
| -0.204429 |
1.169266e-10 |
975 |
GR-127935 |
LSM-2243 |
HTR1A|HTR1B|HTR1D|HTR2A|HTR2C |
10uM |
6h |
LINCSCP_26980 |
LINCSCP_26980 |
HT29 |
| -0.204427 |
1.169701e-10 |
975 |
LDN 193189 |
LSM-1115 |
ACVR1|BMPR1A |
10uM |
6h |
LINCSCP_10508 |
LINCSCP_10508 |
AGS |
| -0.204427 |
1.169786e-10 |
975 |
Ciglitazone |
LSM-1911 |
PPARG |
10uM |
6h |
LINCSCP_7647 |
LINCSCP_7647 |
A549 |
| 0.204425 |
1.170365e-10 |
975 |
Diphenidol |
LSM-2008 |
CHRM1|CHRM3|CHRM4 |
10uM |
6h |
LINCSCP_14539 |
LINCSCP_14539 |
HA1E |
| 0.20442 |
1.171623e-10 |
975 |
BRD-K40240180 |
LSM-10884 |
|
5uM |
24h |
LINCSCP_61231 |
LINCSCP_61231 |
VCAP |
| -0.204415 |
1.172656e-10 |
975 |
BRD-K85642378 |
LSM-41940 |
|
1uM |
24h |
LINCSCP_312561 |
LINCSCP_312561 |
VCAP |
| -0.204411 |
1.173634e-10 |
975 |
VU0365118-1 |
LSM-3189 |
|
10uM |
24h |
LINCSCP_45712 |
LINCSCP_45712 |
PC3 |
| 0.204341 |
1.191429e-10 |
975 |
Nefazodone |
LSM-4031 |
HTR2A|HTR2C|SLC6A2|SLC6A4 |
0.37uM |
24h |
LINCSCP_92191 |
LINCSCP_92191 |
HA1E |
| -0.20434 |
1.191642e-10 |
975 |
CP-724714 |
LSM-42777 |
ERBB2 |
10uM |
6h |
LINCSCP_2209 |
LINCSCP_2209 |
A375 |
| 0.204324 |
1.195515e-10 |
975 |
alizapride |
LSM-45800 |
|
3.33uM |
24h |
LINCSCP_142146 |
LINCSCP_142146 |
MCF7 |
| -0.204315 |
1.197886e-10 |
975 |
IC 261 |
LSM-42870 |
|
1uM |
6h |
LINCSCP_253647 |
LINCSCP_253647 |
MCF7 |
| 0.204314 |
1.198185e-10 |
975 |
BRD-K07004447 |
LSM-6742 |
|
5uM |
24h |
LINCSCP_63053 |
LINCSCP_63053 |
VCAP |
| 0.204303 |
1.200923e-10 |
975 |
CHEMBL2355627 |
LSM-11872 |
|
5uM |
24h |
LINCSCP_61476 |
LINCSCP_61476 |
VCAP |
| -0.204299 |
1.202015e-10 |
975 |
GSK-461364 |
LSM-1013 |
PLK1 |
0.12uM |
24h |
LINCSCP_127652 |
LINCSCP_127652 |
HT29 |
| 0.204299 |
1.202079e-10 |
975 |
Tubocurarine |
LSM-4245 |
CHRNA1|CHRNA2|CHRNB1|CHRND|CHRNE|CHRNG|HTR3A |
10uM |
6h |
LINCSCP_220868 |
LINCSCP_220868 |
HEPG2 |
| 0.204296 |
1.202688e-10 |
975 |
Vorinostat |
LSM-3828 |
HDAC1|HDAC2|HDAC3|HDAC6|HDAC8 |
0.5uM |
24h |
LINCSCP_201015 |
LINCSCP_201015 |
A549 |
| 0.204287 |
1.204954e-10 |
975 |
Benzohydroxamate |
LSM-36789 |
|
0.5uM |
24h |
LINCSCP_49240 |
LINCSCP_49240 |
PC3 |
| 0.204272 |
1.208871e-10 |
975 |
Omacetaxine Mepesuccinate |
LSM-3716 |
|
0.001uM |
24h |
LINCSCP_36004 |
LINCSCP_36004 |
MCF7 |
| -0.20426 |
1.211860e-10 |
975 |
HG-5-88-01 |
LSM-42725 |
COQ8B|EGFR |
10uM |
24h |
LINCSCP_52312 |
LINCSCP_52312 |
SKB |
| -0.204257 |
1.212683e-10 |
975 |
Palbociclib |
LSM-1071 |
CCND1|CDK4|CDK6 |
10uM |
3h |
LINCSCP_130170 |
LINCSCP_130170 |
LNCAP |
| -0.204248 |
1.214994e-10 |
975 |
Chlorprothixene |
LSM-42990 |
DRD2|DRD3|HTR2A|HTR2C |
10uM |
24h |
LINCSCP_47563 |
LINCSCP_47563 |
PC3 |
| -0.204242 |
1.216586e-10 |
975 |
BRD-K65494396 |
LSM-40847 |
|
10uM |
6h |
LINCSCP_49159 |
LINCSCP_49159 |
PC3 |
| 0.204239 |
1.217304e-10 |
975 |
MK-2866 (GTx-024) |
LSM-45447 |
AR |
0.12uM |
24h |
LINCSCP_71317 |
LINCSCP_71317 |
A375 |
| 0.204236 |
1.218045e-10 |
975 |
SA-1925610 |
LSM-38660 |
|
1uM |
6h |
LINCSCP_252417 |
LINCSCP_252417 |
MCF7 |
| -0.204235 |
1.218423e-10 |
975 |
9-Cis retinol |
LSM-5317 |
RARA|RARB|RARG|RORB |
40uM |
6h |
LINCSCP_51181 |
LINCSCP_51181 |
RMUGS |
| -0.20423 |
1.219646e-10 |
975 |
SCHEMBL16226502 |
LSM-43056 |
HSP90AA1 |
10uM |
24h |
LINCSCP_114377 |
LINCSCP_114377 |
HME1 |
| -0.204217 |
1.222951e-10 |
975 |
Nocodazole |
LSM-2260 |
|
10uM |
24h |
LINCSCP_47491 |
LINCSCP_47491 |
PC3 |
| 0.204214 |
1.223860e-10 |
975 |
SMP2_000249 |
LSM-1820 |
ATP1A1 |
10uM |
24h |
LINCSCP_11384 |
LINCSCP_11384 |
ASC |
| 0.204212 |
1.224465e-10 |
975 |
CHEMBL1788383 |
LSM-3875 |
DRD2|SIGMAR1 |
10uM |
24h |
LINCSCP_18322 |
LINCSCP_18322 |
HCC515 |
| 0.204207 |
1.225589e-10 |
975 |
CHEMBL2136735 |
LSM-1152 |
FGFR1|FGFR3|FLT1|FLT4|KDR|PDGFRA|PDGFRB |
0.12uM |
3h |
LINCSCP_145787 |
LINCSCP_145787 |
MDAMB231 |
| 0.204175 |
1.234104e-10 |
975 |
ZINC5751650 |
LSM-43166 |
|
10uM |
24h |
LINCSCP_52206 |
LINCSCP_52206 |
SKB |
| 0.204159 |
1.238105e-10 |
975 |
SCHEMBL16226502 |
LSM-43056 |
HSP90AA1 |
0.001uM |
24h |
LINCSCP_201088 |
LINCSCP_201088 |
A549 |
| -0.204157 |
1.238710e-10 |
975 |
R547 |
LSM-45812 |
|
1.11uM |
24h |
LINCSCP_106605 |
LINCSCP_106605 |
HELA |
| -0.204115 |
1.249769e-10 |
975 |
CHEMBL2144875 |
LSM-6105 |
|
10uM |
24h |
LINCSCP_33848 |
LINCSCP_33848 |
MCF7 |
| 0.204099 |
1.253994e-10 |
975 |
Danazol |
LSM-3073 |
AR|ESR1|GNRHR|PGR |
10uM |
6h |
LINCSCP_3092 |
LINCSCP_3092 |
A375 |
| -0.204064 |
1.263340e-10 |
975 |
Simeprevir |
LSM-45598 |
|
0.04uM |
24h |
LINCSCP_142498 |
LINCSCP_142498 |
MCF7 |
| -0.204051 |
1.266747e-10 |
975 |
SPOX1_000651 |
LSM-4624 |
|
10uM |
24h |
LINCSCP_32174 |
LINCSCP_32174 |
MCF7 |
| -0.204044 |
1.268814e-10 |
975 |
NVP-BHG712 |
LSM-1201 |
|
10uM |
24h |
LINCSCP_148229 |
LINCSCP_148229 |
NPC.CAS9 |
| -0.204039 |
1.270060e-10 |
975 |
GTP 14564 |
LSM-2363 |
FLT3 |
10uM |
6h |
LINCSCP_2691 |
LINCSCP_2691 |
A375 |
| -0.204037 |
1.270495e-10 |
975 |
BRD-K32628102 |
LSM-39067 |
|
10uM |
6h |
LINCSCP_279452 |
LINCSCP_279452 |
PC3 |
| 0.204028 |
1.272946e-10 |
975 |
ALD1-H_000553 |
LSM-45118 |
|
10uM |
24h |
LINCSCP_239532 |
LINCSCP_239532 |
MCF7 |
| 0.204017 |
1.276015e-10 |
975 |
SA-1456734 |
LSM-40148 |
|
0.5uM |
24h |
LINCSCP_37703 |
LINCSCP_37703 |
MCF7 |
| -0.204001 |
1.280350e-10 |
975 |
Vemurafenib |
LSM-42737 |
BRAF |
0.5uM |
6h |
LINCSCP_52 |
LINCSCP_52 |
A375 |
| -0.203969 |
1.289055e-10 |
975 |
Sildenafil |
LSM-3797 |
PDE5A |
0.01uM |
6h |
LINCSCP_9341 |
LINCSCP_9341 |
A549 |
| -0.203942 |
1.296332e-10 |
975 |
I-BET151 |
LSM-6335 |
|
0.12uM |
24h |
LINCSCP_128893 |
LINCSCP_128893 |
HUVEC |
| -0.203939 |
1.297331e-10 |
975 |
GSK 1059615 |
LSM-42799 |
PIK3CA|PIK3CB|PIK3CD|PIK3CG |
10uM |
24h |
LINCSCP_148967 |
LINCSCP_148967 |
NPC |
| -0.203933 |
1.298960e-10 |
975 |
AZ20 |
LSM-36357 |
|
10uM |
24h |
LINCSCP_150183 |
LINCSCP_150183 |
NPC.TAK |
| -0.203917 |
1.303458e-10 |
975 |
ML162 |
LSM-1493 |
|
10uM |
24h |
LINCSCP_31543 |
LINCSCP_31543 |
MCF7 |
| -0.203899 |
1.308312e-10 |
975 |
CHEMBL3187962 |
LSM-6081 |
|
10uM |
6h |
LINCSCP_272230 |
LINCSCP_272230 |
PC3 |
| -0.203895 |
1.309451e-10 |
975 |
BDBM50442904 |
LSM-4418 |
|
10uM |
6h |
LINCSCP_23550 |
LINCSCP_23550 |
HEPG2 |
| -0.20389 |
1.310755e-10 |
975 |
Carbamazepine |
LSM-3610 |
SCN10A|SCN11A|SCN1A|SCN2A|SCN3A|SCN4A|SCN5A|SCN7A|SCN8A|SCN9A |
100uM |
6h |
LINCSCP_15644 |
LINCSCP_15644 |
HA1E |
| -0.203873 |
1.315537e-10 |
975 |
AS-605240 |
LSM-42784 |
PIK3CG |
0.12uM |
3h |
LINCSCP_145949 |
LINCSCP_145949 |
MDAMB231 |
| 0.203871 |
1.315996e-10 |
975 |
AC1MXYGS |
LSM-2620 |
|
10uM |
24h |
LINCSCP_5588 |
LINCSCP_5588 |
A549 |
| -0.203868 |
1.317032e-10 |
975 |
MG-132 |
LSM-1107 |
PSMB1 |
20uM |
24h |
LINCSCP_134817 |
LINCSCP_134817 |
MCF7 |
| -0.203852 |
1.321363e-10 |
975 |
MLS-0315803.0001 |
LSM-3201 |
|
10uM |
6h |
LINCSCP_19754 |
LINCSCP_19754 |
HCC515 |
| -0.203845 |
1.323442e-10 |
975 |
Tyrphostin B7 |
LSM-42938 |
PDGFRB |
10uM |
6h |
LINCSCP_265375 |
LINCSCP_265375 |
PC3 |
| 0.203841 |
1.324481e-10 |
975 |
BRD-K72375447 |
LSM-12869 |
|
5uM |
24h |
LINCSCP_62473 |
LINCSCP_62473 |
VCAP |
| -0.203803 |
1.335022e-10 |
975 |
KUC104493 |
LSM-2344 |
|
10uM |
6h |
LINCSCP_15959 |
LINCSCP_15959 |
HA1E |
| -0.203791 |
1.338643e-10 |
975 |
(3-Isopropoxyphenyl)(1-((5-methyl-1-propyl-1H-pyrazol-4-yl)methyl)piperidin-3-yl)methanone |
LSM-1323 |
|
10uM |
24h |
LINCSCP_177107 |
LINCSCP_177107 |
A375 |
| 0.203767 |
1.345279e-10 |
975 |
BRD-K94177318 |
LSM-14199 |
|
5uM |
24h |
LINCSCP_62067 |
LINCSCP_62067 |
VCAP |
| -0.203749 |
1.350475e-10 |
975 |
Paricalcitol |
LSM-45519 |
VDR |
10uM |
24h |
LINCSCP_105969 |
LINCSCP_105969 |
HELA |
| 0.203742 |
1.352642e-10 |
975 |
DIMETHYL FUMARATE |
LSM-45569 |
KEAP1 |
1.11uM |
24h |
LINCSCP_90041 |
LINCSCP_90041 |
HA1E |
| 0.203715 |
1.360233e-10 |
975 |
Triclosan |
LSM-2929 |
DNMT1 |
0.12uM |
24h |
LINCSCP_171337 |
LINCSCP_171337 |
YAPC |
| -0.203713 |
1.360758e-10 |
975 |
MLS002264481 |
LSM-3043 |
|
10uM |
24h |
LINCSCP_1404 |
LINCSCP_1404 |
A375 |
| -0.203697 |
1.365364e-10 |
975 |
Homatropine hydrobromide |
LSM-46037 |
CHRM1 |
10uM |
6h |
LINCSCP_4315 |
LINCSCP_4315 |
A549 |
| -0.203682 |
1.369675e-10 |
975 |
1-(2,6-Dichlorobenzylideneamino)guanidine |
LSM-3266 |
|
10uM |
6h |
LINCSCP_30391 |
LINCSCP_30391 |
MCF7 |
| -0.203675 |
1.371729e-10 |
975 |
AC1MHNXZ |
LSM-37086 |
|
10uM |
24h |
LINCSCP_263462 |
LINCSCP_263462 |
NPC |
| -0.203671 |
1.372946e-10 |
975 |
Curcumin |
LSM-43083 |
PTGS1|PTGS2 |
0.04uM |
24h |
LINCSCP_76659 |
LINCSCP_76659 |
A375 |
| 0.203624 |
1.386616e-10 |
975 |
THZ-2-98-01 |
LSM-44946 |
|
3.33uM |
24h |
LINCSCP_129979 |
LINCSCP_129979 |
LNCAP |
| -0.203621 |
1.387653e-10 |
975 |
MLS000089581 |
LSM-3886 |
|
10uM |
24h |
LINCSCP_31015 |
LINCSCP_31015 |
MCF7 |
| -0.203604 |
1.392609e-10 |
975 |
Wortmannin |
LSM-3947 |
PIK3CA|PIK3CG|PLK1 |
10uM |
24h |
LINCSCP_67180 |
LINCSCP_67180 |
HT29 |
| -0.203599 |
1.393961e-10 |
975 |
BRD-K85790491 |
LSM-13684 |
|
5uM |
24h |
LINCSCP_230761 |
LINCSCP_230761 |
HT29 |
| 0.203574 |
1.401544e-10 |
975 |
Cytarabine |
LSM-5470 |
POLA1|POLB|POLD1|POLE |
0.04uM |
24h |
LINCSCP_74129 |
LINCSCP_74129 |
A375 |
| -0.203572 |
1.401880e-10 |
975 |
Camostat Mesilate |
LSM-45240 |
|
0.37uM |
24h |
LINCSCP_91603 |
LINCSCP_91603 |
HA1E |
| 0.203544 |
1.410372e-10 |
975 |
TUL_XIX002 |
LSM-36793 |
|
0.01uM |
6h |
LINCSCP_55132 |
LINCSCP_55132 |
THP1 |
| -0.203541 |
1.411197e-10 |
975 |
CHEMBL2141330 |
LSM-39999 |
|
10uM |
6h |
LINCSCP_27215 |
LINCSCP_27215 |
HT29 |
| -0.20353 |
1.414572e-10 |
975 |
Tozasertib |
LSM-1021 |
ABL1|AURKA|AURKB|AURKC|BCR|FLT3|JAK2 |
10uM |
24h |
LINCSCP_4081 |
LINCSCP_4081 |
A375 |
| -0.203497 |
1.424493e-10 |
975 |
MG-132 |
LSM-1107 |
PSMB1 |
20uM |
24h |
LINCSCP_134723 |
LINCSCP_134723 |
MCF7 |
| 0.203495 |
1.424983e-10 |
975 |
BRD-K41087962 |
LSM-42690 |
|
0.5uM |
6h |
LINCSCP_54231 |
LINCSCP_54231 |
SW620 |
| 0.203494 |
1.425326e-10 |
975 |
MLS003128748 |
LSM-10166 |
|
5uM |
24h |
LINCSCP_309135 |
LINCSCP_309135 |
VCAP |
| 0.20348 |
1.429630e-10 |
975 |
Zileuton |
LSM-5084 |
ALOX5 |
10uM |
24h |
LINCSCP_73461 |
LINCSCP_73461 |
A375 |
| -0.203477 |
1.430441e-10 |
975 |
Oxibendazole |
LSM-3153 |
TUBB |
10uM |
24h |
LINCSCP_32910 |
LINCSCP_32910 |
MCF7 |
| -0.203476 |
1.430658e-10 |
975 |
Mitoxantrone |
LSM-2481 |
TOP2A |
1.11uM |
24h |
LINCSCP_131894 |
LINCSCP_131894 |
MCF7 |
| -0.203454 |
1.437274e-10 |
975 |
Carbazole, 9-(4-methylbenzoyl)- |
LSM-3597 |
|
10uM |
6h |
LINCSCP_5148 |
LINCSCP_5148 |
A549 |
| -0.203445 |
1.440257e-10 |
975 |
BRD-K60637442 |
LSM-12093 |
|
5uM |
24h |
LINCSCP_8637 |
LINCSCP_8637 |
A549 |
| -0.203438 |
1.442184e-10 |
975 |
Firategrast |
LSM-45715 |
ITGA4|ITGB1|ITGB7 |
1.11uM |
24h |
LINCSCP_71607 |
LINCSCP_71607 |
A375 |
| -0.203436 |
1.442752e-10 |
975 |
BG-51 |
LSM-45301 |
HDAC3 |
0.5uM |
24h |
LINCSCP_250213 |
LINCSCP_250213 |
MCF7 |
| -0.203436 |
1.442809e-10 |
975 |
331771-20-1 |
LSM-1096 |
AURKA|AURKB |
10uM |
24h |
LINCSCP_149355 |
LINCSCP_149355 |
NPC |
| -0.203432 |
1.444209e-10 |
975 |
MLS003129663 |
LSM-7167 |
|
10uM |
24h |
LINCSCP_249960 |
LINCSCP_249960 |
MCF7 |
| -0.203384 |
1.458864e-10 |
975 |
CHEMBL585951 |
LSM-36386 |
MAPK8 |
1.11uM |
3h |
LINCSCP_131720 |
LINCSCP_131720 |
MCF10A |
| -0.203383 |
1.458974e-10 |
975 |
BRD-K45627302 |
LSM-44774 |
|
10uM |
24h |
LINCSCP_249788 |
LINCSCP_249788 |
MCF7 |
| 0.203368 |
1.463866e-10 |
975 |
MILNACIPRAN HYDROCHLORIDE |
LSM-45870 |
SLC6A2|SLC6A4 |
0.04uM |
24h |
LINCSCP_138059 |
LINCSCP_138059 |
MCF7 |
| -0.203362 |
1.465435e-10 |
975 |
AZ20 |
LSM-36357 |
|
10uM |
24h |
LINCSCP_148025 |
LINCSCP_148025 |
NPC.CAS9 |
| 0.203355 |
1.467892e-10 |
975 |
BRD-K23886631 |
LSM-38573 |
|
5uM |
24h |
LINCSCP_63016 |
LINCSCP_63016 |
VCAP |
| -0.203351 |
1.469054e-10 |
975 |
BRD-A28746609 |
LSM-1102 |
NR1I2|TUBB |
3.33uM |
24h |
LINCSCP_169351 |
LINCSCP_169351 |
YAPC |
| -0.20334 |
1.472540e-10 |
975 |
BRD-K46796516 |
LSM-11286 |
|
5uM |
24h |
LINCSCP_61786 |
LINCSCP_61786 |
VCAP |
| -0.203336 |
1.473667e-10 |
975 |
MLS002460474 |
LSM-3256 |
|
10uM |
6h |
LINCSCP_29146 |
LINCSCP_29146 |
JHUEM2 |
| 0.203335 |
1.473837e-10 |
975 |
Mafenide |
LSM-5445 |
CA6 |
10uM |
24h |
LINCSCP_45690 |
LINCSCP_45690 |
PC3 |
| -0.20331 |
1.481779e-10 |
975 |
Buparlisib |
LSM-1148 |
PIK3CA|PIK3CB|PIK3CD|PIK3CG|PIK3R1|PIK3R2|PIK3R3|PIK3R5 |
3.33uM |
24h |
LINCSCP_136777 |
LINCSCP_136777 |
MCF7 |
| -0.203273 |
1.493413e-10 |
975 |
Dasatinib |
LSM-1020 |
ABL1|BCR|BLK|EPHA2|FGR|FRK|FYN|HCK|KIT|LCK|LYN|PDGFRB|SRC|SRMS|YES1 |
10uM |
24h |
LINCSCP_116673 |
LINCSCP_116673 |
HT29 |
| 0.20327 |
1.494175e-10 |
975 |
Trametinib |
LSM-1143 |
MAP2K1|MAP2K2 |
3.33uM |
3h |
LINCSCP_163476 |
LINCSCP_163476 |
SKBR3 |
| -0.203248 |
1.501317e-10 |
975 |
Totaralolal |
LSM-1625 |
|
10uM |
6h |
LINCSCP_56111 |
LINCSCP_56111 |
VCAP |
| -0.203221 |
1.509727e-10 |
975 |
LY2874455 |
LSM-45659 |
|
10uM |
24h |
LINCSCP_89884 |
LINCSCP_89884 |
HA1E |
| -0.203213 |
1.512523e-10 |
975 |
BRD-K21498052 |
LSM-38435 |
|
5uM |
24h |
LINCSCP_48321 |
LINCSCP_48321 |
PC3 |
| 0.203195 |
1.518187e-10 |
975 |
Carbacyclin |
LSM-42923 |
PPARD|PTGIR |
10uM |
24h |
LINCSCP_43426 |
LINCSCP_43426 |
NPC |
| 0.203187 |
1.520722e-10 |
975 |
MLS000766411 |
LSM-4603 |
|
10uM |
6h |
LINCSCP_46343 |
LINCSCP_46343 |
PC3 |
| -0.203186 |
1.520911e-10 |
975 |
TAE-684 |
LSM-1024 |
ALK |
10uM |
24h |
LINCSCP_11042 |
LINCSCP_11042 |
ASC |
| 0.203182 |
1.522396e-10 |
975 |
Amidate |
LSM-1640 |
GABRA1|GABRA2|GABRA3|GABRA4|GABRA5|GABRA6|GABRB1|GABRB2|GABRB3|GABRD|GABRE|GABRG1|GABRG2|GABRG3|GABRP|GABRQ |
0.04uM |
24h |
LINCSCP_140224 |
LINCSCP_140224 |
MCF7 |
| -0.203177 |
1.523857e-10 |
975 |
CHEMBL1698064 |
LSM-1979 |
APEX1 |
10uM |
24h |
LINCSCP_45659 |
LINCSCP_45659 |
PC3 |
| -0.203173 |
1.525332e-10 |
975 |
Nepafenac |
LSM-45729 |
PTGS1|PTGS2 |
0.04uM |
24h |
LINCSCP_169919 |
LINCSCP_169919 |
YAPC |
| -0.203162 |
1.528714e-10 |
975 |
Androstenol |
LSM-5400 |
NR1I3 |
10uM |
6h |
LINCSCP_2333 |
LINCSCP_2333 |
A375 |
| 0.203162 |
1.528724e-10 |
975 |
Alvelestat |
LSM-45793 |
|
0.12uM |
24h |
LINCSCP_137638 |
LINCSCP_137638 |
MCF7 |
| -0.203155 |
1.530890e-10 |
975 |
Albendazole |
LSM-3782 |
|
1.11uM |
24h |
LINCSCP_143473 |
LINCSCP_143473 |
MCF7 |
| -0.203153 |
1.531532e-10 |
975 |
VGX-1027 |
LSM-45622 |
|
0.37uM |
24h |
LINCSCP_135329 |
LINCSCP_135329 |
MCF7 |
| 0.203137 |
1.536784e-10 |
975 |
Imatinib |
LSM-1023 |
ABL1|BCR|CSF1R|KIT|PDGFRA|PDGFRB |
0.12uM |
3h |
LINCSCP_145937 |
LINCSCP_145937 |
MDAMB231 |
| 0.203136 |
1.537200e-10 |
975 |
GSK-319347A |
LSM-1216 |
IKBKG |
5uM |
24h |
LINCSCP_15337 |
LINCSCP_15337 |
HA1E |
| -0.203131 |
1.538853e-10 |
975 |
CHEMBL520231 |
LSM-43280 |
XPO1 |
10uM |
6h |
LINCSCP_39877 |
LINCSCP_39877 |
NCIH1694 |
| -0.203113 |
1.544696e-10 |
975 |
Sarsasapogenin |
LSM-45816 |
|
0.53uM |
24h |
LINCSCP_172425 |
LINCSCP_172425 |
YAPC |
| -0.203108 |
1.546382e-10 |
975 |
BSPBIO_000981 |
LSM-43126 |
ACTA1 |
10uM |
6h |
LINCSCP_2145 |
LINCSCP_2145 |
A375 |
| -0.203107 |
1.546534e-10 |
975 |
Loperamide |
LSM-3365 |
OPRD1|OPRM1 |
10uM |
6h |
LINCSCP_20742 |
LINCSCP_20742 |
HCC515 |
| 0.203102 |
1.548123e-10 |
975 |
Cobicistat (GS-9350) |
LSM-45771 |
CYP3A4|CYP3A43|CYP3A5|CYP3A7|CYP3A7-CYP3A51P |
0.04uM |
24h |
LINCSCP_136991 |
LINCSCP_136991 |
MCF7 |
| -0.203084 |
1.554170e-10 |
975 |
MLS003126519 |
LSM-3676 |
|
10uM |
6h |
LINCSCP_1616 |
LINCSCP_1616 |
A375 |
| 0.203068 |
1.559306e-10 |
975 |
ST021200 |
LSM-4601 |
|
10uM |
6h |
LINCSCP_12541 |
LINCSCP_12541 |
CL34 |
| -0.203054 |
1.563814e-10 |
975 |
Sertaconazole |
LSM-1938 |
|
10uM |
24h |
LINCSCP_34648 |
LINCSCP_34648 |
MCF7 |
| -0.203042 |
1.567863e-10 |
975 |
CHEMBL1716096 |
LSM-2446 |
|
10uM |
24h |
LINCSCP_31346 |
LINCSCP_31346 |
MCF7 |
| 0.203042 |
1.568061e-10 |
975 |
ZINC01045466 |
LSM-4913 |
|
10uM |
6h |
LINCSCP_295950 |
LINCSCP_295950 |
VCAP |
| -0.203038 |
1.569339e-10 |
975 |
Benzthiazide |
LSM-2474 |
CA2|SLC12A3 |
10uM |
24h |
LINCSCP_153888 |
LINCSCP_153888 |
PC3 |
| -0.203025 |
1.573606e-10 |
975 |
XL888 |
LSM-45553 |
|
0.04uM |
24h |
LINCSCP_104728 |
LINCSCP_104728 |
HELA |
| 0.20302 |
1.575341e-10 |
975 |
Indomethacin |
LSM-3275 |
PPARG|PTGDR2|PTGS1|PTGS2 |
10uM |
6h |
LINCSCP_525 |
LINCSCP_525 |
A375 |
| -0.203011 |
1.578265e-10 |
975 |
MLS000594029 |
LSM-4801 |
|
10uM |
24h |
LINCSCP_31907 |
LINCSCP_31907 |
MCF7 |
| 0.202977 |
1.589615e-10 |
975 |
Ammonium Glycyrrhizinate |
LSM-46003 |
|
1.11uM |
24h |
LINCSCP_156267 |
LINCSCP_156267 |
PC3 |
| -0.202976 |
1.589748e-10 |
975 |
AT-7519 |
LSM-1004 |
CDK1|CDK10|CDK11B|CDK12|CDK13|CDK14|CDK15|CDK16|CDK17|CDK18|CDK19|CDK2|CDK20|CDK3|CDK4|CDK5|CDK6|CDK7|CDK8|CDK9 |
1.11uM |
24h |
LINCSCP_137906 |
LINCSCP_137906 |
MCF7 |
| -0.202966 |
1.593308e-10 |
975 |
M3M3FBS |
LSM-2196 |
PLCB2|PLCB3|PLCD1|PLCG1|PLCG2 |
10uM |
24h |
LINCSCP_52726 |
LINCSCP_52726 |
SKB |
| 0.202963 |
1.594395e-10 |
975 |
Valproic acid |
LSM-4620 |
ABAT|ALDH5A1|HDAC1|SCN1A|SCN3A |
5uM |
48h |
LINCSCP_64536 |
LINCSCP_64536 |
VCAP |
| -0.202956 |
1.596471e-10 |
975 |
Radicicol |
LSM-43303 |
|
5uM |
48h |
LINCSCP_64517 |
LINCSCP_64517 |
VCAP |
| -0.202943 |
1.600933e-10 |
975 |
SYK Inhibitor |
LSM-42930 |
SYK |
10uM |
24h |
LINCSCP_11431 |
LINCSCP_11431 |
ASC |
| -0.20292 |
1.608711e-10 |
975 |
Nevirapine |
LSM-5336 |
CYP1A2|CYP2A6|CYP2B6|CYP2C9|CYP2D6|CYP3A4|CYP3A5 |
0.37uM |
24h |
LINCSCP_101492 |
LINCSCP_101492 |
HELA |
| -0.202919 |
1.609195e-10 |
975 |
GSK-461364 |
LSM-1013 |
PLK1 |
10uM |
24h |
LINCSCP_51488 |
LINCSCP_51488 |
SKBR3 |
| -0.202905 |
1.613681e-10 |
975 |
C24H25CLFN5O3 |
LSM-42794 |
EGFR|ERBB2|ERBB4 |
0.12uM |
3h |
LINCSCP_145781 |
LINCSCP_145781 |
MDAMB231 |
| 0.202904 |
1.614115e-10 |
975 |
MLS002699810 |
LSM-4058 |
|
10uM |
6h |
LINCSCP_21938 |
LINCSCP_21938 |
HEPG2 |
| -0.202874 |
1.624265e-10 |
975 |
CHEMBL1242477 |
LSM-6208 |
PIK3CA|PIK3CB|PIK3CD|PIK3CG |
20uM |
6h |
LINCSCP_21319 |
LINCSCP_21319 |
HEC108 |
| -0.202866 |
1.627226e-10 |
975 |
AC1Q6JJ5 |
LSM-6192 |
TOP2A |
0.01uM |
24h |
LINCSCP_9669 |
LINCSCP_9669 |
A549 |
| 0.202861 |
1.628767e-10 |
975 |
16,16-Dimethyl prostaglandin e2 |
LSM-43285 |
HPGD |
10uM |
6h |
LINCSCP_39827 |
LINCSCP_39827 |
MDST8 |
| -0.202848 |
1.633188e-10 |
975 |
AC1O8PYD |
LSM-1697 |
NR3C1 |
10uM |
24h |
LINCSCP_52713 |
LINCSCP_52713 |
SKB |
| -0.202848 |
1.633329e-10 |
975 |
BRD-K32568627 |
LSM-39061 |
|
10uM |
6h |
LINCSCP_16814 |
LINCSCP_16814 |
HA1E |
| -0.20284 |
1.635958e-10 |
975 |
Dasatinib |
LSM-1020 |
ABL1|BCR|BLK|EPHA2|FGR|FRK|FYN|HCK|KIT|LCK|LYN|PDGFRB|SRC|SRMS|YES1 |
1.11uM |
24h |
LINCSCP_124645 |
LINCSCP_124645 |
HT29 |
| 0.202838 |
1.636919e-10 |
975 |
BUTORPHANOL-(+)-TARTRATE (DEA license) |
LSM-45696 |
OPRK1|OPRM1 |
1.11uM |
24h |
LINCSCP_122490 |
LINCSCP_122490 |
HT29 |
| -0.202805 |
1.648189e-10 |
975 |
BRD-K38586507 |
LSM-39392 |
|
5uM |
24h |
LINCSCP_248965 |
LINCSCP_248965 |
MCF7 |
| -0.202797 |
1.650858e-10 |
975 |
BRD-K63513868 |
LSM-45333 |
|
1uM |
6h |
LINCSCP_43872 |
LINCSCP_43872 |
PC3 |
| -0.202796 |
1.651418e-10 |
975 |
Tolazamide |
LSM-2699 |
ABCC8|KCNJ11 |
10uM |
24h |
LINCSCP_296050 |
LINCSCP_296050 |
VCAP |
| 0.20279 |
1.653461e-10 |
975 |
BRD-K33451389 |
LSM-10456 |
|
5uM |
24h |
LINCSCP_62275 |
LINCSCP_62275 |
VCAP |
| 0.202787 |
1.654534e-10 |
975 |
noscapine |
|
|
1.11uM |
3h |
LINCSCP_164098 |
LINCSCP_164098 |
SKBR3 |
| 0.202777 |
1.657788e-10 |
975 |
BRD-A35207501 |
LSM-45361 |
|
1uM |
24h |
LINCSCP_222093 |
LINCSCP_222093 |
HL60 |
| -0.202768 |
1.660970e-10 |
975 |
MLS001172197 |
LSM-3527 |
|
10uM |
24h |
LINCSCP_25957 |
LINCSCP_25957 |
HT29 |
| 0.20276 |
1.663928e-10 |
975 |
TAK-242 |
LSM-45934 |
|
0.37uM |
24h |
LINCSCP_123310 |
LINCSCP_123310 |
HT29 |
| -0.202754 |
1.666080e-10 |
975 |
PD-0325901 |
LSM-1101 |
MAP2K1|MAP2K2 |
1.11uM |
24h |
LINCSCP_83274 |
LINCSCP_83274 |
ASC.C |
| -0.20275 |
1.667359e-10 |
975 |
GF-109203 |
LSM-2677 |
PRKCA |
10uM |
6h |
LINCSCP_66255 |
LINCSCP_66255 |
WSUDLCL2 |
| 0.202742 |
1.670144e-10 |
975 |
Buparlisib |
LSM-1148 |
PIK3CA|PIK3CB|PIK3CD|PIK3CG|PIK3R1|PIK3R2|PIK3R3|PIK3R5 |
0.12uM |
24h |
LINCSCP_130581 |
LINCSCP_130581 |
MCF10A |
| -0.202741 |
1.670428e-10 |
975 |
BRD-K15973523 |
LSM-9385 |
|
10uM |
24h |
LINCSCP_9002 |
LINCSCP_9002 |
A549 |
| -0.202733 |
1.673407e-10 |
975 |
AZD-1775 |
LSM-1153 |
WEE1 |
1.11uM |
24h |
LINCSCP_140089 |
LINCSCP_140089 |
MCF7 |
| -0.202714 |
1.680106e-10 |
975 |
MG-132 |
LSM-1107 |
PSMB1 |
20uM |
24h |
LINCSCP_72395 |
LINCSCP_72395 |
A375 |
| 0.202708 |
1.682042e-10 |
975 |
MK-8245 |
LSM-45756 |
|
3.33uM |
24h |
LINCSCP_71302 |
LINCSCP_71302 |
A375 |
| 0.202702 |
1.684161e-10 |
975 |
Alizapride |
LSM-4953 |
DRD2 |
0.12uM |
24h |
LINCSCP_75201 |
LINCSCP_75201 |
A375 |
| -0.202689 |
1.688888e-10 |
975 |
Famciclovir |
LSM-2990 |
|
3.33uM |
24h |
LINCSCP_124422 |
LINCSCP_124422 |
HT29 |
| -0.20267 |
1.695690e-10 |
975 |
BRD-A00474148 |
LSM-45242 |
|
3.33uM |
24h |
LINCSCP_135957 |
LINCSCP_135957 |
MCF7 |
| 0.202667 |
1.696728e-10 |
975 |
BRD-K00256608 |
LSM-8440 |
|
5uM |
24h |
LINCSCP_62747 |
LINCSCP_62747 |
VCAP |
| 0.202652 |
1.702097e-10 |
975 |
MK-2866 (GTx-024) |
LSM-45447 |
AR |
0.37uM |
24h |
LINCSCP_71316 |
LINCSCP_71316 |
A375 |
| -0.202647 |
1.703969e-10 |
975 |
BRD-K75111717 |
LSM-13030 |
|
5uM |
24h |
LINCSCP_62033 |
LINCSCP_62033 |
VCAP |
| -0.202645 |
1.704573e-10 |
975 |
BRD-A25736793 |
LSM-43054 |
MTOR |
1.11uM |
24h |
LINCSCP_146225 |
LINCSCP_146225 |
MNEU.E |
| 0.202643 |
1.705356e-10 |
975 |
Fccp |
LSM-2317 |
|
10uM |
6h |
LINCSCP_7436 |
LINCSCP_7436 |
A549 |
| -0.202642 |
1.705541e-10 |
975 |
Chrysin |
LSM-6566 |
|
1.11uM |
24h |
LINCSCP_103191 |
LINCSCP_103191 |
HELA |
| 0.202642 |
1.705665e-10 |
975 |
MLS002276505 |
LSM-2599 |
|
10uM |
24h |
LINCSCP_25908 |
LINCSCP_25908 |
HT29 |
| 0.202638 |
1.707275e-10 |
975 |
Wortmannin |
LSM-3947 |
PIK3CA|PIK3CG|PLK1 |
0.001uM |
24h |
LINCSCP_250724 |
LINCSCP_250724 |
MCF7 |
| -0.202637 |
1.707323e-10 |
975 |
AT-7519 |
LSM-1004 |
CDK1|CDK10|CDK11B|CDK12|CDK13|CDK14|CDK15|CDK16|CDK17|CDK18|CDK19|CDK2|CDK20|CDK3|CDK4|CDK5|CDK6|CDK7|CDK8|CDK9 |
0.12uM |
24h |
LINCSCP_169714 |
LINCSCP_169714 |
YAPC |
| 0.20263 |
1.710130e-10 |
975 |
BRD-K32581454-001-01-5 |
LSM-6827 |
|
0.5uM |
24h |
LINCSCP_37903 |
LINCSCP_37903 |
MCF7 |
| -0.202615 |
1.715364e-10 |
975 |
AC1OCDAW |
LSM-1622 |
TOP2A |
0.37uM |
24h |
LINCSCP_10003 |
LINCSCP_10003 |
A549 |
| -0.202602 |
1.720166e-10 |
975 |
SMR000068650 |
LSM-2859 |
|
100uM |
6h |
LINCSCP_51140 |
LINCSCP_51140 |
RMUGS |
| -0.2026 |
1.720744e-10 |
975 |
SU-4312 |
LSM-2454 |
KDR |
10uM |
24h |
LINCSCP_52625 |
LINCSCP_52625 |
SKB |
| 0.202599 |
1.721329e-10 |
975 |
Foretinib |
LSM-1158 |
FLT1|FLT3|FLT4|KDR|KIT|MET|PDGFRA|PDGFRB|TEK |
0.12uM |
24h |
LINCSCP_69121 |
LINCSCP_69121 |
A375 |
| 0.202596 |
1.722259e-10 |
975 |
BRD-K17741643 |
LSM-14742 |
|
5uM |
24h |
LINCSCP_64169 |
LINCSCP_64169 |
VCAP |
| -0.202589 |
1.724782e-10 |
975 |
SCHEMBL6465902 |
LSM-3544 |
PDE5A |
10uM |
24h |
LINCSCP_42580 |
LINCSCP_42580 |
NPC |
| 0.202588 |
1.725234e-10 |
975 |
Glimepiride |
LSM-44957 |
ABCC8|KCNJ11 |
10uM |
6h |
LINCSCP_226677 |
LINCSCP_226677 |
HT29 |
| -0.20258 |
1.728085e-10 |
975 |
13-Hydroxy-8,14,19-trimethoxy-4,10,12,16-tetramethyl-3,20,22-trioxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18-pentaen-9-yl carbamate |
LSM-42815 |
HSP90AA1 |
0.5uM |
24h |
LINCSCP_43899 |
LINCSCP_43899 |
PC3 |
| 0.202571 |
1.731390e-10 |
975 |
Taurocholate |
LSM-5866 |
CEL |
10uM |
6h |
LINCSCP_20512 |
LINCSCP_20512 |
HCC515 |
| -0.202569 |
1.732078e-10 |
975 |
AZD-1775 |
LSM-1153 |
WEE1 |
1.11uM |
24h |
LINCSCP_112269 |
LINCSCP_112269 |
HEPG2 |
| -0.202559 |
1.735710e-10 |
975 |
BRD-K53501402 |
LSM-40209 |
|
10uM |
24h |
LINCSCP_33877 |
LINCSCP_33877 |
MCF7 |
| -0.202551 |
1.738661e-10 |
975 |
BRD-K67236726 |
LSM-12519 |
|
10uM |
24h |
LINCSCP_310413 |
LINCSCP_310413 |
VCAP |
| 0.202551 |
1.738758e-10 |
975 |
PRESTWICK3_000646 |
LSM-1699 |
|
10uM |
24h |
LINCSCP_4165 |
LINCSCP_4165 |
A549 |
| -0.202549 |
1.739368e-10 |
975 |
SCHEMBL17497408 |
LSM-44607 |
|
3uM |
24h |
LINCSCP_17249 |
LINCSCP_17249 |
HA1E |
| -0.202546 |
1.740346e-10 |
975 |
Antimycin A |
LSM-5076 |
CYCS |
10uM |
24h |
LINCSCP_34253 |
LINCSCP_34253 |
MCF7 |
| 0.202527 |
1.747402e-10 |
975 |
Imatinib |
LSM-1023 |
ABL1|BCR|CSF1R|KIT|PDGFRA|PDGFRB |
0.04uM |
24h |
LINCSCP_163784 |
LINCSCP_163784 |
SKBR3 |
| -0.202496 |
1.758981e-10 |
975 |
PF431396 |
LSM-1116 |
|
0.37uM |
24h |
LINCSCP_144667 |
LINCSCP_144667 |
MDAMB231 |
| -0.20249 |
1.761085e-10 |
975 |
Sildenafil |
LSM-3797 |
PDE5A |
10uM |
24h |
LINCSCP_32933 |
LINCSCP_32933 |
MCF7 |
| -0.202488 |
1.761701e-10 |
975 |
AZD-8055 |
LSM-1007 |
MTOR |
0.12uM |
24h |
LINCSCP_145284 |
LINCSCP_145284 |
MDAMB231 |
| -0.202478 |
1.765456e-10 |
975 |
Itrazole |
LSM-5032 |
|
10uM |
6h |
LINCSCP_257259 |
LINCSCP_257259 |
NCIH508 |
| -0.202477 |
1.765860e-10 |
975 |
Mecamylamine |
LSM-4990 |
CHRNA2|CHRNA3|CHRNB4 |
10uM |
24h |
LINCSCP_102292 |
LINCSCP_102292 |
HELA |
| -0.202475 |
1.766533e-10 |
975 |
BRD-K72853990-066-01-3 |
LSM-5805 |
ADRA2A|ADRA2B|ADRA2C|DRD1|DRD2|DRD3|DRD4|DRD5|HTR1A|HTR1B|HTR1D|HTR2A|HTR2B|HTR2C |
10uM |
24h |
LINCSCP_243541 |
LINCSCP_243541 |
MCF7 |
| 0.202456 |
1.773814e-10 |
975 |
BRD-K97829610 |
LSM-14442 |
|
5uM |
24h |
LINCSCP_62193 |
LINCSCP_62193 |
VCAP |
| -0.202445 |
1.777835e-10 |
975 |
GSK 1059615 |
LSM-42799 |
PIK3CA|PIK3CB|PIK3CD|PIK3CG |
10uM |
24h |
LINCSCP_131922 |
LINCSCP_131922 |
MCF7 |
| -0.202443 |
1.778680e-10 |
975 |
CHEMBL1551506 |
LSM-2315 |
|
10uM |
24h |
LINCSCP_31338 |
LINCSCP_31338 |
MCF7 |
| -0.202433 |
1.782114e-10 |
975 |
PD-0325901 |
LSM-1101 |
MAP2K1|MAP2K2 |
0.12uM |
24h |
LINCSCP_144615 |
LINCSCP_144615 |
MDAMB231 |
| -0.202429 |
1.783939e-10 |
975 |
SCHEMBL5945809 |
LSM-2339 |
HTR2A |
10uM |
24h |
LINCSCP_42852 |
LINCSCP_42852 |
NPC |
| 0.202423 |
1.786050e-10 |
975 |
Meclofenamic acid |
LSM-3108 |
ALOX5|PTGS1|PTGS2 |
10uM |
6h |
LINCSCP_34388 |
LINCSCP_34388 |
MCF7 |
| -0.202422 |
1.786331e-10 |
975 |
Prosteride |
LSM-1842 |
SRD5A1|SRD5A2 |
0.12uM |
24h |
LINCSCP_173139 |
LINCSCP_173139 |
YAPC |
| 0.202406 |
1.792343e-10 |
975 |
K-115 |
LSM-45986 |
|
3.33uM |
24h |
LINCSCP_76529 |
LINCSCP_76529 |
A375 |
| 0.202395 |
1.796523e-10 |
975 |
SCHEMBL618594 |
LSM-1070 |
|
3.33uM |
24h |
LINCSCP_86871 |
LINCSCP_86871 |
CD34 |
| -0.202389 |
1.798721e-10 |
975 |
Milciclib (PHA-848125) |
LSM-45577 |
CDK1|CDK2|CDK4|NTRK1 |
10uM |
24h |
LINCSCP_105999 |
LINCSCP_105999 |
HELA |
| -0.202348 |
1.814286e-10 |
975 |
Mccg |
LSM-37073 |
|
10uM |
24h |
LINCSCP_43237 |
LINCSCP_43237 |
NPC |
| 0.202347 |
1.814744e-10 |
975 |
MLS003568140 |
LSM-2084 |
|
10uM |
6h |
LINCSCP_268325 |
LINCSCP_268325 |
PC3 |
| -0.202344 |
1.815877e-10 |
975 |
Mibefradil |
LSM-2192 |
CACNA1C|CACNA1G|CACNA1H|CACNA1I |
10uM |
24h |
LINCSCP_52725 |
LINCSCP_52725 |
SKB |
| 0.202337 |
1.818697e-10 |
975 |
XAV 939 |
LSM-5303 |
TNKS|TNKS2 |
0.01uM |
6h |
LINCSCP_250873 |
LINCSCP_250873 |
MCF7 |
| 0.202333 |
1.819979e-10 |
975 |
BRD-K71182858 |
LSM-12774 |
|
5uM |
24h |
LINCSCP_63895 |
LINCSCP_63895 |
VCAP |
| -0.20232 |
1.825225e-10 |
975 |
1166227-08-2 |
LSM-1204 |
|
10uM |
24h |
LINCSCP_113701 |
LINCSCP_113701 |
HME1 |
| 0.202296 |
1.834443e-10 |
975 |
L 655240 |
LSM-4003 |
|
10uM |
24h |
LINCSCP_92176 |
LINCSCP_92176 |
HA1E |
| 0.202291 |
1.836122e-10 |
975 |
TL Aurora 09 |
LSM-45304 |
|
10uM |
6h |
LINCSCP_49747 |
LINCSCP_49747 |
PC3 |
| 0.202267 |
1.845626e-10 |
975 |
Imatinib |
LSM-1023 |
ABL1|BCR|CSF1R|KIT|PDGFRA|PDGFRB |
10uM |
3h |
LINCSCP_130374 |
LINCSCP_130374 |
LNCAP |
| 0.202261 |
1.847787e-10 |
975 |
BRD-K65904652 |
LSM-40871 |
|
10uM |
6h |
LINCSCP_59372 |
LINCSCP_59372 |
VCAP |
| -0.202257 |
1.849310e-10 |
975 |
MLS001065858 |
LSM-3606 |
|
10uM |
24h |
LINCSCP_238410 |
LINCSCP_238410 |
MCF7 |
| -0.202215 |
1.865689e-10 |
975 |
BRD-K13079805 |
LSM-9211 |
|
5uM |
24h |
LINCSCP_27649 |
LINCSCP_27649 |
HT29 |
| -0.202214 |
1.866312e-10 |
975 |
CHEMBL2360495 |
LSM-6811 |
|
10uM |
6h |
LINCSCP_27241 |
LINCSCP_27241 |
HT29 |
| 0.202201 |
1.871382e-10 |
975 |
BRD-K95551268 |
LSM-42453 |
|
5uM |
24h |
LINCSCP_64342 |
LINCSCP_64342 |
VCAP |
| -0.202192 |
1.874688e-10 |
975 |
Adenosine |
LSM-28568 |
ADORA1|ADORA2A|ADORA2B|ADORA3 |
1.11uM |
24h |
LINCSCP_75049 |
LINCSCP_75049 |
A375 |
| -0.202165 |
1.885383e-10 |
975 |
Cytochalasin B |
LSM-43278 |
ACTB |
10uM |
6h |
LINCSCP_15574 |
LINCSCP_15574 |
HA1E |
| 0.202127 |
1.900636e-10 |
975 |
Ischemin |
LSM-6336 |
|
1.11uM |
24h |
LINCSCP_133897 |
LINCSCP_133897 |
MCF7 |
| 0.202124 |
1.901821e-10 |
975 |
BRD-K75633187 |
LSM-13054 |
|
5uM |
24h |
LINCSCP_63525 |
LINCSCP_63525 |
VCAP |
| 0.202123 |
1.902322e-10 |
975 |
Tetrahydrobiopterin |
LSM-5120 |
PAH|TH |
10uM |
24h |
LINCSCP_59438 |
LINCSCP_59438 |
VCAP |
| -0.202084 |
1.917807e-10 |
975 |
BRD-K89824424 |
LSM-42166 |
|
10uM |
24h |
LINCSCP_28397 |
LINCSCP_28397 |
HT29 |
| -0.202084 |
1.917883e-10 |
975 |
CI-1040 |
LSM-1048 |
MAP2K1|MAP2K2 |
3.33uM |
24h |
LINCSCP_138181 |
LINCSCP_138181 |
MCF7 |
| -0.202082 |
1.918574e-10 |
975 |
MG-132 |
LSM-1107 |
PSMB1 |
20uM |
24h |
LINCSCP_72393 |
LINCSCP_72393 |
A375 |
| -0.202075 |
1.921313e-10 |
975 |
BRD-K04986062 |
LSM-45341 |
|
1uM |
24h |
LINCSCP_222126 |
LINCSCP_222126 |
HL60 |
| 0.202073 |
1.922325e-10 |
975 |
BRD-K76223260 |
LSM-13084 |
|
5uM |
24h |
LINCSCP_61819 |
LINCSCP_61819 |
VCAP |
| -0.20207 |
1.923421e-10 |
975 |
CI-1040 |
LSM-1048 |
MAP2K1|MAP2K2 |
10uM |
24h |
LINCSCP_99600 |
LINCSCP_99600 |
HCC515 |
| 0.202068 |
1.924027e-10 |
975 |
Yohimbine |
LSM-2779 |
ADRA2A|ADRA2B|ADRA2C|HTR1A|HTR1B|HTR1D|HTR2B |
0.04uM |
24h |
LINCSCP_71998 |
LINCSCP_71998 |
A375 |
| -0.202065 |
1.925333e-10 |
975 |
SPECTRUM_000011 |
LSM-1767 |
|
1.11uM |
24h |
LINCSCP_126168 |
LINCSCP_126168 |
HT29 |
| 0.202064 |
1.925668e-10 |
975 |
FR-180204 |
LSM-42790 |
MAPK1|MAPK3 |
1uM |
24h |
LINCSCP_36828 |
LINCSCP_36828 |
MCF7 |
| -0.202061 |
1.927175e-10 |
975 |
SCHEMBL17857056 |
LSM-5545 |
|
1uM |
24h |
LINCSCP_11702 |
LINCSCP_11702 |
BT20 |
| -0.202046 |
1.933071e-10 |
975 |
PI-103 |
LSM-1126 |
MTOR|PIK3CA|PIK3CB|PIK3CD|PIK3CG |
10uM |
6h |
LINCSCP_289092 |
LINCSCP_289092 |
U937 |
| 0.202039 |
1.935868e-10 |
975 |
BRD-K26653603 |
LSM-8179 |
|
5uM |
24h |
LINCSCP_60744 |
LINCSCP_60744 |
VCAP |
| -0.202039 |
1.935912e-10 |
975 |
CHEMBL2355034 |
LSM-37650 |
|
10uM |
6h |
LINCSCP_33979 |
LINCSCP_33979 |
MCF7 |
| -0.202032 |
1.938972e-10 |
975 |
UNC1215 |
LSM-6338 |
|
3.33uM |
24h |
LINCSCP_86977 |
LINCSCP_86977 |
CD34 |
| 0.202028 |
1.940356e-10 |
975 |
BRD-K83920942 |
LSM-13558 |
|
5uM |
6h |
LINCSCP_62419 |
LINCSCP_62419 |
VCAP |
| -0.202026 |
1.941278e-10 |
975 |
Temoporfin |
LSM-45995 |
|
0.12uM |
24h |
LINCSCP_155239 |
LINCSCP_155239 |
PC3 |
| -0.202022 |
1.942738e-10 |
975 |
Heat |
LSM-1404 |
ADRA1A |
10uM |
6h |
LINCSCP_192859 |
LINCSCP_192859 |
A549 |
| -0.202021 |
1.943297e-10 |
975 |
Tozasertib |
LSM-1021 |
ABL1|AURKA|AURKB|AURKC|BCR|FLT3|JAK2 |
10uM |
3h |
LINCSCP_144951 |
LINCSCP_144951 |
MDAMB231 |
| 0.202012 |
1.946777e-10 |
975 |
AC1Q6JJ5 |
LSM-6192 |
TOP2A |
0.1uM |
6h |
LINCSCP_51061 |
LINCSCP_51061 |
RMUGS |
| -0.201994 |
1.954253e-10 |
975 |
OTSSP167 |
LSM-6340 |
|
10uM |
24h |
LINCSCP_140213 |
LINCSCP_140213 |
MCF7 |
| 0.201985 |
1.957925e-10 |
975 |
SA-243929 |
LSM-37535 |
|
1uM |
24h |
LINCSCP_253446 |
LINCSCP_253446 |
MCF7 |
| 0.201952 |
1.971726e-10 |
975 |
QL47 |
LSM-6019 |
BMX|BTK |
0.5uM |
6h |
LINCSCP_51768 |
LINCSCP_51768 |
SKBR3 |
| 0.201943 |
1.975449e-10 |
975 |
Topiramate |
LSM-5435 |
CA2|CA4|GABRA1|GABRA2|GABRA3|GABRA4|GABRA5|GABRA6|GABRB1|GABRB2|GABRB3|GABRD|GABRE|GABRG1|GABRG2|GABRG3|GABRP|GABRQ|GRIA1|GRIA2|GRIA3|GRIA4|GRIK1|GRIK2|GRIK3|GRIK4|GRIK5|SCN10A|SCN11A|SCN1A|SCN2A|SCN3A|SCN4A|SCN5A|SCN7A|SCN8A|SCN9A |
1.11uM |
24h |
LINCSCP_101401 |
LINCSCP_101401 |
HELA |
| -0.201938 |
1.977406e-10 |
975 |
BRD-K43579410 |
LSM-39667 |
|
0.5uM |
24h |
LINCSCP_312473 |
LINCSCP_312473 |
VCAP |
| -0.201929 |
1.981253e-10 |
975 |
Alvocidib |
LSM-1011 |
CDK1|CDK2|CDK4|CDK5|CDK6|CDK7|CDK8|CDK9|EGFR|PYGM |
0.001uM |
24h |
LINCSCP_9747 |
LINCSCP_9747 |
A549 |
| 0.201915 |
1.986839e-10 |
975 |
BRD-A15501135 |
LSM-45357 |
|
30uM |
24h |
LINCSCP_309961 |
LINCSCP_309961 |
VCAP |
| -0.201893 |
1.996107e-10 |
975 |
Meclofenamic acid |
LSM-3108 |
ALOX5|PTGS1|PTGS2 |
10uM |
24h |
LINCSCP_107927 |
LINCSCP_107927 |
HELA |
| -0.201887 |
1.998569e-10 |
975 |
Moroxydine |
LSM-5675 |
|
10uM |
24h |
LINCSCP_34298 |
LINCSCP_34298 |
MCF7 |
| 0.20185 |
2.014069e-10 |
975 |
Fluoxetine |
LSM-1449 |
SLC6A4 |
10uM |
6h |
LINCSCP_57849 |
LINCSCP_57849 |
VCAP |
| -0.201847 |
2.015633e-10 |
975 |
Tolmetin |
LSM-3852 |
PTGS1|PTGS2 |
10uM |
24h |
LINCSCP_262203 |
LINCSCP_262203 |
NPC |
| -0.201837 |
2.019647e-10 |
975 |
R-7128 |
LSM-45627 |
|
10uM |
24h |
LINCSCP_160748 |
LINCSCP_160748 |
PC3 |
| 0.201832 |
2.021683e-10 |
975 |
Resminostat |
LSM-45663 |
|
0.12uM |
24h |
LINCSCP_169228 |
LINCSCP_169228 |
YAPC |
| -0.201832 |
2.021918e-10 |
975 |
1268524-70-4 |
LSM-6332 |
|
10uM |
24h |
LINCSCP_164641 |
LINCSCP_164641 |
SKL.C |
| 0.201818 |
2.027524e-10 |
975 |
Nateglinide |
LSM-5555 |
ABCC8|KCNJ11 |
0.37uM |
24h |
LINCSCP_139173 |
LINCSCP_139173 |
MCF7 |
| -0.201814 |
2.029459e-10 |
975 |
Apilimod |
LSM-45286 |
|
3.33uM |
24h |
LINCSCP_157236 |
LINCSCP_157236 |
PC3 |
| 0.201813 |
2.029634e-10 |
975 |
Plerixafor |
LSM-36826 |
CXCR4 |
10uM |
6h |
LINCSCP_53272 |
LINCSCP_53272 |
SKM1 |
| 0.201786 |
2.041516e-10 |
975 |
Gefitinib |
LSM-1098 |
EGFR |
0.04uM |
3h |
LINCSCP_133198 |
LINCSCP_133198 |
MCF7 |
| -0.201766 |
2.049798e-10 |
975 |
AC1NUE3V |
LSM-43141 |
DUSP1|DUSP6 |
10uM |
24h |
LINCSCP_37842 |
LINCSCP_37842 |
MCF7 |
| -0.201758 |
2.053347e-10 |
975 |
Mitoxantrone |
LSM-2481 |
TOP2A |
3.33uM |
24h |
LINCSCP_136484 |
LINCSCP_136484 |
MCF7 |
| 0.201753 |
2.055329e-10 |
975 |
Imatinib |
LSM-1023 |
ABL1|BCR|CSF1R|KIT|PDGFRA|PDGFRB |
0.04uM |
3h |
LINCSCP_131789 |
LINCSCP_131789 |
MCF10A |
| -0.201746 |
2.058675e-10 |
975 |
BRD-K49477330 |
LSM-44782 |
|
10uM |
24h |
LINCSCP_35330 |
LINCSCP_35330 |
MCF7 |
| 0.201723 |
2.068570e-10 |
975 |
Ammonium Glycyrrhizinate |
LSM-46003 |
|
3.33uM |
24h |
LINCSCP_138061 |
LINCSCP_138061 |
MCF7 |
| -0.2017 |
2.078395e-10 |
975 |
AT-7519 |
LSM-1004 |
CDK1|CDK10|CDK11B|CDK12|CDK13|CDK14|CDK15|CDK16|CDK17|CDK18|CDK19|CDK2|CDK20|CDK3|CDK4|CDK5|CDK6|CDK7|CDK8|CDK9 |
0.04uM |
24h |
LINCSCP_88127 |
LINCSCP_88127 |
HA1E |
| -0.201686 |
2.084607e-10 |
975 |
GSK 525762A |
LSM-6334 |
|
1.11uM |
24h |
LINCSCP_128849 |
LINCSCP_128849 |
HUVEC |
| 0.201678 |
2.088078e-10 |
975 |
Probenecid |
LSM-4140 |
SLC22A11|SLC22A6|SLC22A8 |
10uM |
24h |
LINCSCP_244090 |
LINCSCP_244090 |
MCF7 |
| 0.201676 |
2.089104e-10 |
975 |
ICI 192,605 |
LSM-45545 |
|
1.11uM |
24h |
LINCSCP_139772 |
LINCSCP_139772 |
MCF7 |
| -0.201672 |
2.090726e-10 |
975 |
CGP 60474 |
LSM-1025 |
CDK1 |
0.04uM |
24h |
LINCSCP_112668 |
LINCSCP_112668 |
HEPG2 |
| 0.201665 |
2.093717e-10 |
975 |
BRD-K67661368 |
LSM-12547 |
|
5uM |
24h |
LINCSCP_62028 |
LINCSCP_62028 |
VCAP |
| -0.201665 |
2.093794e-10 |
975 |
17-DMAG (Alvespimycin) HCl |
LSM-46133 |
|
0.37uM |
24h |
LINCSCP_71738 |
LINCSCP_71738 |
A375 |
| 0.201655 |
2.097959e-10 |
975 |
Lapatinib |
LSM-1051 |
EGFR|ERBB2 |
10uM |
24h |
LINCSCP_81645 |
LINCSCP_81645 |
A549 |
| -0.201644 |
2.102915e-10 |
975 |
Methylnaltrexone (Bromide) |
LSM-45638 |
|
0.37uM |
24h |
LINCSCP_135419 |
LINCSCP_135419 |
MCF7 |
| -0.201634 |
2.107241e-10 |
975 |
179324-69-7 |
LSM-6281 |
ADRM1|PSMA1|PSMA2|PSMA3|PSMA4|PSMA5|PSMA6|PSMA7|PSMA8|PSMB1|PSMB10|PSMB11|PSMB2|PSMB3|PSMB4|PSMB5|PSMB6|PSMB7|PSMB8|PSMB9|PSMC1|PSMC2|PSMC3|PSMC4|PSMC5|PSMC6|PSMD1|PSMD11|PSMD12|PSMD13|PSMD14|PSMD2|PSMD3|PSMD4|PSMD6|PSMD7|PSMD8|SEM1 |
20uM |
24h |
LINCSCP_71064 |
LINCSCP_71064 |
A375 |
| 0.201616 |
2.115169e-10 |
975 |
ZSTK 474 |
LSM-1053 |
PIK3CG |
0.12uM |
3h |
LINCSCP_133179 |
LINCSCP_133179 |
MCF7 |
| -0.20161 |
2.117751e-10 |
975 |
BRD-A41986761 |
LSM-45957 |
|
0.04uM |
24h |
LINCSCP_135199 |
LINCSCP_135199 |
MCF7 |
| 0.201586 |
2.128679e-10 |
975 |
CHEMBL2132289 |
LSM-1044 |
RPS6KA3 |
10uM |
6h |
LINCSCP_39185 |
LINCSCP_39185 |
MDAMB231 |
| -0.201579 |
2.131593e-10 |
975 |
CI-1040 |
LSM-1048 |
MAP2K1|MAP2K2 |
10uM |
24h |
LINCSCP_104807 |
LINCSCP_104807 |
HELA |
| -0.201565 |
2.138088e-10 |
975 |
Tetrahydrouridine |
LSM-45757 |
|
0.12uM |
24h |
LINCSCP_160236 |
LINCSCP_160236 |
PC3 |
| -0.201551 |
2.144033e-10 |
975 |
Mizolastine |
LSM-5377 |
HRH1 |
0.12uM |
24h |
LINCSCP_119933 |
LINCSCP_119933 |
HT29 |
| 0.201547 |
2.146156e-10 |
975 |
BRD-K38459107 |
LSM-39385 |
|
5uM |
6h |
LINCSCP_64397 |
LINCSCP_64397 |
VCAP |
| -0.201542 |
2.148114e-10 |
975 |
CHEMBL1868011 |
LSM-6088 |
CASP3 |
0.5uM |
6h |
LINCSCP_37089 |
LINCSCP_37089 |
MCF7 |
| -0.201532 |
2.152940e-10 |
975 |
GSK 1059615 |
LSM-42799 |
PIK3CA|PIK3CB|PIK3CD|PIK3CG |
3.33uM |
24h |
LINCSCP_131923 |
LINCSCP_131923 |
MCF7 |
| -0.201514 |
2.161116e-10 |
975 |
Bambuterol |
LSM-4346 |
ADRB2 |
10uM |
24h |
LINCSCP_34240 |
LINCSCP_34240 |
MCF7 |
| 0.201511 |
2.162281e-10 |
975 |
Cis-N,N-Dimethyl-9-(3-(1-Piperazinyl)Propylidene)Thioxanthene-2-Sulfonamide |
LSM-43212 |
HTR2A |
10uM |
24h |
LINCSCP_5410 |
LINCSCP_5410 |
A549 |
| -0.20151 |
2.162672e-10 |
975 |
MLS002264428 |
LSM-4143 |
|
10uM |
6h |
LINCSCP_1659 |
LINCSCP_1659 |
A375 |
| -0.201504 |
2.165365e-10 |
975 |
MLS002264411 |
LSM-1873 |
|
10uM |
24h |
LINCSCP_5363 |
LINCSCP_5363 |
A549 |
| -0.201501 |
2.166897e-10 |
975 |
BRD-A25736793 |
LSM-43054 |
MTOR |
1.11uM |
24h |
LINCSCP_147609 |
LINCSCP_147609 |
NPC.CAS9 |
| -0.201491 |
2.171109e-10 |
975 |
BRD-A08662020 |
LSM-45607 |
|
0.12uM |
24h |
LINCSCP_76502 |
LINCSCP_76502 |
A375 |
| -0.201484 |
2.174558e-10 |
975 |
Pimasertib |
LSM-5946 |
MAP2K1|MAP2K2 |
1.11uM |
24h |
LINCSCP_73832 |
LINCSCP_73832 |
A375 |
| -0.201483 |
2.175040e-10 |
975 |
Lomatin |
LSM-1376 |
|
10uM |
6h |
LINCSCP_25317 |
LINCSCP_25317 |
HT29 |
| -0.201467 |
2.182292e-10 |
975 |
179324-69-7 |
LSM-6281 |
ADRM1|PSMA1|PSMA2|PSMA3|PSMA4|PSMA5|PSMA6|PSMA7|PSMA8|PSMB1|PSMB10|PSMB11|PSMB2|PSMB3|PSMB4|PSMB5|PSMB6|PSMB7|PSMB8|PSMB9|PSMC1|PSMC2|PSMC3|PSMC4|PSMC5|PSMC6|PSMD1|PSMD11|PSMD12|PSMD13|PSMD14|PSMD2|PSMD3|PSMD4|PSMD6|PSMD7|PSMD8|SEM1 |
20uM |
24h |
LINCSCP_71063 |
LINCSCP_71063 |
A375 |
| 0.201439 |
2.195015e-10 |
975 |
Loxoprofen |
LSM-5054 |
|
0.12uM |
24h |
LINCSCP_105739 |
LINCSCP_105739 |
HELA |
| 0.201422 |
2.202884e-10 |
975 |
BRD-K01608965 |
LSM-8538 |
|
5uM |
24h |
LINCSCP_63049 |
LINCSCP_63049 |
VCAP |
| 0.201415 |
2.206158e-10 |
975 |
Sulfadoxine |
LSM-5657 |
|
3.33uM |
24h |
LINCSCP_73404 |
LINCSCP_73404 |
A375 |
| -0.201414 |
2.206635e-10 |
975 |
BRD-K73434853 |
LSM-41258 |
|
10uM |
24h |
LINCSCP_312527 |
LINCSCP_312527 |
VCAP |
| -0.201413 |
2.206876e-10 |
975 |
MLS003178531 |
LSM-3273 |
|
10uM |
24h |
LINCSCP_1409 |
LINCSCP_1409 |
A375 |
| -0.201407 |
2.209637e-10 |
975 |
Anastrozole |
LSM-5631 |
CYP19A1 |
3.33uM |
24h |
LINCSCP_91649 |
LINCSCP_91649 |
HA1E |
| -0.201404 |
2.211364e-10 |
975 |
PRESTWICK3_000121 |
LSM-1670 |
ADRA2A|ADRA2B|ADRA2C|DRD1|DRD2|DRD3|DRD4|DRD5|HTR1A|HTR1B|HTR1D|HTR2A|HTR2B|HTR2C |
10uM |
6h |
LINCSCP_443 |
LINCSCP_443 |
A375 |
| -0.201403 |
2.211651e-10 |
975 |
GSK 1059615 |
LSM-42799 |
PIK3CA|PIK3CB|PIK3CD|PIK3CG |
0.04uM |
24h |
LINCSCP_69050 |
LINCSCP_69050 |
A375 |
| -0.201399 |
2.213318e-10 |
975 |
Adarotene |
LSM-45863 |
|
0.37uM |
24h |
LINCSCP_121886 |
LINCSCP_121886 |
HT29 |
| -0.201388 |
2.218700e-10 |
975 |
CC-401 |
LSM-1186 |
|
10uM |
24h |
LINCSCP_152401 |
LINCSCP_152401 |
PC3 |
| -0.201381 |
2.221690e-10 |
975 |
MLS003128690 |
LSM-11578 |
|
5uM |
24h |
LINCSCP_64291 |
LINCSCP_64291 |
VCAP |
| 0.201373 |
2.225602e-10 |
975 |
Taranabant |
LSM-45803 |
CNR1 |
0.04uM |
24h |
LINCSCP_74212 |
LINCSCP_74212 |
A375 |
| -0.201365 |
2.229201e-10 |
975 |
Atomoxetine |
LSM-2452 |
SLC6A2|SLC6A3|SLC6A4 |
1.11uM |
24h |
LINCSCP_153878 |
LINCSCP_153878 |
PC3 |
| -0.201361 |
2.231106e-10 |
975 |
PD-0325901 |
LSM-1101 |
MAP2K1|MAP2K2 |
10uM |
24h |
LINCSCP_99792 |
LINCSCP_99792 |
HCC515 |
| -0.201357 |
2.233219e-10 |
975 |
Mebendazole |
LSM-3749 |
|
3.33uM |
24h |
LINCSCP_123130 |
LINCSCP_123130 |
HT29 |
| -0.201353 |
2.234753e-10 |
975 |
PNU-74654 |
LSM-44945 |
CTNNB1|TCF4 |
80uM |
6h |
LINCSCP_12538 |
LINCSCP_12538 |
CL34 |
| -0.201338 |
2.242005e-10 |
975 |
Fenbendazole |
LSM-3134 |
TUBB |
10uM |
24h |
LINCSCP_42901 |
LINCSCP_42901 |
NPC |
| -0.201326 |
2.247746e-10 |
975 |
BRD-A28746609 |
LSM-1102 |
NR1I2|TUBB |
3.33uM |
24h |
LINCSCP_120966 |
LINCSCP_120966 |
HT29 |
| 0.201321 |
2.249864e-10 |
975 |
Latanoprost |
LSM-43170 |
PTGFR |
10uM |
24h |
LINCSCP_154434 |
LINCSCP_154434 |
PC3 |
| 0.201305 |
2.257348e-10 |
975 |
BRD-K73408523 |
LSM-12925 |
|
10uM |
24h |
LINCSCP_37041 |
LINCSCP_37041 |
MCF7 |
| -0.201294 |
2.262580e-10 |
975 |
MLS002699429 |
LSM-44942 |
|
10uM |
6h |
LINCSCP_15875 |
LINCSCP_15875 |
HA1E |
| 0.201267 |
2.275170e-10 |
975 |
16Beta-hydroxydisitoxigenin |
LSM-1432 |
ATP1A1 |
10uM |
6h |
LINCSCP_44607 |
LINCSCP_44607 |
PC3 |
| 0.201253 |
2.282103e-10 |
975 |
Lapatinib |
LSM-1051 |
EGFR|ERBB2 |
0.37uM |
24h |
LINCSCP_130005 |
LINCSCP_130005 |
LNCAP |
| 0.201244 |
2.286368e-10 |
975 |
BRD-K43931839 |
LSM-11109 |
|
5uM |
24h |
LINCSCP_63223 |
LINCSCP_63223 |
VCAP |
| -0.201243 |
2.286806e-10 |
975 |
Procaine |
LSM-5396 |
HTR3A|SCN10A|SCN11A|SCN1A|SCN2A|SCN3A|SCN4A|SCN5A|SCN7A|SCN8A|SCN9A |
10uM |
24h |
LINCSCP_102423 |
LINCSCP_102423 |
HELA |
| -0.20123 |
2.292994e-10 |
975 |
SKF96365 |
LSM-1766 |
CYP3A4|TRPC1 |
10uM |
24h |
LINCSCP_37853 |
LINCSCP_37853 |
MCF7 |
| -0.201225 |
2.295520e-10 |
975 |
NMS-1286937 |
LSM-45818 |
|
1.11uM |
24h |
LINCSCP_160072 |
LINCSCP_160072 |
PC3 |
| -0.201221 |
2.297259e-10 |
975 |
Mubritinib (TAK 165) |
LSM-45710 |
ERBB2 |
0.04uM |
24h |
LINCSCP_154523 |
LINCSCP_154523 |
PC3 |
| -0.201209 |
2.303317e-10 |
975 |
Cefoperazone |
LSM-15520 |
|
0.04uM |
24h |
LINCSCP_138653 |
LINCSCP_138653 |
MCF7 |
| -0.201184 |
2.315206e-10 |
975 |
13-Methyl-7-[9-(4,4,5,5,5-pentafluoropentylsulfinyl)nonyl]-6,7,8,9,11,12,14,15,16,17-decahydrocyclopenta[a]phenanthrene-3,17-diol |
LSM-1895 |
ESR1 |
10uM |
24h |
LINCSCP_18829 |
LINCSCP_18829 |
HCC515 |
| -0.201165 |
2.324427e-10 |
975 |
LY2874455 |
LSM-45659 |
|
10uM |
24h |
LINCSCP_101693 |
LINCSCP_101693 |
HELA |
| -0.201156 |
2.328926e-10 |
975 |
Aloisine A |
LSM-4110 |
CDK2 |
10uM |
24h |
LINCSCP_33147 |
LINCSCP_33147 |
MCF7 |
| -0.201134 |
2.339538e-10 |
975 |
WH-4-025 |
LSM-44937 |
|
0.37uM |
24h |
LINCSCP_144888 |
LINCSCP_144888 |
MDAMB231 |
| 0.201125 |
2.344073e-10 |
975 |
BRD-K52797126 |
LSM-7532 |
|
5uM |
24h |
LINCSCP_60200 |
LINCSCP_60200 |
VCAP |
| 0.201115 |
2.348962e-10 |
975 |
Tyrphostin A9 |
LSM-4617 |
|
10uM |
24h |
LINCSCP_11034 |
LINCSCP_11034 |
ASC |
| -0.201103 |
2.354402e-10 |
975 |
Wortmannin |
LSM-3947 |
PIK3CA|PIK3CG|PLK1 |
0.5uM |
24h |
LINCSCP_264405 |
LINCSCP_264405 |
PC3 |
| -0.201091 |
2.360583e-10 |
975 |
KW-2449 |
LSM-42803 |
ABL1|AURKA|AURKB|FLT3 |
10uM |
24h |
LINCSCP_149658 |
LINCSCP_149658 |
NPC.TAK |
| 0.201084 |
2.363822e-10 |
975 |
SCHEMBL6874948 |
LSM-5674 |
LCK |
0.37uM |
3h |
LINCSCP_113346 |
LINCSCP_113346 |
HME1 |
| -0.201078 |
2.367043e-10 |
975 |
CGS-15943 |
LSM-3076 |
ADORA1|ADORA2A|ADORA2B |
10uM |
24h |
LINCSCP_67591 |
LINCSCP_67591 |
MCF7 |
| 0.201066 |
2.372888e-10 |
975 |
PLX-4720 |
LSM-1049 |
BRAF |
0.12uM |
24h |
LINCSCP_130647 |
LINCSCP_130647 |
MCF10A |
| -0.201059 |
2.376561e-10 |
975 |
Withaferin A |
LSM-6685 |
IKBKB|NAMPT |
10uM |
24h |
LINCSCP_68541 |
LINCSCP_68541 |
VCAP |
| 0.201054 |
2.378745e-10 |
975 |
PF-04217903 |
LSM-1166 |
MET |
10uM |
24h |
LINCSCP_84136 |
LINCSCP_84136 |
ASC |
| -0.201047 |
2.382350e-10 |
975 |
BRD-K72429558 |
LSM-41196 |
|
10uM |
24h |
LINCSCP_42190 |
LINCSCP_42190 |
NPC |
| -0.201025 |
2.393462e-10 |
975 |
Methixene |
LSM-1467 |
CHRM1|CHRM5|HTR2C |
1.11uM |
24h |
LINCSCP_135394 |
LINCSCP_135394 |
MCF7 |
| -0.201022 |
2.394798e-10 |
975 |
Ifosfamide |
LSM-5118 |
CYP2A6|CYP2B6|CYP2C18|CYP2C19|CYP2C8|CYP2C9|CYP3A4|CYP3A5|CYP3A7|PTGS1 |
1.11uM |
24h |
LINCSCP_124369 |
LINCSCP_124369 |
HT29 |
| -0.201022 |
2.394984e-10 |
975 |
BRD-K30645599 |
LSM-38945 |
|
30uM |
24h |
LINCSCP_310001 |
LINCSCP_310001 |
VCAP |
| -0.201006 |
2.402643e-10 |
975 |
179324-69-7 |
LSM-6281 |
ADRM1|PSMA1|PSMA2|PSMA3|PSMA4|PSMA5|PSMA6|PSMA7|PSMA8|PSMB1|PSMB10|PSMB11|PSMB2|PSMB3|PSMB4|PSMB5|PSMB6|PSMB7|PSMB8|PSMB9|PSMC1|PSMC2|PSMC3|PSMC4|PSMC5|PSMC6|PSMD1|PSMD11|PSMD12|PSMD13|PSMD14|PSMD2|PSMD3|PSMD4|PSMD6|PSMD7|PSMD8|SEM1 |
20uM |
24h |
LINCSCP_71061 |
LINCSCP_71061 |
A375 |
| -0.20099 |
2.410987e-10 |
975 |
CHEMBL607856 |
LSM-3321 |
|
10uM |
6h |
LINCSCP_43777 |
LINCSCP_43777 |
OV7 |
| -0.200987 |
2.412501e-10 |
975 |
Ondansetron |
LSM-1375 |
HTR3A |
10uM |
6h |
LINCSCP_190132 |
LINCSCP_190132 |
A549 |
| -0.200968 |
2.421859e-10 |
975 |
ZINC02419385 |
LSM-4849 |
|
1uM |
6h |
LINCSCP_254400 |
LINCSCP_254400 |
MCF7 |
| -0.200968 |
2.422084e-10 |
975 |
AT-7519 |
LSM-1004 |
CDK1|CDK10|CDK11B|CDK12|CDK13|CDK14|CDK15|CDK16|CDK17|CDK18|CDK19|CDK2|CDK20|CDK3|CDK4|CDK5|CDK6|CDK7|CDK8|CDK9 |
10uM |
24h |
LINCSCP_137904 |
LINCSCP_137904 |
MCF7 |
| 0.200954 |
2.428916e-10 |
975 |
Entinostat |
LSM-4811 |
HDAC1|HDAC10|HDAC11|HDAC2|HDAC3|HDAC4|HDAC5|HDAC6|HDAC7|HDAC8|HDAC9 |
0.37uM |
24h |
LINCSCP_164709 |
LINCSCP_164709 |
SKL.C |
| -0.200946 |
2.433004e-10 |
975 |
Gliclazide |
LSM-5096 |
ABCC8 |
1.11uM |
24h |
LINCSCP_171676 |
LINCSCP_171676 |
YAPC |
| 0.200942 |
2.435107e-10 |
975 |
Phenanthridone |
LSM-2229 |
PARP1 |
0.01uM |
6h |
LINCSCP_9554 |
LINCSCP_9554 |
A549 |
| -0.200931 |
2.440618e-10 |
975 |
Quizartinib |
LSM-1037 |
CSF1R|FLT3|KIT|PDGFRA|PDGFRB|RET |
10uM |
24h |
LINCSCP_148684 |
LINCSCP_148684 |
NPC |
| -0.200925 |
2.443488e-10 |
975 |
13-Hydroxy-8,14,19-trimethoxy-4,10,12,16-tetramethyl-3,20,22-trioxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18-pentaen-9-yl carbamate |
LSM-42815 |
HSP90AA1 |
0.04uM |
3h |
LINCSCP_85757 |
LINCSCP_85757 |
BT20 |
| 0.200914 |
2.449551e-10 |
975 |
Ingenol 3,20-dibenzoate |
LSM-4445 |
PRKCD|PRKCE |
0.001uM |
24h |
LINCSCP_9149 |
LINCSCP_9149 |
A549 |
| -0.200902 |
2.455515e-10 |
975 |
CAY10618 |
LSM-4946 |
NAMPT |
10uM |
24h |
LINCSCP_30646 |
LINCSCP_30646 |
MCF7 |
| -0.200891 |
2.461096e-10 |
975 |
SPECTRUM_001092 |
LSM-1337 |
NR3C1 |
10uM |
6h |
LINCSCP_406 |
LINCSCP_406 |
A375 |
| -0.200889 |
2.462071e-10 |
975 |
Targinine |
LSM-36418 |
|
0.12uM |
24h |
LINCSCP_157533 |
LINCSCP_157533 |
PC3 |
| -0.200888 |
2.462781e-10 |
975 |
QL-XI-92 |
LSM-42736 |
DDR1 |
10uM |
6h |
LINCSCP_47065 |
LINCSCP_47065 |
PC3 |
| 0.200885 |
2.464205e-10 |
975 |
Probucol |
LSM-3617 |
ABCA1 |
3.33uM |
24h |
LINCSCP_142692 |
LINCSCP_142692 |
MCF7 |
| -0.200883 |
2.465015e-10 |
975 |
MK 0893 |
LSM-45875 |
GCGR |
10uM |
24h |
LINCSCP_101615 |
LINCSCP_101615 |
HELA |
| -0.200868 |
2.472836e-10 |
975 |
Palbociclib |
LSM-1071 |
CCND1|CDK4|CDK6 |
10uM |
24h |
LINCSCP_85896 |
LINCSCP_85896 |
BT20 |
| -0.200867 |
2.473412e-10 |
975 |
PD-0325901 |
LSM-1101 |
MAP2K1|MAP2K2 |
1.11uM |
24h |
LINCSCP_83982 |
LINCSCP_83982 |
ASC.C |
| -0.200865 |
2.474539e-10 |
975 |
179324-69-7 |
LSM-6281 |
ADRM1|PSMA1|PSMA2|PSMA3|PSMA4|PSMA5|PSMA6|PSMA7|PSMA8|PSMB1|PSMB10|PSMB11|PSMB2|PSMB3|PSMB4|PSMB5|PSMB6|PSMB7|PSMB8|PSMB9|PSMC1|PSMC2|PSMC3|PSMC4|PSMC5|PSMC6|PSMD1|PSMD11|PSMD12|PSMD13|PSMD14|PSMD2|PSMD3|PSMD4|PSMD6|PSMD7|PSMD8|SEM1 |
20uM |
24h |
LINCSCP_134643 |
LINCSCP_134643 |
MCF7 |
| -0.200848 |
2.483444e-10 |
975 |
SMR000543856 |
LSM-2149 |
|
10uM |
6h |
LINCSCP_272218 |
LINCSCP_272218 |
PC3 |
| -0.200844 |
2.485407e-10 |
975 |
SR57227A |
LSM-2188 |
HTR3A |
3.33uM |
24h |
LINCSCP_167907 |
LINCSCP_167907 |
YAPC |
| -0.200843 |
2.485910e-10 |
975 |
Cytochalasin B |
LSM-43278 |
ACTB |
10uM |
24h |
LINCSCP_25505 |
LINCSCP_25505 |
HT29 |
| 0.200833 |
2.491148e-10 |
975 |
CHEMBL2333339 |
LSM-4809 |
|
10uM |
6h |
LINCSCP_22560 |
LINCSCP_22560 |
HEPG2 |
| -0.200817 |
2.499260e-10 |
975 |
2-(Ethylmercuriothio)benzoic acid |
LSM-5710 |
|
10uM |
24h |
LINCSCP_127300 |
LINCSCP_127300 |
HT29 |
| -0.200803 |
2.506454e-10 |
975 |
Ciglitazone |
LSM-1911 |
PPARG |
10uM |
24h |
LINCSCP_263798 |
LINCSCP_263798 |
NPC |
| -0.200799 |
2.508728e-10 |
975 |
Momelotinib |
LSM-1141 |
JAK1|JAK2 |
0.12uM |
24h |
LINCSCP_132178 |
LINCSCP_132178 |
MCF7 |
| -0.200791 |
2.512715e-10 |
975 |
AC1MGQL6 |
LSM-4334 |
|
10uM |
24h |
LINCSCP_42220 |
LINCSCP_42220 |
NPC |
| -0.200788 |
2.514450e-10 |
975 |
Ichthynone |
LSM-2615 |
|
3uM |
6h |
LINCSCP_28948 |
LINCSCP_28948 |
HUH7 |
| -0.200781 |
2.518268e-10 |
975 |
SMR001318078 |
LSM-1737 |
|
10uM |
6h |
LINCSCP_15832 |
LINCSCP_15832 |
HA1E |
| 0.200758 |
2.530287e-10 |
975 |
Dacarbazine |
LSM-5487 |
|
0.04uM |
24h |
LINCSCP_72016 |
LINCSCP_72016 |
A375 |
| -0.200751 |
2.534030e-10 |
975 |
AS-605240 |
LSM-42784 |
PIK3CG |
3.33uM |
3h |
LINCSCP_133212 |
LINCSCP_133212 |
MCF7 |
| 0.200743 |
2.538014e-10 |
975 |
LRRK2-IN-1 |
LSM-1086 |
LRRK2 |
0.37uM |
24h |
LINCSCP_81702 |
LINCSCP_81702 |
A549 |
| -0.200705 |
2.558135e-10 |
975 |
KUC103875 |
LSM-2801 |
|
10uM |
24h |
LINCSCP_177821 |
LINCSCP_177821 |
A375 |
| -0.200687 |
2.567754e-10 |
975 |
Dasatinib |
LSM-1020 |
ABL1|BCR|BLK|EPHA2|FGR|FRK|FYN|HCK|KIT|LCK|LYN|PDGFRB|SRC|SRMS|YES1 |
3.33uM |
3h |
LINCSCP_164007 |
LINCSCP_164007 |
SKBR3 |
| -0.200681 |
2.571193e-10 |
975 |
Febuxostat |
LSM-3064 |
XDH |
10uM |
24h |
LINCSCP_7605 |
LINCSCP_7605 |
A549 |
| -0.200679 |
2.572448e-10 |
975 |
CHEMBL2361787 |
LSM-13210 |
|
10uM |
24h |
LINCSCP_35247 |
LINCSCP_35247 |
MCF7 |
| -0.20067 |
2.577171e-10 |
975 |
Broad-Sai-424 |
LSM-45346 |
|
3.33uM |
24h |
LINCSCP_9965 |
LINCSCP_9965 |
A549 |
| 0.200666 |
2.579297e-10 |
975 |
PD-173074 |
LSM-1026 |
FGFR1|FGFR3 |
1uM |
6h |
LINCSCP_12074 |
LINCSCP_12074 |
BT20 |
| -0.200666 |
2.579382e-10 |
975 |
AKT Inhibitor VIII |
LSM-1035 |
AKT1|AKT2 |
10uM |
6h |
LINCSCP_17629 |
LINCSCP_17629 |
HCC15 |
| 0.200656 |
2.584449e-10 |
975 |
SCHEMBL3958507 |
LSM-5245 |
COQ8B|EGFR |
0.12uM |
24h |
LINCSCP_151115 |
LINCSCP_151115 |
PC3 |
| 0.200652 |
2.586636e-10 |
975 |
MK-2206 |
LSM-1057 |
AKT1|AKT2|AKT3 |
0.37uM |
3h |
LINCSCP_145744 |
LINCSCP_145744 |
MDAMB231 |
| 0.200645 |
2.590384e-10 |
975 |
EXALAMIDE |
LSM-45860 |
|
0.04uM |
24h |
LINCSCP_155988 |
LINCSCP_155988 |
PC3 |
| 0.200638 |
2.594107e-10 |
975 |
Dacarbazine |
LSM-5487 |
|
1.11uM |
24h |
LINCSCP_102138 |
LINCSCP_102138 |
HELA |
| 0.200628 |
2.599649e-10 |
975 |
Tremorine |
LSM-2171 |
|
10uM |
6h |
LINCSCP_34359 |
LINCSCP_34359 |
MCF7 |
| -0.200619 |
2.604623e-10 |
975 |
NVP-BHG712 |
LSM-1201 |
|
10uM |
24h |
LINCSCP_150381 |
LINCSCP_150381 |
NPC.TAK |
| -0.200611 |
2.609129e-10 |
975 |
BAY 61-3606 |
LSM-1167 |
SYK |
10uM |
24h |
LINCSCP_89117 |
LINCSCP_89117 |
HA1E |
| 0.200605 |
2.611873e-10 |
975 |
SGX-523 |
LSM-1123 |
MET |
1uM |
6h |
LINCSCP_39550 |
LINCSCP_39550 |
MDAMB231 |
| 0.200591 |
2.619673e-10 |
975 |
C21H29NO |
LSM-1495 |
CHRM1 |
10uM |
6h |
LINCSCP_32966 |
LINCSCP_32966 |
MCF7 |
| -0.200586 |
2.622466e-10 |
975 |
Enzastaurin |
LSM-1069 |
PRKCB |
1.11uM |
24h |
LINCSCP_174907 |
LINCSCP_174907 |
YAPC |
| -0.20058 |
2.625546e-10 |
975 |
Mebendazole |
LSM-3749 |
|
10uM |
24h |
LINCSCP_123129 |
LINCSCP_123129 |
HT29 |
| -0.200563 |
2.635197e-10 |
975 |
KUC111774N |
LSM-36810 |
|
0.5uM |
24h |
LINCSCP_38407 |
LINCSCP_38407 |
MCF7 |
| 0.200562 |
2.635880e-10 |
975 |
BRD-K00664012 |
LSM-37319 |
|
10uM |
6h |
LINCSCP_59559 |
LINCSCP_59559 |
VCAP |
| -0.200558 |
2.637795e-10 |
975 |
AZD4547 |
LSM-6308 |
|
1.11uM |
24h |
LINCSCP_149648 |
LINCSCP_149648 |
NPC.TAK |
| 0.200557 |
2.638159e-10 |
975 |
Penfluridol |
LSM-2334 |
|
1.11uM |
24h |
LINCSCP_104713 |
LINCSCP_104713 |
HELA |
| -0.200546 |
2.644562e-10 |
975 |
GSK429286A |
LSM-1012 |
ROCK1 |
1uM |
6h |
LINCSCP_36569 |
LINCSCP_36569 |
MCF7 |
| 0.200537 |
2.649352e-10 |
975 |
MLS000046849 |
LSM-4081 |
|
10uM |
24h |
LINCSCP_31218 |
LINCSCP_31218 |
MCF7 |
| 0.200537 |
2.649610e-10 |
975 |
BRD-K50696746 |
LSM-7498 |
|
5uM |
24h |
LINCSCP_60387 |
LINCSCP_60387 |
VCAP |
| 0.20052 |
2.658510e-10 |
975 |
BX 912 |
LSM-1055 |
PDK1|PDPK1 |
1.11uM |
24h |
LINCSCP_130687 |
LINCSCP_130687 |
MCF10A |
| -0.200517 |
2.660525e-10 |
975 |
SB 242235 |
LSM-45559 |
|
10uM |
24h |
LINCSCP_154542 |
LINCSCP_154542 |
PC3 |
| -0.200501 |
2.669055e-10 |
975 |
Alisertib |
LSM-37184 |
AURKA |
0.12uM |
24h |
LINCSCP_142899 |
LINCSCP_142899 |
MCF7 |
| -0.200501 |
2.669509e-10 |
975 |
Eplerenone |
LSM-42771 |
NR3C2 |
10uM |
24h |
LINCSCP_72905 |
LINCSCP_72905 |
A375 |
| 0.200492 |
2.674419e-10 |
975 |
AC1MQIYX |
LSM-4693 |
|
10uM |
24h |
LINCSCP_31955 |
LINCSCP_31955 |
MCF7 |
| -0.200489 |
2.675781e-10 |
975 |
BRD-K32628102 |
LSM-39067 |
|
10uM |
24h |
LINCSCP_48955 |
LINCSCP_48955 |
PC3 |
| -0.200482 |
2.679904e-10 |
975 |
Ergothioneine |
LSM-45829 |
|
0.37uM |
24h |
LINCSCP_72420 |
LINCSCP_72420 |
A375 |
| -0.20048 |
2.681182e-10 |
975 |
BRD-A80960055-001-01-7 |
LSM-5162 |
|
10uM |
24h |
LINCSCP_52338 |
LINCSCP_52338 |
SKB |
| -0.200449 |
2.698522e-10 |
975 |
MLS000564806 |
LSM-4368 |
|
10uM |
6h |
LINCSCP_39686 |
LINCSCP_39686 |
MDST8 |
| 0.200441 |
2.703008e-10 |
975 |
Sulfadoxine |
LSM-5657 |
|
0.12uM |
24h |
LINCSCP_73407 |
LINCSCP_73407 |
A375 |
| 0.200433 |
2.707472e-10 |
975 |
3,7-Bis(dimethylamino)phenothiazin-5-ium |
LSM-4555 |
ACHE |
0.5uM |
6h |
LINCSCP_253261 |
LINCSCP_253261 |
MCF7 |
| 0.200431 |
2.708163e-10 |
975 |
BRD-K71031872 |
LSM-12762 |
|
5uM |
6h |
LINCSCP_62573 |
LINCSCP_62573 |
VCAP |
| -0.200429 |
2.709455e-10 |
975 |
SCHEMBL12684744 |
LSM-40288 |
|
10uM |
6h |
LINCSCP_20631 |
LINCSCP_20631 |
HCC515 |
| 0.20042 |
2.714685e-10 |
975 |
Enzalutamide |
LSM-6254 |
AR |
0.1uM |
24h |
LINCSCP_747 |
LINCSCP_747 |
A375 |
| -0.200406 |
2.722716e-10 |
975 |
AC1MEVG9 |
LSM-3935 |
PTPN1 |
10uM |
6h |
LINCSCP_54355 |
LINCSCP_54355 |
SW620 |
| -0.200403 |
2.723949e-10 |
975 |
MLS000778276 |
LSM-43118 |
|
3uM |
6h |
LINCSCP_37320 |
LINCSCP_37320 |
MCF7 |
| 0.200392 |
2.730611e-10 |
975 |
Carbacyclin |
LSM-42923 |
PPARD|PTGIR |
0.5uM |
24h |
LINCSCP_288818 |
LINCSCP_288818 |
U937 |
| -0.200387 |
2.733460e-10 |
975 |
BRD-K55343182 |
LSM-7577 |
|
5uM |
24h |
LINCSCP_60210 |
LINCSCP_60210 |
VCAP |
| -0.200384 |
2.735024e-10 |
975 |
L 168049 |
LSM-2394 |
GCGR |
10uM |
24h |
LINCSCP_25260 |
LINCSCP_25260 |
HT29 |
| -0.200354 |
2.752058e-10 |
975 |
BRD-K74842589 |
LSM-41346 |
|
1uM |
24h |
LINCSCP_66018 |
LINCSCP_66018 |
VCAP |
| -0.200338 |
2.761031e-10 |
975 |
BRD-K19919069 |
LSM-38339 |
|
10uM |
6h |
LINCSCP_65783 |
LINCSCP_65783 |
VCAP |
| -0.200334 |
2.763829e-10 |
975 |
PD-0325901 |
LSM-1101 |
MAP2K1|MAP2K2 |
0.12uM |
24h |
LINCSCP_88926 |
LINCSCP_88926 |
HA1E |
| 0.200309 |
2.777884e-10 |
975 |
MLS000536845 |
LSM-4496 |
|
10uM |
6h |
LINCSCP_217018 |
LINCSCP_217018 |
HCC515 |
| -0.200287 |
2.791001e-10 |
975 |
LY 2183240 |
LSM-2839 |
FAAH |
10uM |
24h |
LINCSCP_30544 |
LINCSCP_30544 |
MCF7 |
| 0.200286 |
2.791307e-10 |
975 |
Zaprinast |
LSM-2259 |
PDE5A |
10uM |
6h |
LINCSCP_34365 |
LINCSCP_34365 |
MCF7 |
| 0.20028 |
2.794771e-10 |
975 |
N-(4-METHOXYPHENYL)-1-PHENYL-1H-PYRAZOL-3-AMINE |
LSM-45685 |
|
0.12uM |
24h |
LINCSCP_123228 |
LINCSCP_123228 |
HT29 |
| -0.200279 |
2.795204e-10 |
975 |
CEP-701 |
LSM-45844 |
|
3.33uM |
24h |
LINCSCP_166431 |
LINCSCP_166431 |
YAPC |
| -0.200278 |
2.796073e-10 |
975 |
Lafutidine |
LSM-45448 |
|
1.11uM |
24h |
LINCSCP_172767 |
LINCSCP_172767 |
YAPC |
| -0.200275 |
2.797434e-10 |
975 |
Sitagliptin |
LSM-5363 |
DPP4 |
1.11uM |
24h |
LINCSCP_136360 |
LINCSCP_136360 |
MCF7 |
| -0.200266 |
2.802798e-10 |
975 |
GSK-1070916 |
LSM-1062 |
AURKB|AURKC |
10uM |
24h |
LINCSCP_165640 |
LINCSCP_165640 |
SKL |
| -0.200253 |
2.810571e-10 |
975 |
5-(6-Aminopurin-9-yl)-2-methyltetrahydrofuran-3-ol |
LSM-4354 |
|
0.37uM |
24h |
LINCSCP_73674 |
LINCSCP_73674 |
A375 |
| -0.200251 |
2.811631e-10 |
975 |
BML-259 |
LSM-6266 |
CDK2|CDK5 |
80uM |
6h |
LINCSCP_51201 |
LINCSCP_51201 |
RMUGS |
| -0.200245 |
2.814989e-10 |
975 |
Erythromycin Ethyl Succinate |
LSM-5056 |
MLNR |
10uM |
24h |
LINCSCP_47272 |
LINCSCP_47272 |
PC3 |
| -0.200245 |
2.815209e-10 |
975 |
SB743921 |
LSM-45775 |
|
0.04uM |
24h |
LINCSCP_160309 |
LINCSCP_160309 |
PC3 |
| -0.200243 |
2.816162e-10 |
975 |
Valdecoxib |
LSM-5305 |
PTGS2 |
100uM |
24h |
LINCSCP_25480 |
LINCSCP_25480 |
HT29 |
| -0.200223 |
2.828195e-10 |
975 |
Rivafurazon |
LSM-3779 |
|
10uM |
24h |
LINCSCP_30301 |
LINCSCP_30301 |
MCF7 |
| -0.20022 |
2.829837e-10 |
975 |
Momelotinib |
LSM-1141 |
JAK1|JAK2 |
3.33uM |
24h |
LINCSCP_69297 |
LINCSCP_69297 |
A375 |
| -0.200208 |
2.836861e-10 |
975 |
ARMODAFINIL |
LSM-45603 |
|
0.04uM |
24h |
LINCSCP_103954 |
LINCSCP_103954 |
HELA |
| -0.200205 |
2.838439e-10 |
975 |
Butoconazole |
LSM-1344 |
|
10uM |
24h |
LINCSCP_71469 |
LINCSCP_71469 |
A375 |
| 0.200197 |
2.843362e-10 |
975 |
Dipyridamole |
LSM-3927 |
ADA|PDE10A|PDE1A|PDE1B|PDE1C|PDE2A|PDE3A|PDE3B|PDE4A|PDE4B|PDE4C|PDE4D|PDE5A|PDE6A|PDE6B|PDE6C|PDE6D|PDE6G|PDE6H|PDE7A|PDE7B|PDE8A|PDE8B|PDE9A|SLC29A1 |
10uM |
6h |
LINCSCP_194207 |
LINCSCP_194207 |
A549 |
| 0.200188 |
2.848486e-10 |
975 |
Dicloxacillin |
LSM-5234 |
|
0.04uM |
24h |
LINCSCP_104877 |
LINCSCP_104877 |
HELA |
| 0.200182 |
2.852528e-10 |
975 |
BRD-A69951442-001-01-3 |
LSM-4466 |
NR3C1 |
10uM |
6h |
LINCSCP_12900 |
LINCSCP_12900 |
EFO27 |
| 0.200163 |
2.863574e-10 |
975 |
SCHEMBL17378613 |
LSM-5749 |
CSF1R |
10uM |
24h |
LINCSCP_129524 |
LINCSCP_129524 |
JURKAT |
| 0.200155 |
2.867991e-10 |
975 |
ZK-93426 |
LSM-3530 |
GABRA1 |
10uM |
24h |
LINCSCP_18001 |
LINCSCP_18001 |
HCC515 |
| -0.200154 |
2.869047e-10 |
975 |
Fedratinib |
LSM-1142 |
FLT3|JAK2 |
3uM |
24h |
LINCSCP_253867 |
LINCSCP_253867 |
MCF7 |
| -0.200145 |
2.874464e-10 |
975 |
BCB03_000734 |
LSM-4718 |
|
10uM |
24h |
LINCSCP_31966 |
LINCSCP_31966 |
MCF7 |
| -0.200132 |
2.882058e-10 |
975 |
MLS002699811 |
LSM-3541 |
|
10uM |
6h |
LINCSCP_1606 |
LINCSCP_1606 |
A375 |
| -0.200102 |
2.899839e-10 |
975 |
BRD-K12182524 |
LSM-37898 |
|
10uM |
6h |
LINCSCP_23144 |
LINCSCP_23144 |
HEPG2 |
| 0.200101 |
2.900649e-10 |
975 |
GW-5074 |
LSM-42779 |
RAF1 |
1uM |
24h |
LINCSCP_36457 |
LINCSCP_36457 |
MCF7 |
| -0.2001 |
2.901498e-10 |
975 |
BSPBIO_000981 |
LSM-43126 |
ACTA1 |
10uM |
6h |
LINCSCP_26487 |
LINCSCP_26487 |
HT29 |
| 0.200098 |
2.902523e-10 |
975 |
Tamatinib |
LSM-1040 |
SYK |
1.11uM |
24h |
LINCSCP_129771 |
LINCSCP_129771 |
LNCAP |
| -0.200094 |
2.904904e-10 |
975 |
13-Hydroxy-8,14,19-trimethoxy-4,10,12,16-tetramethyl-3,20,22-trioxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18-pentaen-9-yl carbamate |
LSM-42815 |
HSP90AA1 |
10uM |
6h |
LINCSCP_66914 |
LINCSCP_66914 |
HCC515 |
| -0.200092 |
2.905992e-10 |
975 |
Manumycin-A |
LSM-43075 |
FNTA|IKBKB |
10uM |
24h |
LINCSCP_158367 |
LINCSCP_158367 |
PC3 |
| -0.200087 |
2.908813e-10 |
975 |
WZ-4-145 |
LSM-42716 |
|
10uM |
6h |
LINCSCP_20547 |
LINCSCP_20547 |
HCC515 |
| 0.200086 |
2.909630e-10 |
975 |
FPA1_000042 |
LSM-36684 |
|
10uM |
6h |
LINCSCP_20266 |
LINCSCP_20266 |
HCC515 |
| -0.200083 |
2.911595e-10 |
975 |
Bendamustine HCl |
LSM-45554 |
|
10uM |
24h |
LINCSCP_153265 |
LINCSCP_153265 |
PC3 |
| -0.200076 |
2.915916e-10 |
975 |
TW 37 |
LSM-6236 |
BCL2|BCL2L1|MCL1 |
10uM |
6h |
LINCSCP_12712 |
LINCSCP_12712 |
COV644 |
| -0.200069 |
2.919888e-10 |
975 |
AZ20 |
LSM-36357 |
|
3.33uM |
24h |
LINCSCP_82391 |
LINCSCP_82391 |
A549 |
| -0.200068 |
2.920431e-10 |
975 |
PHA-665752 |
LSM-42793 |
MET |
0.37uM |
24h |
LINCSCP_162891 |
LINCSCP_162891 |
SKBR3 |
| 0.200063 |
2.923572e-10 |
975 |
TR-14035 |
LSM-45616 |
|
0.04uM |
24h |
LINCSCP_72362 |
LINCSCP_72362 |
A375 |
| -0.20006 |
2.925557e-10 |
975 |
Procaterol |
LSM-1391 |
ADRB2 |
1uM |
6h |
LINCSCP_37971 |
LINCSCP_37971 |
MCF7 |
| 0.200058 |
2.926387e-10 |
975 |
FTI276 |
LSM-4727 |
FNTA |
0.001uM |
24h |
LINCSCP_35714 |
LINCSCP_35714 |
MCF7 |
| -0.200053 |
2.929568e-10 |
975 |
Carfilzomib (PR-171) |
LSM-45547 |
ADRM1|PSMA1|PSMA2|PSMA3|PSMA4|PSMA5|PSMA6|PSMA7|PSMA8|PSMB1|PSMB10|PSMB11|PSMB2|PSMB3|PSMB4|PSMB5|PSMB6|PSMB7|PSMB8|PSMB9|PSMC1|PSMC2|PSMC3|PSMC4|PSMC5|PSMC6|PSMD1|PSMD11|PSMD12|PSMD13|PSMD14|PSMD2|PSMD3|PSMD4|PSMD6|PSMD7|PSMD8|SEM1 |
1.11uM |
24h |
LINCSCP_121495 |
LINCSCP_121495 |
HT29 |
| -0.200049 |
2.931986e-10 |
975 |
936890-98-1 |
LSM-42786 |
MTOR |
0.37uM |
24h |
LINCSCP_99801 |
LINCSCP_99801 |
HCC515 |
| 0.200046 |
2.933884e-10 |
975 |
N-[4-(1-Benzoylpiperidin-4-yl)butyl]-3-pyridin-3-ylpropanamide |
LSM-6279 |
|
0.5uM |
6h |
LINCSCP_51231 |
LINCSCP_51231 |
RMUGS |
| -0.200033 |
2.941853e-10 |
975 |
AC1Q6JJ5 |
LSM-6192 |
TOP2A |
0.1uM |
24h |
LINCSCP_44849 |
LINCSCP_44849 |
PC3 |